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Found 36 with Last Name = 'fagnere' and Initial = 'c'
TargetAromatase [1-48](Homo sapiens (Human))
BiomolÉCules Et Cibles Cellulaires Tumorales

LigandPNGBDBM13061(4,4 -(1H-1,2,4-triazol-1-ylmethanediyl)dibenzonitr...)
Affinity DataIC50:  18nMAssay Description:The inhibitory activities of the compounds toward aromatase were determined in vitro using human placental microsomes and [1,2,6,7-3H]-androstenedion...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Upres Ea 1085 BiomoléCules Et Cibles Cellulaires Tumorales

Curated by ChEMBL
LigandPNGBDBM50118965(4-Imidazol-1-yl-2-phenyl-chroman-7-ol | CHEMBL9591...)
Affinity DataIC50:  40nMAssay Description:In vitro inhibition of [1,2,6,7-3H]androstenedione binding to Aromatase of human placental microsomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase [1-48](Homo sapiens (Human))
BiomolÉCules Et Cibles Cellulaires Tumorales

LigandPNGBDBM85252(2,4-Trans-4'-hydroxy-4-imidazolyl-7-methoxyfla...)
Affinity DataIC50:  40nMAssay Description:The inhibitory activities of the compounds toward aromatase were determined in vitro using human placental microsomes and [1,2,6,7-3H]-androstenedion...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Upres Ea 1085 BiomoléCules Et Cibles Cellulaires Tumorales

Curated by ChEMBL
LigandPNGBDBM50118965(4-Imidazol-1-yl-2-phenyl-chroman-7-ol | CHEMBL9591...)
Affinity DataIC50:  41nMAssay Description:Inhibition of aromatase activity in human placental microsomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase [1-48](Homo sapiens (Human))
BiomolÉCules Et Cibles Cellulaires Tumorales

LigandPNGBDBM85253(2,4-Trans-4',7-dihydroxy-4-imidazolyl-7-methox...)
Affinity DataIC50:  77nMAssay Description:The inhibitory activities of the compounds toward aromatase were determined in vitro using human placental microsomes and [1,2,6,7-3H]-androstenedion...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Upres Ea 1085 BiomoléCules Et Cibles Cellulaires Tumorales

Curated by ChEMBL
LigandPNGBDBM50118966(1-(7-Methoxy-2-phenyl-chroman-4-yl)-1H-imidazole |...)
Affinity DataIC50:  90nMAssay Description:In vitro inhibition of [1,2,6,7-3H]androstenedione binding to Aromatase of human placental microsomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Upres Ea 1085 BiomoléCules Et Cibles Cellulaires Tumorales

Curated by ChEMBL
LigandPNGBDBM50118966(1-(7-Methoxy-2-phenyl-chroman-4-yl)-1H-imidazole |...)
Affinity DataIC50:  91nMAssay Description:Inhibition of aromatase activity in human placental microsomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase [1-48](Homo sapiens (Human))
BiomolÉCules Et Cibles Cellulaires Tumorales

LigandPNGBDBM85249(2,4-Trans-3'-hydroxy-4-imidazolyl-7-methoxyfla...)
Affinity DataIC50:  130nMAssay Description:The inhibitory activities of the compounds toward aromatase were determined in vitro using human placental microsomes and [1,2,6,7-3H]-androstenedion...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase [1-48](Homo sapiens (Human))
BiomolÉCules Et Cibles Cellulaires Tumorales

LigandPNGBDBM85251(2,4-Trans-4'-cyano-4-imidazolyl-7-methoxyflava...)
Affinity DataIC50:  133nMAssay Description:The inhibitory activities of the compounds toward aromatase were determined in vitro using human placental microsomes and [1,2,6,7-3H]-androstenedion...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase [1-48](Homo sapiens (Human))
BiomolÉCules Et Cibles Cellulaires Tumorales

LigandPNGBDBM85250(2,4-Trans-4'-chloro-4-imidazolyl-7-methoxyflav...)
Affinity DataIC50:  200nMAssay Description:The inhibitory activities of the compounds toward aromatase were determined in vitro using human placental microsomes and [1,2,6,7-3H]-androstenedion...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Upres Ea 1085 BiomoléCules Et Cibles Cellulaires Tumorales

Curated by ChEMBL
LigandPNGBDBM50153525(2-Phenyl-4-[1,2,4]triazol-1-yl-chroman-7-ol | CHEM...)
Affinity DataIC50:  430nMAssay Description:In vitro inhibition of [1,2,6,7-3H]androstenedione binding to Aromatase of human placental microsomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Upres Ea 1085 BiomoléCules Et Cibles Cellulaires Tumorales

Curated by ChEMBL
LigandPNGBDBM50374254(CHEMBL439241)
Affinity DataIC50:  610nMAssay Description:Inhibition of human aromatase in placental microsomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Upres Ea 1085 BiomoléCules Et Cibles Cellulaires Tumorales

Curated by ChEMBL
LigandPNGBDBM50111269(7-Methoxy-2-phenyl-3-pyridin-4-ylmethylene-chroman...)
Affinity DataIC50:  620nMAssay Description:In vitro inhibition of [1,2,6,7-3H]-androstenedione binding to human placental microsome cytochrome P450 19A1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Upres Ea 1085 BiomoléCules Et Cibles Cellulaires Tumorales

Curated by ChEMBL
LigandPNGBDBM50345188(2-(4-hydroxyphenyl)-2,3-dihydrobenzo[h]chromen-4-o...)
Affinity DataIC50:  630nMAssay Description:Inhibition of human aromatase in placental microsomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Upres Ea 1085 BiomoléCules Et Cibles Cellulaires Tumorales

Curated by ChEMBL
LigandPNGBDBM50111268(2-Phenyl-3-pyridin-4-ylmethylene-chroman-4-one | C...)
Affinity DataIC50:  800nMAssay Description:In vitro inhibition of [1,2,6,7-3H]-androstenedione binding to human placental microsome cytochrome P450 19A1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Upres Ea 1085 BiomoléCules Et Cibles Cellulaires Tumorales

Curated by ChEMBL
LigandPNGBDBM50374255(CHEMBL258257)
Affinity DataIC50:  1.37E+3nMAssay Description:Inhibition of human aromatase in placental microsomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Upres Ea 1085 BiomoléCules Et Cibles Cellulaires Tumorales

Curated by ChEMBL
LigandPNGBDBM50153523(1-(7-Methoxy-2-phenyl-chroman-4-yl)-1H-[1,2,4]tria...)
Affinity DataIC50:  1.40E+3nMAssay Description:In vitro inhibition of [1,2,6,7-3H]androstenedione binding to Aromatase of human placental microsomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Upres Ea 1085 BiomoléCules Et Cibles Cellulaires Tumorales

Curated by ChEMBL
LigandPNGBDBM50345187(4-(4-oxo-3,4-dihydro-2H-benzo[h]chromen-2-yl)benzo...)
Affinity DataIC50:  1.54E+3nMAssay Description:Inhibition of human aromatase in placental microsomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Upres Ea 1085 BiomoléCules Et Cibles Cellulaires Tumorales

Curated by ChEMBL
LigandPNGBDBM50111270(7-Methoxy-2-phenyl-3-pyridin-4-ylmethylene-chroman...)
Affinity DataIC50:  1.60E+3nMAssay Description:In vitro inhibition of [1,2,6,7-3H]-androstenedione binding to human placental microsome cytochrome P450 19A1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Upres Ea 1085 BiomoléCules Et Cibles Cellulaires Tumorales

Curated by ChEMBL
LigandPNGBDBM50014323(2-PHENYL-4H-BENZO[H]CHROMEN-4-ONE | 2-Phenyl-benzo...)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of human aromatase in placental microsomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Upres Ea 1085 BiomoléCules Et Cibles Cellulaires Tumorales

Curated by ChEMBL
LigandPNGBDBM50241408((2S)-liquiritigenin | 7-HYDROXY-2-(4-HYDROXY-PHENY...)
Affinity DataIC50:  2.10E+3nMAssay Description:Inhibition of human aromatase in placental microsomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Upres Ea 1085 BiomoléCules Et Cibles Cellulaires Tumorales

Curated by ChEMBL
LigandPNGBDBM50111271(2-Phenyl-3-pyridin-4-ylmethylene-chroman-4-one | C...)
Affinity DataIC50:  3.30E+3nMAssay Description:In vitro inhibition of [1,2,6,7-3H]-androstenedione binding to human placental microsome cytochrome P450 19A1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Upres Ea 1085 BiomoléCules Et Cibles Cellulaires Tumorales

Curated by ChEMBL
LigandPNGBDBM50374256(CHEMBL255110)
Affinity DataIC50:  3.40E+3nMAssay Description:Inhibition of human aromatase in placental microsomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Upres Ea 1085 BiomoléCules Et Cibles Cellulaires Tumorales

Curated by ChEMBL
LigandPNGBDBM50374258(CHEMBL256407)
Affinity DataIC50:  3.50E+3nMAssay Description:Inhibition of human aromatase in placental microsomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Upres Ea 1085 BiomoléCules Et Cibles Cellulaires Tumorales

Curated by ChEMBL
LigandPNGBDBM50374257(CHEMBL402970)
Affinity DataIC50:  3.70E+3nMAssay Description:Inhibition of human aromatase in placental microsomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Upres Ea 1085 BiomoléCules Et Cibles Cellulaires Tumorales

Curated by ChEMBL
LigandPNGBDBM50104887(2,3-dihydro-7-hydroxy-2-phenyl-4H-1-benzopyran-4-o...)
Affinity DataIC50:  3.80E+3nMAssay Description:Inhibition of human aromatase in placental microsomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Upres Ea 1085 BiomoléCules Et Cibles Cellulaires Tumorales

Curated by ChEMBL
LigandPNGBDBM50104887(2,3-dihydro-7-hydroxy-2-phenyl-4H-1-benzopyran-4-o...)
Affinity DataIC50:  3.80E+3nMAssay Description:Inhibition of aromatase activity in human placental microsomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Upres Ea 1085 BiomoléCules Et Cibles Cellulaires Tumorales

Curated by ChEMBL
LigandPNGBDBM50345186(2-phenyl-2,3-dihydrobenzo[h]chromen-4-one | 2-phen...)
Affinity DataIC50:  4.30E+3nMAssay Description:Inhibition of human aromatase in placental microsomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Upres Ea 1085 BiomoléCules Et Cibles Cellulaires Tumorales

Curated by ChEMBL
LigandPNGBDBM9460(3-(4-aminophenyl)-3-ethyl-piperidine-2,6-dione | 3...)
Affinity DataIC50:  5.20E+3nMAssay Description:Inhibition of aromatase activity in human placental microsomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetAromatase(Homo sapiens (Human))
Upres Ea 1085 BiomoléCules Et Cibles Cellulaires Tumorales

Curated by ChEMBL
LigandPNGBDBM9460(3-(4-aminophenyl)-3-ethyl-piperidine-2,6-dione | 3...)
Affinity DataIC50:  5.20E+3nMAssay Description:In vitro inhibition of [1,2,6,7-3H]-androstenedione binding to human placental microsome cytochrome P450 19A1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetAromatase(Homo sapiens (Human))
Upres Ea 1085 BiomoléCules Et Cibles Cellulaires Tumorales

Curated by ChEMBL
LigandPNGBDBM50106920((+/-)-7-methoxy-2-phenylchroman-4-one | 7-Methoxy-...)
Affinity DataIC50:  8.00E+3nMAssay Description:Inhibition of aromatase activity in human placental microsomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Upres Ea 1085 BiomoléCules Et Cibles Cellulaires Tumorales

Curated by ChEMBL
LigandPNGBDBM50106920((+/-)-7-methoxy-2-phenylchroman-4-one | 7-Methoxy-...)
Affinity DataIC50:  8.00E+3nMAssay Description:In vitro inhibition of [1,2,6,7-3H]-androstenedione binding to human placental microsome cytochrome P450 19A1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Upres Ea 1085 BiomoléCules Et Cibles Cellulaires Tumorales

Curated by ChEMBL
LigandPNGBDBM50106920((+/-)-7-methoxy-2-phenylchroman-4-one | 7-Methoxy-...)
Affinity DataIC50:  8.00E+3nMAssay Description:Inhibition of human aromatase in placental microsomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Upres Ea 1085 BiomoléCules Et Cibles Cellulaires Tumorales

Curated by ChEMBL
LigandPNGBDBM50051358(2,3-Dihydroflavone | 2,3-dihydro-2-phenyl-4H-1-ben...)
Affinity DataIC50:  2.80E+4nMAssay Description:Inhibition of human aromatase in placental microsomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Upres Ea 1085 BiomoléCules Et Cibles Cellulaires Tumorales

Curated by ChEMBL
LigandPNGBDBM50051358(2,3-Dihydroflavone | 2,3-dihydro-2-phenyl-4H-1-ben...)
Affinity DataIC50:  2.85E+4nMAssay Description:In vitro inhibition of [1,2,6,7-3H]-androstenedione binding to human placental microsome cytochrome P450 19A1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Upres Ea 1085 BiomoléCules Et Cibles Cellulaires Tumorales

Curated by ChEMBL
LigandPNGBDBM50153524(4-(7-Methoxy-2-phenyl-chroman-4-yl)-4H-[1,2,4]tria...)
Affinity DataIC50:  3.16E+4nMAssay Description:In vitro inhibition of [1,2,6,7-3H]androstenedione binding to Aromatase of human placental microsomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed