Compile Data Set for Download or QSAR
maximum 50k data
Found 426 with Last Name = 'hallberg' and Initial = 'm'
TargetType-2 angiotensin II receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50030815(CHEMBL404594)
Affinity DataKi:  0.140nMAssay Description:Binding affinity to AT2 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50009338((S)-2-((S)-1-((S)-2-((S)-2-((S)-2-((S)-2-((S)-5-(d...)
Affinity DataKi:  0.220nMAssay Description:Binding affinity to AT1 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Rattus norvegicus (rat))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50436546(CHEMBL2397481)
Affinity DataKi:  0.300nMAssay Description:Binding affinity to substance P receptor (1 to 7 amino acids) binding site in rat spinal cord membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Rattus norvegicus (rat))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50436546(CHEMBL2397481)
Affinity DataKi:  0.300nMAssay Description:Displacement of [3H]SP1-7 from NK1 receptor in Sprague-Dawley rat spinal cord membranes after 60 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-2 angiotensin II receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50009338((S)-2-((S)-1-((S)-2-((S)-2-((S)-2-((S)-2-((S)-5-(d...)
Affinity DataKi:  0.380nMAssay Description:Binding affinity to AT2 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-2 angiotensin II receptor(Sus scrofa)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50156173((1-((2'-(1H-tetrazol-5-yl)biphenyl-4-yl)methyl)-2-...)
Affinity DataKi:  0.400nMAssay Description:Displacement of [I125I]AngII form pig AT2 receptor myometrial membrane incubated for 1.5 hrs by gamma counting methodMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetType-2 angiotensin II receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50156173((1-((2'-(1H-tetrazol-5-yl)biphenyl-4-yl)methyl)-2-...)
Affinity DataKi:  0.400nMAssay Description:Binding affinity to AT2 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-2 angiotensin II receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50199311(CHEMBL215160 | N-butyloxycarbonyl-2-(4-imidazol-1-...)
Affinity DataKi:  0.5nMAssay Description:Displacement of [125I]Ang2 from AT2 receptor in pig uterus membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-2 angiotensin II receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50199326(CHEMBL217673 | N-butyloxycarbonyl-2-(4-imidazol-1-...)
Affinity DataKi:  0.600nMAssay Description:Displacement of [125I]Ang2 from AT2 receptor in pig uterus membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50030815(CHEMBL404594)
Affinity DataKi:  0.650nMAssay Description:Binding affinity to AT1 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-2 angiotensin II receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50199331(CHEMBL216250 | N-(1-butyloxy-methylcarbonyl)-3-(4-...)
Affinity DataKi:  1nMAssay Description:Displacement of [125I]Ang2 from AT2 receptor in pig uterus membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50049189(3-[4-(2-Ethyl-57-dimethyl-imidazo[45-b]pyridin-3-y...)
Affinity DataKi:  1.10nMAssay Description:Displacement of 125I-[Sar1,Ile8]ANGII form AT1 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetType-2 angiotensin II receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50594171(CHEMBL5186237)
Affinity DataKi:  1.20nMAssay Description:Displacement of 125I-[Sar1,Ile8]ANGII form recombinant human full length AT2 receptor expressed in HEK293 cells incubated for 120 mins by scintillati...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetType-2 angiotensin II receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50594186(CHEMBL5174659)
Affinity DataKi:  1.40nMAssay Description:Displacement of 125I-[Sar1,Ile8]ANGII form recombinant human full length AT2 receptor expressed in HEK293 cells incubated for 120 mins by scintillati...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetSubstance-P receptor(Rattus norvegicus (rat))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50188489((S)-2-Amino-N-((S)-1-carbamoyl-2-phenyl-ethyl)-3-p...)
Affinity DataKi:  1.5nMAssay Description:Displacement of [3H]SP1-7 from NK1 receptor in Sprague-Dawley rat spinal cord membranes after 60 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50188489((S)-2-Amino-N-((S)-1-carbamoyl-2-phenyl-ethyl)-3-p...)
Affinity DataKi:  1.5nMAssay Description:Binding affinity to NK1 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50188489((S)-2-Amino-N-((S)-1-carbamoyl-2-phenyl-ethyl)-3-p...)
Affinity DataKi:  1.5nMAssay Description:Displacement of [3H]-SP1-7 from NK1 receptor (unknown origin) by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Rattus norvegicus (rat))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50188489((S)-2-Amino-N-((S)-1-carbamoyl-2-phenyl-ethyl)-3-p...)
