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Found 79 with Last Name = 'braga' and Initial = 'r'
TargetFructose-bisphosphate aldolase class 2(Escherichia coli (strain K12))
Université

Curated by ChEMBL
LigandPNGBDBM50167777(2-(hydroxyamino)-2-oxoethyl dihydrogen phosphate |...)
Affinity DataKi:  10nMAssay Description:Inhibitory activity against class II FBP aldolase from Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFructose-bisphosphate aldolase A(Oryctolagus cuniculus)
Université

Curated by ChEMBL
LigandPNGBDBM50167777(2-(hydroxyamino)-2-oxoethyl dihydrogen phosphate |...)
Affinity DataKi:  1.00E+3nMAssay Description:Inhibitory activity against class I FBP aldolase from rabbitMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFructose-bisphosphate aldolase class 2(Escherichia coli (strain K12))
Université

Curated by ChEMBL
LigandPNGBDBM50175712(2-oxo-2-(phenylsulfonamido)ethyl dihydrogen phosph...)
Affinity DataKi:  1.00E+5nMAssay Description:Inhibitory activity against class II FBP aldolase from Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFructose-bisphosphate aldolase class 2(Escherichia coli (strain K12))
Université

Curated by ChEMBL
LigandPNGBDBM50175714(2-(methylsulfonamido)-2-oxoethyl dihydrogen phosph...)
Affinity DataKi:  3.50E+5nMAssay Description:Inhibitory activity against class II FBP aldolase from Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFructose-bisphosphate aldolase class 2(Escherichia coli (strain K12))
Université

Curated by ChEMBL
LigandPNGBDBM50167776((2-Hydroxycarbamoyl-ethyl)-phosphonic acid | 3-(hy...)
Affinity DataKi: >1.00E+6nMAssay Description:Inhibitory activity against class II FBP aldolase from Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFructose-bisphosphate aldolase A(Oryctolagus cuniculus)
Université

Curated by ChEMBL
LigandPNGBDBM50167776((2-Hydroxycarbamoyl-ethyl)-phosphonic acid | 3-(hy...)
Affinity DataKi: >1.00E+6nMAssay Description:Inhibitory activity against class I FBP aldolase from rabbitMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFructose-bisphosphate aldolase A(Oryctolagus cuniculus)
Université

Curated by ChEMBL
LigandPNGBDBM50175713(3-oxo-3-(phenylsulfonamido)propylphosphonic acid |...)
Affinity DataKi: >1.00E+7nMAssay Description:Inhibitory activity against class I FBP aldolase from rabbitMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFructose-bisphosphate aldolase A(Oryctolagus cuniculus)
Université

Curated by ChEMBL
LigandPNGBDBM50175712(2-oxo-2-(phenylsulfonamido)ethyl dihydrogen phosph...)
Affinity DataKi: >1.00E+7nMAssay Description:Inhibitory activity against class I FBP aldolase from rabbitMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFructose-bisphosphate aldolase class 2(Escherichia coli (strain K12))
Université

Curated by ChEMBL
LigandPNGBDBM50175713(3-oxo-3-(phenylsulfonamido)propylphosphonic acid |...)
Affinity DataKi: >1.00E+7nMAssay Description:Inhibitory activity against class II FBP aldolase from Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFructose-bisphosphate aldolase class 2(Escherichia coli (strain K12))
Université

Curated by ChEMBL
LigandPNGBDBM50175715(3-(methylsulfonamido)-3-oxopropylphosphonic acid |...)
Affinity DataKi: >1.00E+7nMAssay Description:Inhibitory activity against class II FBP aldolase from Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFructose-bisphosphate aldolase A(Oryctolagus cuniculus)
Université

Curated by ChEMBL
LigandPNGBDBM50175715(3-(methylsulfonamido)-3-oxopropylphosphonic acid |...)
Affinity DataKi: >1.00E+7nMAssay Description:Inhibitory activity against class I FBP aldolase from rabbitMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFructose-bisphosphate aldolase A(Oryctolagus cuniculus)
Université

Curated by ChEMBL
LigandPNGBDBM50175714(2-(methylsulfonamido)-2-oxoethyl dihydrogen phosph...)
Affinity DataKi: >1.00E+7nMAssay Description:Inhibitory activity against class I FBP aldolase from rabbitMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDihydrofolate reductase(Homo sapiens (Human))
University Of Torino

