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Found 57 with Last Name = 'boteju' and Initial = 'lw'
TargetGalanin receptor type 3(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50187923(1,3-dihydro-1-phenyl-3-[[3-(trilfluoromethyl)pheny...)
Affinity DataKi:  17nMAssay Description:Displacement of [125I]galanin from human GAL3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 3(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50189598(1-(ethylpropyl)-3-{[3-(trifluoromethyl)phenyl]azam...)
Affinity DataKi:  52nMAssay Description:Displacement of [125I]galanin from human GAL3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50187923(1,3-dihydro-1-phenyl-3-[[3-(trilfluoromethyl)pheny...)
Affinity DataKi:  72nMAssay Description:Binding affinity to human 5HT4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 3(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50189596(1-(2-propynyl)-3-{[3-(trifluoromethyl)phenyl]azame...)
Affinity DataKi:  89nMAssay Description:Displacement of [125I]galanin from human GAL3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 3(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50189600((E)-1-allyl-3-(3,4-dichlorophenylimino)indolin-2-o...)
Affinity DataKi:  150nMAssay Description:Displacement of [125I]galanin from human GAL3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 3(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50189597((E)-3-(2,3-dichlorophenylimino)indolin-2-one | CHE...)
Affinity DataKi:  437nMAssay Description:Displacement of [125I]galanin from human GAL3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 3(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50189595(3-{[3-(trifluoromethyl)phenyl]azamethylene}benzo[d...)
Affinity DataKi:  596nMAssay Description:Displacement of [125I]galanin from human GAL3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 3(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50189599((E)-3-(4-chlorophenylimino)indolin-2-one | CHEMBL2...)
Affinity DataKi:  850nMAssay Description:Displacement of [125I]galanin from human GAL3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 3(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50189601((E)-3-(4-methoxyphenylimino)indolin-2-one | (E/Z)-...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [125I]galanin from human GAL3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50029748((2R,3R)-15-(2-Acetylamino-hexanoylamino)-9-benzyl-...)
Affinity DataIC50:  0.5nMAssay Description:The concentration that inhibits 50% specific binding was determined against the Melanocortin 1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50184359((3S,6S,9R,12S,15S,23S)-15-((S)-2-acetylamino-hexan...)
Affinity DataIC50:  0.5nMAssay Description:The concentration that inhibits 50% specific binding was determined against the Melanocortin 1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM21146((3S)-3-[(2S)-2-[(2S)-2-{2-[(2R)-2-[(2S)-2-[(3S)-3-...)
Affinity DataIC50:  0.790nMAssay Description:Binding affinity towards Cholecystokinin type B receptor was determined in guinea pig cortex using [3H]SNF8702 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50280901((S)-3-({1-[(S)-2-(2-Amino-acetylamino)-3-(S)-1H-in...)
Affinity DataIC50:  1.90nMAssay Description:Compound was tested for its binding affinity towards Cholecystokinin type B receptor in cortical membranes (CNS)More data for this Ligand-Target Pair
In DepthDetails Article
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50454019(CHEMBL2370906)
Affinity DataIC50:  2nMAssay Description:The concentration that inhibits 50% specific binding was determined against the Melanocortin 1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50092394((S)-3-((S)-2-{[(S)-2-(2-Amino-acetylamino)-3-(S)-1...)
Affinity DataIC50:  3.30nMAssay Description:Compound was tested for its binding affinity towards Cholecystokinin type B receptor in cortical membranes (CNS)More data for this Ligand-Target Pair
In DepthDetails Article
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50001683(13-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-7...)
Affinity DataIC50:  4.10nMAssay Description:Binding affinity towards Opioid receptor delta 1 was determined in guinea pig wholebrain using [3H][4''-Cl-Phe4]-DPDPE as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM21146((3S)-3-[(2S)-2-[(2S)-2-{2-[(2R)-2-[(2S)-2-[(3S)-3-...)
Affinity DataIC50:  29nMAssay Description:Binding affinity towards Opioid receptor delta 1 was determined in guinea pig wholebrain using [3H][4''-Cl-Phe4]-DPDPE as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50280900(3-((S)-2-{5-[(S)-1-tert-Butoxycarbonylamino-2-(1H-...)
