Affinity DataKi: 4nMAssay Description:In vitro inhibition of Histamine H2 receptor by measuring its ability to block the histamine-stimulated adenylate cyclase of guinea pig hippocampal h...More data for this Ligand-Target Pair
Affinity DataKi: 6.30nMAssay Description:In vitro inhibition of Histamine H2 receptor by measuring its ability to block the histamine-stimulated adenylate cyclase of guinea pig hippocampal h...More data for this Ligand-Target Pair
Affinity DataKi: 6.30nMAssay Description:In vitro inhibition of Histamine H2 receptor by measuring its ability to block the histamine-stimulated adenylate cyclase of guinea pig hippocampal h...More data for this Ligand-Target Pair
Affinity DataKi: 32nMAssay Description:Evaluated in vitro for Histamine H2 receptor inhibition using the dimaprit stimulated chronotropic response of the guinea pig atriumMore data for this Ligand-Target Pair
Affinity DataKi: 58nMAssay Description:Compound was evaluated for its inhibitory activity against human thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 160nMAssay Description:Compound was evaluated for its inhibitory activity against human thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 200nMAssay Description:Evaluated in vitro for Histamine H2 receptor inhibition using the dimaprit stimulated chronotropic response of the guinea pig atriumMore data for this Ligand-Target Pair
Affinity DataKi: 316nMAssay Description:Evaluated in vitro for Histamine H2 receptor inhibition using the dimaprit stimulated chronotropic response of the guinea pig atriumMore data for this Ligand-Target Pair
Affinity DataKi: 316nMAssay Description:Evaluated in vitro for Histamine H2 receptor inhibition using the dimaprit stimulated chronotropic response of the guinea pig atriumMore data for this Ligand-Target Pair
Affinity DataKi: 398nMAssay Description:Evaluated in vitro for Histamine H2 receptor inhibition using the dimaprit stimulated chronotropic response of the guinea pig atriumMore data for this Ligand-Target Pair
Affinity DataKi: 501nMAssay Description:In vitro inhibition of Histamine H2 receptor by measuring its ability to block the histamine-stimulated adenylate cyclase of guinea pig hippocampal h...More data for this Ligand-Target Pair
Affinity DataKi: 501nMAssay Description:In vitro inhibition of Histamine H2 receptor by measuring its ability to block the histamine-stimulated adenylate cyclase of guinea pig hippocampal h...More data for this Ligand-Target Pair
Affinity DataKi: 501nMAssay Description:Evaluated in vitro for Histamine H2 receptor inhibition using the dimaprit stimulated chronotropic response of the guinea pig atriumMore data for this Ligand-Target Pair
Affinity DataKi: 700nMAssay Description:Compound was evaluated for its inhibitory activity against human thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 794nMAssay Description:Evaluated in vitro for Histamine H2 receptor inhibition using the dimaprit stimulated chronotropic response of the guinea pig atriumMore data for this Ligand-Target Pair
Affinity DataKi: 1.30E+3nMAssay Description:Compound was evaluated for its inhibitory activity against human thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 4.70E+3nMAssay Description:Compound was evaluated for its inhibitory activity against human thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 7.90E+3nMAssay Description:Compound was evaluated for its inhibitory activity against human thrombinMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Compound was evaluated for its inhibitory activity against human thrombinMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Compound was evaluated for its inhibitory activity against trypsinMore data for this Ligand-Target Pair
Affinity DataKi: 1.58E+4nMAssay Description:Evaluated in vitro for Histamine H2 receptor inhibition using the dimaprit stimulated chronotropic response of the guinea pig atriumMore data for this Ligand-Target Pair
Affinity DataKi: 1.60E+4nMAssay Description:Compound was evaluated for its inhibitory activity against trypsinMore data for this Ligand-Target Pair
Affinity DataKi: 3.16E+4nMAssay Description:Evaluated in vitro for Histamine H2 receptor inhibition using the dimaprit stimulated chronotropic response of the guinea pig atriumMore data for this Ligand-Target Pair
Affinity DataKi: 3.98E+4nMAssay Description:Evaluated in vitro for Histamine H2 receptor inhibition using the dimaprit stimulated chronotropic response of the guinea pig atriumMore data for this Ligand-Target Pair
Affinity DataKi: 7.70E+4nMAssay Description:Compound was evaluated for its inhibitory activity against trypsinMore data for this Ligand-Target Pair
Affinity DataKi: 7.70E+4nMAssay Description:Compound was evaluated for its inhibitory activity against trypsinMore data for this Ligand-Target Pair
Affinity DataKi: 2.33E+5nMAssay Description:Compound was evaluated for its inhibitory activity against trypsinMore data for this Ligand-Target Pair
Affinity DataKi: >5.00E+5nMAssay Description:Compound was evaluated for its inhibitory activity against human thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 5.17E+5nMAssay Description:Compound was evaluated for its inhibitory activity against trypsinMore data for this Ligand-Target Pair
Affinity DataKi: 5.68E+5nMAssay Description:Compound was evaluated for its inhibitory activity against trypsinMore data for this Ligand-Target Pair
Affinity DataKi: 5.81E+5nMAssay Description:Compound was evaluated for its inhibitory activity against human thrombinMore data for this Ligand-Target Pair
Affinity DataIC50: 17nMAssay Description:Inhibition of squalene synthase from rat liver microsomesMore data for this Ligand-Target Pair
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Bos taurus (bovine))
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataIC50: 80nMAssay Description:Inhibition of farnesyl protein transferase from bovine brainMore data for this Ligand-Target Pair
Affinity DataIC50: 90nMAssay Description:Inhibition of squalene synthase from rat liver microsomesMore data for this Ligand-Target Pair
Affinity DataIC50: 100nMAssay Description:Compound was evaluated for binding affinity at bovine brain Alpha-1 adrenergic receptor in a filtration-based assay using [3H]prazosin as the radioli...More data for this Ligand-Target Pair
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Bos taurus (bovine))
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataIC50: 170nMAssay Description:Inhibition of farnesyl protein transferase from bovine brainMore data for this Ligand-Target Pair
Affinity DataIC50: 220nMAssay Description:Inhibition of squalene synthase from rat liver microsomesMore data for this Ligand-Target Pair
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Bos taurus (bovine))
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataIC50: 410nMAssay Description:Inhibition of farnesyl protein transferase from bovine brainMore data for this Ligand-Target Pair
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Bos taurus (bovine))
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataIC50: 470nMAssay Description:Inhibition of farnesyl protein transferase from bovine brainMore data for this Ligand-Target Pair
Affinity DataIC50: 480nMAssay Description:Inhibition of squalene synthase from rat liver microsomesMore data for this Ligand-Target Pair
Affinity DataIC50: 500nMAssay Description:Inhibition of squalene synthase from rat liver microsomesMore data for this Ligand-Target Pair
Affinity DataIC50: 500nMAssay Description:Compound was evaluated for binding affinity at bovine brain Alpha-1 adrenergic receptor in a filtration-based assay using [3H]prazosin as the radioli...More data for this Ligand-Target Pair
Affinity DataIC50: 900nMAssay Description:Compound was evaluated for binding affinity at bovine brain Alpha-1 adrenergic receptor determined in a filtration-based assay using [3H]prazosin as ...More data for this Ligand-Target Pair
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Bos taurus (bovine))
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataIC50: 980nMAssay Description:Inhibition of farnesyl protein transferase from bovine brainMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+3nMAssay Description:Compound was evaluated for binding affinity at bovine brain Alpha-1 adrenergic receptor in a filtration-based assay using [3H]prazosin as the radioli...More data for this Ligand-Target Pair
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of squalene synthase from rat liver microsomesMore data for this Ligand-Target Pair
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of squalene synthase from rat liver microsomesMore data for this Ligand-Target Pair
Affinity DataIC50: 1.50E+3nMAssay Description:Compound was evaluated for binding affinity at bovine brain Alpha-1 adrenergic receptor in a filtration-based assay using [3H]prazosin as the radioli...More data for this Ligand-Target Pair
Affinity DataIC50: 2.30E+3nMAssay Description:Inhibition of squalene synthase from rat liver microsomesMore data for this Ligand-Target Pair
Affinity DataIC50: 2.30E+3nMAssay Description:Compound was evaluated for binding affinity at bovine brain Alpha-1 adrenergic receptor in a filtration-based assay using [3H]prazosin as the radioli...More data for this Ligand-Target Pair