Affinity DataKi: 0.240nMpH: 6.8Assay Description:Inhibition of human MMP12 catalytic domain (98 to 266) at pH 6.8 by isothermal titration calorimetryMore data for this Ligand-Target Pair
Affinity DataKi: 0.260nMAssay Description:Binding affinity to human MMP12 catalytic domain (98 to 266) by isothermal titration calorimetryMore data for this Ligand-Target Pair
Affinity DataKi: 0.280nMAssay Description:Binding affinity to human MMP12 catalytic domain (98 to 266) by isothermal titration calorimetryMore data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Inhibition of MMP13 by fluorimetric assayMore data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Inhibition of MMP12 (unknown origin)-mediated Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 by fluorimetric assayMore data for this Ligand-Target Pair
Affinity DataKi: 1.70nMAssay Description:Inhibition of MMP13 by fluorimetric assayMore data for this Ligand-Target Pair
Affinity DataKi: 1.70nMAssay Description:Inhibition of MMP13 by fluorimetric assayMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Inhibition of MMP12 (unknown origin)-mediated Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 by fluorimetric assayMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Inhibition of MMP12 (unknown origin)-mediated Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 by fluorimetric assayMore data for this Ligand-Target Pair
Affinity DataKi: 2.20nMAssay Description:Inhibition of MMP13 by fluorimetric assayMore data for this Ligand-Target Pair
Affinity DataKi: 2.70nMAssay Description:Inhibition of MMP13 by fluorimetric assayMore data for this Ligand-Target Pair
Affinity DataKi: 2.90nMAssay Description:Inhibition of MMP13 by fluorimetric assayMore data for this Ligand-Target Pair
Affinity DataKi: 3.10nMAssay Description:Inhibition of MMP13 by fluorimetric assayMore data for this Ligand-Target Pair
Affinity DataKi: 3.60nMAssay Description:Inhibition of MMP13 by fluorimetric assayMore data for this Ligand-Target Pair
Affinity DataKi: 4.30nMAssay Description:Inhibition of MMP12 by fluorimetric assayMore data for this Ligand-Target Pair
Affinity DataKi: 4.60nMAssay Description:Inhibition of MMP8 by fluorimetric assayMore data for this Ligand-Target Pair
Affinity DataKi: 5nMAssay Description:Inhibition of MMP12 (unknown origin)-mediated Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 by fluorimetric assayMore data for this Ligand-Target Pair
Affinity DataKi: 5nMAssay Description:Inhibition of MMP12 (unknown origin)-mediated Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 by fluorimetric assayMore data for this Ligand-Target Pair
Affinity DataKi: 5.70nMAssay Description:Inhibition of human carbonic anhydrase 12 incubated for 15 mins prior to testing by stopped flow CO2 hydrase assayMore data for this Ligand-Target Pair
Affinity DataKi: 6nMAssay Description:Inhibition of MMP12 by fluorimetric assayMore data for this Ligand-Target Pair
Affinity DataKi: 6nMAssay Description:Inhibition of MMP12 (unknown origin)-mediated Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 by fluorimetric assayMore data for this Ligand-Target Pair
Affinity DataKi: 7nMAssay Description:Inhibition of MMP12 by fluorimetric assayMore data for this Ligand-Target Pair
Affinity DataKi: 7nMAssay Description:Inhibition of MMP12 (unknown origin)-mediated Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 by fluorimetric assayMore data for this Ligand-Target Pair
Affinity DataKi: 7.60nMAssay Description:Inhibition of MMP12 by fluorimetric assayMore data for this Ligand-Target Pair
Affinity DataKi: 8nMAssay Description:Inhibition of MMP8 by fluorimetric assayMore data for this Ligand-Target Pair
Affinity DataKi: 8nMAssay Description:Inhibition of MMP12 by fluorimetric assayMore data for this Ligand-Target Pair
Affinity DataKi: 9nMAssay Description:Inhibition of MMP8 by fluorimetric assayMore data for this Ligand-Target Pair
Affinity DataKi: 9nMAssay Description:Inhibition of MMP12 (unknown origin)-mediated Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 by fluorimetric assayMore data for this Ligand-Target Pair
Affinity DataKi: 9nMAssay Description:Inhibition of MMP8 by fluorimetric assayMore data for this Ligand-Target Pair
Affinity DataKi: 9.10nMAssay Description:Inhibition of MMP8 by fluorimetric assayMore data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Inhibition of MMP8 by fluorimetric assayMore data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Inhibition of MMP12 (unknown origin)-mediated Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 by fluorimetric assayMore data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Inhibition of MMP12 (unknown origin)-mediated Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 by fluorimetric assayMore data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:Inhibition of MMP12 by fluorimetric assayMore data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:Inhibition of MMP8 by fluorimetric assayMore data for this Ligand-Target Pair
Affinity DataKi: 14.3nMAssay Description:Inhibition of MMP12 by fluorimetric assayMore data for this Ligand-Target Pair
Affinity DataKi: 15nMAssay Description:Binding affinity to human MMP12 catalytic domain (98 to 266) by isothermal titration calorimetryMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2(Rattus norvegicus (Rat))
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Curated by ChEMBL
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Curated by ChEMBL
Affinity DataKi: 15nMAssay Description:Displacement of [3H]flumazenil from rat GABAA alpha1beta2gamma2 expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 15nMAssay Description:Inhibition of MMP12 (unknown origin)-mediated Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 by fluorimetric assayMore data for this Ligand-Target Pair
Affinity DataKi: 16nMAssay Description:Inhibition of MMP12 (unknown origin)-mediated Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 by fluorimetric assayMore data for this Ligand-Target Pair
Affinity DataKi: 16nMAssay Description:Binding affinity to human MMP12 catalytic domain (98 to 266) by isothermal titration calorimetryMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2(Rattus norvegicus (Rat))
Università
Curated by ChEMBL
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Curated by ChEMBL
Affinity DataKi: 17nMAssay Description:Displacement of [3H]flumazenil from rat GABAA alpha1beta2gamma2 expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 18nMAssay Description:Inhibition of MMP13 by fluorimetric assayMore data for this Ligand-Target Pair
Affinity DataKi: 20nMAssay Description:Inhibition of MMP12 (unknown origin)-mediated Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 by fluorimetric assayMore data for this Ligand-Target Pair
Affinity DataKi: 23nMAssay Description:Inhibition of MMP12 (unknown origin)-mediated Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 by fluorimetric assayMore data for this Ligand-Target Pair
Affinity DataKi: 24nMAssay Description:Inhibition of MMP8 by fluorimetric assayMore data for this Ligand-Target Pair
Affinity DataKi: 25nMAssay Description:Inhibition of human carbonic anhydrase 9 incubated for 15 mins prior to testing by stopped flow CO2 hydrase assayMore data for this Ligand-Target Pair
Affinity DataKi: 31nMAssay Description:Inhibition of MMP12 by fluorimetric assayMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2(Rattus norvegicus (Rat))
Università
Curated by ChEMBL
Università
Curated by ChEMBL
Affinity DataKi: 31.3nMAssay Description:Displacement of [3H]flumazenil from rat GABAA alpha1beta2gamma2 expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 32nMAssay Description:Inhibition of MMP1 by fluorimetric assayMore data for this Ligand-Target Pair