Affinity DataKi:  1.5nMAssay Description:Displacement of [3H]SP1-7 from NK1 receptor in Sprague-Dawley rat spinal cord membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Rattus norvegicus (rat))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50308381(CHEMBL589979 | H-Arg-Pro-Lys-Pro-Gln-Gln-Phe-OH)
Affinity DataKi:  1.60nMAssay Description:Displacement of [3H]SP1-7 from NK1 receptor in Sprague-Dawley rat spinal cord membranes after 60 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Rattus norvegicus (rat))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50308381(CHEMBL589979 | H-Arg-Pro-Lys-Pro-Gln-Gln-Phe-OH)
Affinity DataKi:  1.60nMAssay Description:Binding affinity to substance P receptor (1 to 7 amino acids) binding site in rat spinal cord membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Rattus norvegicus (rat))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50308381(CHEMBL589979 | H-Arg-Pro-Lys-Pro-Gln-Gln-Phe-OH)
Affinity DataKi:  1.60nMAssay Description:Displacement of [3H]SP1-7 from NK1 receptor in Sprague-Dawley rat spinal cord membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Rattus norvegicus (rat))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50276158(CHEMBL4127872)
Affinity DataKi:  1.80nMAssay Description:Displacement of [3H]SP1-7 from NK1 receptor in Sprague-Dawley rat spinal cord membranes after 60 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucyl-cystinyl aminopeptidase(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50346448(2-(2-(((2S,6S,13S,E)-13-Amino-2-(4-hydroxybenzyl)-...)
Affinity DataKi:  1.80nMAssay Description:Inhibition of catalytic activity of recombinant human IRAP transfected in human HEK-293 cells assessed as clevage of substrate L-leucine-p-nitroanili...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-2 angiotensin II receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50156173((1-((2'-(1H-tetrazol-5-yl)biphenyl-4-yl)methyl)-2-...)
Affinity DataKi:  1.80nMAssay Description:Agonist activity at AT2 receptor in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetType-2 angiotensin II receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50049189(3-[4-(2-Ethyl-57-dimethyl-imidazo[45-b]pyridin-3-y...)
Affinity DataKi:  2nMAssay Description:Displacement of 125I-[Sar1,Ile8]ANGII form AT2 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetType-2 angiotensin II receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50199317(CHEMBL214525 | N-ethyloxycarbonyl-2-(4-imidazol-1-...)
Affinity DataKi:  2nMAssay Description:Displacement of [125I]Ang2 from AT2 receptor in pig uterus membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Rattus norvegicus (rat))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50436553(CHEMBL2396664)
Affinity DataKi:  2.20nMAssay Description:Displacement of [3H]SP1-7 from NK1 receptor in Sprague-Dawley rat spinal cord membranes after 60 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Rattus norvegicus (rat))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50436553(CHEMBL2396664)
Affinity DataKi:  2.20nMAssay Description:Displacement of [3H]SP1-7 from substance P receptor (1 to 7 amino acids) binding site in Sprague-Dawley rat spinal cord membranes after 60 mins by li...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50436553(CHEMBL2396664)
Affinity DataKi:  2.20nMAssay Description:Displacement of [3H]-SP1-7 from NK1 receptor (unknown origin) by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50436553(CHEMBL2396664)
Affinity DataKi:  2.20nMAssay Description:Binding affinity to NK1 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-2 angiotensin II receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50594170(CHEMBL5174923)
Affinity DataKi:  2.70nMAssay Description:Displacement of 125I-[Sar1,Ile8]ANGII form recombinant human full length AT2 receptor expressed in HEK293 cells incubated for 120 mins by scintillati...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetType-2 angiotensin II receptor(Sus scrofa)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50049189(3-[4-(2-Ethyl-57-dimethyl-imidazo[45-b]pyridin-3-y...)
Affinity DataKi:  2.80nMAssay Description:Displacement of [I125I]AngII form pig AT2 receptor myometrial membrane incubated for 1.5 hrs by gamma counting methodMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetType-2 angiotensin II receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50594187(CHEMBL5179119)
Affinity DataKi:  3.20nMAssay Description:Displacement of 125I-[Sar1,Ile8]ANGII form recombinant human full length AT2 receptor expressed in HEK293 cells incubated for 120 mins by scintillati...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetSubstance-P receptor(Rattus norvegicus (rat))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50436547(CHEMBL2397494)
Affinity DataKi:  3.30nMAssay Description:Displacement of [3H]SP1-7 from substance P receptor (1 to 7 amino acids) binding site in Sprague-Dawley rat spinal cord membranes after 60 mins by li...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucyl-cystinyl aminopeptidase(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50331042(2-(2-(((4R,8S,11S)-11-amino-8-(4-hydroxybenzyl)-6,...)
Affinity DataKi:  3.30nMAssay Description:Inhibition of catalytic activity of human recombinant IRAP expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetType-2 angiotensin II receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50156173((1-((2'-(1H-tetrazol-5-yl)biphenyl-4-yl)methyl)-2-...)
Affinity DataKi:  3.60nMAssay Description:Displacement of [125-I]-[Sar1Ile8]-angiotensin II from human AT2R expressed in HEK293 cell membrane assessed as inhibition constant by radioligand bi...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetType-1 angiotensin II receptor A(RAT)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50049189(3-[4-(2-Ethyl-57-dimethyl-imidazo[45-b]pyridin-3-y...)
Affinity DataKi:  3.90nMAssay Description:Displacement of [I125I]AngII form AT1 receptor in rat liver membrane incubated for 1.5 hrs by gamma counting methodMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetType-2 angiotensin II receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50600576(CHEMBL5177359)
Affinity DataKi:  4nMAssay Description:Displacement of [125-I]-[Sar1Ile8]-angiotensin II from human AT2R expressed in HEK293 cell membrane assessed as inhibition constant by radioligand bi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetType-2 angiotensin II receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50199318(CHEMBL384462 | N-(N-butyl-methylaminocarbonyl)-3-(...)
Affinity DataKi:  4nMAssay Description:Displacement of [125I]Ang2 from AT2 receptor in pig uterus membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucyl-cystinyl aminopeptidase(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50346455(2-(2-(((2S,5S,13S,E)-13-Amino-2-(4-hydroxybenzyl)-...)
Affinity DataKi:  4.10nMAssay Description:Inhibition of catalytic activity of recombinant human IRAP transfected in human HEK-293 cells assessed as clevage of substrate L-leucine-p-nitroanili...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-2 angiotensin II receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50600590(CHEMBL5207511)
Affinity DataKi:  4.5nMAssay Description:Displacement of [125-I]-[Sar1Ile8]-angiotensin II from human AT2R expressed in HEK293 cell membrane assessed as inhibition constant by radioligand bi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetType-2 angiotensin II receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50199312(CHEMBL217249 | N-butyloxycarbonyl-3-(4-imidazol-1-...)
Affinity DataKi:  5nMAssay Description:Displacement of [125I]Ang2 from AT2 receptor in pig uterus membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-2 angiotensin II receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50199321(CHEMBL214592 | N-butyloxycarbonyl-2-(4-imidazol-1-...)
Affinity DataKi:  5nMAssay Description:Displacement of [125I]Ang2 from AT2 receptor in pig uterus membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-2 angiotensin II receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50600586(CHEMBL5170220)
Affinity DataKi:  5.10nMAssay Description:Displacement of [125-I]-[Sar1Ile8]-angiotensin II from human AT2R expressed in HEK293 cell membrane assessed as inhibition constant by radioligand bi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetLeucyl-cystinyl aminopeptidase(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50331046(2-(2-(((5S,9S,12S)-12-amino-9-(4-hydroxybenzyl)-7,...)
Affinity DataKi:  5.20nMAssay Description:Inhibition of catalytic activity of human recombinant IRAP expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50041558(CHEMBL2042018)
Affinity DataKi:  5.20nMAssay Description:Displacement of [3H]-SP1-7 from NK1 receptor (unknown origin) by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50041558(CHEMBL2042018)
Affinity DataKi:  5.20nMAssay Description:Binding affinity to NK1 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Rattus norvegicus (rat))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50041558(CHEMBL2042018)
Affinity DataKi:  5.20nMAssay Description:Displacement of [3H]SP1-7 from NK1 receptor in Sprague-Dawley rat spinal cord membranes after 60 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-2 angiotensin II receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50600578(CHEMBL5176951)
Affinity DataKi:  5.30nMAssay Description:Displacement of [125-I]-[Sar1Ile8]-angiotensin II from human AT2R expressed in HEK293 cell membrane assessed as inhibition constant by radioligand bi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetType-2 angiotensin II receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50594184(CHEMBL5178751)
Affinity DataKi:  5.70nMAssay Description:Displacement of 125I-[Sar1,Ile8]ANGII form recombinant human full length AT2 receptor expressed in HEK293 cells incubated for 120 mins by scintillati...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
Displayed 1 to 50 (of 426 total ) | Next | Last >>
Jump to: