Affinity DataKi: 0.710nMAssay Description:Displacement of [3H]-NPA from rat brain Dopamine receptor D2More data for this Ligand-Target Pair
Affinity DataKi: 1.20nMAssay Description:Binding affinity for Adenosine A1 receptor in cerebral cortices of Sprague-Dawley male rats using [3H]-CHAMore data for this Ligand-Target Pair
Affinity DataKi: 1.30nMAssay Description:Binding affinity for Adenosine A1 receptor in corpora striata of rats using [3H]NECAMore data for this Ligand-Target Pair
Affinity DataKi: 2.10nMAssay Description:Displacement of [3H]-NPA from rat brain Dopamine receptor D2More data for this Ligand-Target Pair
Affinity DataKi: 3nMAssay Description:Evaluated for the binding affinity towards the Adenosine A1 receptor in corpora striata of rats using [3H]CHA as radioligand.More data for this Ligand-Target Pair
Affinity DataKi: 3nMAssay Description:Binding affinity for Adenosine A1 receptor in cerebral cortices of Sprague-Dawley male rats using [3H]CHAMore data for this Ligand-Target Pair
Affinity DataKi: 3nMAssay Description:Displacement of [3H]-NPA from rat brain Dopamine receptor D2More data for this Ligand-Target Pair
Affinity DataKi: 3nMAssay Description:Evaluated for the binding affinity towards the Adenosine A1 receptor in corpora striata of rats using [3H]CHA as radioligand.More data for this Ligand-Target Pair
Affinity DataKi: 3.10nMAssay Description:Displacement of [3H]-NPA from rat brain Dopamine receptor D2More data for this Ligand-Target Pair
Affinity DataKi: 3.70nMAssay Description:Displacement of [3H]-NPA from rat brain Dopamine receptor D2More data for this Ligand-Target Pair
Affinity DataKi: 3.80nMAssay Description:Displacement of [3H]-NPA from rat brain Dopamine receptor D2More data for this Ligand-Target Pair
Affinity DataKi: 4.20nMAssay Description:Displacement of [3H]-NPA from rat brain Dopamine receptor D2More data for this Ligand-Target Pair
Affinity DataKi: 4.20nMAssay Description:Displacement of [3H]-NPA from rat brain Dopamine receptor D2More data for this Ligand-Target Pair
Affinity DataKi: 4.60nMAssay Description:Binding affinity for Adenosine A1 receptor in corpora striata of rats using [3H]NECAMore data for this Ligand-Target Pair
Affinity DataKi: 4.80nMAssay Description:Displacement of [3H]-NPA from rat brain Dopamine receptor D2More data for this Ligand-Target Pair
Affinity DataKi: 5nMAssay Description:Binding affinity for Adenosine A2 receptor in corpora striata of rats using [3H]NECAMore data for this Ligand-Target Pair
Affinity DataKi: 5.10nMAssay Description:Displacement of [3H]-NPA from rat brain Dopamine receptor D2More data for this Ligand-Target Pair
Affinity DataKi: 6.30nMAssay Description:Displacement of [3H]-NPA from rat brain Dopamine receptor D2More data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Evaluated for the binding affinity towards the Adenosine A1 receptor in corpora striata of rats using [3H]CHA as radioligand.More data for this Ligand-Target Pair
Affinity DataKi: 15.5nMAssay Description:Ki determinations were generously provided by the National Institute of Mental Health's Psychoactive Drug Screening Program (PDSP).More data for this Ligand-Target Pair
Affinity DataKi: 17.3nMAssay Description:Ki determinations were generously provided by the National Institute of Mental Health's Psychoactive Drug Screening Program (PDSP).More data for this Ligand-Target Pair
Affinity DataKi: 17.3nMAssay Description:Procedures employed by the PDSP as described in the NIMH-PDSP Assay Protocol Book, Version II. The standard drug used in both Sigma subtype assays is...More data for this Ligand-Target Pair
Affinity DataKi: 18nMAssay Description:Ki determinations were generously provided by the National Institute of Mental Health's Psychoactive Drug Screening Program (PDSP).More data for this Ligand-Target Pair
Affinity DataKi: 30nMAssay Description:The compounds were tested for activity vs. opioid receptor subtypes Kappa (KOR), Delta (DOR) and Mu (MOR) at an initial concentration of 10 μM e...More data for this Ligand-Target Pair
Affinity DataKi: 35.4nMAssay Description:Ki determinations were generously provided by the National Institute of Mental Health's Psychoactive Drug Screening Program (PDSP).More data for this Ligand-Target Pair
Affinity DataKi: 35.4nMAssay Description:Procedures employed by the PDSP as described in the NIMH-PDSP Assay Protocol Book, Version II. The standard drug used in both Sigma subtype assays is...More data for this Ligand-Target Pair
Affinity DataKi: 37.2nMAssay Description:Ki determinations were generously provided by the National Institute of Mental Health's Psychoactive Drug Screening Program (PDSP).More data for this Ligand-Target Pair
Affinity DataKi: 37.2nMAssay Description:Procedures employed by the PDSP as described in the NIMH-PDSP Assay Protocol Book, Version II. The standard drug used in both Sigma subtype assays is...More data for this Ligand-Target Pair
Affinity DataKi: 45nMAssay Description:In vitro ability of the compound to displace [3H]-ketanserin from 5-hydroxytryptamine 2A receptor in rat brain.More data for this Ligand-Target Pair
Affinity DataKi: 47nMAssay Description:The compounds were tested for activity vs. opioid receptor subtypes Kappa (KOR), Delta (DOR) and Mu (MOR) at an initial concentration of 10 μM e...More data for this Ligand-Target Pair
Affinity DataKi: 49nMAssay Description:Binding affinity for Adenosine A1 receptor in cerebral cortices of Sprague-Dawley male rats using [3H]-CHAMore data for this Ligand-Target Pair
Affinity DataKi: 59.8nMAssay Description:Ki determinations were generously provided by the National Institute of Mental Health's Psychoactive Drug Screening Program (PDSP).More data for this Ligand-Target Pair
Affinity DataKi: 70nMAssay Description:Ki determinations were generously provided by the National Institute of Mental Health's Psychoactive Drug Screening Program (PDSP).More data for this Ligand-Target Pair
Affinity DataKi: 70nMAssay Description:Procedures employed by the PDSP as described in the NIMH-PDSP Assay Protocol Book, Version II. The standard drug used in both Sigma subtype assays is...More data for this Ligand-Target Pair
Affinity DataKi: 83nMAssay Description:Displacement of [3H]-NPA from rat brain Dopamine receptor D2More data for this Ligand-Target Pair
Affinity DataKi: 97.2nMAssay Description:Ki determinations were generously provided by the National Institute of Mental Health's Psychoactive Drug Screening Program (PDSP).More data for this Ligand-Target Pair
Affinity DataKi: 97.2nMAssay Description:Procedures employed by the PDSP as described in the NIMH-PDSP Assay Protocol Book, Version II. The standard drug used in both Sigma subtype assays is...More data for this Ligand-Target Pair
Affinity DataKi: 98nMAssay Description:Ki determinations were generously provided by the National Institute of Mental Health's Psychoactive Drug Screening Program (PDSP).More data for this Ligand-Target Pair
Affinity DataKi: 146nMAssay Description:Ki determinations were generously provided by the National Institute of Mental Health's Psychoactive Drug Screening Program (PDSP).More data for this Ligand-Target Pair
Affinity DataKi: 146nMAssay Description:Procedures employed by the PDSP as described in the NIMH-PDSP Assay Protocol Book, Version II. The standard drug used in both Sigma subtype assays is...More data for this Ligand-Target Pair
Affinity DataKi: 200nMAssay Description:Evaluated for the binding affinity towards the Adenosine A1 receptor in corpora striata of rats using [3H]CHA as radioligand.More data for this Ligand-Target Pair
Affinity DataKi: 217nMAssay Description:Procedures employed by the PDSP as described in the NIMH-PDSP Assay Protocol Book, Version II. The standard drug used in both Sigma subtype assays is...More data for this Ligand-Target Pair
Affinity DataKi: 217nMAssay Description:Ki determinations were generously provided by the National Institute of Mental Health's Psychoactive Drug Screening Program (PDSP).More data for this Ligand-Target Pair
Affinity DataKi: 249nMAssay Description:The compounds were tested for activity vs. opioid receptor subtypes Kappa (KOR), Delta (DOR) and Mu (MOR) at an initial concentration of 10 μM e...More data for this Ligand-Target Pair
Affinity DataKi: 305nMAssay Description:Ki determinations were generously provided by the National Institute of Mental Health's Psychoactive Drug Screening Program (PDSP).More data for this Ligand-Target Pair