Affinity DataIC50:  37nMAssay Description:Compound was tested for its binding affinity towards Cholecystokinin type A receptor in pancreatic membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50422178(CHEMBL2112688)
Affinity DataIC50:  65nMAssay Description:Binding affinity towards Opioid receptor delta 1 was determined in guinea pig wholebrain using [3H][4''-Cl-Phe4]-DPDPE as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50422175(CHEMBL2112689)
Affinity DataIC50:  88nMAssay Description:Binding affinity towards Cholecystokinin type B receptor was determined in guinea pig cortex using [3H]SNF8702 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50422175(CHEMBL2112689)
Affinity DataIC50:  140nMAssay Description:Binding affinity towards Opioid receptor delta 1 was determined in guinea pig wholebrain using [3H][4''-Cl-Phe4]-DPDPE as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50280904((S)-3-{(S)-2-[(S)-2-(2-Amino-acetylamino)-3-(S)-1H...)
Affinity DataIC50:  169nMAssay Description:Compound was tested for its binding affinity towards Cholecystokinin type B receptor in cortical membranes (CNS)More data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50280903(3-((S)-2-{5-[(S)-1-(2-tert-Butoxycarbonylamino-ace...)
Affinity DataIC50:  364nMAssay Description:Compound was tested for its binding affinity towards Cholecystokinin type A receptor in pancreatic membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetMu-type opioid receptor(GUINEA PIG)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM21146((3S)-3-[(2S)-2-[(2S)-2-{2-[(2R)-2-[(2S)-2-[(3S)-3-...)
Affinity DataIC50:  700nMAssay Description:Binding affinity towards Opioid receptor mu 1 was determined in guinea pig wholebrain using [3H]CTOP radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50422177(CHEMBL2111881)
Affinity DataIC50:  820nMAssay Description:Binding affinity towards Opioid receptor delta 1 was determined in guinea pig wholebrain using [3H][4''-Cl-Phe4]-DPDPE as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Cavia porcellus)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50422178(CHEMBL2112688)
Affinity DataIC50:  1.00E+3nMAssay Description:Binding affinity towards Cholecystokinin type A receptor was determined in guinea pig pancreatic membranes using [125I]-BH-CCK-8 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50422176(CHEMBL2111882)
Affinity DataIC50:  1.05E+3nMAssay Description:Binding affinity towards Opioid receptor delta 1 was determined in guinea pig wholebrain using [3H][4''-Cl-Phe4]-DPDPE as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Cavia porcellus)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50422175(CHEMBL2112689)
Affinity DataIC50: >1.20E+3nMAssay Description:Binding affinity towards Cholecystokinin type A receptor was determined in guinea pig pancreatic membranes using [125I]-BH-CCK-8 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50280900(3-((S)-2-{5-[(S)-1-tert-Butoxycarbonylamino-2-(1H-...)
Affinity DataIC50:  1.88E+3nMAssay Description:Compound was tested for its binding affinity towards Cholecystokinin type B receptor in cortical membranes (CNS)More data for this Ligand-Target Pair
In DepthDetails Article
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50422178(CHEMBL2112688)
Affinity DataIC50:  1.90E+3nMAssay Description:Binding affinity towards Cholecystokinin type B receptor was determined in guinea pig cortex using [3H]SNF8702 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50280904((S)-3-{(S)-2-[(S)-2-(2-Amino-acetylamino)-3-(S)-1H...)
Affinity DataIC50:  2.18E+3nMAssay Description:Compound was tested for its binding affinity towards Cholecystokinin type A receptor in pancreatic membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50280901((S)-3-({1-[(S)-2-(2-Amino-acetylamino)-3-(S)-1H-in...)
Affinity DataIC50:  2.70E+3nMAssay Description:Compound was tested for its binding affinity towards Cholecystokinin type A receptor in pancreatic membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetMu-type opioid receptor(GUINEA PIG)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50422178(CHEMBL2112688)
Affinity DataIC50:  3.05E+3nMAssay Description:Binding affinity towards Opioid receptor mu 1 was determined in guinea pig wholebrain using [3H]CTOP radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50280903(3-((S)-2-{5-[(S)-1-(2-tert-Butoxycarbonylamino-ace...)
Affinity DataIC50:  4.25E+3nMAssay Description:Compound was tested for its binding affinity towards Cholecystokinin type B receptor in cortical membranes (CNS)More data for this Ligand-Target Pair
In DepthDetails Article
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50280898((3S,4R)-3-((S)-2-{5-[(S)-1-(2-Amino-acetylamino)-2...)
