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Found 262 with Last Name = 'hudson' and Initial = 'al'
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of Bristol

Curated by ChEMBL
LigandPNGBDBM21864((21R)-22-(cyclopropylmethyl)-14-oxa-11,22-diazahep...)
Affinity DataKi:  0.150nMAssay Description:Binding affinity to Opioid receptor delta 1 using [3H]DPDPE as a radioligand in guinea pigMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of Bristol

Curated by ChEMBL
LigandPNGBDBM50098195(22-cyclopropylmethyl-11-(2-fluoroethyl)-14-oxa-11,...)
Affinity DataKi:  0.240nMAssay Description:Binding affinity to Opioid receptor delta 1 using [3H]DPDPE as a radioligand in guinea pigMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of Bristol

Curated by ChEMBL
LigandPNGBDBM50098192(22-cyclopropylmethyl-11-ethyl-14-oxa-11,22-diazahe...)
Affinity DataKi:  0.260nMAssay Description:Binding affinity to Opioid receptor delta 1 using [3H]DPDPE as a radioligand in guinea pigMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of Bristol

Curated by ChEMBL
LigandPNGBDBM50098196(22-cyclopropylmethyl-11-(3-fluoropropyl)-14-oxa-11...)
Affinity DataKi:  0.400nMAssay Description:Binding affinity to Opioid receptor delta 1 using [3H]DPDPE as a radioligand in guinea pigMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of Bristol

Curated by ChEMBL
LigandPNGBDBM50098199(22-cyclopropylmethyl-11-propyl-14-oxa-11,22-diazah...)
Affinity DataKi:  0.440nMAssay Description:Binding affinity to Opioid receptor delta 1 using [3H]DPDPE as a radioligand in guinea pigMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of Bristol

Curated by ChEMBL
LigandPNGBDBM50451343(CHEMBL477154)
Affinity DataKi:  0.490nMAssay Description:Binding affinity to Opioid receptor delta 1 using [3H]DPDPE as a radioligand in guinea pigMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of Bristol

Curated by ChEMBL
LigandPNGBDBM50098201(CHEMBL367962 | N-[22-cyclopropylmethyl-11-(2-fluor...)
Affinity DataKi:  0.550nMAssay Description:Binding affinity to Opioid receptor delta 1 using [3H]DPDPE as a radioligand in guinea pigMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of Bristol

Curated by ChEMBL
LigandPNGBDBM50098186(22-cyclopropylmethyl-2-ethylamino-14-oxa-11,22-dia...)
Affinity DataKi:  0.770nMAssay Description:Binding affinity to Opioid receptor delta 1 using [3H]DPDPE as a radioligand in guinea pigMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of Bristol

Curated by ChEMBL
LigandPNGBDBM50098198(CHEMBL170399 | N-[22-cyclopropylmethyl-11-(3-fluor...)
Affinity DataKi:  0.820nMAssay Description:Binding affinity to Opioid receptor delta 1 using [3H]DPDPE as a radioligand in guinea pigMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of Bristol

Curated by ChEMBL
LigandPNGBDBM50098188(CHEMBL176537 | N-[22-cyclopropylmethyl-16-hydroxy-...)
Affinity DataKi:  0.890nMAssay Description:Binding affinity to Opioid receptor delta 1 using [3H]DPDPE as a radioligand in guinea pigMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of Bristol

Curated by ChEMBL
LigandPNGBDBM50098187(22-cyclopropylmethyl-2-(3-propylsulfanylpropylamin...)
Affinity DataKi:  1.80nMAssay Description:Binding affinity to Opioid receptor delta 1 using [3H]DPDPE as a radioligand in guinea pigMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of Bristol

Curated by ChEMBL
LigandPNGBDBM50098193(22-cyclopropylmethyl-2-propylamino-14-oxa-11,22-di...)
Affinity DataKi:  2.40nMAssay Description:Binding affinity to Opioid receptor delta 1 using [3H]DPDPE as a radioligand in guinea pigMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of Bristol

Curated by ChEMBL
LigandPNGBDBM50098202(11-(3-fluoropropyl)-22-methyl-14-oxa-11,22-diazahe...)
Affinity DataKi:  2.70nMAssay Description:Binding affinity to Opioid receptor delta 1 using [3H]DPDPE as a radioligand in guinea pigMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of Bristol

Curated by ChEMBL
LigandPNGBDBM50098194(11-(2-fluoroethyl)-22-methyl-(2S)-14-oxa-11,22-dia...)
Affinity DataKi:  6.40nMAssay Description:Binding affinity to Opioid receptor delta 1 using [3H]DPDPE as a radioligand in guinea pigMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50019848(2-(2,3-dihydro-1,4-benzodioxin-2-yl)-4,5-dihydro-1...)
Affinity DataKi:  7.10nMAssay Description:Displacement of [3H]RX821002 from human alpha2A adrenergic receptor expressed in CHO cells after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
University Of Bristol

Curated by ChEMBL
LigandPNGBDBM50098187(22-cyclopropylmethyl-2-(3-propylsulfanylpropylamin...)
Affinity DataKi:  8.10nMAssay Description:Binding affinity to Opioid receptor mu 1 by using [3H]DAMGO as a radioligand from guinea pigMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Bristol

Curated by ChEMBL
LigandPNGBDBM50451343(CHEMBL477154)
Affinity DataKi:  8.30nMAssay Description:Binding affinity to Opioid receptor kappa 1 by using [3H]U-69593 as a radioligand from guinea pigMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Bristol

Curated by ChEMBL
LigandPNGBDBM50098195(22-cyclopropylmethyl-11-(2-fluoroethyl)-14-oxa-11,...)
Affinity DataKi:  8.30nMAssay Description:Binding affinity to Opioid receptor kappa 1 by using [3H]U-69593 as a radioligand from guinea pigMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Bristol

Curated by ChEMBL
LigandPNGBDBM50098196(22-cyclopropylmethyl-11-(3-fluoropropyl)-14-oxa-11...)
Affinity DataKi:  9.80nMAssay Description:Binding affinity to Opioid receptor kappa 1 by using [3H]U-69593 as a radioligand from guinea pigMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of Bristol

Curated by ChEMBL
LigandPNGBDBM50098200(2N-(2-fluoroethyl)-22-cyclopropylmethyl-16-methoxy...)
Affinity DataKi:  10nMAssay Description:Binding affinity to Opioid receptor delta 1 using [3H]DPDPE as a radioligand in guinea pigMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNischarin(Homo sapiens (Human))
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50138500(2-((E)-Styryl)-4,5-dihydro-1H-imidazole | 2-styryl...)
Affinity DataKi:  10nMAssay Description:Binding affinity for rat imidazoline receptor I-1 from crude P2 membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Bristol

Curated by ChEMBL
LigandPNGBDBM50098199(22-cyclopropylmethyl-11-propyl-14-oxa-11,22-diazah...)
Affinity DataKi:  12nMAssay Description:Binding affinity to Opioid receptor kappa 1 by using [3H]U-69593 as a radioligand from guinea pigMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of Bristol

Curated by ChEMBL
LigandPNGBDBM50098191(2N-(3-fluoropropyl)-22-cyclopropylmethyl-16-methox...)
Affinity DataKi:  13nMAssay Description:Binding affinity to Opioid receptor delta 1 using [3H]DPDPE as a radioligand in guinea pigMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Bristol

Curated by ChEMBL
LigandPNGBDBM50098192(22-cyclopropylmethyl-11-ethyl-14-oxa-11,22-diazahe...)
Affinity DataKi:  14nMAssay Description:Binding affinity to Opioid receptor kappa 1 by using [3H]U-69593 as a radioligand from guinea pigMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50271255(1-[(Imidazolidin-2-yl)imino]indazole hydrochloride...)
Affinity DataKi:  14nMAssay Description:Displacement of [3H]RX821002 from alpha2-adrenoceptor in Sprague-Dawley rat brain membranes after 45 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Bristol

