TargetHistone deacetylase 1(Homo sapiens (Human))
Broad Institute Of Mit And Harvard
Curated by ChEMBL
Broad Institute Of Mit And Harvard
Curated by ChEMBL
Affinity DataKi: <0.200nMAssay Description:Inhibition of C-terminal His-tagged and C-terminal FLAG-tagged full length human recombinant HDAC1 expressed in baculovirus coexpressed in fall armyw...More data for this Ligand-Target Pair
Affinity DataKi: 0.447nMAssay Description:Inhibition of N/OFQ binding to human Orphanin FQ receptor (Nociceptin/Orphanin)More data for this Ligand-Target Pair
Affinity DataKi: 0.525nMAssay Description:Inhibition of N/OFQ binding to human Orphanin FQ receptor (Nociceptin/Orphanin)More data for this Ligand-Target Pair
Affinity DataKi: 0.646nMAssay Description:Inhibition of N/OFQ binding to human Orphanin FQ receptor (Nociceptin/Orphanin)More data for this Ligand-Target Pair
Affinity DataKi: 0.661nMAssay Description:Inhibition of N/OFQ binding to human Orphanin FQ receptor (Nociceptin/Orphanin)More data for this Ligand-Target Pair
Affinity DataKi: 0.776nMAssay Description:Inhibition of N/OFQ binding to human Orphanin FQ receptor (Nociceptin/Orphanin)More data for this Ligand-Target Pair
Affinity DataKi: 1.20nMAssay Description:Inhibition of N/OFQ binding to human Orphanin FQ receptor (Nociceptin/Orphanin)More data for this Ligand-Target Pair
Affinity DataKi: 1.20nMAssay Description:Inhibition of N/OFQ binding to human Orphanin FQ receptor (Nociceptin/Orphanin)More data for this Ligand-Target Pair
TargetHistone deacetylase 2(Homo sapiens (Human))
Broad Institute Of Mit And Harvard
Curated by ChEMBL
Broad Institute Of Mit And Harvard
Curated by ChEMBL
Affinity DataKi: 1.5nMAssay Description:Inhibition full length human recombinant HDAC2 expressed in baculovirus coexpressed in fall armyworm Sf9 cells using carboxyfluorescein (FAM)-labeled...More data for this Ligand-Target Pair
Affinity DataKi: 1.70nMAssay Description:Inhibition of N/OFQ binding to human Orphanin FQ receptor (Nociceptin/Orphanin)More data for this Ligand-Target Pair
Affinity DataKi: 1.70nMAssay Description:Inhibition of N/OFQ binding to human Orphanin FQ receptor (Nociceptin/Orphanin)More data for this Ligand-Target Pair
Affinity DataKi: 2.10nMAssay Description:Inhibition of N/OFQ binding to human Orphanin FQ receptor (Nociceptin/Orphanin)More data for this Ligand-Target Pair
Affinity DataKi: 2.10nMAssay Description:Inhibition of N/OFQ binding to human Orphanin FQ receptor (Nociceptin/Orphanin)More data for this Ligand-Target Pair
Affinity DataKi: 2.20nMAssay Description:Inhibition of N/OFQ binding to human Orphanin FQ receptor (Nociceptin/Orphanin)More data for this Ligand-Target Pair
Affinity DataKi: 11nM IC50: 15nMAssay Description:DPP-IV inhibitors were measured for their ability to inhibit DPP-IV mediated cleavage of Ala-Pro-7-amido-4-trifluoromethylcoumarin in a fluorogenic a...More data for this Ligand-Target Pair
Affinity DataKi: 27nMAssay Description:Inhibition of naloxone binding to human Opioid receptor kappa 1More data for this Ligand-Target Pair
Affinity DataKi: 56nMAssay Description:Inhibition of naloxone binding to human Opioid receptor kappa 1More data for this Ligand-Target Pair
TargetHistone deacetylase 1(Homo sapiens (Human))
Broad Institute Of Mit And Harvard
Curated by ChEMBL
Broad Institute Of Mit And Harvard
Curated by ChEMBL
Affinity DataKi: 84nMAssay Description:Inhibition of C-terminal His-tagged and C-terminal FLAG-tagged full length human recombinant HDAC1 expressed in baculovirus coexpressed in fall armyw...More data for this Ligand-Target Pair
Affinity DataKi: 87nMAssay Description:Inhibition of DAMGO binding to human Opioid receptor mu 1More data for this Ligand-Target Pair
Affinity DataKi: 132nMAssay Description:Inhibition of naloxone binding to human Opioid receptor kappa 1More data for this Ligand-Target Pair
Affinity DataKi: 132nMAssay Description:Inhibition of naloxone binding to human Opioid receptor kappa 1More data for this Ligand-Target Pair
Affinity DataKi: 135nMAssay Description:Inhibition of DAMGO binding to human Opioid receptor mu 1More data for this Ligand-Target Pair
Affinity DataKi: 148nMAssay Description:Inhibition of naloxone binding to human Opioid receptor kappa 1More data for this Ligand-Target Pair
Affinity DataKi: 155nMAssay Description:Inhibition of DAMGO binding to human Opioid receptor mu 1More data for this Ligand-Target Pair
Affinity DataKi: 155nMAssay Description:Inhibition of naloxone binding to human Opioid receptor kappa 1More data for this Ligand-Target Pair
Affinity DataKi: 170nMAssay Description:Inhibition of naloxone binding to human Opioid receptor kappa 1More data for this Ligand-Target Pair
Affinity DataKi: 174nMAssay Description:Inhibition of DAMGO binding to human Opioid receptor mu 1More data for this Ligand-Target Pair
TargetHistone deacetylase 1(Homo sapiens (Human))
Broad Institute Of Mit And Harvard
Curated by ChEMBL
Broad Institute Of Mit And Harvard
Curated by ChEMBL
Affinity DataKi: 176nMAssay Description:Inhibition of C-terminal His-tagged and C-terminal FLAG-tagged full length human recombinant HDAC1 expressed in baculovirus coexpressed in fall armyw...More data for this Ligand-Target Pair
Affinity DataKi: 178nMAssay Description:Inhibition of DAMGO binding to human Opioid receptor mu 1More data for this Ligand-Target Pair
Affinity DataKi: 219nMAssay Description:Inhibition of deltorphin II binding to human Opioid receptor delta 1More data for this Ligand-Target Pair
Affinity DataKi: 251nMAssay Description:Inhibition of naloxone binding to human Opioid receptor kappa 1More data for this Ligand-Target Pair
Affinity DataKi: 257nMAssay Description:Inhibition of naloxone binding to human Opioid receptor kappa 1More data for this Ligand-Target Pair
Affinity DataKi: 275nMAssay Description:Inhibition of DAMGO binding to human Opioid receptor mu 1More data for this Ligand-Target Pair
Affinity DataKi: 282nMAssay Description:Inhibition of naloxone binding to human Opioid receptor kappa 1More data for this Ligand-Target Pair
Affinity DataKi: 309nMAssay Description:Inhibition of naloxone binding to human Opioid receptor kappa 1More data for this Ligand-Target Pair
Affinity DataKi: 338nMAssay Description:Inhibition of DAMGO binding to human Opioid receptor mu 1More data for this Ligand-Target Pair
Affinity DataKi: 339nMAssay Description:Inhibition of DAMGO binding to human Opioid receptor mu 1More data for this Ligand-Target Pair
Affinity DataKi: 372nMAssay Description:Inhibition of deltorphin II binding to human Opioid receptor delta 1More data for this Ligand-Target Pair
Affinity DataKi: 389nMAssay Description:Inhibition of deltorphin II binding to human Opioid receptor delta 1More data for this Ligand-Target Pair
Affinity DataKi: 417nMAssay Description:Inhibition of DAMGO binding to human Opioid receptor mu 1More data for this Ligand-Target Pair
TargetHistone deacetylase 3(Homo sapiens (Human))
Broad Institute Of Mit And Harvard
Curated by ChEMBL
Broad Institute Of Mit And Harvard
Curated by ChEMBL
Affinity DataKi: 500nMAssay Description:Inhibition full length human recombinant HDAC3 expressed in baculovirus using carboxyfluorescein (FAM)-labeled acetylated/ trifluoroacetylated peptid...More data for this Ligand-Target Pair
Affinity DataKi: 501nMAssay Description:Inhibition of DAMGO binding to human Opioid receptor mu 1More data for this Ligand-Target Pair
Affinity DataKi: 513nMAssay Description:Inhibition of naloxone binding to human Opioid receptor kappa 1More data for this Ligand-Target Pair
TargetHistone deacetylase 2(Homo sapiens (Human))
Broad Institute Of Mit And Harvard
Curated by ChEMBL
Broad Institute Of Mit And Harvard
Curated by ChEMBL
Affinity DataKi: 519nMAssay Description:Inhibition full length human recombinant HDAC2 expressed in baculovirus coexpressed in fall armyworm Sf9 cells using carboxyfluorescein (FAM)-labeled...More data for this Ligand-Target Pair
Affinity DataKi: 661nMAssay Description:Inhibition of DAMGO binding to human Opioid receptor mu 1More data for this Ligand-Target Pair
Affinity DataKi: 724nMAssay Description:Inhibition of DAMGO binding to human Opioid receptor mu 1More data for this Ligand-Target Pair
Affinity DataKi: 891nMAssay Description:Inhibition of deltorphin II binding to human Opioid receptor delta 1More data for this Ligand-Target Pair
Affinity DataKi: 912nMAssay Description:Inhibition of deltorphin II binding to human Opioid receptor delta 1More data for this Ligand-Target Pair
Affinity DataKi: 933nMAssay Description:Inhibition of deltorphin II binding to human Opioid receptor delta 1More data for this Ligand-Target Pair
Affinity DataKi: 1.02E+3nMAssay Description:Inhibition of deltorphin II binding to human Opioid receptor delta 1More data for this Ligand-Target Pair