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Found 14 with Last Name = 'burnelli' and Initial = 's'
TargetCholinesterase(Equus caballus (Horse))
Università

Curated by ChEMBL
LigandPNGBDBM8961(1,2,3,4-tetrahydro-9-acridinamine | 1,2,3,4-tetrah...)
Affinity DataIC50:  4nMAssay Description:Inhibition of horse serum butyrylcholine esterase in presence of acetylcholine substrate by chemiluminescent assayChecked by AuthorMore data for this Ligand-Target Pair
TargetCarboxylic ester hydrolase(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM8961(1,2,3,4-tetrahydro-9-acridinamine | 1,2,3,4-tetrah...)
Affinity DataIC50:  9nMAssay Description:Inhibition of rat plasma butyrylcholine esterase in presence of butyrylcholine substrate by chemiluminescent assayChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM8960((+/-)-2-[(1-benzylpiperidin-4-yl)methyl]-5,6-dimet...)
Affinity DataIC50:  40nMAssay Description:Inhibition of rat brain acetylcholine esterase in presence of acetylcholine substrate by chemiluminescent assayChecked by AuthorMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM8961(1,2,3,4-tetrahydro-9-acridinamine | 1,2,3,4-tetrah...)
Affinity DataIC50:  200nMAssay Description:Inhibition of rat brain acetylcholine esterase in presence of acetylcholine substrate by chemiluminescent assayChecked by AuthorMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
University Of Bologna

Curated by ChEMBL
LigandPNGBDBM50071171(9-Methoxy-2-methyl-11,12-dihydro-3H,6aH,13H-6-oxa-...)
Affinity DataIC50: >1.00E+3nMAssay Description:Antagonist activity at human muscarinic M4 receptor expressed in CHO cells assessed as blockade of carbachol-induced inhibition of forskolin-stimulat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
University Of Bologna

Curated by ChEMBL
LigandPNGBDBM50376590(CHEMBL402207)
Affinity DataIC50: >1.00E+3nMAssay Description:Antagonist activity at human muscarinic M4 receptor expressed in CHO cells assessed as blockade of carbachol-induced inhibition of forskolin-stimulat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Equus caballus (Horse))
Università

Curated by ChEMBL
LigandPNGBDBM8960((+/-)-2-[(1-benzylpiperidin-4-yl)methyl]-5,6-dimet...)
Affinity DataIC50:  2.70E+3nMAssay Description:Inhibition of horse serum butyrylcholine esterase in presence of acetylcholine substrate by chemiluminescent assayChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Università

Curated by ChEMBL
LigandPNGBDBM50270498(1-benzoyl-3-((6-chloroimidazo[2,1-b]thiazol-5-yl)m...)
Affinity DataIC50:  4.20E+3nMAssay Description:Inhibition of electric eel acetylcholine esterase type V-S in presence of acetylcholine substrate by chemiluminescent assayChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxylic ester hydrolase(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM8960((+/-)-2-[(1-benzylpiperidin-4-yl)methyl]-5,6-dimet...)
Affinity DataIC50:  5.30E+3nMAssay Description:Inhibition of rat plasma butyrylcholine esterase in presence of butyrylcholine substrate by chemiluminescent assayChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Università

Curated by ChEMBL
LigandPNGBDBM50270499(1-acetyl-3-((6-methylimidazo[2,1-b]thiazol-5-yl)me...)
Affinity DataIC50:  3.50E+4nMAssay Description:Inhibition of electric eel acetylcholine esterase type V-S in presence of acetylcholine substrate by chemiluminescent assayChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Università

Curated by ChEMBL
LigandPNGBDBM50270497(1-acetyl-3-((6-chloroimidazo[2,1-b]thiazol-5-yl)me...)
Affinity DataIC50:  6.00E+4nMAssay Description:Inhibition of electric eel acetylcholine esterase type V-S in presence of acetylcholine substrate by chemiluminescent assayChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
University Of Bologna

Curated by ChEMBL
LigandPNGBDBM50376590(CHEMBL402207)
Affinity DataEC50:  67nMAssay Description:Antagonist activity at human muscarinic M4 receptor expressed in CHO cells assessed as blockade of carbachol-induced inhibition of forskolin-stimulat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
University Of Bologna

Curated by ChEMBL
LigandPNGBDBM50376591(CHEMBL403773)
Affinity DataEC50:  138nMAssay Description:Antagonist activity at human muscarinic M4 receptor expressed in CHO cells assessed as blockade of carbachol-induced inhibition of forskolin-stimulat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
University Of Bologna

Curated by ChEMBL
LigandPNGBDBM50071171(9-Methoxy-2-methyl-11,12-dihydro-3H,6aH,13H-6-oxa-...)
Affinity DataEC50:  54nMAssay Description:Antagonist activity at human muscarinic M4 receptor expressed in CHO cells assessed as blockade of carbachol-induced inhibition of forskolin-stimulat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed