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Found 40 with Last Name = 'brinen' and Initial = 'ls'
TargetCruzipain(Trypanosoma cruzi)
University Of California

Curated by ChEMBL
LigandPNGBDBM50306596(3-(4-((S)-4-methyl-2-(quinolin-6-ylmethylamino)pen...)
Affinity DataKi:  100nMAssay Description:Inhibition of Trypanosoma cruzi cruzainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCruzipain(Trypanosoma cruzi)
University Of California

Curated by ChEMBL
LigandPNGBDBM50306600(3-(4-((S)-1-cyclopentyl-1-(quinolin-6-ylmethylamin...)
Affinity DataKi:  110nMAssay Description:Inhibition of Trypanosoma cruzi cruzainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCruzipain(Trypanosoma cruzi)
University Of California

Curated by ChEMBL
LigandPNGBDBM50306598(3-(4-((S)-1-cyclobutyl-1-(quinolin-6-ylmethylamino...)
Affinity DataKi:  130nMAssay Description:Inhibition of Trypanosoma cruzi cruzainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCruzipain(Trypanosoma cruzi)
University Of California

Curated by ChEMBL
LigandPNGBDBM50306597(3-(4-((S)-4-methyl-2-(quinolin-6-ylmethylamino)pen...)
Affinity DataKi:  190nMAssay Description:Inhibition of Trypanosoma cruzi cruzainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
University Of California

Curated by ChEMBL
LigandPNGBDBM50311245((S)-4-methyl-2-phenyl-N-(5-phenyl-1-(phenylsulfony...)
Affinity DataKi:  320nMAssay Description:Inhibition of Trypanosoma brucei rhodesiense rhodesain preincubated after 5 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCruzipain(Trypanosoma cruzi)
University Of California

Curated by ChEMBL
LigandPNGBDBM50306599(3-(4-((S)-1-cyclobutyl-1-(quinolin-6-ylmethylamino...)
Affinity DataKi:  350nMAssay Description:Inhibition of Trypanosoma cruzi cruzainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCruzipain(Trypanosoma cruzi)
University Of California

Curated by ChEMBL
LigandPNGBDBM50306592(3-(4-((S)-3-methyl-2-(quinolin-6-ylmethylamino)but...)
Affinity DataKi:  460nMAssay Description:Inhibition of Trypanosoma cruzi cruzainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCruzipain(Trypanosoma cruzi)
University Of California

Curated by ChEMBL
LigandPNGBDBM50306595(3-(4-((S)-1-cyclopropyl-1-(quinolin-6-ylmethylamin...)
Affinity DataKi:  940nMAssay Description:Inhibition of Trypanosoma cruzi cruzainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCruzipain(Trypanosoma cruzi)
University Of California

Curated by ChEMBL
LigandPNGBDBM50306593(3-(4-((S)-3-methyl-2-(quinolin-6-ylmethylamino)but...)
Affinity DataKi:  1.04E+3nMAssay Description:Inhibition of Trypanosoma cruzi cruzainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCruzipain(Trypanosoma cruzi)
University Of California

Curated by ChEMBL
LigandPNGBDBM50306601(3-(4-((S)-1-cyclohexyl-1-(quinolin-6-ylmethylamino...)
Affinity DataKi:  1.22E+3nMAssay Description:Inhibition of Trypanosoma cruzi cruzainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCruzipain(Trypanosoma cruzi)
University Of California

Curated by ChEMBL
LigandPNGBDBM50306594(3-(4-((S)-3-methyl-2-(quinolin-6-ylmethylamino)but...)
Affinity DataKi:  6.76E+3nMAssay Description:Inhibition of Trypanosoma cruzi cruzainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCruzipain(Trypanosoma cruzi)
University Of California

Curated by ChEMBL
LigandPNGBDBM50229129(4-Methyl-piperazine-1-carboxylic acid [(S)-1-((E)-...)
Affinity DataIC50:  4nMAssay Description:Inhibition of Trypanosoma cruzi cruzain after 5 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
University Of California

Curated by ChEMBL
LigandPNGBDBM50229129(4-Methyl-piperazine-1-carboxylic acid [(S)-1-((E)-...)
Affinity DataIC50:  7nMAssay Description:Inhibition of Trypanosoma brucei rhodesiense rhodesain preincubated after 5 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
University Of California

Curated by ChEMBL
LigandPNGBDBM50311248((S)-3-phenyl-N-(5-phenyl-1-(phenylsulfonyl)pent-1-...)
Affinity DataIC50:  10nMAssay Description:Inhibition of Trypanosoma brucei rhodesiense rhodesain preincubated after 5 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
University Of California

Curated by ChEMBL
LigandPNGBDBM50311250((S)-N-(5-phenyl-1-(phenylsulfonyl)pent-1-en-3-yl)-...)
Affinity DataIC50:  10nMAssay Description:Inhibition of Trypanosoma brucei rhodesiense rhodesain preincubated after 5 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
University Of California

Curated by ChEMBL
LigandPNGBDBM50311247((S)-4-methyl-N-(5-phenyl-1-(phenylsulfonyl)pent-1-...)
Affinity DataIC50:  10nMAssay Description:Inhibition of Trypanosoma brucei rhodesiense rhodesain preincubated after 5 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
University Of California

Curated by ChEMBL
LigandPNGBDBM50311246((S)-4-methyl-N-(5-phenyl-1-(phenylsulfonyl)pent-1-...)
Affinity DataIC50:  30nMAssay Description:Inhibition of Trypanosoma brucei rhodesiense rhodesain preincubated after 5 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
University Of California

Curated by ChEMBL
LigandPNGBDBM50311251((S)-N-(5-phenyl-1-(phenylsulfonyl)pent-1-en-3-yl)-...)
Affinity DataIC50:  50nMAssay Description:Inhibition of Trypanosoma brucei rhodesiense rhodesain preincubated after 5 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
University Of California

Curated by ChEMBL
LigandPNGBDBM50311249((S)-N-(5-phenyl-1-(phenylsulfonyl)pent-1-en-3-yl)-...)
Affinity DataIC50:  50nMAssay Description:Inhibition of Trypanosoma brucei rhodesiense rhodesain preincubated after 5 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCruzipain(Trypanosoma cruzi)
University Of California

Curated by ChEMBL
LigandPNGBDBM50311252((1R,2R)-2-(4-chlorobenzoyl)-N-((S)-5-phenyl-1-(phe...)
Affinity DataIC50:  50nMAssay Description:Inhibition of Trypanosoma cruzi cruzain after 5 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
University Of California

Curated by ChEMBL
LigandPNGBDBM50311252((1R,2R)-2-(4-chlorobenzoyl)-N-((S)-5-phenyl-1-(phe...)
Affinity DataIC50:  100nMAssay Description:Inhibition of Trypanosoma brucei rhodesiense rhodesain preincubated after 5 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCruzipain(Trypanosoma cruzi)
University Of California

Curated by ChEMBL
LigandPNGBDBM50311250((S)-N-(5-phenyl-1-(phenylsulfonyl)pent-1-en-3-yl)-...)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of Trypanosoma cruzi cruzain after 5 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCruzipain(Trypanosoma cruzi)
University Of California

Curated by ChEMBL
LigandPNGBDBM50311247((S)-4-methyl-N-(5-phenyl-1-(phenylsulfonyl)pent-1-...)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of Trypanosoma cruzi cruzain after 5 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCruzipain(Trypanosoma cruzi)
University Of California

Curated by ChEMBL
LigandPNGBDBM50311248((S)-3-phenyl-N-(5-phenyl-1-(phenylsulfonyl)pent-1-...)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of Trypanosoma cruzi cruzain after 5 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCruzipain(Trypanosoma cruzi)
University Of California

Curated by ChEMBL
LigandPNGBDBM50311246((S)-4-methyl-N-(5-phenyl-1-(phenylsulfonyl)pent-1-...)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of Trypanosoma cruzi cruzain after 5 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin B-like cysteine protease(Trypanosoma brucei)
University Of California

Curated by ChEMBL
LigandPNGBDBM50229129(4-Methyl-piperazine-1-carboxylic acid [(S)-1-((E)-...)
Affinity DataIC50:  4.00E+3nMAssay Description:Inhibition of Trypanosoma brucei Cathepsin B-like protease after 5 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCruzipain(Trypanosoma cruzi)
University Of California