Curated by ChEMBL
LigandPNGBDBM21864((21R)-22-(cyclopropylmethyl)-14-oxa-11,22-diazahep...)
Affinity DataKi:  14nMAssay Description:Binding affinity to Opioid receptor kappa 1 by using [3H]U-69593 as a radioligand from guinea pigMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Bristol

Curated by ChEMBL
LigandPNGBDBM50098187(22-cyclopropylmethyl-2-(3-propylsulfanylpropylamin...)
Affinity DataKi:  15nMAssay Description:Binding affinity to Opioid receptor kappa 1 by using [3H]U-69593 as a radioligand from guinea pigMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
University Of Bristol

Curated by ChEMBL
LigandPNGBDBM50098199(22-cyclopropylmethyl-11-propyl-14-oxa-11,22-diazah...)
Affinity DataKi:  16nMAssay Description:Binding affinity to Opioid receptor mu 1 by using [3H]DAMGO as a radioligand from guinea pigMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
University Of Bristol

Curated by ChEMBL
LigandPNGBDBM50098195(22-cyclopropylmethyl-11-(2-fluoroethyl)-14-oxa-11,...)
Affinity DataKi:  17nMAssay Description:Binding affinity to Opioid receptor mu 1 by using [3H]DAMGO as a radioligand from guinea pigMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50019848(2-(2,3-dihydro-1,4-benzodioxin-2-yl)-4,5-dihydro-1...)
Affinity DataKi:  18nMAssay Description:Displacement of [3H]RX821002 from human Alpha-2C adrenergic receptor expressed in CHO cells after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Bristol

Curated by ChEMBL
LigandPNGBDBM50098201(CHEMBL367962 | N-[22-cyclopropylmethyl-11-(2-fluor...)
Affinity DataKi:  18nMAssay Description:Binding affinity to Opioid receptor kappa 1 by using [3H]U-69593 as a radioligand from guinea pigMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Bristol

Curated by ChEMBL
LigandPNGBDBM50098198(CHEMBL170399 | N-[22-cyclopropylmethyl-11-(3-fluor...)
Affinity DataKi:  18nMAssay Description:Binding affinity to Opioid receptor kappa 1 by using [3H]U-69593 as a radioligand from guinea pigMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
University Of Bristol

Curated by ChEMBL
LigandPNGBDBM50098196(22-cyclopropylmethyl-11-(3-fluoropropyl)-14-oxa-11...)
Affinity DataKi:  19nMAssay Description:Binding affinity to Opioid receptor mu 1 by using [3H]DAMGO as a radioligand from guinea pigMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of Bristol

Curated by ChEMBL
LigandPNGBDBM50098197(2N-propyl-22-cyclopropylmethyl-16-methoxy-(13R)-14...)
Affinity DataKi:  19nMAssay Description:Binding affinity to Opioid receptor delta 1 using [3H]DPDPE as a radioligand in guinea pigMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
University Of Bristol

Curated by ChEMBL
LigandPNGBDBM50098198(CHEMBL170399 | N-[22-cyclopropylmethyl-11-(3-fluor...)
Affinity DataKi:  21nMAssay Description:Binding affinity to Opioid receptor mu 1 by using [3H]DAMGO as a radioligand from guinea pigMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50136494(8-Bromo-2,3,4,9-tetrahydro-1H-beta-carboline | CHE...)
Affinity DataKi:  22nMAssay Description:Binding affinity at 5-hydroxytryptamine 2A receptor of rat.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
University Of Bristol

