Affinity DataKi: 0.0100nMAssay Description:Displacement of [125I]-Ghrelin from human GHSR membranes overexpressing GSH-R1a by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 0.0100nMAssay Description:Displacement of [125I]-Ghrelin from human GHSR membranes overexpressing GSH-R1a by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 0.0380nMAssay Description:Inhibition of collagenase (Matrix metalloprotease-13)More data for this Ligand-Target Pair
Affinity DataKi: 0.0500nMAssay Description:Displacement of [125I]-Ghrelin from human GHSR membranes overexpressing GSH-R1a by scintillation countingMore data for this Ligand-Target Pair
Target72 kDa type IV collagenase(Homo sapiens (Human))
Procter And Gamble Pharmaceuticals
Curated by ChEMBL
Procter And Gamble Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: 0.0830nMAssay Description:Inhibition of gelatinase-A (Matrix metalloprotease-2)More data for this Ligand-Target Pair
Affinity DataKi: 0.100nMAssay Description:Displacement of [125I]-Ghrelin from human GHSR membranes overexpressing GSH-R1a by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 0.160nMAssay Description:Displacement of [125I]-Ghrelin from human GHSR membranes overexpressing GSH-R1a by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 0.200nMAssay Description:Displacement of [125I]-Ghrelin from human GHSR membranes overexpressing GSH-R1a by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 0.200nMAssay Description:Displacement of [125I]-Ghrelin from human GHSR membranes overexpressing GSH-R1a by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 0.260nMAssay Description:Displacement of [125I]-Ghrelin from human GHSR membranes overexpressing GSH-R1a by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 0.270nMAssay Description:Displacement of [125I]-Ghrelin from human GHSR membranes overexpressing GSH-R1a by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 0.270nMAssay Description:Inhibition of Matrix metalloprotease-3More data for this Ligand-Target Pair
Affinity DataKi: 0.300nMAssay Description:Displacement of [125I]-Ghrelin from human GHSR membranes overexpressing GSH-R1a by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 0.400nMAssay Description:Displacement of [125I]-Ghrelin from human GHSR membranes overexpressing GSH-R1a by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 0.5nMAssay Description:Displacement of [125I]-Ghrelin from human GHSR membranes overexpressing GSH-R1a by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 0.600nMAssay Description:Displacement of [125I]-Ghrelin from human GHSR membranes overexpressing GSH-R1a by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 0.640nMAssay Description:Displacement of [125I]SS-14 from human SST3 receptor expressed in CHO cells after 60 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 0.900nMAssay Description:Displacement of [125I]-Ghrelin from human GHSR membranes overexpressing GSH-R1a by scintillation countingMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Acadia Pharmaceuticals
Curated by PDSP Ki Database
Acadia Pharmaceuticals
Curated by PDSP Ki Database
Affinity DataKi: 1.5nMAssay Description:Displacement of [125I]-Ghrelin from human GHSR membranes overexpressing GSH-R1a by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 1.70nMAssay Description:Binding affinity to human SST3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.70nMAssay Description:Displacement of [125I]-Ghrelin from human GHSR membranes overexpressing GSH-R1a by scintillation countingMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Acadia Pharmaceuticals
Curated by PDSP Ki Database
Acadia Pharmaceuticals
Curated by PDSP Ki Database
Affinity DataKi: 1.90nMAssay Description:Displacement of [125I]-Ghrelin from human GHSR membranes overexpressing GSH-R1a by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Displacement of [125I]-Ghrelin from human GHSR membranes overexpressing GSH-R1a by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 2.60nMAssay Description:Displacement of [125I]-Ghrelin from human GHSR membranes overexpressing GSH-R1a by scintillation countingMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Acadia Pharmaceuticals
Curated by PDSP Ki Database
Acadia Pharmaceuticals
Curated by PDSP Ki Database
Affinity DataKi: 3.10nMAssay Description:Displacement of [125I]-Ghrelin from human GHSR membranes overexpressing GSH-R1a by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 3.10nMAssay Description:Displacement of [125I]-Ghrelin from human GHSR membranes overexpressing GSH-R1a by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 3.40nMAssay Description:Displacement of [125I]-Ghrelin from human GHSR membranes overexpressing GSH-R1a by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Displacement of [125I]-Ghrelin from human GHSR membranes overexpressing GSH-R1a by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 5nMAssay Description:Displacement of [125I]-Ghrelin from human GHSR membranes overexpressing GSH-R1a by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 6.60nMAssay Description:Displacement of [125I]-Ghrelin from human GHSR membranes overexpressing GSH-R1a by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 6.70nMAssay Description:Displacement of [125I]-Ghrelin from human GHSR membranes overexpressing GSH-R1a by scintillation countingMore data for this Ligand-Target Pair
TargetInterstitial collagenase(Homo sapiens (Human))
Procter And Gamble Pharmaceuticals
Curated by ChEMBL
Procter And Gamble Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: 8.20nMAssay Description:Inhibition of collagenase-1 (Matrix metalloprotease-1)More data for this Ligand-Target Pair
Target72 kDa type IV collagenase(Homo sapiens (Human))
Procter And Gamble Pharmaceuticals
Curated by ChEMBL
Procter And Gamble Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: 20nMAssay Description:Inhibition of gelatinase-A (Matrix metalloprotease-2)More data for this Ligand-Target Pair
TargetInterstitial collagenase(Homo sapiens (Human))
Procter And Gamble Pharmaceuticals
Curated by ChEMBL
Procter And Gamble Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: 33nMAssay Description:Inhibition of collagenase-1 (Matrix metalloprotease-1)More data for this Ligand-Target Pair
Affinity DataKi: 43nMAssay Description:Inhibition of Matrix metalloprotease-3More data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataKi: 44nMAssay Description:Displacement of radiolabeled MK-499 from human ERG channelMore data for this Ligand-Target Pair
Affinity DataKi: 54nMAssay Description:Inhibition of matrilysin (Matrix metalloprotease-7)More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Acadia Pharmaceuticals
Curated by PDSP Ki Database
Acadia Pharmaceuticals
Curated by PDSP Ki Database
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataKi: 300nMAssay Description:Displacement of radiolabeled MK-499 from human ERG channelMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataKi: 369nMAssay Description:Displacement of radiolabeled MK-499 from human ERG channelMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataKi: 377nMAssay Description:Displacement of radiolabeled MK-499 from human ERG channelMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataKi: 385nMAssay Description:Displacement of radiolabeled MK-499 from human ERG channelMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataKi: 462nMAssay Description:Displacement of radiolabeled MK-499 from human ERG channelMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataKi: 543nMAssay Description:Displacement of radiolabeled MK-499 from human ERG channelMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataKi: 1.40E+3nMAssay Description:Displacement of radiolabeled MK-499 from human ERG channelMore data for this Ligand-Target Pair