Affinity DataKi: 1.60nMAssay Description:Inhibition of [3H]-kainate binding at rat forebrain ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
Affinity DataKi: 1.90nMAssay Description:Inhibition of [3H]-kainate binding at rat forebrain ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
Affinity DataKi: 2.10nMAssay Description:Inhibition of [3H]-kainate binding at rat forebrain ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
Affinity DataKi: 2.20nMAssay Description:Inhibition of [3H]-kainate binding at rat forebrain ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
Affinity DataKi: 2.30nMAssay Description:Inhibition of [3H]-kainate binding at rat forebrain ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
Affinity DataKi: 2.60nMAssay Description:Inhibition of [3H]-kainate binding at rat forebrain ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
Affinity DataKi: 2.70nMAssay Description:Inhibition of [3H]-kainate binding at rat forebrain ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
Affinity DataKi: 2.80nMAssay Description:Inhibition of [3H]-kainate binding at rat forebrain ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
Affinity DataKi: 3nMAssay Description:Displacement of [3H]AMPA from homomeric recombinant GluA2 receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 3.5nMAssay Description:Inhibition of [3H]-kainate binding at rat forebrain ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
Affinity DataKi: 3.60nMAssay Description:Inhibition of [3H]-kainate binding at rat forebrain ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
Affinity DataKi: 3.60nMAssay Description:Inhibition of [3H]-kainate binding at rat forebrain ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
Affinity DataKi: 3.70nMAssay Description:Inhibition of [3H]-kainate binding at rat forebrain ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
Affinity DataKi: 3.90nMAssay Description:Inhibition of [3H]-kainate binding at rat forebrain ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
Affinity DataKi: 3.90nMAssay Description:Inhibition of [3H]-kainate binding at rat forebrain ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
Affinity DataKi: 4.80nMAssay Description:Inhibition of [3H]-kainate binding at rat forebrain ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
Affinity DataKi: 6.20nMAssay Description:Inhibition of [3H]-kainate binding at rat forebrain ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
Affinity DataKi: 7.70nMAssay Description:Inhibition of [3H]-kainate binding at rat forebrain ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
Affinity DataKi: 9nMAssay Description:Inhibition of [3H]-kainate binding at rat forebrain ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
Affinity DataKi: 9.10nMAssay Description:Inhibition of [3H]-kainate binding at rat forebrain ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
Affinity DataKi: 9.5nMAssay Description:Inhibition of [3H]-kainate binding at rat forebrain ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
Affinity DataKi: 11.9nMAssay Description:Inhibition of [3H]-kainate binding at rat forebrain ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
Affinity DataKi: 16nMAssay Description:Inhibition of [3H]-kainate binding at rat forebrain ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
Affinity DataKi: 18.3nMAssay Description:Inhibition of [3H]-kainate binding at ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
Affinity DataKi: 18.5nMAssay Description:Inhibition of [3H]-kainate binding at rat forebrain ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, kainate 1(Homo sapiens (Human))
Centro De Investigaci�N Lilly
Curated by ChEMBL
Centro De Investigaci�N Lilly
Curated by ChEMBL
Affinity DataKi: 20nMAssay Description:Displacement of [3H]ATPA from human Gluk1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 23.3nMAssay Description:Inhibition of [3H]-kainate binding at rat forebrain ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
Affinity DataKi: 29.8nMAssay Description:Inhibition of [3H]-kainate binding at ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
Affinity DataKi: 31.7nMAssay Description:Inhibition of [3H]-kainate binding at ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
Affinity DataKi: 38.4nMAssay Description:Inhibition of [3H]-kainate binding at ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
Affinity DataKi: 41.1nMAssay Description:Inhibition of [3H]-kainate binding at ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, kainate 5(Homo sapiens (Human))
Eli Lilly
Curated by PDSP Ki Database
Eli Lilly
Curated by PDSP Ki Database
Affinity DataKi: 53nMAssay Description:Inhibition of [3H]-kainate binding at ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
Affinity DataKi: 54.3nMAssay Description:Inhibition of [3H]-kainate binding at ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
Affinity DataKi: 57.4nMAssay Description:Inhibition of [3H]-kainate binding at ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
TargetInhibitor of nuclear factor kappa-B kinase subunit alpha(Homo sapiens (Human))
University of Strathclyde
Curated by ChEMBL
University of Strathclyde
Curated by ChEMBL
Affinity DataKi: 80nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged IKKalpha (1 to 745 residues) expressed in baculovirus expression system using biotinylated IkBa...More data for this Ligand-Target Pair
Affinity DataKi: 82.2nMAssay Description:Inhibition of [3H]-kainate binding at ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, kainate 1(Homo sapiens (Human))
Centro De Investigaci�N Lilly
Curated by ChEMBL
Centro De Investigaci�N Lilly
Curated by ChEMBL
Affinity DataKi: 90nMAssay Description:Displacement of [3H]ATPA from human Gluk1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 90.6nMAssay Description:Inhibition of [3H]-kainate binding at ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
Affinity DataKi: 93.5nMAssay Description:Inhibition of [3H]-kainate binding at ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, kainate 1(Homo sapiens (Human))
Centro De Investigaci�N Lilly
Curated by ChEMBL
Centro De Investigaci�N Lilly
Curated by ChEMBL
Affinity DataKi: 100nMAssay Description:Displacement of [3H]ATPA from human Gluk1 receptorMore data for this Ligand-Target Pair
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
University of Strathclyde
Curated by ChEMBL
University of Strathclyde
Curated by ChEMBL
Affinity DataKi: 100nMAssay Description:Inhibition of recombinant full length human IKKbeta expressed in baculovirus infected sf9 insect cells using biotinylated IkBalpha as substrate after...More data for this Ligand-Target Pair
Affinity DataKi: 108nMAssay Description:Inhibition of [3H]-kainate binding at ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
Affinity DataKi: 113nMAssay Description:Inhibition of human t-PAMore data for this Ligand-Target Pair
Affinity DataKi: 123nMAssay Description:Inhibition of [3H]-kainate binding at ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
Affinity DataKi: 126nMAssay Description:Inhibition of [3H]-kainate binding at rat forebrain ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
Affinity DataKi: 126nMAssay Description:Inhibition of [3H]-kainate binding at ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
Affinity DataKi: 129nMAssay Description:Inhibition of [3H]-kainate binding at ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
Affinity DataKi: 131nMAssay Description:Inhibition of [3H]-kainate binding at ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
Affinity DataKi: 132nMAssay Description:Inhibition of [3H]-kainate binding at ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair