TargetVascular endothelial growth factor receptor 3(Homo sapiens (Human))
Qilu Pharmaceutical
Curated by ChEMBL
Qilu Pharmaceutical
Curated by ChEMBL
Affinity DataKi: <0.300nMAssay Description:Binding affinity to VEGFR3 (unknown origin)More data for this Ligand-Target Pair
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
Qilu Pharmaceutical
Curated by ChEMBL
Qilu Pharmaceutical
Curated by ChEMBL
Affinity DataKi: <0.300nMAssay Description:Binding affinity to FLT3 (unknown origin)More data for this Ligand-Target Pair
TargetVascular endothelial growth factor receptor 1(Homo sapiens (Human))
Qilu Pharmaceutical
Curated by ChEMBL
Qilu Pharmaceutical
Curated by ChEMBL
Affinity DataKi: 2nMAssay Description:Binding affinity to VEGFR1 (unknown origin)More data for this Ligand-Target Pair
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Qilu Pharmaceutical
Curated by ChEMBL
Qilu Pharmaceutical
Curated by ChEMBL
Affinity DataKi: 3.80nMAssay Description:Binding affinity to VEGFR2 (unknown origin)More data for this Ligand-Target Pair
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
Qilu Pharmaceutical
Curated by ChEMBL
Qilu Pharmaceutical
Curated by ChEMBL
Affinity DataKi: 4nMAssay Description:Binding affinity to c-KIT (unknown origin)More data for this Ligand-Target Pair
TargetPlatelet-derived growth factor receptor beta(Homo sapiens (Human))
Qilu Pharmaceutical
Curated by ChEMBL
Qilu Pharmaceutical
Curated by ChEMBL
Affinity DataKi: 8nMAssay Description:Binding affinity to PDGFR-beta (unknown origin)More data for this Ligand-Target Pair
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Qilu Pharmaceutical
Curated by ChEMBL
Qilu Pharmaceutical
Curated by ChEMBL
Affinity DataKi: 9nMAssay Description:Binding affinity to VEGFR2 (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 12.9nMAssay Description:Inhibition of Yes kinaseMore data for this Ligand-Target Pair
TargetVascular endothelial growth factor receptor 3(Homo sapiens (Human))
Qilu Pharmaceutical
Curated by ChEMBL
Qilu Pharmaceutical
Curated by ChEMBL
Affinity DataKi: 17nMAssay Description:Binding affinity to VEGFR3 (unknown origin)More data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase receptor Ret(Homo sapiens (Human))
Qilu Pharmaceutical
Curated by ChEMBL
Qilu Pharmaceutical
Curated by ChEMBL
Affinity DataKi: 18nMAssay Description:Binding affinity to RET (unknown origin)More data for this Ligand-Target Pair
TargetPlatelet-derived growth factor receptor beta(Homo sapiens (Human))
Qilu Pharmaceutical
Curated by ChEMBL
Qilu Pharmaceutical
Curated by ChEMBL
Affinity DataKi: 19nMAssay Description:Binding affinity to PDGFR-beta (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 19.4nMAssay Description:Inhibition of Abl kinaseMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase receptor UFO(Homo sapiens (Human))
Qilu Pharmaceutical
Curated by ChEMBL
Qilu Pharmaceutical
Curated by ChEMBL
Affinity DataKi: 63nMAssay Description:Binding affinity to AXL (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 89nMAssay Description:Binding affinity to FGFR3 (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 95nMAssay Description:Binding affinity to ALK (unknown origin)More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Qilu Pharmaceutical
Curated by ChEMBL
Qilu Pharmaceutical
Curated by ChEMBL
Affinity DataKi: 110nMAssay Description:Binding affinity to CHK1 (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 120nMAssay Description:Binding affinity to ABL (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 180nMAssay Description:Binding affinity to ARG (unknown origin)More data for this Ligand-Target Pair
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
Qilu Pharmaceutical
Curated by ChEMBL
Qilu Pharmaceutical
Curated by ChEMBL
Affinity DataKi: 200nMAssay Description:Binding affinity to c-KIT (unknown origin)More data for this Ligand-Target Pair
TargetMacrophage colony-stimulating factor 1 receptor(Homo sapiens (Human))
Qilu Pharmaceutical
Curated by ChEMBL
Qilu Pharmaceutical
Curated by ChEMBL
Affinity DataKi: 230nMAssay Description:Binding affinity to FMS (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 340nMAssay Description:Binding affinity to PYK2 (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 350nMAssay Description:Binding affinity to FGFR1 (unknown origin)More data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase receptor Ret(Homo sapiens (Human))
Qilu Pharmaceutical
Curated by ChEMBL
Qilu Pharmaceutical
Curated by ChEMBL
Affinity DataKi: 530nMAssay Description:Binding affinity to FAK (unknown origin)More data for this Ligand-Target Pair
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Qilu Pharmaceutical
Curated by ChEMBL
Qilu Pharmaceutical
Curated by ChEMBL
TargetPhosphorylase b kinase gamma catalytic chain, liver/testis isoform(Homo sapiens (Human))
Qilu Pharmaceutical
Curated by ChEMBL
Qilu Pharmaceutical
Curated by ChEMBL
Affinity DataKi: 840nMAssay Description:Binding affinity to PHKgamma2 (unknown origin)More data for this Ligand-Target Pair
TargetVascular endothelial growth factor receptor 1(Homo sapiens (Human))
Qilu Pharmaceutical
Curated by ChEMBL
Qilu Pharmaceutical
Curated by ChEMBL
Affinity DataKi: 1.10E+3nMAssay Description:Binding affinity to VEGFR1 (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 1.80E+3nMAssay Description:Binding affinity to FYN (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 2.00E+3nMAssay Description:Binding affinity to LCK (unknown origin)More data for this Ligand-Target Pair
TargetPlatelet-derived growth factor receptor beta(Homo sapiens (Human))
Qilu Pharmaceutical
Curated by ChEMBL
Qilu Pharmaceutical
Curated by ChEMBL
Affinity DataKi: 2.09E+3nMAssay Description:Inhibition of PDGFRbetaMore data for this Ligand-Target Pair
Affinity DataIC50: 0.0100nMAssay Description:Inhibition of TrKC (unknown origin) incubated for 120 mins in presence of 33P-ATPMore data for this Ligand-Target Pair
Affinity DataIC50: 0.0500nMAssay Description:Inhibition of human TRKB using poly[Glu:Tyr] (4:1) as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase ROS(Homo sapiens (Human))
Yantai University
Curated by ChEMBL
Yantai University
Curated by ChEMBL
Affinity DataIC50: 0.0700nMAssay Description:Inhibition of human ROS1 using KKKSPGEYVNIEFG as substrate in presence of ATP by radiometric HotSpot kinase assayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.100nMAssay Description:Inhibition of human TRKC using poly[Glu:Tyr] (4:1) as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase ROS(Homo sapiens (Human))
Yantai University
Curated by ChEMBL
Yantai University
Curated by ChEMBL
Affinity DataIC50: 0.170nMAssay Description:Inhibition of ROS1 (unknown origin) incubated for 120 mins in presence of 33P-ATPMore data for this Ligand-Target Pair
Affinity DataIC50: 0.200nMAssay Description:Inhibition of TrKC (unknown origin) incubated for 120 mins in presence of 33P-ATPMore data for this Ligand-Target Pair
Affinity DataIC50: 0.200nMAssay Description:Inhibition of TrKC (unknown origin) incubated for 120 mins in presence of 33P-ATPMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase ROS(Homo sapiens (Human))
Yantai University
Curated by ChEMBL
Yantai University
Curated by ChEMBL
Affinity DataIC50: 0.200nMAssay Description:Inhibition of ROS1 (unknown origin) incubated for 120 mins in presence of 33P-ATPMore data for this Ligand-Target Pair
Affinity DataIC50: 0.200nMAssay Description:Inhibition of TrKC (unknown origin) incubated for 120 mins in presence of 33P-ATPMore data for this Ligand-Target Pair
Affinity DataIC50: 0.5nMAssay Description:Inhibition of TrKC (unknown origin) incubated for 120 mins in presence of 33P-ATPMore data for this Ligand-Target Pair
Affinity DataIC50: 0.5nMT: 2°CAssay Description:Testing of inhibition of kinases in vitro using luciferase-based assay from KinaseGlo, Promega Corp.More data for this Ligand-Target Pair
Affinity DataIC50: 0.5nMAssay Description:Displacement of 125I-dY-peptide from human BRS3 expressed in NFAT-CHO cells after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 0.5nMAssay Description:Displacement of 125I-dY-peptide from human BRS3 expressed in NFAT-CHO cells after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Homo sapiens (Human))
Chinese Academy Of Sciences
Curated by ChEMBL
Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 0.540nMAssay Description:Inhibition of N-terminal GST-tagged human PDE5A1 expressed in baculovirus infected sf9 cells using [3H]cGMP as substrate measured after 30 mins by sc...More data for this Ligand-Target Pair
Affinity DataIC50: 0.542nMT: 2°CAssay Description:Testing of inhibition of kinases in vitro using luciferase-based assay from KinaseGlo, Promega Corp.More data for this Ligand-Target Pair