Affinity DataIC50: 4.5nMAssay Description:Inhibition of recombinant human HDAC6 using fluorogenic substrate by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 6.90nMAssay Description:Inhibition of recombinant human HDAC1 using fluorogenic substrate by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 6.90nMAssay Description:Inhibition of human HDAC1 using RHKK(Ac) as substrateMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Inhibition of human HDAC3 using RHKK(Ac) as substrateMore data for this Ligand-Target Pair
Affinity DataIC50: 19.4nMAssay Description:Inhibition of recombinant human HDAC9 using fluorogenic substrate by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 20.5nMAssay Description:Inhibition of recombinant human HDAC2 using fluorogenic substrate by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 37.5nMAssay Description:Inhibition of recombinant human HDAC3 using fluorogenic substrate by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 38.1nMAssay Description:Inhibition of recombinant human HDAC10 using fluorogenic substrate by fluorescence assayMore data for this Ligand-Target Pair
TargetHeat shock protein HSP 90-alpha(Homo sapiens (Human))
Taipei Medical University
Curated by ChEMBL
Taipei Medical University
Curated by ChEMBL
Affinity DataIC50: 40nMAssay Description:Inhibition of FITC-geldanamycin binding to HSP90alpha (unknown origin) after 3 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetHeat shock protein HSP 90-alpha(Homo sapiens (Human))
Taipei Medical University
Curated by ChEMBL
Taipei Medical University
Curated by ChEMBL
Affinity DataIC50: 46nMAssay Description:Inhibition of FITC-geldanamycin binding to HSP90alpha (unknown origin) after 3 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetHeat shock protein HSP 90-alpha(Homo sapiens (Human))
Taipei Medical University
Curated by ChEMBL
Taipei Medical University
Curated by ChEMBL
Affinity DataIC50: 49nMAssay Description:Inhibition of FITC-geldanamycin binding to HSP90alpha (unknown origin) after 3 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetHeat shock protein HSP 90-alpha(Homo sapiens (Human))
Taipei Medical University
Curated by ChEMBL
Taipei Medical University
Curated by ChEMBL
Affinity DataIC50: 52nMAssay Description:Inhibition of FITC-geldanamycin binding to HSP90alpha (unknown origin) after 3 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetHeat shock protein HSP 90-alpha(Homo sapiens (Human))
Taipei Medical University
Curated by ChEMBL
Taipei Medical University
Curated by ChEMBL
Affinity DataIC50: 56nMAssay Description:Inhibition of FITC-geldanamycin binding to HSP90alpha (unknown origin) after 3 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetHeat shock protein HSP 90-alpha(Homo sapiens (Human))
Taipei Medical University
Curated by ChEMBL
Taipei Medical University
Curated by ChEMBL
Affinity DataIC50: 59nMAssay Description:Inhibition of FITC-geldanamycin binding to HSP90alpha (unknown origin) after 3 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataIC50: 61nMAssay Description:Inhibition of HDAC in human HeLa nuclear extract using Ac-Lys(Ac)-pNA as substrate measured after 30 mins by fluorometric analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 65nMAssay Description:Inhibition of recombinant human HDAC6 using fluorogenic substrate by fluorescence assayMore data for this Ligand-Target Pair
TargetHeat shock protein HSP 90-alpha(Homo sapiens (Human))
Taipei Medical University
Curated by ChEMBL
Taipei Medical University
Curated by ChEMBL
Affinity DataIC50: 66nMAssay Description:Inhibition of FITC-geldanamycin binding to HSP90alpha (unknown origin) after 3 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataIC50: 70nMAssay Description:Inhibition of recombinant human HDAC6 using fluorogenic substrate by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 72nMAssay Description:Inhibition of recombinant human HDAC6 using fluorogenic substrate by fluorescence assayMore data for this Ligand-Target Pair
TargetHeat shock protein HSP 90-alpha(Homo sapiens (Human))
Taipei Medical University
Curated by ChEMBL
Taipei Medical University
Curated by ChEMBL
