Affinity DataKi: 0.150nMAssay Description:Binding affinity to Opioid receptor delta 1 using [3H]DPDPE as a radioligand in guinea pigMore data for this Ligand-Target Pair
Affinity DataKi: 0.240nMAssay Description:Binding affinity to Opioid receptor delta 1 using [3H]DPDPE as a radioligand in guinea pigMore data for this Ligand-Target Pair
Affinity DataKi: 0.260nMAssay Description:Binding affinity to Opioid receptor delta 1 using [3H]DPDPE as a radioligand in guinea pigMore data for this Ligand-Target Pair
Affinity DataKi: 0.400nMAssay Description:Binding affinity to Opioid receptor delta 1 using [3H]DPDPE as a radioligand in guinea pigMore data for this Ligand-Target Pair
Affinity DataKi: 0.440nMAssay Description:Binding affinity to Opioid receptor delta 1 using [3H]DPDPE as a radioligand in guinea pigMore data for this Ligand-Target Pair
Affinity DataKi: 0.490nMAssay Description:Binding affinity to Opioid receptor delta 1 using [3H]DPDPE as a radioligand in guinea pigMore data for this Ligand-Target Pair
Affinity DataKi: 0.550nMAssay Description:Binding affinity to Opioid receptor delta 1 using [3H]DPDPE as a radioligand in guinea pigMore data for this Ligand-Target Pair
Affinity DataKi: 0.770nMAssay Description:Binding affinity to Opioid receptor delta 1 using [3H]DPDPE as a radioligand in guinea pigMore data for this Ligand-Target Pair
Affinity DataKi: 0.820nMAssay Description:Binding affinity to Opioid receptor delta 1 using [3H]DPDPE as a radioligand in guinea pigMore data for this Ligand-Target Pair
Affinity DataKi: 0.890nMAssay Description:Binding affinity to Opioid receptor delta 1 using [3H]DPDPE as a radioligand in guinea pigMore data for this Ligand-Target Pair
Affinity DataKi: 1.80nMAssay Description:Binding affinity to Opioid receptor delta 1 using [3H]DPDPE as a radioligand in guinea pigMore data for this Ligand-Target Pair
Affinity DataKi: 2.40nMAssay Description:Binding affinity to Opioid receptor delta 1 using [3H]DPDPE as a radioligand in guinea pigMore data for this Ligand-Target Pair
Affinity DataKi: 2.70nMAssay Description:Binding affinity to Opioid receptor delta 1 using [3H]DPDPE as a radioligand in guinea pigMore data for this Ligand-Target Pair
Affinity DataKi: 6.40nMAssay Description:Binding affinity to Opioid receptor delta 1 using [3H]DPDPE as a radioligand in guinea pigMore data for this Ligand-Target Pair
Affinity DataKi: 7.10nMAssay Description:Displacement of [3H]RX821002 from human alpha2A adrenergic receptor expressed in CHO cells after 30 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 8.10nMAssay Description:Binding affinity to Opioid receptor mu 1 by using [3H]DAMGO as a radioligand from guinea pigMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Bristol
Curated by ChEMBL
University Of Bristol
Curated by ChEMBL
Affinity DataKi: 8.30nMAssay Description:Binding affinity to Opioid receptor kappa 1 by using [3H]U-69593 as a radioligand from guinea pigMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Bristol
Curated by ChEMBL
University Of Bristol
Curated by ChEMBL
Affinity DataKi: 8.30nMAssay Description:Binding affinity to Opioid receptor kappa 1 by using [3H]U-69593 as a radioligand from guinea pigMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Bristol
Curated by ChEMBL
University Of Bristol
Curated by ChEMBL
Affinity DataKi: 9.80nMAssay Description:Binding affinity to Opioid receptor kappa 1 by using [3H]U-69593 as a radioligand from guinea pigMore data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Binding affinity to Opioid receptor delta 1 using [3H]DPDPE as a radioligand in guinea pigMore data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Binding affinity for rat imidazoline receptor I-1 from crude P2 membranesMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Bristol
Curated by ChEMBL
University Of Bristol
Curated by ChEMBL
Affinity DataKi: 12nMAssay Description:Binding affinity to Opioid receptor kappa 1 by using [3H]U-69593 as a radioligand from guinea pigMore data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:Binding affinity to Opioid receptor delta 1 using [3H]DPDPE as a radioligand in guinea pigMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Bristol
Curated by ChEMBL
University Of Bristol
Curated by ChEMBL
Affinity DataKi: 14nMAssay Description:Binding affinity to Opioid receptor kappa 1 by using [3H]U-69593 as a radioligand from guinea pigMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor(RAT)
Medical University Of Gdansk
Curated by ChEMBL
Medical University Of Gdansk
Curated by ChEMBL
Affinity DataKi: 14nMAssay Description:Displacement of [3H]RX821002 from alpha2-adrenoceptor in Sprague-Dawley rat brain membranes after 45 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Bristol
Curated by ChEMBL
University Of Bristol
Curated by ChEMBL
Affinity DataKi: 14nMAssay Description:Binding affinity to Opioid receptor kappa 1 by using [3H]U-69593 as a radioligand from guinea pigMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Bristol
Curated by ChEMBL
University Of Bristol
Curated by ChEMBL
Affinity DataKi: 15nMAssay Description:Binding affinity to Opioid receptor kappa 1 by using [3H]U-69593 as a radioligand from guinea pigMore data for this Ligand-Target Pair
Affinity DataKi: 16nMAssay Description:Binding affinity to Opioid receptor mu 1 by using [3H]DAMGO as a radioligand from guinea pigMore data for this Ligand-Target Pair
Affinity DataKi: 17nMAssay Description:Binding affinity to Opioid receptor mu 1 by using [3H]DAMGO as a radioligand from guinea pigMore data for this Ligand-Target Pair
Affinity DataKi: 18nMAssay Description:Displacement of [3H]RX821002 from human Alpha-2C adrenergic receptor expressed in CHO cells after 30 mins by scintillation countingMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Bristol
Curated by ChEMBL
University Of Bristol
Curated by ChEMBL
Affinity DataKi: 18nMAssay Description:Binding affinity to Opioid receptor kappa 1 by using [3H]U-69593 as a radioligand from guinea pigMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Bristol
Curated by ChEMBL
University Of Bristol
Curated by ChEMBL
Affinity DataKi: 18nMAssay Description:Binding affinity to Opioid receptor kappa 1 by using [3H]U-69593 as a radioligand from guinea pigMore data for this Ligand-Target Pair
Affinity DataKi: 19nMAssay Description:Binding affinity to Opioid receptor mu 1 by using [3H]DAMGO as a radioligand from guinea pigMore data for this Ligand-Target Pair
Affinity DataKi: 19nMAssay Description:Binding affinity to Opioid receptor delta 1 using [3H]DPDPE as a radioligand in guinea pigMore data for this Ligand-Target Pair
Affinity DataKi: 21nMAssay Description:Binding affinity to Opioid receptor mu 1 by using [3H]DAMGO as a radioligand from guinea pigMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Virginia Commonwealth University
Curated by ChEMBL
Virginia Commonwealth University
Curated by ChEMBL
Affinity DataKi: 22nMAssay Description:Binding affinity at 5-hydroxytryptamine 2A receptor of rat.More data for this Ligand-Target Pair
Affinity DataKi: 22nMAssay Description:Binding affinity to Opioid receptor mu 1 by using [3H]DAMGO as a radioligand from guinea pigMore data for this Ligand-Target Pair
Affinity DataKi: 23nMAssay Description:Displacement of [3H]RX821002 from human alpha2B adrenergic receptor expressed in CHO cells after 30 mins by scintillation countingMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor(RAT)
Medical University Of Gdansk
Curated by ChEMBL
Medical University Of Gdansk
Curated by ChEMBL
Affinity DataKi: 26nMAssay Description:Displacement of [3H]RX821002 from alpha2-adrenoceptor in Sprague-Dawley rat brain membranes after 45 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 27nMAssay Description:Binding affinity to Opioid receptor delta 1 using [3H]DPDPE as a radioligand in guinea pigMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Bristol
Curated by ChEMBL
University Of Bristol
Curated by ChEMBL
Affinity DataKi: 27nMAssay Description:Binding affinity to Opioid receptor kappa 1 by using [3H]U-69593 as a radioligand from guinea pigMore data for this Ligand-Target Pair
Affinity DataKi: 28nMAssay Description:Binding affinity to Opioid receptor mu 1 by using [3H]DAMGO as a radioligand from guinea pigMore data for this Ligand-Target Pair
Affinity DataKi: 30nMAssay Description:Binding affinity to Opioid receptor mu 1 by using [3H]DAMGO as a radioligand from guinea pigMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor(RAT)
Medical University Of Gdansk
Curated by ChEMBL
Medical University Of Gdansk
Curated by ChEMBL
Affinity DataKi: 30nMAssay Description:Displacement of [3H]RX821002 from alpha2-adrenoceptor in Sprague-Dawley rat brain membranes after 45 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 30.8nMAssay Description:Displacement of [3H]2BFI from imidazoline I1 receptor in Sprague-Dawley rat brain membrane after 45 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor(RAT)
Medical University Of Gdansk
Curated by ChEMBL
Medical University Of Gdansk
Curated by ChEMBL
Affinity DataKi: 31nMAssay Description:Displacement of [3H]RX821002 from alpha2-adrenoceptor in Sprague-Dawley rat brain membranes after 45 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 32nMAssay Description:Binding affinity to Opioid receptor mu 1 by using [3H]DAMGO as a radioligand from guinea pigMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor(RAT)
Medical University Of Gdansk
Curated by ChEMBL
Medical University Of Gdansk
Curated by ChEMBL
Affinity DataKi: 32nMAssay Description:Displacement of [3H]RX821002 from alpha2-adrenoceptor in Sprague-Dawley rat brain membranes after 45 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 33nMAssay Description:Displacement of [3H]RS-79948-197 from human alpha2A adrenoceptor expressed in CHO-K1 cells after 45 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 36nMAssay Description:Binding affinity to Opioid receptor mu 1 by using [3H]DAMGO as a radioligand from guinea pigMore data for this Ligand-Target Pair