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Found 986 with Last Name = 'ho' and Initial = 'kh'
TargetGlutamate receptor ionotropic, kainate 2(Rattus norvegicus)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50053067((2S,3S,4S)-3-Carboxymethyl-4-(1-phenyl-vinyl)-pyrr...)
Affinity DataKi:  1.60nMAssay Description:Inhibition of [3H]-kainate binding at rat forebrain ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 2(Rattus norvegicus)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50053071((2S,3S,4S)-3-Carboxymethyl-4-[1-(4-fluoro-3-methyl...)
Affinity DataKi:  1.90nMAssay Description:Inhibition of [3H]-kainate binding at rat forebrain ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 2(Rattus norvegicus)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50053075((2S,3S,4S)-4-(1-Biphenyl-3-yl-vinyl)-3-carboxymeth...)
Affinity DataKi:  2.10nMAssay Description:Inhibition of [3H]-kainate binding at rat forebrain ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 2(Rattus norvegicus)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50053083((2S,3S,4S)-3-Carboxymethyl-4-(1-m-tolyl-vinyl)-pyr...)
Affinity DataKi:  2.20nMAssay Description:Inhibition of [3H]-kainate binding at rat forebrain ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 2(Rattus norvegicus)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50053080((2S,3S,4S)-3-Carboxymethyl-4-[1-(3,4-dimethyl-phen...)
Affinity DataKi:  2.30nMAssay Description:Inhibition of [3H]-kainate binding at rat forebrain ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 2(Rattus norvegicus)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50053088((2S,3S,4S)-3-Carboxymethyl-4-(1-p-tolyl-vinyl)-pyr...)
Affinity DataKi:  2.60nMAssay Description:Inhibition of [3H]-kainate binding at rat forebrain ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 2(Rattus norvegicus)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50053087((2S,3S,4S)-3-Carboxymethyl-4-[1-(4-fluoro-phenyl)-...)
Affinity DataKi:  2.70nMAssay Description:Inhibition of [3H]-kainate binding at rat forebrain ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 2(Rattus norvegicus)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50053064((2S,3S,4S)-4-[1-(4-Butoxy-phenyl)-vinyl]-3-carboxy...)
Affinity DataKi:  2.80nMAssay Description:Inhibition of [3H]-kainate binding at rat forebrain ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 2(Homo sapiens (Human))
Centro De Investigaci�N Lilly

Curated by ChEMBL
LigandPNGBDBM50494356(CHEMBL3088070)
Affinity DataKi:  3nMAssay Description:Displacement of [3H]AMPA from homomeric recombinant GluA2 receptor (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 2(Rattus norvegicus)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50053063((2S,3S,4S)-3-Carboxymethyl-4-[1-(3-methoxy-phenyl)...)
Affinity DataKi:  3.5nMAssay Description:Inhibition of [3H]-kainate binding at rat forebrain ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 2(Rattus norvegicus)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50053059((2S,3S,4S)-3-Carboxymethyl-4-[1-(4-propyl-phenyl)-...)
Affinity DataKi:  3.60nMAssay Description:Inhibition of [3H]-kainate binding at rat forebrain ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 2(Rattus norvegicus)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50053068((2S,3S,4S)-3-Carboxymethyl-4-[1-(4-isopropenyl-phe...)
Affinity DataKi:  3.60nMAssay Description:Inhibition of [3H]-kainate binding at rat forebrain ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 2(Rattus norvegicus)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50002369((2S-(2alpha,3beta,4beta))-2-carboxy-4-(1-methyleth...)
Affinity DataKi:  3.70nMAssay Description:Inhibition of [3H]-kainate binding at rat forebrain ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, kainate 2(Rattus norvegicus)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50053073((2S,3S,4S)-3-Carboxymethyl-4-[1-(4-methoxy-phenyl)...)
Affinity DataKi:  3.90nMAssay Description:Inhibition of [3H]-kainate binding at rat forebrain ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 2(Rattus norvegicus)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50053061((2S,3S,4S)-3-Carboxymethyl-4-[1-(4-chloro-phenyl)-...)
Affinity DataKi:  3.90nMAssay Description:Inhibition of [3H]-kainate binding at rat forebrain ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 2(Rattus norvegicus)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50053082((2S,3S,4S)-4-[1-(4-Butyl-phenyl)-vinyl]-3-carboxym...)
Affinity DataKi:  4.80nMAssay Description:Inhibition of [3H]-kainate binding at rat forebrain ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 2(Rattus norvegicus)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50053065((2S,3S,4S)-3-Carboxymethyl-4-[1-(4-phenethyloxy-ph...)
Affinity DataKi:  6.20nMAssay Description:Inhibition of [3H]-kainate binding at rat forebrain ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 2(Rattus norvegicus)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50053089((2S,3S,4S)-3-Carboxymethyl-4-[1-(4-ethyl-phenyl)-v...)
Affinity DataKi:  7.70nMAssay Description:Inhibition of [3H]-kainate binding at rat forebrain ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 2(Rattus norvegicus)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50053070((2S,3S,4S)-3-Carboxymethyl-4-{1-[4-(1-methylene-pr...)
Affinity DataKi:  9nMAssay Description:Inhibition of [3H]-kainate binding at rat forebrain ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 2(Rattus norvegicus)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50053076((2S,3S,4S)-4-(1-Biphenyl-4-yl-vinyl)-3-carboxymeth...)
Affinity DataKi:  9.10nMAssay Description:Inhibition of [3H]-kainate binding at rat forebrain ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 2(Rattus norvegicus)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50053062((2S,3S,4S)-3-Carboxymethyl-4-[1-(3,5-dimethyl-phen...)
Affinity DataKi:  9.5nMAssay Description:Inhibition of [3H]-kainate binding at rat forebrain ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 2(Rattus norvegicus)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50053074((2S,3S,4S)-3-Carboxymethyl-4-[1-(4-phenoxy-phenyl)...)
Affinity DataKi:  11.9nMAssay Description:Inhibition of [3H]-kainate binding at rat forebrain ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 2(Rattus norvegicus)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50053077((2S,3S,4S)-3-Carboxymethyl-4-[1-(3-phenethyloxy-ph...)
Affinity DataKi:  16nMAssay Description:Inhibition of [3H]-kainate binding at rat forebrain ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 2(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50053058((4E,6E)-(R)-7-[4,5-Bis-(1-hydroxy-vinyl)-pyrrolidi...)
Affinity DataKi:  18.3nMAssay Description:Inhibition of [3H]-kainate binding at ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 2(Rattus norvegicus)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50053060((2S,3S,4S)-4-[1-(4-tert-Butyl-phenyl)-vinyl]-3-car...)
Affinity DataKi:  18.5nMAssay Description:Inhibition of [3H]-kainate binding at rat forebrain ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 1(Homo sapiens (Human))
Centro De Investigaci�N Lilly

Curated by ChEMBL
LigandPNGBDBM50494356(CHEMBL3088070)
Affinity DataKi:  20nMAssay Description:Displacement of [3H]ATPA from human Gluk1 receptorMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 2(Rattus norvegicus)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50053079((2S,3S,4S)-4-[1-(3-Butoxy-phenyl)-vinyl]-3-carboxy...)
Affinity DataKi:  23.3nMAssay Description:Inhibition of [3H]-kainate binding at rat forebrain ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 2(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50053067((2S,3S,4S)-3-Carboxymethyl-4-(1-phenyl-vinyl)-pyrr...)
Affinity DataKi:  29.8nMAssay Description:Inhibition of [3H]-kainate binding at ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 2(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50053061((2S,3S,4S)-3-Carboxymethyl-4-[1-(4-chloro-phenyl)-...)
Affinity DataKi:  31.7nMAssay Description:Inhibition of [3H]-kainate binding at ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 2(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50053087((2S,3S,4S)-3-Carboxymethyl-4-[1-(4-fluoro-phenyl)-...)
Affinity DataKi:  38.4nMAssay Description:Inhibition of [3H]-kainate binding at ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 2(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50053088((2S,3S,4S)-3-Carboxymethyl-4-(1-p-tolyl-vinyl)-pyr...)
Affinity DataKi:  41.1nMAssay Description:Inhibition of [3H]-kainate binding at ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 5(Homo sapiens (Human))
Eli Lilly

Curated by PDSP Ki Database
LigandPNGBDBM86754(LY 466195 | LY-466195)
Affinity DataKi:  50nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 2(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50002369((2S-(2alpha,3beta,4beta))-2-carboxy-4-(1-methyleth...)
Affinity DataKi:  53nMAssay Description:Inhibition of [3H]-kainate binding at ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, kainate 2(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50053071((2S,3S,4S)-3-Carboxymethyl-4-[1-(4-fluoro-3-methyl...)
Affinity DataKi:  54.3nMAssay Description:Inhibition of [3H]-kainate binding at ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 2(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50053073((2S,3S,4S)-3-Carboxymethyl-4-[1-(4-methoxy-phenyl)...)
Affinity DataKi:  57.4nMAssay Description:Inhibition of [3H]-kainate binding at ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit alpha(Homo sapiens (Human))
University of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50257823(CHEMBL4089551)
Affinity DataKi:  80nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged IKKalpha (1 to 745 residues) expressed in baculovirus expression system using biotinylated IkBa...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 2(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50053089((2S,3S,4S)-3-Carboxymethyl-4-[1-(4-ethyl-phenyl)-v...)
Affinity DataKi:  82.2nMAssay Description:Inhibition of [3H]-kainate binding at ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 1(Homo sapiens (Human))
Centro De Investigaci�N Lilly

Curated by ChEMBL
LigandPNGBDBM50494342(CHEMBL3088072)
Affinity DataKi:  90nMAssay Description:Displacement of [3H]ATPA from human Gluk1 receptorMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 2(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50053075((2S,3S,4S)-4-(1-Biphenyl-3-yl-vinyl)-3-carboxymeth...)
Affinity DataKi:  90.6nMAssay Description:Inhibition of [3H]-kainate binding at ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 2(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50053063((2S,3S,4S)-3-Carboxymethyl-4-[1-(3-methoxy-phenyl)...)
Affinity DataKi:  93.5nMAssay Description:Inhibition of [3H]-kainate binding at ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 1(Homo sapiens (Human))
Centro De Investigaci�N Lilly

Curated by ChEMBL
LigandPNGBDBM50494350(CHEMBL3088064)
Affinity DataKi:  100nMAssay Description:Displacement of [3H]ATPA from human Gluk1 receptorMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
University of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50257884(CHEMBL4065551)
Affinity DataKi:  100nMAssay Description:Inhibition of recombinant full length human IKKbeta expressed in baculovirus infected sf9 insect cells using biotinylated IkBalpha as substrate after...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 2(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50053080((2S,3S,4S)-3-Carboxymethyl-4-[1-(3,4-dimethyl-phen...)
Affinity DataKi:  108nMAssay Description:Inhibition of [3H]-kainate binding at ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTissue-type plasminogen activator(Homo sapiens (Human))
Lg Life Sciences

Curated by ChEMBL
LigandPNGBDBM50439332(CHEMBL2419745)
Affinity DataKi:  113nMAssay Description:Inhibition of human t-PAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 2(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50053083((2S,3S,4S)-3-Carboxymethyl-4-(1-m-tolyl-vinyl)-pyr...)
Affinity DataKi:  123nMAssay Description:Inhibition of [3H]-kainate binding at ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 2(Rattus norvegicus)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50053066((2S,3S,4S)-3-Carboxymethyl-4-{1-[4-(5-phenyl-penty...)
Affinity DataKi:  126nMAssay Description:Inhibition of [3H]-kainate binding at rat forebrain ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 2(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50053065((2S,3S,4S)-3-Carboxymethyl-4-[1-(4-phenethyloxy-ph...)
Affinity DataKi:  126nMAssay Description:Inhibition of [3H]-kainate binding at ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 2(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50053084((2S,3S,4S)-3-Carboxymethyl-4-[1-(3-methyl-4-phenet...)
Affinity DataKi:  129nMAssay Description:Inhibition of [3H]-kainate binding at ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 2(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50053076((2S,3S,4S)-4-(1-Biphenyl-4-yl-vinyl)-3-carboxymeth...)
Affinity DataKi:  131nMAssay Description:Inhibition of [3H]-kainate binding at ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 2(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50053068((2S,3S,4S)-3-Carboxymethyl-4-[1-(4-isopropenyl-phe...)
Affinity DataKi:  132nMAssay Description:Inhibition of [3H]-kainate binding at ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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