Curated by ChEMBL
LigandPNGBDBM50311249((S)-N-(5-phenyl-1-(phenylsulfonyl)pent-1-en-3-yl)-...)
Affinity DataIC50:  5.00E+3nMAssay Description:Inhibition of Trypanosoma cruzi cruzain after 5 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCruzipain(Trypanosoma cruzi)
University Of California

Curated by ChEMBL
LigandPNGBDBM50311251((S)-N-(5-phenyl-1-(phenylsulfonyl)pent-1-en-3-yl)-...)
Affinity DataIC50:  6.00E+3nMAssay Description:Inhibition of Trypanosoma cruzi cruzain after 5 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCruzipain(Trypanosoma cruzi)
University Of California

Curated by ChEMBL
LigandPNGBDBM50311245((S)-4-methyl-2-phenyl-N-(5-phenyl-1-(phenylsulfony...)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibition of Trypanosoma cruzi cruzain after 5 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin B-like cysteine protease(Trypanosoma brucei)
University Of California

Curated by ChEMBL
LigandPNGBDBM50311252((1R,2R)-2-(4-chlorobenzoyl)-N-((S)-5-phenyl-1-(phe...)
Affinity DataIC50:  1.60E+4nMAssay Description:Inhibition of Trypanosoma brucei Cathepsin B-like protease after 5 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin B-like cysteine protease(Trypanosoma brucei)
University Of California

Curated by ChEMBL
LigandPNGBDBM50311248((S)-3-phenyl-N-(5-phenyl-1-(phenylsulfonyl)pent-1-...)
Affinity DataIC50:  4.00E+4nMAssay Description:Inhibition of Trypanosoma brucei Cathepsin B-like protease after 5 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
University Of California

Curated by ChEMBL
LigandPNGBDBM50311253((1S,2S)-2-(4-chlorobenzoyl)-N-((S,E)-5-phenyl-1-(p...)
Affinity DataIC50:  5.60E+4nMAssay Description:Inhibition of Trypanosoma brucei rhodesiense rhodesain preincubated after 5 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin B-like cysteine protease(Trypanosoma brucei)
University Of California

Curated by ChEMBL
LigandPNGBDBM50311250((S)-N-(5-phenyl-1-(phenylsulfonyl)pent-1-en-3-yl)-...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of Trypanosoma brucei Cathepsin B-like protease after 5 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin B-like cysteine protease(Trypanosoma brucei)
University Of California

Curated by ChEMBL
LigandPNGBDBM50311249((S)-N-(5-phenyl-1-(phenylsulfonyl)pent-1-en-3-yl)-...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of Trypanosoma brucei Cathepsin B-like protease after 5 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin B-like cysteine protease(Trypanosoma brucei)
University Of California

Curated by ChEMBL
LigandPNGBDBM50311253((1S,2S)-2-(4-chlorobenzoyl)-N-((S,E)-5-phenyl-1-(p...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of Trypanosoma brucei Cathepsin B-like protease after 5 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCruzipain(Trypanosoma cruzi)
University Of California

Curated by ChEMBL
LigandPNGBDBM50311253((1S,2S)-2-(4-chlorobenzoyl)-N-((S,E)-5-phenyl-1-(p...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of Trypanosoma cruzi cruzain after 5 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin B-like cysteine protease(Trypanosoma brucei)
University Of California

Curated by ChEMBL
LigandPNGBDBM50311245((S)-4-methyl-2-phenyl-N-(5-phenyl-1-(phenylsulfony...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of Trypanosoma brucei Cathepsin B-like protease after 5 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin B-like cysteine protease(Trypanosoma brucei)
University Of California

Curated by ChEMBL
LigandPNGBDBM50311246((S)-4-methyl-N-(5-phenyl-1-(phenylsulfonyl)pent-1-...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of Trypanosoma brucei Cathepsin B-like protease after 5 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin B-like cysteine protease(Trypanosoma brucei)
University Of California

Curated by ChEMBL
LigandPNGBDBM50311251((S)-N-(5-phenyl-1-(phenylsulfonyl)pent-1-en-3-yl)-...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of Trypanosoma brucei Cathepsin B-like protease after 5 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin B-like cysteine protease(Trypanosoma brucei)
University Of California

Curated by ChEMBL
LigandPNGBDBM50311247((S)-4-methyl-N-(5-phenyl-1-(phenylsulfonyl)pent-1-...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of Trypanosoma brucei Cathepsin B-like protease after 5 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed