Affinity DataKi: 0.00800nMAssay Description:Potency of inhibition against human leukocyte elastase (HLE) expressed as an apparent binding constantMore data for this Ligand-Target Pair
Affinity DataKi: 0.0110nMAssay Description:Potency of inhibition against human leukocyte elastase (HLE) expressed as an apparent binding constantMore data for this Ligand-Target Pair
Affinity DataKi: 0.0110nMAssay Description:Potency of inhibition against human leukocyte elastase (HLE) expressed as an apparent binding constantMore data for this Ligand-Target Pair
Affinity DataKi: 0.0130nMAssay Description:Potency of inhibition against human leukocyte elastase (HLE) expressed as an apparent binding constantMore data for this Ligand-Target Pair
Affinity DataKi: 0.0130nMAssay Description:Potency of inhibition against human leukocyte elastase (HLE) expressed as an apparent binding constantMore data for this Ligand-Target Pair
Affinity DataKi: 0.0140nMAssay Description:Potency of inhibition against human leukocyte elastase (HLE) expressed as an apparent binding constantMore data for this Ligand-Target Pair
Affinity DataKi: 0.0230nMAssay Description:Evaluated for inhibitory activity against Human leukocyte elastase (HLE)More data for this Ligand-Target Pair
Affinity DataKi: 0.0300nMAssay Description:Evaluated for inhibitory activity against Human leukocyte elastase (HLE)More data for this Ligand-Target Pair
Affinity DataKi: 0.0300nMAssay Description:Evaluated for inhibitory activity against Human leukocyte elastase (HLE)More data for this Ligand-Target Pair
Affinity DataKi: 0.200nMAssay Description:Evaluated for inhibitory activity against Human leukocyte elastase (HLE)More data for this Ligand-Target Pair
Affinity DataKi: 0.200nMAssay Description:Potency of inhibition against human leukocyte elastase (HLE) expressed as an apparent binding constantMore data for this Ligand-Target Pair
Affinity DataKi: 0.270nMAssay Description:Evaluated for inhibitory activity against Human leukocyte elastase (HLE)More data for this Ligand-Target Pair
Affinity DataKi: 0.300nMAssay Description:Ratio of Koff to that of Kon was determined on human leukocyte elastase(HLE)More data for this Ligand-Target Pair
Affinity DataKi: 0.600nMAssay Description:Ratio of Koff to that of Kon was determined on human leukocyte elastase(HLE)More data for this Ligand-Target Pair
Affinity DataKi: 0.600nMAssay Description:Ratio of Koff to that of Kon was determined on human leukocyte elastase(HLE)More data for this Ligand-Target Pair
Affinity DataKi: 0.700nMAssay Description:Ratio of Koff to that of Kon was determined on human leukocyte elastase(HLE)More data for this Ligand-Target Pair
Affinity DataKi: 1.10nMAssay Description:Evaluated for inhibitory activity against Human leukocyte elastase (HLE)More data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Ratio of Koff to that of Kon was determined on human leukocyte elastase(HLE)More data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Ratio of Koff to that of Kon was determined on human leukocyte elastase(HLE)More data for this Ligand-Target Pair
Affinity DataKi: 2.20nMAssay Description:Evaluated for inhibitory activity against Human leukocyte elastase (HLE)More data for this Ligand-Target Pair
Affinity DataKi: 5.20nMAssay Description:Evaluated for inhibitory activity against Human leukocyte elastase (HLE)More data for this Ligand-Target Pair
Affinity DataKi: 14nMAssay Description:Evaluated for inhibitory activity against Human leukocyte elastase (HLE)More data for this Ligand-Target Pair
Affinity DataKi: 15nMAssay Description:Ratio of Koff to that of Kon was determined on human leukocyte elastase(HLE)More data for this Ligand-Target Pair
Affinity DataKi: 15nMAssay Description:Potency of inhibition against human leukocyte elastase (HLE) expressed as an apparent binding constantMore data for this Ligand-Target Pair
Affinity DataKi: 15nMAssay Description:Evaluated for inhibitory activity against Human leukocyte elastase (HLE)More data for this Ligand-Target Pair
Affinity DataKi: 60nMAssay Description:Ratio of Koff to that of Kon was determined on human leukocyte elastase(HLE)More data for this Ligand-Target Pair
Affinity DataKi: >2.00E+3nMAssay Description:Evaluated for inhibitory activity against Human leukocyte elastase (HLE)More data for this Ligand-Target Pair
TargetPolyunsaturated fatty acid 5-lipoxygenase(Rattus norvegicus)
Sterling Research Group
Curated by ChEMBL
Sterling Research Group
Curated by ChEMBL
Affinity DataIC50: 60nMAssay Description:In vitro inhibition of rat 5-LipoxygenaseMore data for this Ligand-Target Pair
TargetPolyunsaturated fatty acid 5-lipoxygenase(Rattus norvegicus)
Sterling Research Group
Curated by ChEMBL
Sterling Research Group
Curated by ChEMBL
Affinity DataIC50: 120nMAssay Description:In vitro inhibition of rat 5-LipoxygenaseMore data for this Ligand-Target Pair
TargetPolyunsaturated fatty acid 5-lipoxygenase(Rattus norvegicus)
Sterling Research Group
Curated by ChEMBL
Sterling Research Group
Curated by ChEMBL
Affinity DataIC50: 140nMAssay Description:In vitro inhibition of rat 5-LipoxygenaseMore data for this Ligand-Target Pair
TargetPolyunsaturated fatty acid 5-lipoxygenase(Rattus norvegicus)
Sterling Research Group
Curated by ChEMBL
Sterling Research Group
Curated by ChEMBL
Affinity DataIC50: 150nMAssay Description:In vitro inhibition of rat 5-LipoxygenaseMore data for this Ligand-Target Pair
TargetPolyunsaturated fatty acid 5-lipoxygenase(Rattus norvegicus)
Sterling Research Group
Curated by ChEMBL
Sterling Research Group
Curated by ChEMBL
Affinity DataIC50: 180nMAssay Description:In vitro inhibition of rat 5-LipoxygenaseMore data for this Ligand-Target Pair
TargetPolyunsaturated fatty acid 5-lipoxygenase(Rattus norvegicus)
Sterling Research Group
Curated by ChEMBL
Sterling Research Group
Curated by ChEMBL
Affinity DataIC50: 190nMAssay Description:In vitro inhibition of rat 5-LipoxygenaseMore data for this Ligand-Target Pair
TargetPolyunsaturated fatty acid 5-lipoxygenase(Rattus norvegicus)
Sterling Research Group
Curated by ChEMBL
Sterling Research Group
Curated by ChEMBL
Affinity DataIC50: 220nMAssay Description:In vitro inhibition of rat 5-LipoxygenaseMore data for this Ligand-Target Pair
TargetPolyunsaturated fatty acid 5-lipoxygenase(Rattus norvegicus)
Sterling Research Group
Curated by ChEMBL
Sterling Research Group
Curated by ChEMBL
Affinity DataIC50: 250nMAssay Description:In vitro inhibition of rat 5-LipoxygenaseMore data for this Ligand-Target Pair
TargetPolyunsaturated fatty acid 5-lipoxygenase(Rattus norvegicus)
Sterling Research Group
Curated by ChEMBL
Sterling Research Group
Curated by ChEMBL
Affinity DataIC50: 260nMAssay Description:In vitro inhibition of rat 5-LipoxygenaseMore data for this Ligand-Target Pair
TargetPolyunsaturated fatty acid 5-lipoxygenase(Rattus norvegicus)
Sterling Research Group
Curated by ChEMBL
Sterling Research Group
Curated by ChEMBL
Affinity DataIC50: 280nMAssay Description:In vitro inhibition of rat 5-LipoxygenaseMore data for this Ligand-Target Pair
TargetPolyunsaturated fatty acid 5-lipoxygenase(Rattus norvegicus)
Sterling Research Group
Curated by ChEMBL
Sterling Research Group
Curated by ChEMBL
Affinity DataIC50: 320nMAssay Description:In vitro inhibition of rat 5-LipoxygenaseMore data for this Ligand-Target Pair
TargetPolyunsaturated fatty acid 5-lipoxygenase(Rattus norvegicus)
Sterling Research Group
Curated by ChEMBL
Sterling Research Group
Curated by ChEMBL
Affinity DataIC50: 440nMAssay Description:In vitro inhibition of rat 5-LipoxygenaseMore data for this Ligand-Target Pair
TargetPolyunsaturated fatty acid 5-lipoxygenase(Rattus norvegicus)
Sterling Research Group
Curated by ChEMBL
Sterling Research Group
Curated by ChEMBL
Affinity DataIC50: 480nMAssay Description:In vitro inhibition of rat 5-LipoxygenaseMore data for this Ligand-Target Pair
TargetPolyunsaturated fatty acid 5-lipoxygenase(Rattus norvegicus)
Sterling Research Group
Curated by ChEMBL
Sterling Research Group
Curated by ChEMBL
Affinity DataIC50: 480nMAssay Description:In vitro inhibition of rat 5-LipoxygenaseMore data for this Ligand-Target Pair
TargetPolyunsaturated fatty acid 5-lipoxygenase(Rattus norvegicus)
Sterling Research Group
Curated by ChEMBL
Sterling Research Group
Curated by ChEMBL
Affinity DataIC50: 500nMAssay Description:In vitro inhibition of rat 5-LipoxygenaseMore data for this Ligand-Target Pair
TargetPolyunsaturated fatty acid 5-lipoxygenase(Rattus norvegicus)
Sterling Research Group
Curated by ChEMBL
Sterling Research Group
Curated by ChEMBL
Affinity DataIC50: 500nMAssay Description:In vitro inhibition of rat 5-LipoxygenaseMore data for this Ligand-Target Pair
TargetPolyunsaturated fatty acid 5-lipoxygenase(Rattus norvegicus)
Sterling Research Group
Curated by ChEMBL
Sterling Research Group
Curated by ChEMBL
Affinity DataIC50: 520nMAssay Description:In vitro inhibition of rat 5-LipoxygenaseMore data for this Ligand-Target Pair
TargetPolyunsaturated fatty acid 5-lipoxygenase(Rattus norvegicus)
Sterling Research Group
Curated by ChEMBL
Sterling Research Group
Curated by ChEMBL
Affinity DataIC50: 520nMAssay Description:In vitro inhibition of rat 5-LipoxygenaseMore data for this Ligand-Target Pair
TargetPolyunsaturated fatty acid 5-lipoxygenase(Rattus norvegicus)
Sterling Research Group
Curated by ChEMBL
Sterling Research Group
Curated by ChEMBL
Affinity DataIC50: 530nMAssay Description:In vitro inhibition of rat 5-LipoxygenaseMore data for this Ligand-Target Pair
TargetPolyunsaturated fatty acid 5-lipoxygenase(Rattus norvegicus)
Sterling Research Group
Curated by ChEMBL
Sterling Research Group
Curated by ChEMBL
Affinity DataIC50: 590nMAssay Description:In vitro inhibition of rat 5-LipoxygenaseMore data for this Ligand-Target Pair
TargetPolyunsaturated fatty acid 5-lipoxygenase(Rattus norvegicus)
Sterling Research Group
Curated by ChEMBL
Sterling Research Group
Curated by ChEMBL
Affinity DataIC50: 670nMAssay Description:In vitro inhibition of rat 5-LipoxygenaseMore data for this Ligand-Target Pair
TargetPolyunsaturated fatty acid 5-lipoxygenase(Rattus norvegicus)
Sterling Research Group
Curated by ChEMBL
Sterling Research Group
Curated by ChEMBL
Affinity DataIC50: <1.00E+3nMAssay Description:In vitro inhibition of rat 5-LipoxygenaseMore data for this Ligand-Target Pair
TargetPolyunsaturated fatty acid 5-lipoxygenase(Rattus norvegicus)
Sterling Research Group
Curated by ChEMBL
Sterling Research Group
Curated by ChEMBL
Affinity DataIC50: >1.00E+3nMAssay Description:In vitro inhibition of rat 5-LipoxygenaseMore data for this Ligand-Target Pair