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Found 71 with Last Name = 'hill' and Initial = 'bt'
TargetHistamine H2 receptor(Cavia porcellus (domestic guinea pig))
TBA

Curated by ChEMBL
LigandPNGBDBM50404821(CHEMBL306465)
Affinity DataKi:  4nMAssay Description:In vitro inhibition of Histamine H2 receptor by measuring its ability to block the histamine-stimulated adenylate cyclase of guinea pig hippocampal h...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H2 receptor(Cavia porcellus (domestic guinea pig))
TBA

Curated by ChEMBL
LigandPNGBDBM50404823(CHEMBL63299)
Affinity DataKi:  6.30nMAssay Description:In vitro inhibition of Histamine H2 receptor by measuring its ability to block the histamine-stimulated adenylate cyclase of guinea pig hippocampal h...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H2 receptor(Cavia porcellus (domestic guinea pig))
TBA

Curated by ChEMBL
LigandPNGBDBM50404822(CHEMBL8982)
Affinity DataKi:  6.30nMAssay Description:In vitro inhibition of Histamine H2 receptor by measuring its ability to block the histamine-stimulated adenylate cyclase of guinea pig hippocampal h...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H2 receptor(Cavia porcellus (domestic guinea pig))
TBA

Curated by ChEMBL
LigandPNGBDBM22568(1-cyano-3-{2-[({2-[(diaminomethylidene)amino]-1,3-...)
Affinity DataKi:  32nMAssay Description:Evaluated in vitro for Histamine H2 receptor inhibition using the dimaprit stimulated chronotropic response of the guinea pig atriumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50070791(4-Amino-1-(4-benzhydryloxy-benzyl)-pyridinium | CH...)
Affinity DataKi:  58nMAssay Description:Compound was evaluated for its inhibitory activity against human thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50070787(4-Amino-1-[4-(1,3-diphenyl-propoxy)-benzyl]-pyridi...)
Affinity DataKi:  160nMAssay Description:Compound was evaluated for its inhibitory activity against human thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H2 receptor(Cavia porcellus (domestic guinea pig))
TBA

Curated by ChEMBL
LigandPNGBDBM50404962(CHEMBL33850)
Affinity DataKi:  200nMAssay Description:Evaluated in vitro for Histamine H2 receptor inhibition using the dimaprit stimulated chronotropic response of the guinea pig atriumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H2 receptor(Cavia porcellus (domestic guinea pig))
TBA

Curated by ChEMBL
LigandPNGBDBM50404955(CHEMBL441965)
Affinity DataKi:  316nMAssay Description:Evaluated in vitro for Histamine H2 receptor inhibition using the dimaprit stimulated chronotropic response of the guinea pig atriumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H2 receptor(Cavia porcellus (domestic guinea pig))
TBA

Curated by ChEMBL
LigandPNGBDBM50404958(CHEMBL284743)
Affinity DataKi:  316nMAssay Description:Evaluated in vitro for Histamine H2 receptor inhibition using the dimaprit stimulated chronotropic response of the guinea pig atriumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H2 receptor(Cavia porcellus (domestic guinea pig))
TBA

Curated by ChEMBL
LigandPNGBDBM50404956(CHEMBL284556)
Affinity DataKi:  398nMAssay Description:Evaluated in vitro for Histamine H2 receptor inhibition using the dimaprit stimulated chronotropic response of the guinea pig atriumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H2 receptor(Cavia porcellus (domestic guinea pig))
TBA

Curated by ChEMBL
LigandPNGBDBM50403559(Brumetadina | CIMETIDINE)
Affinity DataKi:  501nMAssay Description:In vitro inhibition of Histamine H2 receptor by measuring its ability to block the histamine-stimulated adenylate cyclase of guinea pig hippocampal h...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H2 receptor(Cavia porcellus (domestic guinea pig))
TBA

Curated by ChEMBL
LigandPNGBDBM22893(CHEMBL512 | Ranitidine | ZANTAC | dimethyl[(5-{[(2...)
Affinity DataKi:  501nMAssay Description:In vitro inhibition of Histamine H2 receptor by measuring its ability to block the histamine-stimulated adenylate cyclase of guinea pig hippocampal h...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H2 receptor(Cavia porcellus (domestic guinea pig))
TBA

Curated by ChEMBL
LigandPNGBDBM50403559(Brumetadina | CIMETIDINE)
Affinity DataKi:  501nMAssay Description:Evaluated in vitro for Histamine H2 receptor inhibition using the dimaprit stimulated chronotropic response of the guinea pig atriumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50070786(4-Amino-1-(4-benzyloxy-benzyl)-pyridinium | CHEMBL...)
Affinity DataKi:  700nMAssay Description:Compound was evaluated for its inhibitory activity against human thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H2 receptor(Cavia porcellus (domestic guinea pig))
TBA

Curated by ChEMBL
LigandPNGBDBM50404961(CHEMBL284379)
Affinity DataKi:  794nMAssay Description:Evaluated in vitro for Histamine H2 receptor inhibition using the dimaprit stimulated chronotropic response of the guinea pig atriumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50070793((4-Benzhydryloxy-benzyl)-pyridin-4-yl-amine | CHEM...)
Affinity DataKi:  1.30E+3nMAssay Description:Compound was evaluated for its inhibitory activity against human thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50070790((4-Benzyloxy-benzyl)-pyridin-4-yl-amine | CHEMBL47...)
Affinity DataKi:  4.70E+3nMAssay Description:Compound was evaluated for its inhibitory activity against human thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50070788(CHEMBL48029 | N-(4-(benzyloxy)phenethyl)pyridin-4-...)
Affinity DataKi:  7.90E+3nMAssay Description:Compound was evaluated for its inhibitory activity against human thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50070792(4-(4-Benzyloxy-benzyl)-phenylamine | CHEMBL45648)
Affinity DataKi: >1.00E+4nMAssay Description:Compound was evaluated for its inhibitory activity against human thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50070792(4-(4-Benzyloxy-benzyl)-phenylamine | CHEMBL45648)
Affinity DataKi: >1.00E+4nMAssay Description:Compound was evaluated for its inhibitory activity against trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H2 receptor(Cavia porcellus (domestic guinea pig))
TBA

Curated by ChEMBL
LigandPNGBDBM50404957(CHEMBL33996)
Affinity DataKi:  1.58E+4nMAssay Description:Evaluated in vitro for Histamine H2 receptor inhibition using the dimaprit stimulated chronotropic response of the guinea pig atriumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50070787(4-Amino-1-[4-(1,3-diphenyl-propoxy)-benzyl]-pyridi...)
Affinity DataKi:  1.60E+4nMAssay Description:Compound was evaluated for its inhibitory activity against trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H2 receptor(Cavia porcellus (domestic guinea pig))
TBA

Curated by ChEMBL
LigandPNGBDBM50404959(CHEMBL33108)
Affinity DataKi:  3.16E+4nMAssay Description:Evaluated in vitro for Histamine H2 receptor inhibition using the dimaprit stimulated chronotropic response of the guinea pig atriumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H2 receptor(Cavia porcellus (domestic guinea pig))
TBA

Curated by ChEMBL
LigandPNGBDBM50404960(CHEMBL32409)
Affinity DataKi:  3.98E+4nMAssay Description:Evaluated in vitro for Histamine H2 receptor inhibition using the dimaprit stimulated chronotropic response of the guinea pig atriumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50070786(4-Amino-1-(4-benzyloxy-benzyl)-pyridinium | CHEMBL...)
Affinity DataKi:  7.70E+4nMAssay Description:Compound was evaluated for its inhibitory activity against trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50070793((4-Benzhydryloxy-benzyl)-pyridin-4-yl-amine | CHEM...)
Affinity DataKi:  7.70E+4nMAssay Description:Compound was evaluated for its inhibitory activity against trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50070790((4-Benzyloxy-benzyl)-pyridin-4-yl-amine | CHEMBL47...)
Affinity DataKi:  2.33E+5nMAssay Description:Compound was evaluated for its inhibitory activity against trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50070789(1-(4-Benzyloxy-benzyl)-pyridinium | CHEMBL296280)
Affinity DataKi: >5.00E+5nMAssay Description:Compound was evaluated for its inhibitory activity against human thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50070791(4-Amino-1-(4-benzhydryloxy-benzyl)-pyridinium | CH...)
Affinity DataKi:  5.17E+5nMAssay Description:Compound was evaluated for its inhibitory activity against trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50070788(CHEMBL48029 | N-(4-(benzyloxy)phenethyl)pyridin-4-...)
Affinity DataKi:  5.68E+5nMAssay Description:Compound was evaluated for its inhibitory activity against trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50070794(1-(4-Benzyloxy-benzyl)-piperidin-4-ylamine | CHEMB...)
Affinity DataKi:  5.81E+5nMAssay Description:Compound was evaluated for its inhibitory activity against human thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSqualene synthase(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50031839(((E)-6,10-Dimethyl-1-phosphono-undeca-5,9-dienyl)-...)
Affinity DataIC50:  17nMAssay Description:Inhibition of squalene synthase from rat liver microsomesMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50059875((S)-3-Phenyl-2-((4E,8E)-5,9,13-trimethyl-2-phospho...)
Affinity DataIC50:  80nMAssay Description:Inhibition of farnesyl protein transferase from bovine brainMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSqualene synthase(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50287113((S)-3-Phenyl-2-((4E,8E)-5,9,13-trimethyl-2-phospho...)
Affinity DataIC50:  90nMAssay Description:Inhibition of squalene synthase from rat liver microsomesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetAlpha-1A adrenergic receptor(CALF)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50368446(CHEMBL1203299)
Affinity DataIC50:  100nMAssay Description:Compound was evaluated for binding affinity at bovine brain Alpha-1 adrenergic receptor in a filtration-based assay using [3H]prazosin as the radioli...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50287113((S)-3-Phenyl-2-((4E,8E)-5,9,13-trimethyl-2-phospho...)
Affinity DataIC50:  170nMAssay Description:Inhibition of farnesyl protein transferase from bovine brainMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSqualene synthase(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50287115((S)-3-Phenyl-2-((5E,9E)-6,10,14-trimethyl-3-phosph...)
Affinity DataIC50:  220nMAssay Description:Inhibition of squalene synthase from rat liver microsomesMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50059860(((2E,6E)-1-Hydroxy-3,7,11-trimethyl-dodeca-2,6,10-...)
Affinity DataIC50:  410nMAssay Description:Inhibition of farnesyl protein transferase from bovine brainMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50287115((S)-3-Phenyl-2-((5E,9E)-6,10,14-trimethyl-3-phosph...)
Affinity DataIC50:  470nMAssay Description:Inhibition of farnesyl protein transferase from bovine brainMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSqualene synthase(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50287116(((3E,7E)-4,8,12-Trimethyl-1-phenethylcarbamoyl-tri...)
Affinity DataIC50:  480nMAssay Description:Inhibition of squalene synthase from rat liver microsomesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSqualene synthase(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50287118((R)-3-Phenyl-2-((4E,8E)-5,9,13-trimethyl-2-phospho...)
Affinity DataIC50:  500nMAssay Description:Inhibition of squalene synthase from rat liver microsomesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetAlpha-1A adrenergic receptor(CALF)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50003331(CHEMBL101322 | CHEMBL1204312 | N-[4-oxo-1'-[2-(2-p...)
Affinity DataIC50:  500nMAssay Description:Compound was evaluated for binding affinity at bovine brain Alpha-1 adrenergic receptor in a filtration-based assay using [3H]prazosin as the radioli...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(CALF)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50368441(CHEMBL1203302)
Affinity DataIC50:  900nMAssay Description:Compound was evaluated for binding affinity at bovine brain Alpha-1 adrenergic receptor determined in a filtration-based assay using [3H]prazosin as ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50287118((R)-3-Phenyl-2-((4E,8E)-5,9,13-trimethyl-2-phospho...)
Affinity DataIC50:  980nMAssay Description:Inhibition of farnesyl protein transferase from bovine brainMore data for this Ligand-Target Pair
In DepthDetails Article
TargetAlpha-1A adrenergic receptor(CALF)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50368442(CHEMBL1203297)
Affinity DataIC50:  1.00E+3nMAssay Description:Compound was evaluated for binding affinity at bovine brain Alpha-1 adrenergic receptor in a filtration-based assay using [3H]prazosin as the radioli...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSqualene synthase(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50059875((S)-3-Phenyl-2-((4E,8E)-5,9,13-trimethyl-2-phospho...)
Affinity DataIC50:  1.30E+3nMAssay Description:Inhibition of squalene synthase from rat liver microsomesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSqualene synthase(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50287117((S)-3-Phenyl-2-((4E,8E)-5,9,13-trimethyl-2-phospho...)
Affinity DataIC50:  1.40E+3nMAssay Description:Inhibition of squalene synthase from rat liver microsomesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetAlpha-1A adrenergic receptor(CALF)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50003335(CHEMBL1204345 | CHEMBL129583 | L-691121 | N-[1''-(...)
Affinity DataIC50:  1.50E+3nMAssay Description:Compound was evaluated for binding affinity at bovine brain Alpha-1 adrenergic receptor in a filtration-based assay using [3H]prazosin as the radioli...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSqualene synthase(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50059860(((2E,6E)-1-Hydroxy-3,7,11-trimethyl-dodeca-2,6,10-...)
Affinity DataIC50:  2.30E+3nMAssay Description:Inhibition of squalene synthase from rat liver microsomesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetAlpha-1A adrenergic receptor(CALF)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50368447(CHEMBL1203301)
Affinity DataIC50:  2.30E+3nMAssay Description:Compound was evaluated for binding affinity at bovine brain Alpha-1 adrenergic receptor in a filtration-based assay using [3H]prazosin as the radioli...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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