Compile Data Set for Download or QSAR
maximum 50k data
Found 27 with Last Name = 'dewar' and Initial = 'd'
TargetTransporter(Rattus norvegicus (rat))
University Of Glasgow

Curated by ChEMBL
LigandPNGBDBM50198230((S)-2-((S)-(2-iodophenoxy)(phenyl)methyl)morpholin...)
Affinity DataKi:  0.840nMAssay Description:Displacement of [3H]nisoxetine from NAT in Sprague-Dawley rat brain after 4 hrs by liquid scintillation analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus (rat))
University Of Glasgow

Curated by ChEMBL
LigandPNGBDBM50301211((2R,3S)-2-[(2-Iodophenoxy)phenylmethyl]morpholine ...)
Affinity DataKi:  8.40nMAssay Description:Displacement of [3H]nisoxetine from NAT in Sprague-Dawley rat brain after 4 hrs by liquid scintillation analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
University Of Glasgow

Curated by ChEMBL
LigandPNGBDBM22032(1-(2-chlorophenyl)-N-methyl-N-(1-methylpropyl)isoq...)
Affinity DataKi:  9.80nMAssay Description:Displacement of [3H]PK11195 from TSPO in Sprague-Dawley rat brain homogenates by liquid scintillation countingMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
University Of Glasgow

Curated by ChEMBL
LigandPNGBDBM50310140(CHEMBL605154 | N,N-Diethyl-3-iodomethyl-4-phenylqu...)
Affinity DataKi:  12nMAssay Description:Displacement of [3H]PK11195 from TSPO in Sprague-Dawley rat brain homogenates by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
University Of Glasgow

Curated by ChEMBL
LigandPNGBDBM50310139(CHEMBL601203 | N-Benzyl-3-iodomethyl-N-methyl-4-ph...)
Affinity DataKi:  26.1nMAssay Description:Displacement of [3H]PK11195 from TSPO in Sprague-Dawley rat brain homogenates by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
University Of Glasgow

Curated by ChEMBL
LigandPNGBDBM50301213((2R,3S)-2-[(4-Iodophenoxy)phenylmethyl]morpholine ...)
Affinity DataKi:  34.5nMAssay Description:Displacement of [3H]citalopram from SERT in Sprague-Dawley rat brain after 2 hrs by liquid scintillation analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
University Of Glasgow

Curated by ChEMBL
LigandPNGBDBM50301211((2R,3S)-2-[(2-Iodophenoxy)phenylmethyl]morpholine ...)
Affinity DataKi:  51.5nMAssay Description:Displacement of [3H]citalopram from SERT in Sprague-Dawley rat brain after 2 hrs by liquid scintillation analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus (rat))
University Of Glasgow

Curated by ChEMBL
LigandPNGBDBM50264064((2S,3S)-iodoreboxetine | (S)-2-((S)-(2-ethoxypheno...)
Affinity DataKi:  53.8nMAssay Description:Displacement of [3H]nisoxetine from NAT in Sprague-Dawley rat brain after 4 hrs by liquid scintillation analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus (rat))
University Of Glasgow

Curated by ChEMBL
LigandPNGBDBM50264063((2R,3S)-iodoreboxetine | (R)-2-((S)-(2-ethoxypheno...)
Affinity DataKi:  58.2nMAssay Description:Displacement of [3H]nisoxetine from NAT in Sprague-Dawley rat brain after 4 hrs by liquid scintillation analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
University Of Glasgow

Curated by ChEMBL
LigandPNGBDBM50301212((2R,3S)-2-[(3-Iodophenoxy)phenylmethyl]morpholine ...)
Affinity DataKi:  154nMAssay Description:Displacement of [3H]citalopram from SERT in Sprague-Dawley rat brain after 2 hrs by liquid scintillation analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
University Of Glasgow

Curated by ChEMBL
LigandPNGBDBM50310141(4-Phenyl-3-iodomethylquinoline-2-N-methyl-N-sec-bu...)
Affinity DataKi:  173nMAssay Description:Displacement of [3H]PK11195 from TSPO in Sprague-Dawley rat brain homogenates by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
University Of Glasgow

Curated by ChEMBL
LigandPNGBDBM50310138(3-Iodomethyl-N-methyl-N-phenethyl-4-phenylquinolin...)
Affinity DataKi:  411nMAssay Description:Displacement of [3H]PK11195 from TSPO in Sprague-Dawley rat brain homogenates by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
University Of Glasgow

Curated by ChEMBL
LigandPNGBDBM50310137(3-Methyl-4-phenylquinoline-2-N-methyl-N-(3-iodoben...)
Affinity DataKi:  455nMAssay Description:Displacement of [3H]PK11195 from TSPO in Sprague-Dawley rat brain homogenates by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Of Glasgow

Curated by ChEMBL
LigandPNGBDBM50301211((2R,3S)-2-[(2-Iodophenoxy)phenylmethyl]morpholine ...)
Affinity DataKi:  526nMAssay Description:Displacement of [3H]WIN-35,428 from DAT in Sprague-Dawley rat brain after 2 hrs by liquid scintillation analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
University Of Glasgow

Curated by ChEMBL
LigandPNGBDBM50263316((2R,3R)-iodoreboxetine | CHEMBL477406)
Affinity DataKi:  646nMAssay Description:Displacement of [3H]citalopram from rat brain SERTMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Of Glasgow

Curated by ChEMBL
LigandPNGBDBM50263316((2R,3R)-iodoreboxetine | CHEMBL477406)
Affinity DataKi:  716nMAssay Description:Displacement of [3H]WIN-35428 from rat brain DATMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
University Of Glasgow

Curated by ChEMBL
LigandPNGBDBM50310132(4-(4-Fluorophenyl)quinoline-2-N-methyl-N-(4-iodobe...)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]PK11195 from TSPO in Sprague-Dawley rat brain homogenates by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
University Of Glasgow

Curated by ChEMBL
LigandPNGBDBM50310133(4-(4-Fluorophenyl)quinoline-2-N-methyl-N-(3-iodobe...)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]PK11195 from TSPO in Sprague-Dawley rat brain homogenates by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
University Of Glasgow

Curated by ChEMBL
LigandPNGBDBM50310136(3-Methyl-4-phenylquinoline-2-N-methyl-N-(4-iodoben...)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]PK11195 from TSPO in Sprague-Dawley rat brain homogenates by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
University Of Glasgow

Curated by ChEMBL
LigandPNGBDBM50310135(4-Phenylquinoline-2-N-methyl-N-(3-iodobenzyl)carbo...)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]PK11195 from TSPO in Sprague-Dawley rat brain homogenates by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
University Of Glasgow

Curated by ChEMBL
LigandPNGBDBM50310134(4-Phenylquinoline-2-N-methyl-N-(4-iodobenzyl)carbo...)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]PK11195 from TSPO in Sprague-Dawley rat brain homogenates by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus (rat))
University Of Glasgow

Curated by ChEMBL
LigandPNGBDBM50301213((2R,3S)-2-[(4-Iodophenoxy)phenylmethyl]morpholine ...)
Affinity DataKi:  1.10E+3nMAssay Description:Displacement of [3H]nisoxetine from NAT in Sprague-Dawley rat brain after 4 hrs by liquid scintillation analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Of Glasgow

Curated by ChEMBL
LigandPNGBDBM50264064((2S,3S)-iodoreboxetine | (S)-2-((S)-(2-ethoxypheno...)
Affinity DataKi:  1.46E+3nMAssay Description:Displacement of [3H]WIN-35428 from rat brain DATMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus (rat))
University Of Glasgow

Curated by ChEMBL
LigandPNGBDBM50301212((2R,3S)-2-[(3-Iodophenoxy)phenylmethyl]morpholine ...)
Affinity DataKi:  1.70E+3nMAssay Description:Displacement of [3H]nisoxetine from NAT in Sprague-Dawley rat brain after 4 hrs by liquid scintillation analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Of Glasgow

Curated by ChEMBL
LigandPNGBDBM50301212((2R,3S)-2-[(3-Iodophenoxy)phenylmethyl]morpholine ...)
Affinity DataKi:  1.90E+3nMAssay Description:Displacement of [3H]WIN-35,428 from DAT in Sprague-Dawley rat brain after 2 hrs by liquid scintillation analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Of Glasgow

Curated by ChEMBL
LigandPNGBDBM50301213((2R,3S)-2-[(4-Iodophenoxy)phenylmethyl]morpholine ...)
Affinity DataKi:  2.10E+3nMAssay Description:Displacement of [3H]WIN-35,428 from DAT in Sprague-Dawley rat brain after 2 hrs by liquid scintillation analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
University Of Glasgow

Curated by ChEMBL
LigandPNGBDBM50264064((2S,3S)-iodoreboxetine | (S)-2-((S)-(2-ethoxypheno...)
Affinity DataKi:  2.79E+3nMAssay Description:Displacement of [3H]citalopram from rat brain SERTMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed