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Found 55 with Last Name = 'dumas' and Initial = 'p'
TargetReverse transcriptase(Human immunodeficiency virus 1)
University Of Siena

Curated by ChEMBL
LigandPNGBDBM2483((4S)-6-chloro-4-(2-cyclopropylethynyl)-4-(trifluor...)
Affinity DataKi:  4nMAssay Description:Inhibition of wild type HIV1 reverse transcriptase-DNA-dNTP ternary complexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
University Of Siena

Curated by ChEMBL
LigandPNGBDBM50479681(CHEMBL478258)
Affinity DataKi:  8nMAssay Description:Inhibition of wild type HIV1 reverse transcriptase-DNA binary complexMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
University Of Siena

Curated by ChEMBL
LigandPNGBDBM50479681(CHEMBL478258)
Affinity DataKi:  9nMAssay Description:Inhibition of wild type HIV1 reverse transcriptase-DNA-dNTP ternary complexMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
University Of Siena

Curated by ChEMBL
LigandPNGBDBM50479681(CHEMBL478258)
Affinity DataKi:  10nMAssay Description:Inhibition of wild type HIV1 free reverse transcriptaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTissue alpha-L-fucosidase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50065258((2S,3R,4S,5R)-2-Methyl-piperidine-3,4,5-triol | (2...)
Affinity DataKi:  29nMAssay Description:Inhibition constant against Alpha-FucosidaseMore data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
University Of Siena

Curated by ChEMBL
LigandPNGBDBM2483((4S)-6-chloro-4-(2-cyclopropylethynyl)-4-(trifluor...)
Affinity DataKi:  30nMAssay Description:Inhibition of wild type HIV1 free reverse transcriptaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase protein(Human immunodeficiency virus 1)
University Of Siena

Curated by ChEMBL
LigandPNGBDBM50479681(CHEMBL478258)
Affinity DataKi:  30nMAssay Description:Inhibition of HIV1 recombinant reverse transcriptase K103N mutant-DNA-dNTP ternary complex expressed in Escherichia coli BL21More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
University Of Siena

Curated by ChEMBL
LigandPNGBDBM50479680(CHEMBL459082)
Affinity DataKi:  30nMAssay Description:Inhibition of wild type HIV1 reverse transcriptase-DNA binary complexMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
University Of Siena

Curated by ChEMBL
LigandPNGBDBM2483((4S)-6-chloro-4-(2-cyclopropylethynyl)-4-(trifluor...)
Affinity DataKi:  30nMAssay Description:Inhibition of wild type HIV1 reverse transcriptase-DNA binary complexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase protein(Human immunodeficiency virus 1)
University Of Siena

Curated by ChEMBL
LigandPNGBDBM50479681(CHEMBL478258)
Affinity DataKi:  40nMAssay Description:Inhibition of HIV1 recombinant reverse transcriptase K103N mutant-DNA binary complex expressed in Escherichia coli BL21More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
University Of Siena

Curated by ChEMBL
LigandPNGBDBM50479680(CHEMBL459082)
Affinity DataKi:  40nMAssay Description:Inhibition of wild type HIV1 free reverse transcriptaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
University Of Siena

Curated by ChEMBL
LigandPNGBDBM50479680(CHEMBL459082)
Affinity DataKi:  40nMAssay Description:Inhibition of wild type HIV1 reverse transcriptase-DNA-dNTP ternary complexMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase protein(Human immunodeficiency virus 1)
University Of Siena

Curated by ChEMBL
LigandPNGBDBM50479681(CHEMBL478258)
Affinity DataKi:  65nMAssay Description:Inhibition of HIV1 recombinant free reverse transcriptase K103N mutant expressed in Escherichia coli BL21More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase protein(Human immunodeficiency virus 1)
University Of Siena

Curated by ChEMBL
LigandPNGBDBM2483((4S)-6-chloro-4-(2-cyclopropylethynyl)-4-(trifluor...)
Affinity DataKi:  200nMAssay Description:Inhibition of HIV1 recombinant reverse transcriptase K103N mutant-DNA-dNTP ternary complex expressed in Escherichia coli BL21More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase protein(Human immunodeficiency virus 1)
University Of Siena

Curated by ChEMBL
LigandPNGBDBM50479680(CHEMBL459082)
Affinity DataKi:  300nMAssay Description:Inhibition of HIV1 recombinant reverse transcriptase K103N mutant-DNA-dNTP ternary complex expressed in Escherichia coli BL21More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
University Of Siena

Curated by ChEMBL
LigandPNGBDBM1434(11-cyclopropyl-5,11-dihydro-4-methyl-6H-dipyrido[3...)
Affinity DataKi:  400nMAssay Description:Inhibition of wild type HIV1 reverse transcriptase-DNA-dNTP ternary complexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
University Of Siena

