TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataIC50: 2nMAssay Description:Inhibition of Kv1.3 potassium channel expressed in mouse L929 cells by whole cell patch clampMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataIC50: 17nMAssay Description:Inhibition of Kv1.3 potassium channel expressed in mouse L929 cells by whole cell patch clampMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataIC50: 150nMAssay Description:Inhibition of Kv1.3 potassium channel expressed in mouse L929 cells by whole cell patch clampMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataIC50: 150nMAssay Description:Inhibition of Kv1.3 potassium channel expressed in mouse L929 cells by whole cell patch clampMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataIC50: 165nMAssay Description:Inhibition of Kv1.3 potassium channel expressed in mouse L929 cells by whole cell patch clampMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataIC50: 170nMAssay Description:Inhibition of Kv1.3 potassium channel expressed in mouse L929 cells by whole cell patch clampMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataIC50: 200nMAssay Description:Inhibition of Kv1.3 potassium channel expressed in mouse L929 cells by whole cell patch clampMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily A member 3(Mus musculus)
University Of Kiel
Curated by ChEMBL
University Of Kiel
Curated by ChEMBL
Affinity DataIC50: 230nMAssay Description:Blockade of peak steady-state K+ currents of voltage-gated potassium channel subunit Kv1.3 in mouse fibroblasts L929 at 50 uMMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataIC50: 233nMAssay Description:Inhibition of Kv1.3 potassium channel expressed in mouse L929 cells by whole cell patch clampMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily A member 3(Mus musculus)
University Of Kiel
Curated by ChEMBL
University Of Kiel
Curated by ChEMBL
Affinity DataIC50: 280nMAssay Description:Blockade of peak steady-state K+ currents of voltage-gated potassium channel subunit Kv1.3 in mouse fibroblasts L929 at 50 uMMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataIC50: 318nMAssay Description:Inhibition of Kv1.3 potassium channel expressed in mouse L929 cells by whole cell patch clampMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataIC50: 450nMAssay Description:Inhibition of Kv1.3 potassium channel expressed in mouse L929 cells by whole cell patch clampMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataIC50: 520nMAssay Description:Inhibition of Kv1.3 potassium channel expressed in mouse L929 cells by whole cell patch clampMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataIC50: 650nMAssay Description:Inhibition of Kv1.3 potassium channel expressed in mouse L929 cells by whole cell patch clampMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataIC50: 670nMAssay Description:Inhibition of Kv1.3 potassium channel expressed in mouse L929 cells by whole cell patch clampMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataIC50: 890nMAssay Description:Inhibition of Kv1.3 potassium channel expressed in mouse L929 cells by whole cell patch clampMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of Kv1.3 potassium channel expressed in mouse L929 cells by whole cell patch clampMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of Kv1.3 potassium channel expressed in mouse L929 cells by whole cell patch clampMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of Kv1.3 potassium channel expressed in mouse L929 cells by whole cell patch clampMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of Kv1.3 potassium channel expressed in mouse L929 cells by whole cell patch clampMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of Kv1.3 potassium channel expressed in mouse L929 cells by whole cell patch clampMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of Kv1.3 potassium channel expressed in mouse L929 cells by whole cell patch clampMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily A member 3(Mus musculus)
University Of Kiel
Curated by ChEMBL
University Of Kiel
Curated by ChEMBL
Affinity DataIC50: 5.00E+3nMAssay Description:Blockade of peak steady-state K+ currents of voltage-gated potassium channel subunit Kv1.3 in mouse fibroblasts L929 at 50 uMMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataIC50: 6.00E+3nMAssay Description:Inhibition of Kv1.3 potassium channel expressed in mouse L929 cells by whole cell patch clampMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataIC50: 7.00E+3nMAssay Description:Inhibition of Kv1.3 potassium channel expressed in mouse L929 cells by whole cell patch clampMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily A member 3(Mus musculus)
University Of Kiel
Curated by ChEMBL
University Of Kiel
Curated by ChEMBL
Affinity DataIC50: 1.00E+4nMAssay Description:Blockade of peak steady-state K+ currents of voltage-gated potassium channel subunit Kv1.3 in mouse fibroblasts L929 at 50 uMMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of Kv1.3 potassium channel expressed in mouse L929 cells by whole cell patch clampMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataIC50: 1.20E+4nMAssay Description:Inhibition of Kv1.3 potassium channel expressed in mouse L929 cells by whole cell patch clampMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataIC50: 1.50E+4nMAssay Description:Inhibition of Kv1.3 potassium channel expressed in mouse L929 cells by whole cell patch clampMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily A member 3(Mus musculus)
