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Found 119 with Last Name = 'cao' and Initial = 't'
TargetBreakpoint cluster region protein/Tyrosine-protein kinase ABL1(Homo sapiens (Human))
Beijing University Of Technology

Curated by ChEMBL
LigandPNGBDBM50558788(CHEMBL4762806)
Affinity DataIC50:  8.5nMAssay Description:Inhibition of BCR (unknown origin)/recombinant human N-terminal His-tagged ABL1 (27 to end residues) expressed in baculovirus infected Sf9 cells usin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50609911(CHEMBL5284397)
Affinity DataIC50:  10nMAssay Description:Inhibition of wild type EGFR (unknown origin) autophosphorylation by Kinase-Glo luminescent assayMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetGrowth factor receptor-bound protein 2(Homo sapiens (Human))
National Cancer Institute-Bethesda

Curated by ChEMBL
LigandPNGBDBM50072869(CHEMBL331463 | Phosphoric acid mono-{4-[(S)-2-acet...)
Affinity DataIC50:  11nMAssay Description:Inhibition of Grb2 SH2 domain bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))TBA
LigandPNGBDBM5447(CHEMBL939 | GEFITINIB | Iressa | N-(3-Chloro-4-flu...)
Affinity DataIC50:  12nMAssay Description:Inhibition of wild type EGFR (unknown origin) autophosphorylation by Kinase-Glo luminescent assayMore data for this Ligand-Target Pair
TargetBreakpoint cluster region protein/Tyrosine-protein kinase ABL1(Homo sapiens (Human))
Beijing University Of Technology

Curated by ChEMBL
LigandPNGBDBM50558784(CHEMBL4791681)
Affinity DataIC50:  19nMAssay Description:Inhibition of BCR (unknown origin)/recombinant human N-terminal His-tagged ABL1 (27 to end residues) expressed in baculovirus infected Sf9 cells usin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBreakpoint cluster region protein/Tyrosine-protein kinase ABL1(Homo sapiens (Human))
Beijing University Of Technology

Curated by ChEMBL
LigandPNGBDBM50558785(CHEMBL4760801)
Affinity DataIC50:  22nMAssay Description:Inhibition of BCR (unknown origin)/recombinant human N-terminal His-tagged ABL1 (27 to end residues) expressed in baculovirus infected Sf9 cells usin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBreakpoint cluster region protein/Tyrosine-protein kinase ABL1(Homo sapiens (Human))
Beijing University Of Technology

Curated by ChEMBL
LigandPNGBDBM50558782(CHEMBL4781579)
Affinity DataIC50:  26nMAssay Description:Inhibition of BCR (unknown origin)/recombinant human N-terminal His-tagged ABL1 (27 to end residues) expressed in baculovirus infected Sf9 cells usin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50609908(CHEMBL5286368)
Affinity DataIC50:  26nMAssay Description:Inhibition of wild type EGFR (unknown origin) autophosphorylation by Kinase-Glo luminescent assayMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50609909(CHEMBL5276304)
Affinity DataIC50:  41nMAssay Description:Inhibition of wild type EGFR (unknown origin) autophosphorylation by Kinase-Glo luminescent assayMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50609903(CHEMBL5275916)
Affinity DataIC50:  46nMAssay Description:Inhibition of wild type EGFR (unknown origin) autophosphorylation by Kinase-Glo luminescent assayMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50609902(CHEMBL5269684)
Affinity DataIC50:  47nMAssay Description:Inhibition of wild type EGFR (unknown origin) autophosphorylation by Kinase-Glo luminescent assayMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetGrowth factor receptor-bound protein 2(Homo sapiens (Human))
National Cancer Institute-Bethesda

Curated by ChEMBL
LigandPNGBDBM50072862(CHEMBL117807 | Phosphoric acid mono-[4-((S)-2-acet...)
Affinity DataIC50:  70nMAssay Description:Inhibition of Grb2 SH2 domain binding by surface plasmon resonanceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50609906(CHEMBL5271937)
Affinity DataIC50:  70nMAssay Description:Inhibition of wild type EGFR (unknown origin) autophosphorylation by Kinase-Glo luminescent assayMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50609905(CHEMBL5278452)
Affinity DataIC50:  71nMAssay Description:Inhibition of wild type EGFR (unknown origin) autophosphorylation by Kinase-Glo luminescent assayMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetBreakpoint cluster region protein/Tyrosine-protein kinase ABL1(Homo sapiens (Human))
Beijing University Of Technology

Curated by ChEMBL
LigandPNGBDBM50558787(CHEMBL4750498)
Affinity DataIC50:  74nMAssay Description:Inhibition of BCR (unknown origin)/recombinant human N-terminal His-tagged ABL1 (27 to end residues) expressed in baculovirus infected Sf9 cells usin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 2(Homo sapiens (Human))
National Cancer Institute-Bethesda

Curated by ChEMBL
LigandPNGBDBM50072864(CHEMBL115699 | {[4-((S)-2-Acetylamino-2-{1-[(S)-2-...)
Affinity DataIC50:  80nMAssay Description:Inhibition of Growth factor receptor bound protein 2 SH2 domain binding in plasmon resonance binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 2(Homo sapiens (Human))
National Cancer Institute-Bethesda

Curated by ChEMBL
LigandPNGBDBM50072861(CHEMBL19417 | [(S)-4-(2-Acetylamino-2-{1-[2-carbam...)
Affinity DataIC50:  80nMAssay Description:Inhibition of Growth factor receptor bound protein 2 SH2 domain binding in plasmon resonance binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 2(Homo sapiens (Human))
National Cancer Institute-Bethesda

Curated by ChEMBL
LigandPNGBDBM50072861(CHEMBL19417 | [(S)-4-(2-Acetylamino-2-{1-[2-carbam...)
Affinity DataIC50:  80nMAssay Description:Inhibition of Growth factor receptor bound protein 2 SH2 domain binding in plasmon resonance binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBreakpoint cluster region protein/Tyrosine-protein kinase ABL1(Homo sapiens (Human))
Beijing University Of Technology

Curated by ChEMBL
LigandPNGBDBM50558786(CHEMBL4744950)
Affinity DataIC50:  81nMAssay Description:Inhibition of BCR (unknown origin)/recombinant human N-terminal His-tagged ABL1 (27 to end residues) expressed in baculovirus infected Sf9 cells usin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50609899(CHEMBL5269391)
Affinity DataIC50:  87nMAssay Description:Inhibition of wild type EGFR (unknown origin) autophosphorylation by Kinase-Glo luminescent assayMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetBreakpoint cluster region protein/Tyrosine-protein kinase ABL1(Homo sapiens (Human))
Beijing University Of Technology

Curated by ChEMBL
LigandPNGBDBM50558783(CHEMBL4780376)
Affinity DataIC50:  109nMAssay Description:Inhibition of BCR (unknown origin)/recombinant human N-terminal His-tagged ABL1 (27 to end residues) expressed in baculovirus infected Sf9 cells usin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50609900(CHEMBL5287505)
Affinity DataIC50:  121nMAssay Description:Inhibition of wild type EGFR (unknown origin) autophosphorylation by Kinase-Glo luminescent assayMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetBreakpoint cluster region protein/Tyrosine-protein kinase ABL1(Homo sapiens (Human))
Beijing University Of Technology

Curated by ChEMBL
LigandPNGBDBM2579((2S,3R,4R,6R)-3-methoxy-2-methyl-4-(methylamino)-2...)
Affinity DataIC50:  122nMAssay Description:Inhibition of BCR (unknown origin)/recombinant human N-terminal His-tagged ABL1 (27 to end residues) expressed in baculovirus infected Sf9 cells usin...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50609910(CHEMBL5290595)
Affinity DataIC50:  148nMAssay Description:Inhibition of wild type EGFR (unknown origin) autophosphorylation by Kinase-Glo luminescent assayMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetGrowth factor receptor-bound protein 2(Homo sapiens (Human))
National Cancer Institute-Bethesda