Curated by ChEMBL
LigandPNGBDBM15339(6-fluoro-2-[4-(2-fluorophenyl)phenyl]-3-methyl-qui...)
Affinity DataIC50:  1.80nMAssay Description:Inhibition of recombinant human N-terminal truncated GST-tagged DHFR (31 to 395 residues) expressed in Escherichia coli BL21(DE3) pyrD using DHO as s...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Argenta Discovery

Curated by ChEMBL
LigandPNGBDBM50198484(5-(5-((2-(benzofuran-4-yl)ethylamino)methyl)pyridi...)
Affinity DataIC50:  4nMAssay Description:Inhibition of HDAC activity measured by HDAC Fluorescent Activity Assay (mean of two experiments)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Argenta Discovery

Curated by ChEMBL
LigandPNGBDBM50198461(5-(5-((2-chlorophenethylamino)methyl)pyridin-2-yl)...)
Affinity DataIC50:  6nMAssay Description:Inhibition of HDAC activity measured by HDAC Fluorescent Activity Assay (mean of two experiments)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Argenta Discovery

Curated by ChEMBL
LigandPNGBDBM50198462(5-(5-((biphenyl-4-ylmethylamino)methyl)pyridin-2-y...)
Affinity DataIC50:  7nMAssay Description:Inhibition of HDAC activity measured by HDAC Fluorescent Activity Assay (mean of two experiments)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Argenta Discovery

Curated by ChEMBL
LigandPNGBDBM50198480(5-(5-((2-chlorobenzylamino)methyl)pyridin-2-yl)-N-...)
Affinity DataIC50:  7nMAssay Description:Inhibition of HDAC activity measured by HDAC Fluorescent Activity Assay (mean of two experiments)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Argenta Discovery

Curated by ChEMBL
LigandPNGBDBM50198469(CHEMBL441699 | N-hydroxy-5-(5-((2-methylphenethyla...)
Affinity DataIC50:  8nMAssay Description:Inhibition of HDAC activity measured by HDAC Fluorescent Activity Assay (mean of two experiments)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Argenta Discovery

Curated by ChEMBL
LigandPNGBDBM50198473(5-(5-((2-(1H-indol-3-yl)ethylamino)methyl)pyridin-...)
Affinity DataIC50:  8nMAssay Description:Inhibition of HDAC activity measured by HDAC Fluorescent Activity Assay (mean of two experiments)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Argenta Discovery

Curated by ChEMBL
LigandPNGBDBM50198475(5-(5-((benzo[d][1,3]dioxol-5-ylmethylamino)methyl)...)
Affinity DataIC50:  8nMAssay Description:Inhibition of HDAC activity measured by HDAC Fluorescent Activity Assay (mean of two experiments)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Argenta Discovery

Curated by ChEMBL
LigandPNGBDBM50198478(5-(5-(2-(benzylamino)ethyl)pyridin-2-yl)-N-hydroxy...)
Affinity DataIC50:  9nMAssay Description:Inhibition of HDAC activity measured by HDAC Fluorescent Activity Assay (mean of two experiments)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Argenta Discovery

Curated by ChEMBL
LigandPNGBDBM50198454(5-(5-((4-chlorobenzylamino)methyl)pyridin-2-yl)-N-...)
Affinity DataIC50:  9nMAssay Description:Inhibition of HDAC activity measured by HDAC Fluorescent Activity Assay (mean of two experiments)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Argenta Discovery

Curated by ChEMBL
LigandPNGBDBM50198472(5-(5-(2-(benzo[d][1,3]dioxol-5-ylmethylamino)ethyl...)
Affinity DataIC50:  9nMAssay Description:Inhibition of HDAC activity measured by HDAC Fluorescent Activity Assay (mean of two experiments)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Argenta Discovery

Curated by ChEMBL
LigandPNGBDBM50198470(CHEMBL436964 | N-hydroxy-5-(5-((3-methylphenethyla...)
Affinity DataIC50:  9nMAssay Description:Inhibition of HDAC activity measured by HDAC Fluorescent Activity Assay (mean of two experiments)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Argenta Discovery

Curated by ChEMBL
LigandPNGBDBM50198463(5-(5-((4-fluorophenethylamino)methyl)pyridin-2-yl)...)
Affinity DataIC50:  9nMAssay Description:Inhibition of HDAC activity measured by HDAC Fluorescent Activity Assay (mean of two experiments)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Argenta Discovery

Curated by ChEMBL
LigandPNGBDBM50198465(CHEMBL387247 | N-hydroxy-5-(5-((2-phenoxyethylamin...)
Affinity DataIC50:  11nMAssay Description:Inhibition of HDAC activity measured by HDAC Fluorescent Activity Assay (mean of two experiments)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Argenta Discovery

Curated by ChEMBL
LigandPNGBDBM50198453(5-(5-(((2,3-dihydrobenzo[b][1,4]dioxin-6-yl)methyl...)
Affinity DataIC50:  11nMAssay Description:Inhibition of HDAC activity measured by HDAC Fluorescent Activity Assay (mean of two experiments)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Argenta Discovery

Curated by ChEMBL
LigandPNGBDBM50198455(CHEMBL217531 | N-hydroxy-5-(5-((phenethylamino)met...)
Affinity DataIC50:  12nMAssay Description:Inhibition of HDAC activity measured by HDAC Fluorescent Activity Assay (mean of two experiments)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Argenta Discovery

Curated by ChEMBL
LigandPNGBDBM50198466(5-(5-((2-fluorophenethylamino)methyl)pyridin-2-yl)...)
Affinity DataIC50:  12nMAssay Description:Inhibition of HDAC activity measured by HDAC Fluorescent Activity Assay (mean of two experiments)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Argenta Discovery

Curated by ChEMBL
LigandPNGBDBM50198464(5-(5-(2-(4-fluorobenzylamino)ethyl)pyridin-2-yl)-N...)
Affinity DataIC50:  13nMAssay Description:Inhibition of HDAC activity measured by HDAC Fluorescent Activity Assay (mean of two experiments)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Argenta Discovery

Curated by ChEMBL
LigandPNGBDBM50198468(CHEMBL216896 | N-hydroxy-5-(5-((4-methylphenethyla...)
Affinity DataIC50:  14nMAssay Description:Inhibition of HDAC activity measured by HDAC Fluorescent Activity Assay (mean of two experiments)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Argenta Discovery

Curated by ChEMBL
LigandPNGBDBM50198483(5-(5-((benzylamino)methyl)pyridin-2-yl)-N-hydroxyt...)
Affinity DataIC50:  16nMAssay Description:Inhibition of HDAC activity measured by HDAC Fluorescent Activity Assay (mean of two experiments)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDihydrofolate reductase(Homo sapiens (Human))
University Of Torino

Curated by ChEMBL
LigandPNGBDBM50235594(CHEMBL4105330)
Affinity DataIC50:  16nMAssay Description:Inhibition of recombinant human N-terminal truncated GST-tagged DHFR (31 to 395 residues) expressed in Escherichia coli BL21(DE3) pyrD using DHO as s...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Argenta Discovery

Curated by ChEMBL
LigandPNGBDBM50198474(CHEMBL263570 | N-hydroxy-5-(5-((phenylamino)methyl...)
Affinity DataIC50:  16nMAssay Description:Inhibition of HDAC activity measured by HDAC Fluorescent Activity Assay (mean of two experiments)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Argenta Discovery

Curated by ChEMBL
LigandPNGBDBM50198458(CHEMBL385934 | N-hydroxy-5-(5-((2-methoxyphenethyl...)
Affinity DataIC50:  17nMAssay Description:Inhibition of HDAC activity measured by HDAC Fluorescent Activity Assay (mean of two experiments)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDihydrofolate reductase(Homo sapiens (Human))
University Of Torino

Curated by ChEMBL
LigandPNGBDBM50235596(CHEMBL4098306)
Affinity DataIC50:  18nMAssay Description:Inhibition of recombinant human N-terminal truncated GST-tagged DHFR (31 to 395 residues) expressed in Escherichia coli BL21(DE3) pyrD using DHO as s...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Argenta Discovery

Curated by ChEMBL
LigandPNGBDBM50198456(CHEMBL217529 | N-hydroxy-5-(5-((3-phenylpropylamin...)
Affinity DataIC50:  18nMAssay Description:Inhibition of HDAC activity measured by HDAC Fluorescent Activity Assay (mean of two experiments)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Argenta Discovery

Curated by ChEMBL
LigandPNGBDBM50198218(5-(1-(2-(benzo[d][1,3]dioxol-5-ylmethylamino)ethyl...)
Affinity DataIC50:  29nMAssay Description:Inhibition of HDAC activity measured by HDAC Fluorescent Activity Assay (mean of two experiments)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Argenta Discovery