Affinity DataIC50: 86nMAssay Description:Inhibition of FITC-geldanamycin binding to HSP90alpha (unknown origin) after 3 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataIC50: 87nMAssay Description:Inhibition of HDAC in human HeLa nuclear extract using Ac-Lys(Ac)-pNA as substrate measured after 30 mins by fluorometric analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 99nMAssay Description:Inhibition of HDAC in human HeLa nuclear extract using Ac-Lys(Ac)-pNA as substrate measured after 30 mins by fluorometric analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 102nMAssay Description:Inhibition of recombinant human HDAC1 using fluorogenic substrate by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 105nMAssay Description:Inhibition of HDAC in human HeLa nuclear extract using Ac-Lys(Ac)-pNA as substrate measured after 30 mins by fluorometric analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 108nMAssay Description:Inhibition of recombinant human HDAC6 using fluorogenic substrate by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 112nMAssay Description:Inhibition of recombinant human HDAC7 using fluorogenic substrate by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 127nMAssay Description:Inhibition of recombinant human HDAC4 using fluorogenic substrate by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 130nMAssay Description:Inhibition of human HDAC1 using RHKK(Ac) as substrateMore data for this Ligand-Target Pair
Affinity DataIC50: 130nMAssay Description:Inhibition of recombinant human HDAC1 using fluorogenic substrate by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 138nMAssay Description:Inhibition of recombinant human HDAC6 using fluorogenic substrate by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 139nMAssay Description:Inhibition of recombinant human HDAC1 using fluorogenic substrate by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 141nMAssay Description:Inhibition of recombinant human HDAC1 using fluorogenic substrate by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 158nMAssay Description:Inhibition of recombinant human HDAC1 using fluorogenic substrate by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 160nMAssay Description:Inhibition of human HDAC3 using RHKK(Ac) as substrateMore data for this Ligand-Target Pair
Affinity DataIC50: 174nMAssay Description:Inhibition of HDAC in human HeLa nuclear extract using Ac-Lys(Ac)-pNA as substrate measured after 30 mins by fluorometric analysisMore data for this Ligand-Target Pair
TargetMAP kinase-interacting serine/threonine-protein kinase 1(Homo sapiens (Human))
The Chinese University Of Hong Kong (Shenzhen)
Curated by ChEMBL
The Chinese University Of Hong Kong (Shenzhen)
Curated by ChEMBL
Affinity DataIC50: 179nMAssay Description:Inhibition of GST-tagged recombinant human full length MNK1 expressed in insect cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 209nMAssay Description:Inhibition of recombinant human HDAC2 using fluorogenic substrate by fluorescence assayMore data for this Ligand-Target Pair
TargetMAP kinase-interacting serine/threonine-protein kinase 2(Homo sapiens (Human))
The Chinese University Of Hong Kong (Shenzhen)
Curated by ChEMBL
The Chinese University Of Hong Kong (Shenzhen)
Curated by ChEMBL
Affinity DataIC50: 252nMAssay Description:Inhibition of N-terminal GST-tagged recombinant human full length MNK2 expressed in baculovirus expression system incubated for 1 hr by Kinase Tracer...More data for this Ligand-Target Pair
Affinity DataIC50: 263nMAssay Description:Inhibition of recombinant human HDAC5 using fluorogenic substrate by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 275nMAssay Description:Inhibition of recombinant human HDAC6 using fluorogenic substrate by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 284nMAssay Description:Inhibition of human HDAC8 using RHKAcKAc as substrateMore data for this Ligand-Target Pair
Affinity DataIC50: 288nMAssay Description:Inhibition of recombinant human HDAC2 using fluorogenic substrate by fluorescence assayMore data for this Ligand-Target Pair
TargetMAP kinase-interacting serine/threonine-protein kinase 2(Homo sapiens (Human))
The Chinese University Of Hong Kong (Shenzhen)
Curated by ChEMBL
The Chinese University Of Hong Kong (Shenzhen)
Curated by ChEMBL
Affinity DataIC50: 308nMAssay Description:Inhibition of N-terminal GST-tagged recombinant human full length MNK2 expressed in baculovirus expression system incubated for 1 hr by Kinase Tracer...More data for this Ligand-Target Pair
Affinity DataIC50: 314nMAssay Description:Inhibition of recombinant human HDAC8 using fluorogenic substrate by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 333nMAssay Description:Inhibition of recombinant human HDAC2 using fluorogenic substrate by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 340nMAssay Description:Inhibition of human HDAC3 using RHKK(Ac) as substrateMore data for this Ligand-Target Pair
Affinity DataIC50: 386nMAssay Description:Inhibition of recombinant human HDAC2 using fluorogenic substrate by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 390nMAssay Description:Inhibition of recombinant human HDAC8 using fluorogenic substrate by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 440nMAssay Description:Inhibition of human HDAC1 using RHKK(Ac) as substrateMore data for this Ligand-Target Pair
Affinity DataIC50: 468nMAssay Description:Inhibition of recombinant human HDAC1 using fluorogenic substrate by fluorescence assayMore data for this Ligand-Target Pair