Curated by ChEMBL
LigandPNGBDBM50072866(CHEMBL2370501 | Phosphoric acid mono-[4-((4R,7S,10...)
Affinity DataIC50:  370nMAssay Description:Inhibition of Grb2 SH2 domain bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 2(Homo sapiens (Human))
National Cancer Institute-Bethesda

Curated by ChEMBL
LigandPNGBDBM50072865(CHEMBL55627 | N-[(S)-1-{1-[(S)-2-Carbamoyl-1-(3-na...)
Affinity DataIC50:  500nMAssay Description:Inhibition of Grb2 SH2 domain binding in MDA-MB-453 human breast carcinoma cell lysatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 2(Homo sapiens (Human))
National Cancer Institute-Bethesda

Curated by ChEMBL
LigandPNGBDBM50072864(CHEMBL115699 | {[4-((S)-2-Acetylamino-2-{1-[(S)-2-...)
Affinity DataIC50:  500nMAssay Description:Inhibition of Grb2 SH2 domain binding in MDA-MB-453 human breast carcinoma cell lysatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 2(Homo sapiens (Human))
National Cancer Institute-Bethesda

Curated by ChEMBL
LigandPNGBDBM50072868(5-[(S)-2-{1-[(S)-2-Carbamoyl-1-(3-naphthalen-1-yl-...)
Affinity DataIC50:  500nMAssay Description:Inhibition of Grb2 SH2 domain binding in MDA-MB-453 human breast carcinoma cell lysatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50609904(CHEMBL5267140)
Affinity DataIC50:  534nMAssay Description:Inhibition of wild type EGFR (unknown origin) autophosphorylation by Kinase-Glo luminescent assayMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetBreakpoint cluster region protein/Tyrosine-protein kinase ABL1(Homo sapiens (Human))
Beijing University Of Technology

Curated by ChEMBL
LigandPNGBDBM50558789(CHEMBL4753215)
Affinity DataIC50:  621nMAssay Description:Inhibition of BCR (unknown origin)/recombinant human N-terminal His-tagged ABL1 (27 to end residues) expressed in baculovirus infected Sf9 cells usin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBreakpoint cluster region protein/Tyrosine-protein kinase ABL1(Homo sapiens (Human))
Beijing University Of Technology

Curated by ChEMBL
LigandPNGBDBM50558793(CHEMBL4741331)
Affinity DataIC50:  767nMAssay Description:Inhibition of BCR (unknown origin)/recombinant human N-terminal His-tagged ABL1 (27 to end residues) expressed in baculovirus infected Sf9 cells usin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBreakpoint cluster region protein/Tyrosine-protein kinase ABL1(Homo sapiens (Human))
Beijing University Of Technology

Curated by ChEMBL
LigandPNGBDBM50558792(CHEMBL4743038)
Affinity DataIC50:  804nMAssay Description:Inhibition of BCR (unknown origin)/recombinant human N-terminal His-tagged ABL1 (27 to end residues) expressed in baculovirus infected Sf9 cells usin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50609907(CHEMBL5271978)
Affinity DataIC50:  838nMAssay Description:Inhibition of wild type EGFR (unknown origin) autophosphorylation by Kinase-Glo luminescent assayMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50609901(CHEMBL5280531)
Affinity DataIC50:  938nMAssay Description:Inhibition of wild type EGFR (unknown origin) autophosphorylation by Kinase-Glo luminescent assayMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetAndrogen receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50404432(CHEMBL5273071)
Affinity DataIC50:  1.23E+3nMAssay Description:Inhibition of [3H]naloxone receptor binding to opioid receptor in the absence of NaClMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetGrowth factor receptor-bound protein 2(Homo sapiens (Human))
National Cancer Institute-Bethesda

