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Found 245 with Last Name = 'henning' and Initial = 'r'
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Department of Veterans Affairs Medical Center

Curated by PDSP Ki Database
LigandPNGBDBM21397(8-[4-(4-fluorophenyl)-4-keto-butyl]-1-phenyl-1,3,8...)
Affinity DataKi:  0.100nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Department of Veterans Affairs Medical Center

Curated by PDSP Ki Database
LigandPNGBDBM21397(8-[4-(4-fluorophenyl)-4-keto-butyl]-1-phenyl-1,3,8...)
Affinity DataKi:  0.110nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Department of Veterans Affairs Medical Center

Curated by PDSP Ki Database
LigandPNGBDBM21397(8-[4-(4-fluorophenyl)-4-keto-butyl]-1-phenyl-1,3,8...)
Affinity DataKi:  0.120nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Department of Veterans Affairs Medical Center

Curated by PDSP Ki Database
LigandPNGBDBM50008735((+)-3-(tert-butyl)-(3S,4aS,13bS)-2,3,4,4a,8,9,13b,...)
In DepthDetails PubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Department of Veterans Affairs Medical Center

Curated by PDSP Ki Database
LigandPNGBDBM50008735((+)-3-(tert-butyl)-(3S,4aS,13bS)-2,3,4,4a,8,9,13b,...)
Affinity DataKi:  2.20nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Department of Veterans Affairs Medical Center

Curated by PDSP Ki Database
LigandPNGBDBM50008735((+)-3-(tert-butyl)-(3S,4aS,13bS)-2,3,4,4a,8,9,13b,...)
Affinity DataKi:  2.5nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Department of Veterans Affairs Medical Center

Curated by PDSP Ki Database
LigandPNGBDBM21398(4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1...)
Affinity DataKi:  5.40nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAlpha-2C adrenergic receptor(RAT)
Department of Veterans Affairs Medical Center

Curated by PDSP Ki Database
LigandPNGBDBM50019848(2-(2,3-dihydro-1,4-benzodioxin-2-yl)-4,5-dihydro-1...)
Affinity DataKi:  7.90nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetD(2) dopamine receptor(BOVINE)
TBA

Curated by ChEMBL
LigandPNGBDBM50019719(5-Fluoro-1-[1-(5-methyl-2,3-dihydro-benzo[1,4]diox...)
Affinity DataKi:  8nMAssay Description:Displacement of [3H]-spiroperidol from bovine caudate nucleus membrane Dopamine receptor D2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(BOVINE)
TBA

Curated by ChEMBL
LigandPNGBDBM21398(4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1...)
Affinity DataKi:  20nMAssay Description:Binding affinity towards dopamine receptor D2 was determined by displacement of [3H]-spiroperidol from bovine nucleus caudate membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Department of Veterans Affairs Medical Center

Curated by PDSP Ki Database
LigandPNGBDBM11638(CHEMBL26 | Compound 7 | N-[(1-ethylpyrrolidin-2-yl...)
Affinity DataKi:  23nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetD(2) dopamine receptor(BOVINE)
TBA

Curated by ChEMBL
LigandPNGBDBM50019721(1-[1-(6,7-Dimethyl-2,3-dihydro-benzo[1,4]dioxin-2-...)
Affinity DataKi:  25nMAssay Description:Displacement of [3H]-spiroperidol from bovine caudate nucleus membrane Dopamine receptor D2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(BOVINE)
TBA

Curated by ChEMBL
LigandPNGBDBM50019726(1-[1-(7-Chloro-2,3-dihydro-benzo[1,4]dioxin-2-ylme...)
Affinity DataKi:  30nMAssay Description:Binding affinity towards dopamine receptor D2 was determined by displacement of [3H]-spiroperidol from bovine nucleus caudate membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(BOVINE)
TBA

Curated by ChEMBL
LigandPNGBDBM50019717(5-Chloro-1-[1-(2,3-dihydro-benzo[1,4]dioxin-2-ylme...)
Affinity DataKi:  30nMAssay Description:Displacement of [3H]-spiroperidol from bovine caudate nucleus membrane Dopamine receptor D2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2C adrenergic receptor(RAT)
Department of Veterans Affairs Medical Center

Curated by PDSP Ki Database
LigandPNGBDBM35256((S)-mianserin | Lerivon | MIANSERIN | MIANSERIN (+...)
Affinity DataKi:  40nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetD(2) dopamine receptor(BOVINE)
TBA

Curated by ChEMBL
LigandPNGBDBM50019725(5-Methyl-1-[1-(6-methyl-2,3-dihydro-benzo[1,4]diox...)
Affinity DataKi:  40nMAssay Description:Displacement of [3H]-spiroperidol from bovine caudate nucleus membrane Dopamine receptor D2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Department of Veterans Affairs Medical Center

Curated by PDSP Ki Database
LigandPNGBDBM11638(CHEMBL26 | Compound 7 | N-[(1-ethylpyrrolidin-2-yl...)
Affinity DataKi:  42nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Department of Veterans Affairs Medical Center

Curated by PDSP Ki Database
LigandPNGBDBM11638(CHEMBL26 | Compound 7 | N-[(1-ethylpyrrolidin-2-yl...)
Affinity DataKi:  42nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetD(2) dopamine receptor(BOVINE)
TBA

Curated by ChEMBL
LigandPNGBDBM50019727(1-[1-(6,7-Dimethyl-2,3-dihydro-benzo[1,4]dioxin-2-...)
Affinity DataKi:  45nMAssay Description:Displacement of [3H]-spiroperidol from bovine caudate nucleus membrane Dopamine receptor D2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2C adrenergic receptor(RAT)
Department of Veterans Affairs Medical Center

Curated by PDSP Ki Database
LigandPNGBDBM50016897(2-(2,6-dichloroanilino)-1,3-diazacyclopentene-(2) ...)
Affinity DataKi:  47nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetD(2) dopamine receptor(BOVINE)
TBA

Curated by ChEMBL
LigandPNGBDBM50019724(5-Chloro-1-[1-(6-methyl-2,3-dihydro-benzo[1,4]diox...)
Affinity DataKi:  60nMAssay Description:Displacement of [3H]-spiroperidol from bovine caudate nucleus membrane Dopamine receptor D2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(BOVINE)
TBA

Curated by ChEMBL
LigandPNGBDBM50019728(5-Bromo-1-[1-(2,3-dihydro-benzo[1,4]dioxin-2-ylmet...)
Affinity DataKi:  70nMAssay Description:Displacement of [3H]-spiroperidol from bovine caudate nucleus membrane Dopamine receptor D2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(BOVINE)
TBA

Curated by ChEMBL
LigandPNGBDBM50019718(5-Fluoro-1-[1-(6-fluoro-2,3-dihydro-benzo[1,4]diox...)
Affinity DataKi:  70nMAssay Description:Displacement of [3H]-spiroperidol from bovine caudate nucleus membrane Dopamine receptor D2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(BOVINE)
TBA

Curated by ChEMBL
LigandPNGBDBM50019723(1-[1-(2,3-Dihydro-benzo[1,4]dioxin-2-ylmethyl)-pip...)
Affinity DataKi:  120nMAssay Description:Displacement of [3H]-spiroperidol from bovine caudate nucleus membrane Dopamine receptor D2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(BOVINE)
TBA

Curated by ChEMBL
LigandPNGBDBM50019720(1-[1-(7-Fluoro-2,3-dihydro-benzo[1,4]dioxin-2-ylme...)
Affinity DataKi:  150nMAssay Description:Displacement of [3H]-spiroperidol from bovine caudate nucleus membrane Dopamine receptor D2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(BOVINE)
TBA

Curated by ChEMBL
LigandPNGBDBM50019722(1-[1-(2,3-Dihydro-benzo[1,4]dioxin-2-ylmethyl)-pip...)
Affinity DataKi:  150nMAssay Description:Displacement of [3H]-spiroperidol from bovine caudate nucleus membrane Dopamine receptor D2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2C adrenergic receptor(RAT)
Department of Veterans Affairs Medical Center

Curated by PDSP Ki Database
LigandPNGBDBM50008735((+)-3-(tert-butyl)-(3S,4aS,13bS)-2,3,4,4a,8,9,13b,...)
Affinity DataKi:  158nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Department of Veterans Affairs Medical Center

Curated by PDSP Ki Database
LigandPNGBDBM35256((S)-mianserin | Lerivon | MIANSERIN | MIANSERIN (+...)
Affinity DataKi:  3.20E+3nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAlpha-2C adrenergic receptor(RAT)
Department of Veterans Affairs Medical Center

Curated by PDSP Ki Database
LigandPNGBDBM11638(CHEMBL26 | Compound 7 | N-[(1-ethylpyrrolidin-2-yl...)
Affinity DataKi:  4.30E+3nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAlpha-2C adrenergic receptor(RAT)
Department of Veterans Affairs Medical Center

Curated by PDSP Ki Database
LigandPNGBDBM21398(4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1...)
Affinity DataKi:  7.10E+3nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Department of Veterans Affairs Medical Center

Curated by PDSP Ki Database
LigandPNGBDBM81926(Aminoclonidine, p | CAS_66711-21-5 | NSC_51763 | p...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Department of Veterans Affairs Medical Center

Curated by PDSP Ki Database
LigandPNGBDBM50016897(2-(2,6-dichloroanilino)-1,3-diazacyclopentene-(2) ...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Department of Veterans Affairs Medical Center

Curated by PDSP Ki Database
LigandPNGBDBM50019848(2-(2,3-dihydro-1,4-benzodioxin-2-yl)-4,5-dihydro-1...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAlpha-2C adrenergic receptor(RAT)
Department of Veterans Affairs Medical Center

Curated by PDSP Ki Database
LigandPNGBDBM21397(8-[4-(4-fluorophenyl)-4-keto-butyl]-1-phenyl-1,3,8...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetRenin(Homo sapiens (Human))
Hoechst

Curated by ChEMBL
LigandPNGBDBM50045686(4-(4-Amino-piperidin-1-yl)-N-[1-(1-cyclohexylmethy...)
Affinity DataIC50:  0.130nMAssay Description:In vitro inhibition of purified human kidney reninMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Homo sapiens (Human))
Hoechst

Curated by ChEMBL
LigandPNGBDBM50045691(CHEMBL94827 | Methyl-{2-[methyl-(morpholine-4-carb...)
Affinity DataIC50:  0.160nMAssay Description:In vitro inhibition of purified human kidney reninMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Homo sapiens (Human))
Hoechst

Curated by ChEMBL
LigandPNGBDBM50045691(CHEMBL94827 | Methyl-{2-[methyl-(morpholine-4-carb...)
Affinity DataIC50:  0.160nMAssay Description:In vitro inhibition of renin in human plasmaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Homo sapiens (Human))
Hoechst

Curated by ChEMBL
LigandPNGBDBM50045687(2-Benzyl-N-[1-(1-cyclohexylmethyl-2,3-dihydroxy-5-...)
Affinity DataIC50:  0.170nMAssay Description:In vitro inhibition of renin in human plasmaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Homo sapiens (Human))
Hoechst

Curated by ChEMBL
LigandPNGBDBM50045683(4-(4-Amino-piperidin-1-yl)-2-benzyl-N-[1-(1-cycloh...)
Affinity DataIC50:  0.240nMAssay Description:In vitro inhibition of renin in human plasmaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Homo sapiens (Human))
Hoechst

Curated by ChEMBL
LigandPNGBDBM50045685(4-(4-Amino-piperidin-1-yl)-2-benzyl-N-[1-(1-cycloh...)
Affinity DataIC50:  0.25nMAssay Description:In vitro inhibition of purified human kidney reninMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50426601(CHEMBL2325895)
Affinity DataIC50:  0.260nMAssay Description:Inhibition of JAK3 (unknown origin)-mediated phosphorylation of Biotin-KAIETDKEYYTVKD incubated for 10 mins prior to substrate addition measured afte...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Homo sapiens (Human))
Hoechst

Curated by ChEMBL
LigandPNGBDBM50045685(4-(4-Amino-piperidin-1-yl)-2-benzyl-N-[1-(1-cycloh...)
Affinity DataIC50:  0.260nMAssay Description:In vitro inhibition of purified human kidney reninMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Homo sapiens (Human))
Hoechst

Curated by ChEMBL
LigandPNGBDBM50045692(3-(4-Amino-cyclohexanesulfonyl)-2-benzyl-N-[1-(1-c...)
Affinity DataIC50:  0.310nMAssay Description:In vitro inhibition of purified human kidney reninMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Homo sapiens (Human))
Hoechst

Curated by ChEMBL
LigandPNGBDBM50045692(3-(4-Amino-cyclohexanesulfonyl)-2-benzyl-N-[1-(1-c...)
Affinity DataIC50:  0.310nMAssay Description:In vitro inhibition of purified human kidney reninMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Homo sapiens (Human))
Hoechst

Curated by ChEMBL
LigandPNGBDBM50045693(4-Amino-piperidine-1-carboxylic acid 1-[1-(1-cyclo...)
Affinity DataIC50:  0.370nMAssay Description:In vitro inhibition of renin in human plasmaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Homo sapiens (Human))
Hoechst

Curated by ChEMBL
LigandPNGBDBM50045693(4-Amino-piperidine-1-carboxylic acid 1-[1-(1-cyclo...)
Affinity DataIC50:  0.370nMAssay Description:In vitro inhibition of renin in human plasmaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Homo sapiens (Human))
Hoechst

Curated by ChEMBL
LigandPNGBDBM50045683(4-(4-Amino-piperidin-1-yl)-2-benzyl-N-[1-(1-cycloh...)
Affinity DataIC50:  0.380nMAssay Description:In vitro inhibition of purified human kidney reninMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Homo sapiens (Human))
Hoechst

Curated by ChEMBL
LigandPNGBDBM50045683(4-(4-Amino-piperidin-1-yl)-2-benzyl-N-[1-(1-cycloh...)
Affinity DataIC50:  0.390nMAssay Description:In vitro inhibition of purified human kidney reninMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Homo sapiens (Human))
Hoechst

Curated by ChEMBL
LigandPNGBDBM50045687(2-Benzyl-N-[1-(1-cyclohexylmethyl-2,3-dihydroxy-5-...)
Affinity DataIC50:  0.430nMAssay Description:In vitro inhibition of renin in human plasmaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50426599(CHEMBL2325898)
Affinity DataIC50:  0.440nMAssay Description:Inhibition of JAK3 (unknown origin)-mediated phosphorylation of Biotin-KAIETDKEYYTVKD incubated for 10 mins prior to substrate addition measured afte...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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