Affinity DataKi: 0.770nMAssay Description:Evaluated for its ability to displace [3H]-clonidine from alpha-2 adrenergic receptor of calf cerebral cortexMore data for this Ligand-Target Pair
Affinity DataKi: 0.890nMAssay Description:Binding affinity against oxytocin receptor in rat uterusMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor(RAT)
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataKi: 1.10nMAssay Description:Compound was tested for inhibition of human plasma reninMore data for this Ligand-Target Pair
Affinity DataKi: 1.10nMAssay Description:Binding affinity against oxytocin receptor in rat uterusMore data for this Ligand-Target Pair
TargetOxytocin receptor(Homo sapiens (Human))
Merck Sharp & Dohme Research Laboratories
Curated by PDSP Ki Database
Merck Sharp & Dohme Research Laboratories
Curated by PDSP Ki Database
Affinity DataKi: 1.40nMAssay Description:Evaluated for its ability to displace [3H]-clonidine from alpha-2 adrenergic receptor of calf cerebral cortexMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor(RAT)
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataKi: 1.60nMAssay Description:Compound was tested for inhibition of hog kidney reninMore data for this Ligand-Target Pair
Affinity DataKi: 3.40nMAssay Description:Binding affinity against oxytocin receptor in rat uterusMore data for this Ligand-Target Pair
Affinity DataKi: 3.70nMAssay Description:Binding affinity was evaluated by measuring the displacement of [3H]-AVP (arginine vasopressin) from specific binding sites in rat liverMore data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:In vitro inhibition of Histamine H2 receptor by measuring its ability to block the histamine-stimulated adenylate cyclase of guinea pig hippocampal h...More data for this Ligand-Target Pair
TargetOxytocin receptor(Homo sapiens (Human))
Merck Sharp & Dohme Research Laboratories
Curated by PDSP Ki Database
Merck Sharp & Dohme Research Laboratories
Curated by PDSP Ki Database
Affinity DataKi: 4.20nMAssay Description:Inhibition of [3H]- oxytocin binding to rat uterine Oxytocin receptorMore data for this Ligand-Target Pair
TargetOxytocin receptor(Homo sapiens (Human))
Merck Sharp & Dohme Research Laboratories
Curated by PDSP Ki Database
Merck Sharp & Dohme Research Laboratories
Curated by PDSP Ki Database
TargetOxytocin receptor(Homo sapiens (Human))
Merck Sharp & Dohme Research Laboratories
Curated by PDSP Ki Database
Merck Sharp & Dohme Research Laboratories
Curated by PDSP Ki Database
Affinity DataKi: 4.60nMAssay Description:Binding affinity was evaluated by measuring the displacement of [3H]-OT (oxytocin) from specific binding sites in uterine tissue obtained from humanMore data for this Ligand-Target Pair
TargetOxytocin receptor(Homo sapiens (Human))
Merck Sharp & Dohme Research Laboratories
Curated by PDSP Ki Database
Merck Sharp & Dohme Research Laboratories
Curated by PDSP Ki Database
Affinity DataKi: 5.30nMAssay Description:Inhibition of [3H]- oxytocin binding to rat uterine Oxytocin receptorMore data for this Ligand-Target Pair
Affinity DataKi: 5.60nMAssay Description:Binding affinity was evaluated by measuring the displacement of [3H]-AVP (arginine vasopressin) from specific binding sites in rat liverMore data for this Ligand-Target Pair
Affinity DataKi: 5.90nMAssay Description:Inhibition of [3H]- oxytocin binding to rat uterine Oxytocin receptorMore data for this Ligand-Target Pair
Affinity DataKi: 6.30nMAssay Description:In vitro inhibition of Histamine H2 receptor by measuring its ability to block the histamine-stimulated adenylate cyclase of guinea pig hippocampal h...More data for this Ligand-Target Pair
Affinity DataKi: 6.30nMAssay Description:In vitro inhibition of Histamine H2 receptor by measuring its ability to block the histamine-stimulated adenylate cyclase of guinea pig hippocampal h...More data for this Ligand-Target Pair
Affinity DataKi: 7.30nMAssay Description:Inhibition of [3H]- oxytocin binding to rat uterine Oxytocin receptorMore data for this Ligand-Target Pair
Affinity DataKi: 7.30nMAssay Description:Binding affinity against oxytocin receptor in rat uterusMore data for this Ligand-Target Pair
Affinity DataKi: 7.80nMAssay Description:Inhibition of [3H]- oxytocin binding to rat uterine Oxytocin receptorMore data for this Ligand-Target Pair
Affinity DataKi: 8.10nMAssay Description:Inhibition of [3H]- oxytocin binding to rat uterine Oxytocin receptorMore data for this Ligand-Target Pair
Affinity DataKi: 8.10nMAssay Description:Binding affinity against oxytocin receptor in rat uterusMore data for this Ligand-Target Pair
TargetOxytocin receptor(Homo sapiens (Human))
Merck Sharp & Dohme Research Laboratories
Curated by PDSP Ki Database
Merck Sharp & Dohme Research Laboratories
Curated by PDSP Ki Database
Affinity DataKi: 9.60nMAssay Description:Binding affinity against oxytocin receptor in rat uterusMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor(RAT)
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataKi: 10nMAssay Description:Compound was tested for inhibition of hog kidney reninMore data for this Ligand-Target Pair
Affinity DataKi: 15nMAssay Description:Binding affinity was evaluated by measuring the displacement of [3H]-AVP (arginine vasopressin) from specific binding sites in rat liverMore data for this Ligand-Target Pair
Affinity DataKi: 17nMAssay Description:Inhibition of [3H]- oxytocin binding to rat uterine Oxytocin receptorMore data for this Ligand-Target Pair