Curated by ChEMBL
LigandPNGBDBM50072868(5-[(S)-2-{1-[(S)-2-Carbamoyl-1-(3-naphthalen-1-yl-...)
Affinity DataIC50:  1.30E+3nMAssay Description:Inhibition of Growth factor receptor bound protein 2 SH2 domain binding in plasmon resonance binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 2(Homo sapiens (Human))
National Cancer Institute-Bethesda

Curated by ChEMBL
LigandPNGBDBM50072860(Asp-Asp-Pro-Ser-pTyr-Val-Asn-Val-Gln | CHEMBL41223...)
Affinity DataIC50:  1.30E+3nMAssay Description:Inhibition of Grb2 SH2 domain bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50404469(CHEMBL5287380)
Affinity DataIC50:  2.05E+3nMAssay Description:Binding affinity towards 5-hydroxytryptamine 3 receptor by displacement of radioligand [3H]GR-65630.More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAndrogen receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50404450(CHEMBL5281425)
Affinity DataIC50:  2.09E+3nMAssay Description:Compound was tested for its direct effect on cell-free reverse transcriptase (RT) activity of HIV-1 (LAV-1)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAndrogen receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50404452(CHEMBL5290281)
Affinity DataIC50:  2.09E+3nMAssay Description:Compound was tested for its direct effect on cell-free reverse transcriptase (RT) activity of HIV-1 (LAV-1)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAndrogen receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50404449(CHEMBL5266054)
Affinity DataIC50:  2.14E+3nMAssay Description:Compound was tested for its direct effect on cell-free reverse transcriptase (RT) activity of HIV-1 (LAV-1)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAndrogen receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50404470(CHEMBL5286595)
Affinity DataIC50:  2.19E+3nMAssay Description:Binding affinity towards 5-hydroxytryptamine 3 receptor by displacement of radioligand [3H]GR-65630.More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAndrogen receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50404467(CHEMBL5287623)
Affinity DataIC50:  2.30E+3nMAssay Description:Binding affinity towards 5-hydroxytryptamine 3 receptor by displacement of radioligand [3H]GR-65630.More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAndrogen receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50404435(CHEMBL5268639)
Affinity DataIC50:  2.38E+3nMAssay Description:Inhibition of [3H]naloxone receptor binding to opioid receptor in the absence of NaClMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAndrogen receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50404447(CHEMBL5276723)
Affinity DataIC50:  2.41E+3nMAssay Description:Melanin concentrating hormone(MCH) activity, causes melanosome aggregation within integumental fish melanocytes and lightening of the skinMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetBreakpoint cluster region protein/Tyrosine-protein kinase ABL1(Homo sapiens (Human))
Beijing University Of Technology

Curated by ChEMBL
LigandPNGBDBM50558790(CHEMBL4779313)
Affinity DataIC50:  2.44E+3nMAssay Description:Inhibition of BCR (unknown origin)/recombinant human N-terminal His-tagged ABL1 (27 to end residues) expressed in baculovirus infected Sf9 cells usin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50404451(CHEMBL5288135)
Affinity DataIC50:  2.52E+3nMAssay Description:Compound was tested for its direct effect on cell-free reverse transcriptase (RT) activity of HIV-1 (LAV-1)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAndrogen receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50404445(CHEMBL5279893)
Affinity DataIC50:  2.54E+3nMAssay Description:Effective dose (10 nM) to determine muscarinic nature of the contractile response in guinea pig ileum, when methylatropine was competitively anatgoni...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAndrogen receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50404832(CHEMBL5287211)
Affinity DataIC50:  2.58E+3nMAssay Description:Binding affinity towards 5-hydroxytryptamine 3 receptor by displacement of radioligand [3H]GR-65630.More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAndrogen receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50404446(CHEMBL5277025)
Affinity DataIC50:  2.72E+3nMAssay Description:Melanin concentrating hormone(MCH) activity, causes melanosome aggregation within integumental fish melanocytes and lightening of the skinMore data for this Ligand-Target Pair
In DepthDetails PubMed
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