Affinity DataIC50:  4.53E+3nMAssay Description:Compound was tested for its binding affinity towards Cholecystokinin type B receptor in cortical membranes (CNS)More data for this Ligand-Target Pair
In DepthDetails Article
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50422177(CHEMBL2111881)
Affinity DataIC50:  6.50E+3nMAssay Description:Binding affinity towards Cholecystokinin type B receptor was determined in guinea pig cortex using [3H]SNF8702 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50422176(CHEMBL2111882)
Affinity DataIC50:  6.50E+3nMAssay Description:Binding affinity towards Cholecystokinin type B receptor was determined in guinea pig cortex using [3H]SNF8702 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50422175(CHEMBL2112689)
Affinity DataIC50:  6.80E+3nMAssay Description:Binding affinity towards Opioid receptor mu 1 was determined in guinea pig wholebrain using [3H]CTOP radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50001683(13-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-7...)
Affinity DataIC50:  7.30E+3nMAssay Description:Binding affinity towards Opioid receptor mu 1 was determined in guinea pig wholebrain using [3H]CTOP radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Cavia porcellus)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50422177(CHEMBL2111881)
Affinity DataIC50:  8.60E+3nMAssay Description:Binding affinity towards Cholecystokinin type A receptor was determined in guinea pig pancreatic membranes using [125I]-BH-CCK-8 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Cavia porcellus)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50422176(CHEMBL2111882)
Affinity DataIC50:  8.60E+3nMAssay Description:Binding affinity towards Cholecystokinin type A receptor was determined in guinea pig pancreatic membranes using [125I]-BH-CCK-8 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50280899((S)-N-((S)-1-Carbamoyl-2-phenyl-ethyl)-3-{(S)-2-[3...)
Affinity DataIC50: >1.00E+4nMAssay Description:Compound was tested for its binding affinity towards Cholecystokinin type B receptor in cortical membranes (CNS)More data for this Ligand-Target Pair
In DepthDetails Article
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50280902(3-{2-Benzyloxycarbonylamino-2-[1-(1-benzyloxycarbo...)
Affinity DataIC50: >1.00E+4nMAssay Description:Compound was tested for its binding affinity towards Cholecystokinin type B receptor in cortical membranes (CNS)More data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50092394((S)-3-((S)-2-{[(S)-2-(2-Amino-acetylamino)-3-(S)-1...)
Affinity DataIC50: >1.00E+4nMAssay Description:Compound was tested for its binding affinity towards Cholecystokinin type A receptor in pancreatic membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50280902(3-{2-Benzyloxycarbonylamino-2-[1-(1-benzyloxycarbo...)
Affinity DataIC50: >1.00E+4nMAssay Description:Compound was tested for its binding affinity towards Cholecystokinin type A receptor in pancreatic membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50280898((3S,4R)-3-((S)-2-{5-[(S)-1-(2-Amino-acetylamino)-2...)
Affinity DataIC50: >1.00E+4nMAssay Description:Compound was tested for its binding affinity towards Cholecystokinin type A receptor in pancreatic membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(Cavia porcellus)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM21146((3S)-3-[(2S)-2-[(2S)-2-{2-[(2R)-2-[(2S)-2-[(3S)-3-...)
Affinity DataIC50: >1.20E+4nMAssay Description:Binding affinity towards Cholecystokinin type A receptor was determined in guinea pig pancreatic membranes using [125I]-BH-CCK-8 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50422177(CHEMBL2111881)
Affinity DataIC50: >3.00E+4nMAssay Description:Binding affinity towards Opioid receptor mu 1 was determined in guinea pig wholebrain using [3H]CTOP radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50422176(CHEMBL2111882)
Affinity DataIC50: >3.00E+4nMAssay Description:Binding affinity towards Opioid receptor mu 1 was determined in guinea pig wholebrain using [3H]CTOP radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50184359((3S,6S,9R,12S,15S,23S)-15-((S)-2-acetylamino-hexan...)
Affinity DataEC50:  0.150nMAssay Description:Effective concentration against Melanocortin 1 receptor transfected into L-cells was determined by concentration of peptide for 50% maximal cAMP gene...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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