Curated by ChEMBL
LigandPNGBDBM50198482(5-(5-((3,4-dihydroisoquinolin-2(1H)-yl)methyl)pyri...)
Affinity DataIC50:  30nMAssay Description:Inhibition of HDAC activity measured by HDAC Fluorescent Activity Assay (mean of two experiments)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Argenta Discovery

Curated by ChEMBL
LigandPNGBDBM50198471(CHEMBL279353 | N-hydroxy-5-(5-(2-(phenethylamino)e...)
Affinity DataIC50:  31nMAssay Description:Inhibition of HDAC activity measured by HDAC Fluorescent Activity Assay (mean of two experiments)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Argenta Discovery

Curated by ChEMBL
LigandPNGBDBM50198459(5-(5-((benzyl(methyl)amino)methyl)pyridin-2-yl)-N-...)
Affinity DataIC50:  35nMAssay Description:Inhibition of HDAC activity measured by HDAC Fluorescent Activity Assay (mean of two experiments)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDihydrofolate reductase(Homo sapiens (Human))
University Of Torino

Curated by ChEMBL
LigandPNGBDBM50235589(CHEMBL4090575)
Affinity DataIC50:  36nMAssay Description:Inhibition of recombinant human N-terminal truncated GST-tagged DHFR (31 to 395 residues) expressed in Escherichia coli BL21(DE3) pyrD using DHO as s...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDihydrofolate reductase(Homo sapiens (Human))
University Of Torino

Curated by ChEMBL
LigandPNGBDBM50235597(CHEMBL4088968)
Affinity DataIC50:  41nMAssay Description:Inhibition of recombinant human N-terminal truncated GST-tagged DHFR (31 to 395 residues) expressed in Escherichia coli BL21(DE3) pyrD using DHO as s...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDihydrofolate reductase(Homo sapiens (Human))
University Of Torino

Curated by ChEMBL
LigandPNGBDBM50235595(CHEMBL4081077)
Affinity DataIC50:  44nMAssay Description:Inhibition of recombinant human N-terminal truncated GST-tagged DHFR (31 to 395 residues) expressed in Escherichia coli BL21(DE3) pyrD using DHO as s...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDihydrofolate reductase(Homo sapiens (Human))
University Of Torino

Curated by ChEMBL
LigandPNGBDBM50235593(CHEMBL4062046)
Affinity DataIC50:  45nMAssay Description:Inhibition of recombinant human N-terminal truncated GST-tagged DHFR (31 to 395 residues) expressed in Escherichia coli BL21(DE3) pyrD using DHO as s...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Argenta Discovery

Curated by ChEMBL
LigandPNGBDBM50198457(CHEMBL425971 | N-hydroxy-5-(5-(phenethylamino)pyri...)
Affinity DataIC50:  80nMAssay Description:Inhibition of HDAC activity measured by HDAC Fluorescent Activity Assay (mean of two experiments)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThioredoxin glutathione reductase(Schistosoma mansoni)
Universidade Federal De Goi£S

Curated by ChEMBL
LigandPNGBDBM50532918(CHEMBL1325877)
Affinity DataIC50:  100nMAssay Description:Inhibition of Schistosoma mansoni TGRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThioredoxin glutathione reductase(Schistosoma mansoni)
Universidade Federal De Goi£S

Curated by ChEMBL
LigandPNGBDBM50532918(CHEMBL1325877)
Affinity DataIC50:  100nMAssay Description:Inhibition of Schistosoma mansoni TGRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDihydrofolate reductase(Homo sapiens (Human))
University Of Torino

Curated by ChEMBL
LigandPNGBDBM50235590(CHEMBL4071260)
Affinity DataIC50:  108nMAssay Description:Inhibition of recombinant human N-terminal truncated GST-tagged DHFR (31 to 395 residues) expressed in Escherichia coli BL21(DE3) pyrD using DHO as s...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Argenta Discovery

Curated by ChEMBL
LigandPNGBDBM19149(CHEMBL98 | N-hydroxy-N'-phenyloctanediamide | SAHA...)
Affinity DataIC50:  125nMAssay Description:Inhibition of HDAC activity measured by HDAC Fluorescent Activity Assay (mean of two experiments)More data for this Ligand-Target Pair
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