University Of Kiel
Curated by ChEMBL
University Of Kiel
Curated by ChEMBL
Affinity DataIC50: 1.80E+4nMAssay Description:Inhibition of voltage-gated potassium channel subunit Kv1.3 expressed in L929 cellsMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of Kv1.3 potassium channel expressed in mouse L929 cells by whole cell patch clampMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily A member 3(Mus musculus)
University Of Kiel
Curated by ChEMBL
University Of Kiel
Curated by ChEMBL
Affinity DataIC50: 4.90E+4nMAssay Description:Blockade of peak steady-state K+ currents of voltage-gated potassium channel subunit Kv1.3 in mouse fibroblasts L929 at 50 uMMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataIC50: 1.01E+5nMAssay Description:Inhibition of Kv1.3 potassium channel expressed in mouse L929 cells by whole cell patch clampMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily A member 2(Homo sapiens (Human))
University Of Kiel
Curated by ChEMBL
University Of Kiel
Curated by ChEMBL
Affinity DataKd: 5.90E+5nMAssay Description:Blockade of peak K+ currents against Kv1.2 geneMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily A member 5(Homo sapiens (Human))
University Of Kiel
Curated by ChEMBL
University Of Kiel
Curated by ChEMBL
Affinity DataKd: 2.70E+5nMAssay Description:Blockade of peak K+ currents against Kv1.5 geneMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily A member 3(Mus musculus)
University Of Kiel
Curated by ChEMBL
University Of Kiel
Curated by ChEMBL
Affinity DataKd: 9.00E+4nMAssay Description:Blockade of peak Kv1.3 potassium currentsMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily A member 1(Homo sapiens (Human))
University Of Kiel
Curated by ChEMBL
University Of Kiel
Curated by ChEMBL
Affinity DataKd: >2.00E+5nMAssay Description:Blockade of peak K+ currents against Kv1.1 geneMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily A member 3(Mus musculus)
University Of Kiel
Curated by ChEMBL
University Of Kiel
Curated by ChEMBL
Affinity DataKd: 1.95E+5nMAssay Description:Blockade of peak Kv1.3 potassium currentsMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily A member 3(Mus musculus)
University Of Kiel
Curated by ChEMBL
University Of Kiel
Curated by ChEMBL
Affinity DataKd: 1.01E+5nMAssay Description:Blockade of peak Kv1.3 potassium currentsMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily C member 1(Homo sapiens (Human))
University Of Kiel
Curated by ChEMBL
University Of Kiel
Curated by ChEMBL
Affinity DataKd: 1.11E+5nMAssay Description:Blockade of peak K+ currents against Kv3.1 geneMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily A member 3(Mus musculus)
University Of Kiel
Curated by ChEMBL
University Of Kiel
Curated by ChEMBL
Affinity DataKd: 2.80E+4nMAssay Description:Blockade of peak Kv1.3 potassium currentsMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily A member 3(Mus musculus)
University Of Kiel
Curated by ChEMBL
University Of Kiel
Curated by ChEMBL
Affinity DataKd: 2.80E+4nMAssay Description:Blockade of peak Kv1.3 potassium currentsMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily C member 1(Homo sapiens (Human))
University Of Kiel
Curated by ChEMBL
University Of Kiel
Curated by ChEMBL
Affinity DataKd: 1.78E+5nMAssay Description:Blockade of peak K+ currents against Kv3.1 geneMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily A member 1(Homo sapiens (Human))
University Of Kiel
Curated by ChEMBL
University Of Kiel
Curated by ChEMBL
Affinity DataKd: 2.90E+5nMAssay Description:Blockade of peak K+ currents against Kv1.1 geneMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily A member 2(Homo sapiens (Human))
University Of Kiel
Curated by ChEMBL
University Of Kiel
Curated by ChEMBL
Affinity DataKd: 4.10E+4nMAssay Description:Blockade of peak K+ currents against Kv1.2 geneMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily A member 1(Homo sapiens (Human))
University Of Kiel
Curated by ChEMBL
University Of Kiel
Curated by ChEMBL
Affinity DataKd: 1.67E+5nMAssay Description:Blockade of peak K+ currents against Kv1.1 geneMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily A member 6(Homo sapiens (Human))
University Of Kiel
Curated by ChEMBL
University Of Kiel
Curated by ChEMBL
Affinity DataKd: 1.87E+5nMAssay Description:Blockade of peak K+ currents against Kv1.6 geneMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily A member 1(Homo sapiens (Human))
University Of Kiel
Curated by ChEMBL
University Of Kiel
Curated by ChEMBL
Affinity DataKd: 5.60E+4nMAssay Description:Blockade of peak K+ currents against Kv1.1 geneMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily A member 2(Homo sapiens (Human))
University Of Kiel
Curated by ChEMBL
University Of Kiel
Curated by ChEMBL
Affinity DataKd: 2.30E+4nMAssay Description:Blockade of peak K+ currents against Kv1.2 geneMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily C member 1(Homo sapiens (Human))
University Of Kiel
Curated by ChEMBL
University Of Kiel
Curated by ChEMBL
Affinity DataKd: 2.90E+4nMAssay Description:Blockade of peak K+ currents against Kv3.1 geneMore data for this Ligand-Target Pair