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Found 78 with Last Name = 'giorgi' and Initial = 'r'
TargetType-1 angiotensin II receptor A/B(RAT)
Laboratori Guidotti

Curated by ChEMBL
LigandPNGBDBM50470323(CHEMBL327505)
Affinity DataKi:  2.5nMAssay Description:Inhibition of [3H]angiotensin II binding to rat adrenal cortex membrane containing angiotensin II receptor, type 1More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A/B(RAT)
Laboratori Guidotti

Curated by ChEMBL
LigandPNGBDBM50470328(CHEMBL317300)
Affinity DataKi:  4.40nMAssay Description:Inhibition of [3H]angiotensin II binding to rat adrenal cortex membrane containing angiotensin II receptor, type 1More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A/B(RAT)
Laboratori Guidotti

Curated by ChEMBL
LigandPNGBDBM50470310(CHEMBL98592)
Affinity DataKi:  4.5nMAssay Description:Inhibition of [3H]angiotensin II binding to rat adrenal cortex membrane containing angiotensin II receptor, type 1More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A/B(RAT)
Laboratori Guidotti

Curated by ChEMBL
LigandPNGBDBM50470321(CHEMBL99008)
Affinity DataKi:  7.70nMAssay Description:Inhibition of [3H]angiotensin II binding to rat adrenal cortex membrane containing angiotensin II receptor, type 1More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A/B(RAT)
Laboratori Guidotti

Curated by ChEMBL
LigandPNGBDBM50470340(CHEMBL98370)
Affinity DataKi:  8.80nMAssay Description:Inhibition of [3H]angiotensin II binding to rat adrenal cortex membrane containing angiotensin II receptor, type 1More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A/B(RAT)
Laboratori Guidotti

Curated by ChEMBL
LigandPNGBDBM50470326(CHEMBL319990)
Affinity DataKi:  9.10nMAssay Description:Inhibition of [3H]angiotensin II binding to rat adrenal cortex membrane containing angiotensin II receptor, type 1More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A/B(RAT)
Laboratori Guidotti

Curated by ChEMBL
LigandPNGBDBM50470330(CHEMBL318194)
Affinity DataKi:  12nMAssay Description:Inhibition of [3H]angiotensin II binding to rat adrenal cortex membrane containing angiotensin II receptor, type 1More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A/B(RAT)
Laboratori Guidotti

Curated by ChEMBL
LigandPNGBDBM50470313(CHEMBL441640)
Affinity DataKi:  12nMAssay Description:Inhibition of [3H]angiotensin II binding to rat adrenal cortex membrane containing angiotensin II receptor, type 1More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A/B(RAT)
Laboratori Guidotti

Curated by ChEMBL
LigandPNGBDBM50470317(CHEMBL319370)
Affinity DataKi:  19nMAssay Description:Inhibition of [3H]angiotensin II binding to rat adrenal cortex membrane containing angiotensin II receptor, type 1More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A/B(RAT)
Laboratori Guidotti

Curated by ChEMBL
LigandPNGBDBM50470309(CHEMBL318898)
Affinity DataKi:  25nMAssay Description:Inhibition of [3H]angiotensin II binding to rat adrenal cortex membrane containing angiotensin II receptor, type 1More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A/B(RAT)
Laboratori Guidotti

Curated by ChEMBL
LigandPNGBDBM50470336(CHEMBL317205)
Affinity DataKi:  25nMAssay Description:Inhibition of [3H]angiotensin II binding to rat adrenal cortex membrane containing angiotensin II receptor, type 1More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A/B(RAT)
Laboratori Guidotti

Curated by ChEMBL
LigandPNGBDBM50470338(CHEMBL101952)
Affinity DataKi:  27nMAssay Description:Inhibition of [3H]angiotensin II binding to rat adrenal cortex membrane containing angiotensin II receptor, type 1More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A/B(RAT)
Laboratori Guidotti

Curated by ChEMBL
LigandPNGBDBM50470337(CHEMBL275324)
Affinity DataKi:  29nMAssay Description:Inhibition of [3H]angiotensin II binding to rat adrenal cortex membrane containing angiotensin II receptor, type 1More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A/B(RAT)
Laboratori Guidotti

Curated by ChEMBL
LigandPNGBDBM50470334(CHEMBL101982)
Affinity DataKi:  30nMAssay Description:Inhibition of [3H]angiotensin II binding to rat adrenal cortex membrane containing angiotensin II receptor, type 1More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A/B(RAT)
Laboratori Guidotti

Curated by ChEMBL
LigandPNGBDBM50470322(CHEMBL100598)
Affinity DataKi:  32nMAssay Description:Inhibition of [3H]angiotensin II binding to rat adrenal cortex membrane containing angiotensin II receptor, type 1More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A/B(RAT)
Laboratori Guidotti

Curated by ChEMBL
LigandPNGBDBM50470335(CHEMBL318567)
Affinity DataKi:  38nMAssay Description:Inhibition of [3H]angiotensin II binding to rat adrenal cortex membrane containing angiotensin II receptor, type 1More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A/B(RAT)
Laboratori Guidotti

Curated by ChEMBL
LigandPNGBDBM50470320(CHEMBL421579)
Affinity DataKi:  40nMAssay Description:Inhibition of [3H]angiotensin II binding to rat adrenal cortex membrane containing angiotensin II receptor, type 1More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A/B(RAT)
Laboratori Guidotti

Curated by ChEMBL
LigandPNGBDBM50470319(CHEMBL99690)
Affinity DataKi:  40nMAssay Description:Inhibition of [3H]angiotensin II binding to rat adrenal cortex membrane containing angiotensin II receptor, type 1More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A/B(RAT)
Laboratori Guidotti

Curated by ChEMBL
LigandPNGBDBM50470333(CHEMBL98205)
Affinity DataKi:  40nMAssay Description:Inhibition of [3H]angiotensin II binding to rat adrenal cortex membrane containing angiotensin II receptor, type 1More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A/B(RAT)
Laboratori Guidotti

Curated by ChEMBL
LigandPNGBDBM50470327(CHEMBL327293)
Affinity DataKi:  41nMAssay Description:Inhibition of [3H]angiotensin II binding to rat adrenal cortex membrane containing angiotensin II receptor, type 1More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A/B(RAT)
Laboratori Guidotti

Curated by ChEMBL
LigandPNGBDBM50470311(CHEMBL97996)
Affinity DataKi:  42nMAssay Description:Inhibition of [3H]angiotensin II binding to rat adrenal cortex membrane containing angiotensin II receptor, type 1More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A/B(RAT)
Laboratori Guidotti

Curated by ChEMBL
LigandPNGBDBM50470318(CHEMBL101385)
Affinity DataKi:  44nMAssay Description:Inhibition of [3H]angiotensin II binding to rat adrenal cortex membrane containing angiotensin II receptor, type 1More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A/B(RAT)
Laboratori Guidotti

Curated by ChEMBL
LigandPNGBDBM50470329(CHEMBL101704)
Affinity DataKi:  45nMAssay Description:Inhibition of [3H]angiotensin II binding to rat adrenal cortex membrane containing angiotensin II receptor, type 1More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A/B(RAT)
Laboratori Guidotti

Curated by ChEMBL
LigandPNGBDBM50470315(CHEMBL98850)
Affinity DataKi:  53nMAssay Description:Inhibition of [3H]angiotensin II binding to rat adrenal cortex membrane containing angiotensin II receptor, type 1More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A/B(RAT)
Laboratori Guidotti

Curated by ChEMBL
LigandPNGBDBM50470306(CHEMBL98961)
Affinity DataKi:  54nMAssay Description:Inhibition of [3H]angiotensin II binding to rat adrenal cortex membrane containing angiotensin II receptor, type 1More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A/B(RAT)
Laboratori Guidotti

Curated by ChEMBL
LigandPNGBDBM50470312(CHEMBL100453)
Affinity DataKi:  59nMAssay Description:Inhibition of [3H]angiotensin II binding to rat adrenal cortex membrane containing angiotensin II receptor, type 1More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A/B(RAT)
Laboratori Guidotti

Curated by ChEMBL
LigandPNGBDBM50470307(CHEMBL99207)
Affinity DataKi:  61nMAssay Description:Inhibition of [3H]angiotensin II binding to rat adrenal cortex membrane containing angiotensin II receptor, type 1More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A/B(RAT)
Laboratori Guidotti

Curated by ChEMBL
LigandPNGBDBM50470308(CHEMBL318883)
Affinity DataKi:  67nMAssay Description:Inhibition of [3H]angiotensin II binding to rat adrenal cortex membrane containing angiotensin II receptor, type 1More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A/B(RAT)
Laboratori Guidotti

Curated by ChEMBL
LigandPNGBDBM50470316(CHEMBL98421)
Affinity DataKi:  70nMAssay Description:Inhibition of [3H]angiotensin II binding to rat adrenal cortex membrane containing angiotensin II receptor, type 1More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A/B(RAT)
Laboratori Guidotti

Curated by ChEMBL
LigandPNGBDBM50470324(CHEMBL327729)
Affinity DataKi:  90nMAssay Description:Inhibition of [3H]angiotensin II binding to rat adrenal cortex membrane containing angiotensin II receptor, type 1More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A/B(RAT)
Laboratori Guidotti

Curated by ChEMBL
LigandPNGBDBM50470331(CHEMBL100786)
Affinity DataKi:  180nMAssay Description:Inhibition of [3H]angiotensin II binding to rat adrenal cortex membrane containing angiotensin II receptor, type 1More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A/B(RAT)
Laboratori Guidotti

Curated by ChEMBL
LigandPNGBDBM50470314(CHEMBL101597)
Affinity DataKi:  243nMAssay Description:Inhibition of [3H]angiotensin II binding to rat adrenal cortex membrane containing angiotensin II receptor, type 1More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A/B(RAT)
Laboratori Guidotti

Curated by ChEMBL
LigandPNGBDBM50470339(CHEMBL328605)
Affinity DataKi:  250nMAssay Description:Inhibition of [3H]angiotensin II binding to rat adrenal cortex membrane containing angiotensin II receptor, type 1More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A/B(RAT)
Laboratori Guidotti

Curated by ChEMBL
LigandPNGBDBM50470332(CHEMBL101939)
Affinity DataKi:  290nMAssay Description:Inhibition of [3H]angiotensin II binding to rat adrenal cortex membrane containing angiotensin II receptor, type 1More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A/B(RAT)
Laboratori Guidotti

Curated by ChEMBL
LigandPNGBDBM50470325(CHEMBL316509)
Affinity DataKi:  1.66E+3nMAssay Description:Inhibition of [3H]angiotensin II binding to rat adrenal cortex membrane containing angiotensin II receptor, type 1More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAngiotensin-converting enzyme(Rattus norvegicus)
Laboratori Guidotti

Curated by ChEMBL
LigandPNGBDBM21642((2S)-1-[(2S)-2-methyl-3-sulfanylpropanoyl]pyrrolid...)
Affinity DataIC50:  3nMAssay Description:In vitro inhibitory activity against rat serum angiotensin I converting enzyme using hippuryl-glycyl-glycine as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAngiotensin-converting enzyme(Rattus norvegicus)
Laboratori Guidotti

Curated by ChEMBL
LigandPNGBDBM50046641(1R,2R-trans-2-(Ethyl-hydroxycarbamoylmethyl-carbam...)
Affinity DataIC50:  14nMAssay Description:In vitro inhibitory activity against rat serum angiotensin I converting enzyme using hippuryl-glycyl-glycine as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Menarini Ricerche

Curated by ChEMBL
LigandPNGBDBM50070307((1R,2S)-2-(2-Methylamino-3-naphthalen-2-yl-propion...)
Affinity DataIC50:  22nMAssay Description:Compound was evaluated for the inhibition of thrombin using the synthetic substrate chromozym THMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAngiotensin-converting enzyme(Rattus norvegicus)
Laboratori Guidotti

Curated by ChEMBL
LigandPNGBDBM50046633(1R,2R-trans-2-(Hydroxycarbamoylmethyl-methyl-carba...)
Affinity DataIC50:  45nMAssay Description:In vitro inhibitory activity against rat serum angiotensin I converting enzyme using hippuryl-glycyl-glycine as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAngiotensin-converting enzyme(Rattus norvegicus)
Laboratori Guidotti

Curated by ChEMBL
LigandPNGBDBM50046633(1R,2R-trans-2-(Hydroxycarbamoylmethyl-methyl-carba...)
Affinity DataIC50:  45nMAssay Description:In vitro inhibitory activity against rat serum angiotensin I converting enzyme using hippuryl-glycyl-glycine as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Menarini Ricerche

Curated by ChEMBL
LigandPNGBDBM50228863((S)-1-((R)-2-Methylamino-3-phenyl-propionyl)-pyrro...)
Affinity DataIC50:  46nMAssay Description:Compound was evaluated for the inhibition of thrombin using the synthetic substrate chromozym THMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAngiotensin-converting enzyme(Rattus norvegicus)
Laboratori Guidotti

Curated by ChEMBL
LigandPNGBDBM50046632(CHEMBL159829 | Cis-2-(Hydroxycarbamoylmethyl-propy...)
Affinity DataIC50:  400nMAssay Description:In vitro inhibitory activity against rat serum angiotensin I converting enzyme using hippuryl-glycyl-glycine as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAngiotensin-converting enzyme(Rattus norvegicus)
Laboratori Guidotti

Curated by ChEMBL
LigandPNGBDBM50046632(CHEMBL159829 | Cis-2-(Hydroxycarbamoylmethyl-propy...)
Affinity DataIC50:  400nMAssay Description:In vitro inhibitory activity against rat serum angiotensin I converting enzyme using hippuryl-glycyl-glycine as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAngiotensin-converting enzyme(Rattus norvegicus)
Laboratori Guidotti

Curated by ChEMBL
LigandPNGBDBM50046621(CHEMBL352453 | Trans-2-(Hydroxycarbamoylmethyl-iso...)
Affinity DataIC50:  500nMAssay Description:In vitro inhibitory activity against rat serum angiotensin I converting enzyme using hippuryl-glycyl-glycine as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAngiotensin-converting enzyme(Rattus norvegicus)
Laboratori Guidotti

Curated by ChEMBL
LigandPNGBDBM50046629(1-(3-Hydroxycarbamoyl-2-methyl-propionyl)-pyrrolid...)
Affinity DataIC50:  600nMAssay Description:In vitro inhibitory activity against rat serum angiotensin I converting enzyme using hippuryl-glycyl-glycine as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAngiotensin-converting enzyme(Rattus norvegicus)
Laboratori Guidotti

Curated by ChEMBL
LigandPNGBDBM50046628(CHEMBL434293 | Trans-2-(Hydroxycarbamoylmethyl-met...)
Affinity DataIC50:  1.40E+3nMAssay Description:In vitro inhibitory activity against rat serum angiotensin I converting enzyme using hippuryl-glycyl-glycine as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAngiotensin-converting enzyme(Rattus norvegicus)
Laboratori Guidotti

Curated by ChEMBL
LigandPNGBDBM50046631(CHEMBL159791 | Cis-2-(3-Mercapto-propionyl)-cycloh...)
Affinity DataIC50:  1.70E+3nMAssay Description:In vitro inhibitory activity against rat serum angiotensin I converting enzyme using hippuryl-glycyl-glycine as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAngiotensin-converting enzyme(Rattus norvegicus)
Laboratori Guidotti

Curated by ChEMBL
LigandPNGBDBM50046631(CHEMBL159791 | Cis-2-(3-Mercapto-propionyl)-cycloh...)
Affinity DataIC50:  1.70E+3nMAssay Description:In vitro inhibitory activity against rat serum angiotensin I converting enzyme using hippuryl-glycyl-glycine as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAngiotensin-converting enzyme(Rattus norvegicus)
Laboratori Guidotti

Curated by ChEMBL
LigandPNGBDBM50046641(1R,2R-trans-2-(Ethyl-hydroxycarbamoylmethyl-carbam...)
Affinity DataIC50:  2.90E+3nMAssay Description:In vitro inhibitory activity against rat serum angiotensin I converting enzyme using hippuryl-glycyl-glycine as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAngiotensin-converting enzyme(Rattus norvegicus)
Laboratori Guidotti

Curated by ChEMBL
LigandPNGBDBM50046634(CHEMBL161968 | Cis-2-(Hydroxycarbamoylmethyl-carba...)
Affinity DataIC50:  3.00E+3nMAssay Description:In vitro inhibitory activity against rat serum angiotensin I converting enzyme using hippuryl-glycyl-glycine as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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