Affinity DataKi: 7nMAssay Description:Binding affinity for adenosine A1 receptor in vitro using rat brain membranes.More data for this Ligand-Target Pair
Affinity DataKi: 7.5nMAssay Description:Binding affinity for adenosine A1 receptor in vitro using rat brain membranes.More data for this Ligand-Target Pair
Affinity DataKi: 7.90nMAssay Description:Binding affinity for adenosine A1 receptor in rat brain membraneMore data for this Ligand-Target Pair
Affinity DataKi: 8.30nMAssay Description:Binding affinity for adenosine A1 receptor in vitro using rat brain membranes.More data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:Binding affinity for adenosine A1 receptor in vitro using rat brain membranes.More data for this Ligand-Target Pair
Affinity DataKi: 14nMAssay Description:Binding affinity for adenosine A1 receptor in vitro using rat brain membranes.More data for this Ligand-Target Pair
Affinity DataKi: 14nMAssay Description:Binding affinity for adenosine A1 receptor in vitro using rat brain membranes.More data for this Ligand-Target Pair
Affinity DataKi: 23nMAssay Description:Binding affinity for adenosine A1 receptor in vitro using rat brain membranes.More data for this Ligand-Target Pair
Affinity DataKi: 26nMAssay Description:Binding affinity for adenosine A1 receptor in vitro using rat brain membranes.More data for this Ligand-Target Pair
Affinity DataKi: 29nMAssay Description:Binding affinity for adenosine A1 receptor in vitro using rat brain membranes.More data for this Ligand-Target Pair
Affinity DataKi: 39nMAssay Description:Binding affinity for adenosine A1 receptor in vitro using rat brain membranes.More data for this Ligand-Target Pair
Affinity DataKi: 39nMAssay Description:Binding affinity for adenosine A1 receptor in vitro using rat brain membranes.More data for this Ligand-Target Pair
Affinity DataKi: 50nMAssay Description:Binding affinity for adenosine A1 receptor in vitro using rat brain membranes.More data for this Ligand-Target Pair
Affinity DataKi: 50nMAssay Description:Binding affinity for adenosine A1 receptor in vitro using rat brain membranes.More data for this Ligand-Target Pair
Affinity DataKi: 62nMAssay Description:Binding affinity for adenosine A1 receptor in vitro using rat brain membranes.More data for this Ligand-Target Pair
Affinity DataKi: 110nMAssay Description:Binding affinity for adenosine A1 receptor in vitro using rat brain membranes.More data for this Ligand-Target Pair
Affinity DataKi: 120nMAssay Description:Binding affinity for adenosine A1 receptor in vitro using rat brain membranes.More data for this Ligand-Target Pair
Affinity DataKi: 130nMAssay Description:Binding affinity for adenosine A1 receptor in vitro using rat brain membranes.More data for this Ligand-Target Pair
Affinity DataKi: 140nMAssay Description:Binding affinity for adenosine A1 receptor in vitro using rat brain membranes.More data for this Ligand-Target Pair
Affinity DataKi: 140nMAssay Description:Binding affinity for adenosine A1 receptor in vitro using rat brain membranes.More data for this Ligand-Target Pair
Affinity DataKi: 150nMAssay Description:Binding affinity for adenosine A1 receptor in vitro using rat brain membranes.More data for this Ligand-Target Pair
Affinity DataKi: 160nMAssay Description:Binding affinity for adenosine A1 receptor in vitro using rat brain membranes.More data for this Ligand-Target Pair
Affinity DataKi: 160nMAssay Description:Binding affinity for adenosine A1 receptor in vitro using rat brain membranes.More data for this Ligand-Target Pair
Affinity DataKi: 170nMAssay Description:Binding affinity for adenosine A1 receptor in vitro using rat brain membranes.More data for this Ligand-Target Pair
Affinity DataKi: 170nMAssay Description:Binding affinity for adenosine A1 receptor in vitro using rat brain membranes.More data for this Ligand-Target Pair
Affinity DataKi: 180nMAssay Description:Binding affinity for adenosine A1 receptor in vitro using rat brain membranes.More data for this Ligand-Target Pair
Affinity DataKi: 200nMAssay Description:Binding affinity for adenosine A1 receptor in vitro using rat brain membranes.More data for this Ligand-Target Pair
Affinity DataKi: 370nMAssay Description:Binding affinity for adenosine A1 receptor in rat brain membraneMore data for this Ligand-Target Pair
Affinity DataKi: 510nMAssay Description:Binding affinity for adenosine A1 receptor in vitro using rat brain membranes.More data for this Ligand-Target Pair
Affinity DataKi: 890nMAssay Description:Binding affinity for adenosine A1 receptor in vitro using rat brain membranes.More data for this Ligand-Target Pair
Affinity DataKi: 895nMAssay Description:Binding affinity for adenosine A1 receptor in vitro using rat brain membranes.More data for this Ligand-Target Pair
Affinity DataKi: 1.40E+3nMAssay Description:Binding affinity for adenosine A1 receptor in vitro using rat brain membranes.More data for this Ligand-Target Pair
TargetEstrogen receptor(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by ChEMBL
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by ChEMBL
Affinity DataIC50: 11nMAssay Description:Binding affinity towards estrogen receptor alpha by [3H]17-beta-estradiol displacement.More data for this Ligand-Target Pair
TargetEstrogen receptor beta(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by ChEMBL
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by ChEMBL
Affinity DataIC50: 19nMAssay Description:Binding affinity towards estrogen receptor beta by [3H]17-beta-estradiol displacement.More data for this Ligand-Target Pair
TargetEstrogen receptor beta(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by ChEMBL
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by ChEMBL
Affinity DataIC50: 90nMAssay Description:Binding affinity towards estrogen receptor beta by [3H]17-beta-estradiol displacement.More data for this Ligand-Target Pair
TargetEstrogen receptor beta(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by ChEMBL
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by ChEMBL
Affinity DataIC50: 90nMAssay Description:Binding affinity towards estrogen receptor beta by [3H]17-beta-estradiol displacement.More data for this Ligand-Target Pair
TargetEstrogen receptor beta(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by ChEMBL
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by ChEMBL
Affinity DataIC50: 120nMAssay Description:Binding affinity towards estrogen receptor beta by [3H]17-beta-estradiol displacement.More data for this Ligand-Target Pair
TargetEstrogen receptor(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by ChEMBL
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by ChEMBL
Affinity DataIC50: 180nMAssay Description:Binding affinity towards estrogen receptor alpha by [3H]17-beta-estradiol displacement.More data for this Ligand-Target Pair
TargetEstrogen receptor beta(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by ChEMBL
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by ChEMBL
Affinity DataIC50: 200nMAssay Description:Binding affinity towards estrogen receptor beta by [3H]17-beta-estradiol displacement.More data for this Ligand-Target Pair
TargetEstrogen receptor(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by ChEMBL
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by ChEMBL
Affinity DataIC50: 210nMAssay Description:Binding affinity towards estrogen receptor alpha by [3H]17-beta-estradiol displacement.More data for this Ligand-Target Pair
TargetEstrogen receptor beta(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by ChEMBL
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by ChEMBL
Affinity DataIC50: 240nMAssay Description:Binding affinity towards estrogen receptor beta by [3H]17-beta-estradiol displacement.More data for this Ligand-Target Pair
TargetEstrogen receptor beta(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by ChEMBL
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by ChEMBL
Affinity DataIC50: 240nMAssay Description:Binding affinity towards estrogen receptor beta by [3H]17-beta-estradiol displacement.More data for this Ligand-Target Pair
TargetEstrogen receptor beta(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by ChEMBL
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by ChEMBL
Affinity DataIC50: 320nMAssay Description:Binding affinity towards estrogen receptor beta by [3H]17-beta-estradiol displacement.More data for this Ligand-Target Pair
TargetEstrogen receptor(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by ChEMBL
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by ChEMBL
Affinity DataIC50: 320nMAssay Description:Binding affinity towards estrogen receptor alpha by [3H]17-beta-estradiol displacement.More data for this Ligand-Target Pair
TargetEstrogen receptor beta(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by ChEMBL
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by ChEMBL
Affinity DataIC50: 330nMAssay Description:Binding affinity towards estrogen receptor beta by [3H]17-beta-estradiol displacement.More data for this Ligand-Target Pair
TargetEstrogen receptor beta(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by ChEMBL
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by ChEMBL
Affinity DataIC50: 390nMAssay Description:Binding affinity towards estrogen receptor beta by [3H]17-beta-estradiol displacement.More data for this Ligand-Target Pair
TargetEstrogen receptor beta(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by ChEMBL
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by ChEMBL
Affinity DataIC50: 540nMAssay Description:Binding affinity towards estrogen receptor beta by [3H]17-beta-estradiol displacement.More data for this Ligand-Target Pair
TargetEstrogen receptor(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by ChEMBL
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by ChEMBL
Affinity DataIC50: 850nMAssay Description:Binding affinity towards estrogen receptor alpha by [3H]17-beta-estradiol displacement.More data for this Ligand-Target Pair
TargetEstrogen receptor beta(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by ChEMBL
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by ChEMBL
Affinity DataIC50: 1.10E+3nMAssay Description:Binding affinity towards estrogen receptor beta by [3H]17-beta-estradiol displacement.More data for this Ligand-Target Pair
TargetEstrogen receptor beta(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by ChEMBL
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by ChEMBL
Affinity DataIC50: 1.10E+3nMAssay Description:Binding affinity towards estrogen receptor beta by [3H]17-beta-estradiol displacement.More data for this Ligand-Target Pair