Curated by ChEMBL
LigandPNGBDBM1434(11-cyclopropyl-5,11-dihydro-4-methyl-6H-dipyrido[3...)
Affinity DataKi:  400nMAssay Description:Inhibition of wild type HIV1 free reverse transcriptaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase protein(Human immunodeficiency virus 1)
University Of Siena

Curated by ChEMBL
LigandPNGBDBM50479680(CHEMBL459082)
Affinity DataKi:  400nMAssay Description:Inhibition of HIV1 recombinant reverse transcriptase K103N mutant-DNA binary complex expressed in Escherichia coli BL21More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
University Of Siena

Curated by ChEMBL
LigandPNGBDBM1434(11-cyclopropyl-5,11-dihydro-4-methyl-6H-dipyrido[3...)
Affinity DataKi:  500nMAssay Description:Inhibition of wild type HIV1 reverse transcriptase-DNA binary complexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase protein(Human immunodeficiency virus 1)
University Of Siena

Curated by ChEMBL
LigandPNGBDBM50479680(CHEMBL459082)
Affinity DataKi:  600nMAssay Description:Inhibition of HIV1 recombinant free reverse transcriptase K103N mutant expressed in Escherichia coli BL21More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase protein(Human immunodeficiency virus 1)
University Of Siena

Curated by ChEMBL
LigandPNGBDBM2483((4S)-6-chloro-4-(2-cyclopropylethynyl)-4-(trifluor...)
Affinity DataKi:  1.50E+3nMAssay Description:Inhibition of HIV1 recombinant free reverse transcriptase K103N mutant expressed in Escherichia coli BL21More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase protein(Human immunodeficiency virus 1)
University Of Siena

Curated by ChEMBL
LigandPNGBDBM2483((4S)-6-chloro-4-(2-cyclopropylethynyl)-4-(trifluor...)
Affinity DataKi:  1.60E+3nMAssay Description:Inhibition of HIV1 recombinant reverse transcriptase K103N mutant-DNA binary complex expressed in Escherichia coli BL21More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase protein(Human immunodeficiency virus 1)
University Of Siena

Curated by ChEMBL
LigandPNGBDBM1434(11-cyclopropyl-5,11-dihydro-4-methyl-6H-dipyrido[3...)
Affinity DataKi:  4.00E+3nMAssay Description:Inhibition of HIV1 recombinant reverse transcriptase K103N mutant-DNA binary complex expressed in Escherichia coli BL21More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTissue alpha-L-fucosidase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50403111(CHEMBL1289015)
Affinity DataKi:  4.00E+3nMAssay Description:Inhibition constant against Alpha-FucosidaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetReverse transcriptase protein(Human immunodeficiency virus 1)
University Of Siena

Curated by ChEMBL
LigandPNGBDBM1434(11-cyclopropyl-5,11-dihydro-4-methyl-6H-dipyrido[3...)
Affinity DataKi:  4.00E+3nMAssay Description:Inhibition of HIV1 recombinant free reverse transcriptase K103N mutant expressed in Escherichia coli BL21More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase protein(Human immunodeficiency virus 1)
University Of Siena

Curated by ChEMBL
LigandPNGBDBM1434(11-cyclopropyl-5,11-dihydro-4-methyl-6H-dipyrido[3...)
Affinity DataKi:  5.00E+3nMAssay Description:Inhibition of HIV1 recombinant reverse transcriptase K103N mutant-DNA-dNTP ternary complex expressed in Escherichia coli BL21More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTissue alpha-L-fucosidase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50285247((2R,3R,4R,5R)-2-Methyl-piperidine-3,4,5-triol | CH...)
Affinity DataKi:  1.10E+4nMAssay Description:Inhibition constant against Alpha-FucosidaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetTissue alpha-L-fucosidase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50065259((2R,3R,4R,5R)-2-(Hydroxymethyl)piperidine-3,4,5-tr...)
Affinity DataKi:  3.00E+4nMAssay Description:Inhibition constant against Alpha-FucosidaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetTissue alpha-L-fucosidase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50403112(CHEMBL2115566)
Affinity DataKi:  5.00E+4nMAssay Description:Inhibition constant against Alpha-FucosidaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetTissue alpha-L-fucosidase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50403114(CHEMBL1337303)
Affinity DataKi:  5.30E+4nMAssay Description:Inhibition constant against Alpha-FucosidaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetTissue alpha-L-fucosidase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50104411((R)-6-Methyl-tetrahydro-thiopyran-2,3,4,5-tetraol ...)
Affinity DataKi:  8.00E+4nMAssay Description:Inhibition constant against Alpha-FucosidaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetTissue alpha-L-fucosidase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50280035(1-(4-Hydroxy-2-methyl-3,4-dihydro-2H-pyran-3-yl)-e...)
Affinity DataKi:  9.00E+4nMAssay Description:Inhibition constant against Alpha-FucosidaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetTissue alpha-L-fucosidase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50242419(6-Deoxy-L-galactose | 6-deoxy-L-galactopyranoseL-f...)
Affinity DataKi:  3.00E+5nMAssay Description:Inhibition constant against Alpha-FucosidaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetTissue alpha-L-fucosidase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50037814(2,5-Bis-hydroxymethyl-pyrrolidine-3,4-diol | CHEMB...)
Affinity DataKi:  9.10E+5nMAssay Description:Inhibition constant against Alpha-FucosidaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetTissue alpha-L-fucosidase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50403113(CHEMBL2115524)
Affinity DataKi:  1.00E+6nMAssay Description:Inhibition constant against Alpha-FucosidaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetTissue alpha-L-fucosidase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50280032((2R,3R,4R,5S)-2-Methyl-piperidine-3,4,5-triol | 1,...)
Affinity DataKi:  1.70E+6nMAssay Description:Inhibition constant against Alpha-FucosidaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetTissue alpha-L-fucosidase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50076963((3R,5R)-2-Hydroxymethyl-1-methyl-piperidine-3,4,5-...)
Affinity DataKi:  5.30E+6nMAssay Description:Inhibition constant against Alpha-FucosidaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetTissue alpha-L-fucosidase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50179480((2R,3S,4R,5S)-2-methylpiperidine-3,4,5-triol | CHE...)
Affinity DataKi:  7.90E+6nMAssay Description:Inhibition constant against Alpha-FucosidaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetTissue alpha-L-fucosidase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50280035(1-(4-Hydroxy-2-methyl-3,4-dihydro-2H-pyran-3-yl)-e...)
Affinity DataKi:  2.60E+7nMAssay Description:Inhibition constant against Alpha-FucosidaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetTissue alpha-L-fucosidase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50163440((2R,3S,4R,5S)-2-(hydroxymethyl)piperidine-3,4,5-tr...)
Affinity DataKi:  3.40E+7nMAssay Description:Inhibition constant against Alpha-FucosidaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetTissue alpha-L-fucosidase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50403109(CHEMBL2115527)
Affinity DataKi:  3.50E+7nMAssay Description:Inhibition constant against Alpha-Fucosidase; Uncompetitive inhibitionMore data for this Ligand-Target Pair
In DepthDetails Article
TargetTissue alpha-L-fucosidase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50403109(CHEMBL2115527)
Affinity DataKi:  3.50E+7nMAssay Description:Inhibition constant against Alpha-Fucosidase; Uncompetitive inhibitionMore data for this Ligand-Target Pair
In DepthDetails Article
TargetTissue alpha-L-fucosidase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50280039(2-Phenyl-3,4-dihydro-2H-pyran-3,4-diol | CHEMBL120...)
Affinity DataKi:  8.30E+7nMAssay Description:Inhibition constant against Alpha-Fucosidase; Uncompetitive inhibitionMore data for this Ligand-Target Pair
In DepthDetails Article
TargetTissue alpha-L-fucosidase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50280039(2-Phenyl-3,4-dihydro-2H-pyran-3,4-diol | CHEMBL120...)
Affinity DataKi:  8.30E+7nMAssay Description:Inhibition constant against Alpha-Fucosidase; Uncompetitive inhibitionMore data for this Ligand-Target Pair
In DepthDetails Article
TargetTissue alpha-L-fucosidase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50403110(CHEMBL179085)
Affinity DataKi:  9.00E+7nMAssay Description:Inhibition constant against Alpha-FucosidaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetTissue alpha-L-fucosidase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50280034(1-(4-Hydroxy-2-phenyl-3,4-dihydro-2H-pyran-3-yl)-e...)
Affinity DataKi: >1.00E+8nMAssay Description:Inhibition constant against Alpha-FucosidaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetTissue alpha-L-fucosidase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50280038(3,5-Dimethyl-2-phenyl-3,4-dihydro-2H-pyran-4-ol | ...)
Affinity DataKi: >1.00E+8nMAssay Description:Inhibition constant against Alpha-FucosidaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetTissue alpha-L-fucosidase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50280038(3,5-Dimethyl-2-phenyl-3,4-dihydro-2H-pyran-4-ol | ...)
Affinity DataKi: >1.00E+8nMAssay Description:Inhibition constant against Alpha-FucosidaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetTissue alpha-L-fucosidase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM18351((2R,3R,4R,5S)-2-(Hydroxymethyl)piperidine-3,4,5-tr...)
Affinity DataKi: >1.00E+8nMAssay Description:Inhibition constant against Alpha-FucosidaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetTissue alpha-L-fucosidase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50280037(3-Benzyloxy-2-phenyl-3,4-dihydro-2H-pyran-4-ol | C...)
Affinity DataKi: >1.00E+8nMAssay Description:Inhibition constant against Alpha-FucosidaseMore data for this Ligand-Target Pair
In DepthDetails Article
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