Curated by ChEMBL
LigandPNGBDBM50098192(22-cyclopropylmethyl-11-ethyl-14-oxa-11,22-diazahe...)
Affinity DataKi:  22nMAssay Description:Binding affinity to Opioid receptor mu 1 by using [3H]DAMGO as a radioligand from guinea pigMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50019848(2-(2,3-dihydro-1,4-benzodioxin-2-yl)-4,5-dihydro-1...)
Affinity DataKi:  23nMAssay Description:Displacement of [3H]RX821002 from human alpha2B adrenergic receptor expressed in CHO cells after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50497435(CHEMBL3343699)
Affinity DataKi:  26nMAssay Description:Displacement of [3H]RX821002 from alpha2-adrenoceptor in Sprague-Dawley rat brain membranes after 45 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of Bristol

Curated by ChEMBL
LigandPNGBDBM50098185(2N-ethyl-22-cyclopropylmethyl-16-methoxy-(13R)-14-...)
Affinity DataKi:  27nMAssay Description:Binding affinity to Opioid receptor delta 1 using [3H]DPDPE as a radioligand in guinea pigMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Bristol

Curated by ChEMBL
LigandPNGBDBM50098188(CHEMBL176537 | N-[22-cyclopropylmethyl-16-hydroxy-...)
Affinity DataKi:  27nMAssay Description:Binding affinity to Opioid receptor kappa 1 by using [3H]U-69593 as a radioligand from guinea pigMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
University Of Bristol

Curated by ChEMBL
LigandPNGBDBM21864((21R)-22-(cyclopropylmethyl)-14-oxa-11,22-diazahep...)
Affinity DataKi:  28nMAssay Description:Binding affinity to Opioid receptor mu 1 by using [3H]DAMGO as a radioligand from guinea pigMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
University Of Bristol

Curated by ChEMBL
LigandPNGBDBM50098194(11-(2-fluoroethyl)-22-methyl-(2S)-14-oxa-11,22-dia...)
Affinity DataKi:  30nMAssay Description:Binding affinity to Opioid receptor mu 1 by using [3H]DAMGO as a radioligand from guinea pigMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50497438(CHEMBL3343704)
Affinity DataKi:  30nMAssay Description:Displacement of [3H]RX821002 from alpha2-adrenoceptor in Sprague-Dawley rat brain membranes after 45 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNischarin(RAT)
Medical University Of Gdansk

Curated by ChEMBL
LigandPNGBDBM50334197(7-Chloro-3-[(imidazolidin-2-yl)imino]indazole hydr...)
Affinity DataKi:  30.8nMAssay Description:Displacement of [3H]2BFI from imidazoline I1 receptor in Sprague-Dawley rat brain membrane after 45 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50497439(CHEMBL3343700)
Affinity DataKi:  31nMAssay Description:Displacement of [3H]RX821002 from alpha2-adrenoceptor in Sprague-Dawley rat brain membranes after 45 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
University Of Bristol

Curated by ChEMBL
LigandPNGBDBM50098201(CHEMBL367962 | N-[22-cyclopropylmethyl-11-(2-fluor...)
Affinity DataKi:  32nMAssay Description:Binding affinity to Opioid receptor mu 1 by using [3H]DAMGO as a radioligand from guinea pigMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50497436(CHEMBL3343703)
Affinity DataKi:  32nMAssay Description:Displacement of [3H]RX821002 from alpha2-adrenoceptor in Sprague-Dawley rat brain membranes after 45 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50497435(CHEMBL3343699)
Affinity DataKi:  33nMAssay Description:Displacement of [3H]RS-79948-197 from human alpha2A adrenoceptor expressed in CHO-K1 cells after 45 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
University Of Bristol

Curated by ChEMBL
LigandPNGBDBM50098188(CHEMBL176537 | N-[22-cyclopropylmethyl-16-hydroxy-...)
Affinity DataKi:  36nMAssay Description:Binding affinity to Opioid receptor mu 1 by using [3H]DAMGO as a radioligand from guinea pigMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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