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Found 166 with Last Name = 'gray' and Initial = 'c'
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM15131(5-indazolyl pyridine 3 | 5-{5-[(2S)-2-amino-3-(1H-...)
Affinity DataKi:  0.160nMAssay Description:Inhibition of AKT1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM15131(5-indazolyl pyridine 3 | 5-{5-[(2S)-2-amino-3-(1H-...)
Affinity DataIC50:  2.5nMAssay Description:Inhibition of myristoylated wild type AKT1 expressed in HEK293T cells by in-vitro immunoprecipitation kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRibosomal protein S6 kinase beta-1(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50326705(3-bromo-4-(4-(2-methoxyphenyl)piperazin-1-yl)-1H-p...)
Affinity DataIC50:  9.10nMAssay Description:Inhibition of S6K1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelial lipase(Homo sapiens (Human))
Xenon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50444153(CHEMBL3093304)
Affinity DataIC50:  25nMAssay Description:Inhibition of recombinant human endothelial lipase using bis-BODIPY-FL C11-PC as substrate preincubated for 30 mins followed by substrate addition by...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-beta serine/threonine-protein kinase(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM15131(5-indazolyl pyridine 3 | 5-{5-[(2S)-2-amino-3-(1H-...)
Affinity DataIC50:  30nMAssay Description:Inhibition of myristoylated wild type AKT2 expressed in HEK293T cells by in-vitro immunoprecipitation kinase assayMore data for this Ligand-Target Pair
TargetIsoprenyl transferase(Streptococcus pneumoniae)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50372752(CHEMBL272547)
Affinity DataIC50:  40nMAssay Description:Inhibition of Streptococcus pneumoniae UPPSMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-gamma serine/threonine-protein kinase(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM15131(5-indazolyl pyridine 3 | 5-{5-[(2S)-2-amino-3-(1H-...)
Affinity DataIC50:  51nMAssay Description:Inhibition of myristoylated wild type AKT3 expressed in HEK293T cells by in-vitro immunoprecipitation kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIsoprenyl transferase(Streptococcus pneumoniae)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50372771(CHEMBL404127)
Affinity DataIC50:  60nMAssay Description:Inhibition of Streptococcus pneumoniae UPPSMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIsoprenyl transferase(Streptococcus pneumoniae)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50372754(CHEMBL272054)
Affinity DataIC50:  70nMAssay Description:Inhibition of Streptococcus pneumoniae UPPSMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIsoprenyl transferase(Streptococcus pneumoniae)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50372766(CHEMBL271482)
Affinity DataIC50:  70nMAssay Description:Inhibition of Streptococcus pneumoniae UPPSMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelial lipase(Homo sapiens (Human))
Xenon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50444147(CHEMBL3093396)
Affinity DataIC50:  88nMAssay Description:Inhibition of recombinant human endothelial lipase using bis-BODIPY-FL C11-PC as substrate preincubated for 30 mins followed by substrate addition by...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIsoprenyl transferase(Streptococcus pneumoniae)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50372750(CHEMBL272914)
Affinity DataIC50:  110nMAssay Description:Inhibition of Streptococcus pneumoniae UPPSMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIsoprenyl transferase(Streptococcus pneumoniae)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50372751(CHEMBL256222)
Affinity DataIC50:  110nMAssay Description:Inhibition of Streptococcus pneumoniae UPPSMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelial lipase(Homo sapiens (Human))
Xenon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50444138(CHEMBL3093392)
Affinity DataIC50:  110nMAssay Description:Inhibition of human endothelial lipase using HDL as substrate assessed as release of free fatty acids preincubated for 30 mins followed by substrate ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIsoprenyl transferase(Streptococcus pneumoniae)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50372760(CHEMBL257948)
Affinity DataIC50:  120nMAssay Description:Inhibition of Streptococcus pneumoniae UPPSMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelial lipase(Homo sapiens (Human))
Xenon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50444140(CHEMBL3093394)
Affinity DataIC50:  120nMAssay Description:Inhibition of human endothelial lipase using HDL as substrate assessed as release of free fatty acids preincubated for 30 mins followed by substrate ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelial lipase(Homo sapiens (Human))
Xenon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50444141(CHEMBL3093393)
Affinity DataIC50:  130nMAssay Description:Inhibition of human endothelial lipase using HDL as substrate assessed as release of free fatty acids preincubated for 30 mins followed by substrate ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelial lipase(Homo sapiens (Human))
Xenon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50444150(CHEMBL3093307)
Affinity DataIC50:  131nMAssay Description:Inhibition of recombinant human endothelial lipase using bis-BODIPY-FL C11-PC as substrate preincubated for 30 mins followed by substrate addition by...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIsoprenyl transferase(Streptococcus pneumoniae)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50372767(CHEMBL272913)
Affinity DataIC50:  140nMAssay Description:Inhibition of Streptococcus pneumoniae UPPSMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelial lipase(Homo sapiens (Human))
Xenon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50444148(CHEMBL3093309)
Affinity DataIC50:  156nMAssay Description:Inhibition of recombinant human endothelial lipase using bis-BODIPY-FL C11-PC as substrate preincubated for 30 mins followed by substrate addition by...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIsoprenyl transferase(Streptococcus pneumoniae)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50372762(CHEMBL272162)
Affinity DataIC50:  160nMAssay Description:Inhibition of Streptococcus pneumoniae UPPSMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIsoprenyl transferase(Streptococcus pneumoniae)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50372753(CHEMBL271845)
Affinity DataIC50:  180nMAssay Description:Inhibition of Streptococcus pneumoniae UPPSMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelial lipase(Homo sapiens (Human))
Xenon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50444144(CHEMBL3093302)
Affinity DataIC50:  184nMAssay Description:Inhibition of recombinant human endothelial lipase using bis-BODIPY-FL C11-PC as substrate preincubated for 30 mins followed by substrate addition by...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIsoprenyl transferase(Streptococcus pneumoniae)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50372753(CHEMBL271845)
Affinity DataIC50:  200nMAssay Description:Inhibition of Streptococcus pneumoniae UPPSMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIsoprenyl transferase(Streptococcus pneumoniae)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50372780(CHEMBL404126)
Affinity DataIC50:  200nMAssay Description:Inhibition of Streptococcus pneumoniae UPPSMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelial lipase(Homo sapiens (Human))
Xenon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50444158(CHEMBL3093401)
Affinity DataIC50:  209nMAssay Description:Inhibition of recombinant human endothelial lipase using bis-BODIPY-FL C11-PC as substrate preincubated for 30 mins followed by substrate addition by...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelial lipase(Homo sapiens (Human))
Xenon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50444139(CHEMBL3093395)
Affinity DataIC50:  214nMAssay Description:Inhibition of recombinant human endothelial lipase using bis-BODIPY-FL C11-PC as substrate preincubated for 30 mins followed by substrate addition by...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelial lipase(Homo sapiens (Human))
Xenon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50444141(CHEMBL3093393)
Affinity DataIC50:  219nMAssay Description:Inhibition of recombinant human endothelial lipase using bis-BODIPY-FL C11-PC as substrate preincubated for 30 mins followed by substrate addition by...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelial lipase(Homo sapiens (Human))
Xenon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50444149(CHEMBL3093308)
Affinity DataIC50:  236nMAssay Description:Inhibition of recombinant human endothelial lipase using bis-BODIPY-FL C11-PC as substrate preincubated for 30 mins followed by substrate addition by...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelial lipase(Homo sapiens (Human))
Xenon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50444151(CHEMBL3093306)
Affinity DataIC50:  236nMAssay Description:Inhibition of recombinant human endothelial lipase using bis-BODIPY-FL C11-PC as substrate preincubated for 30 mins followed by substrate addition by...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelial lipase(Homo sapiens (Human))
Xenon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50444138(CHEMBL3093392)
Affinity DataIC50:  237nMAssay Description:Inhibition of recombinant human endothelial lipase using bis-BODIPY-FL C11-PC as substrate preincubated for 30 mins followed by substrate addition by...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFascin(Homo sapiens (human))
Cruk Beatson Institute

Curated by ChEMBL
LigandPNGBDBM50526225(CHEMBL4452711)
Affinity DataIC50:  240nMAssay Description:Inhibition of human (His8)2-tagged fascin (1 to 493 residues) expressed in Escherichia coli BL21(DE3) pLysS assessed as reduction in F-actin bundling...More data for this Ligand-Target Pair
TargetEndothelial lipase(Homo sapiens (Human))
Xenon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50444138(CHEMBL3093392)
Affinity DataIC50:  250nMAssay Description:Inhibition of full length human endothelial lipase transfected in HEK293 cells using PED-A1 as substrate preincubated for 30 mins followed by substra...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelial lipase(Homo sapiens (Human))
Xenon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50444140(CHEMBL3093394)
Affinity DataIC50:  252nMAssay Description:Inhibition of recombinant human endothelial lipase using bis-BODIPY-FL C11-PC as substrate preincubated for 30 mins followed by substrate addition by...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelial lipase(Homo sapiens (Human))
Xenon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50444154(CHEMBL3093303)
Affinity DataIC50:  259nMAssay Description:Inhibition of recombinant human endothelial lipase using bis-BODIPY-FL C11-PC as substrate preincubated for 30 mins followed by substrate addition by...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIsoprenyl transferase(Streptococcus pneumoniae)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50372758(CHEMBL269960)
Affinity DataIC50:  300nMAssay Description:Inhibition of Streptococcus pneumoniae UPPSMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFascin(Homo sapiens (human))
Cruk Beatson Institute

Curated by ChEMBL
LigandPNGBDBM50526241(CHEMBL4461540)
Affinity DataIC50:  330nMAssay Description:Inhibition of human (His8)2-tagged fascin (1 to 493 residues) expressed in Escherichia coli BL21(DE3) pLysS assessed as reduction in F-actin bundling...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEndothelial lipase(Homo sapiens (Human))
Xenon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50444139(CHEMBL3093395)
Affinity DataIC50:  330nMAssay Description:Inhibition of human endothelial lipase using HDL as substrate assessed as release of free fatty acids preincubated for 30 mins followed by substrate ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelial lipase(Homo sapiens (Human))
Xenon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50444143(CHEMBL3093391)
Affinity DataIC50:  366nMAssay Description:Inhibition of recombinant human endothelial lipase using bis-BODIPY-FL C11-PC as substrate preincubated for 30 mins followed by substrate addition by...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelial lipase(Homo sapiens (Human))
Xenon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50444152(CHEMBL3093305)
Affinity DataIC50:  372nMAssay Description:Inhibition of recombinant human endothelial lipase using bis-BODIPY-FL C11-PC as substrate preincubated for 30 mins followed by substrate addition by...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelial lipase(Homo sapiens (Human))
Xenon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50444146(CHEMBL3093398)
Affinity DataIC50:  499nMAssay Description:Inhibition of recombinant human endothelial lipase using bis-BODIPY-FL C11-PC as substrate preincubated for 30 mins followed by substrate addition by...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIsoprenyl transferase(Streptococcus pneumoniae)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50372755(CHEMBL255828)
Affinity DataIC50:  500nMAssay Description:Inhibition of Streptococcus pneumoniae UPPSMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFascin(Homo sapiens (human))
Cruk Beatson Institute

Curated by ChEMBL
LigandPNGBDBM50526227(CHEMBL4574198)
Affinity DataIC50:  510nMAssay Description:Inhibition of human (His8)2-tagged fascin (1 to 493 residues) expressed in Escherichia coli BL21(DE3) pLysS assessed as reduction in F-actin bundling...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEndothelial lipase(Homo sapiens (Human))
Xenon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50444142(CHEMBL3093399)
Affinity DataIC50:  551nMAssay Description:Inhibition of recombinant human endothelial lipase using bis-BODIPY-FL C11-PC as substrate preincubated for 30 mins followed by substrate addition by...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelial lipase(Homo sapiens (Human))
Xenon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50444160(CHEMBL3093397)
Affinity DataIC50:  570nMAssay Description:Inhibition of recombinant human endothelial lipase using bis-BODIPY-FL C11-PC as substrate preincubated for 30 mins followed by substrate addition by...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFascin(Homo sapiens (human))
Cruk Beatson Institute

Curated by ChEMBL
LigandPNGBDBM50526240(CHEMBL4566108)
Affinity DataIC50:  630nMAssay Description:Inhibition of human (His8)2-tagged fascin (1 to 493 residues) expressed in Escherichia coli BL21(DE3) pLysS assessed as reduction in F-actin bundling...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIsoprenyl transferase(Streptococcus pneumoniae)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50372768(CHEMBL272696)
Affinity DataIC50:  630nMAssay Description:Inhibition of Streptococcus pneumoniae UPPSMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFascin(Homo sapiens (human))
Cruk Beatson Institute

Curated by ChEMBL
LigandPNGBDBM50526226(CHEMBL4559691)
Affinity DataIC50:  630nMAssay Description:Inhibition of human (His8)2-tagged fascin (1 to 493 residues) expressed in Escherichia coli BL21(DE3) pLysS assessed as reduction in F-actin bundling...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetEndothelial lipase(Homo sapiens (Human))
Xenon Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50444159(CHEMBL3093400)
Affinity DataIC50:  659nMAssay Description:Inhibition of recombinant human endothelial lipase using bis-BODIPY-FL C11-PC as substrate preincubated for 30 mins followed by substrate addition by...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIsoprenyl transferase(Streptococcus pneumoniae)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50372759(CHEMBL256476)
Affinity DataIC50:  800nMAssay Description:Inhibition of Streptococcus pneumoniae UPPSMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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