TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
Eisai
Curated by ChEMBL
Eisai
Curated by ChEMBL
Affinity DataKi: 9.5nMAssay Description:Inhibitory activity against AcetylcholinesteraseMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
Eisai
Curated by ChEMBL
Eisai
Curated by ChEMBL
Affinity DataKi: 9.5nMAssay Description:Inhibitory activity against AcetylcholinesteraseMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
Eisai
Curated by ChEMBL
Eisai
Curated by ChEMBL
Affinity DataKi: 17.5nMAssay Description:Inhibitory activity was calculated for the model Acetylcholinesterase (Expt-1)More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
Eisai
Curated by ChEMBL
Eisai
Curated by ChEMBL
Affinity DataKi: 18nMAssay Description:Inhibitory activity was calculated for the model Acetylcholinesterase (Expt-1)More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
Eisai
Curated by ChEMBL
Eisai
Curated by ChEMBL
Affinity DataKi: 19nMAssay Description:Inhibitory activity was calculated for the model Acetylcholinesterase (Expt-1)More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
Eisai
Curated by ChEMBL
Eisai
Curated by ChEMBL
Affinity DataKi: 27nMAssay Description:Inhibitory activity against AcetylcholinesteraseMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
Eisai
Curated by ChEMBL
Eisai
Curated by ChEMBL
Affinity DataKi: 37.6nMAssay Description:Inhibitory activity was calculated for the model Acetylcholinesterase (Expt-2)More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
Eisai
Curated by ChEMBL
Eisai
Curated by ChEMBL
Affinity DataKi: 38nMAssay Description:Inhibitory activity was calculated for the model Acetylcholinesterase (Expt-2)More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
Eisai
Curated by ChEMBL
Eisai
Curated by ChEMBL
Affinity DataKi: 47nMAssay Description:Inhibitory activity was calculated for the model Acetylcholinesterase (Expt-2)More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
Eisai
Curated by ChEMBL
Eisai
Curated by ChEMBL
Affinity DataKi: 54nMAssay Description:Inhibitory activity against AcetylcholinesteraseMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
Eisai
Curated by ChEMBL
Eisai
Curated by ChEMBL
Affinity DataKi: 54nMAssay Description:Inhibitory activity was calculated for the model Acetylcholinesterase (Expt-2)More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
Eisai
Curated by ChEMBL
Eisai
Curated by ChEMBL
Affinity DataKi: 122nMAssay Description:Inhibitory activity was calculated for the model Acetylcholinesterase (Expt-1)More data for this Ligand-Target Pair
Affinity DataIC50: 0.300nMAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. The amount of a yellow substance formed after incubation was d...More data for this Ligand-Target Pair
Affinity DataIC50: 0.430nMAssay Description:In vitro inhibitory activity of the compound against acetylcholinesteraseMore data for this Ligand-Target Pair
Affinity DataIC50: 0.560nMAssay Description:In vitro inhibitory concentration against acetylcholinesterase (AChE) obtained from mouse brain homogenate.More data for this Ligand-Target Pair
Affinity DataIC50: 0.600nMAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. The amount of a yellow substance formed after incubation was d...More data for this Ligand-Target Pair
Affinity DataIC50: 0.600nMAssay Description:Inhibitory activity against acetylcholinesteraseMore data for this Ligand-Target Pair
Affinity DataIC50: 0.600nMAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. The amount of a yellow substance formed after incubation was d...More data for this Ligand-Target Pair
Affinity DataIC50: 0.680nMAssay Description:Inhibitory activity against acetylcholinesteraseMore data for this Ligand-Target Pair
Affinity DataIC50: 0.680nMAssay Description:Inhibitory concentration of the compound was determined in vitro and ex vivo for anti-AChE activity in rat brainMore data for this Ligand-Target Pair
Affinity DataIC50: 0.690nMAssay Description:In vitro inhibitory concentration against acetylcholinesterase (AChE) obtained from mouse brain homogenate.More data for this Ligand-Target Pair
Affinity DataIC50: 0.820nMAssay Description:Inhibition of acetylcholinesterase activityMore data for this Ligand-Target Pair
Affinity DataIC50: 0.900nMAssay Description:Inhibition of acetylcholinesterase activityMore data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Inhibition of acetylcholinesterase.More data for this Ligand-Target Pair
Affinity DataIC50: 1.20nMAssay Description:In vitro inhibitory concentration against acetylcholinesterase (AChE) obtained from mouse brain homogenate.More data for this Ligand-Target Pair
Affinity DataIC50: 1.20nMAssay Description:Inhibitory activity against acetylcholinesteraseMore data for this Ligand-Target Pair
Affinity DataIC50: 1.30nMAssay Description:Inhibition of acetylcholinesterase.More data for this Ligand-Target Pair
Affinity DataIC50: 1.5nMAssay Description:Inhibition of acetylcholinesterase activityMore data for this Ligand-Target Pair
Affinity DataIC50: 1.5nMAssay Description:Inhibitory activity against acetylcholinesteraseMore data for this Ligand-Target Pair
Affinity DataIC50: 1.80nMAssay Description:IC50 against acetylcholinesterase; value ranges from 1.3-380 nM.More data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:Inhibition of acetylcholinesterase.More data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:Inhibitory activity against acetylcholinesteraseMore data for this Ligand-Target Pair
Affinity DataIC50: 2.20nMAssay Description:In vitro inhibitory concentration against acetylcholinesterase (AChE) obtained from mouse brain homogenate.More data for this Ligand-Target Pair
Affinity DataIC50: 2.40nMAssay Description:In vitro inhibitory concentration against acetylcholinesterase (AChE) obtained from mouse brain homogenate.More data for this Ligand-Target Pair
Affinity DataIC50: 2.70nMAssay Description:Inhibition of Acetylcholinesterase activity in mouse brain homogenateMore data for this Ligand-Target Pair
Affinity DataIC50: 2.80nMAssay Description:In vitro inhibitory concentration against acetylcholinesterase (AChE) obtained from mouse brain homogenate.More data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:Inhibition of acetylcholinesterase activityMore data for this Ligand-Target Pair
Affinity DataIC50: 4nMAssay Description:Inhibition of Acetylcholinesterase activity in mouse brain homogenateMore data for this Ligand-Target Pair
Affinity DataIC50: 4nMAssay Description:Inhibition of acetylcholinesterase.More data for this Ligand-Target Pair
Affinity DataIC50: 4nMAssay Description:Inhibitory activity against acetylcholinesteraseMore data for this Ligand-Target Pair
Affinity DataIC50: 4.20nMAssay Description:Inhibition of acetylcholinesterase activityMore data for this Ligand-Target Pair
Affinity DataIC50: 4.20nMAssay Description:In vitro inhibitory concentration against acetylcholinesterase (AChE) obtained from mouse brain homogenate.More data for this Ligand-Target Pair
Affinity DataIC50: 4.5nMAssay Description:In vitro inhibitory concentration against acetylcholinesterase (AChE) obtained from mouse brain homogenate.More data for this Ligand-Target Pair
Affinity DataIC50: 5.20nMAssay Description:Inhibition of acetylcholinesterase.More data for this Ligand-Target Pair
Affinity DataIC50: 5.20nMAssay Description:Inhibition of acetylcholinesterase.More data for this Ligand-Target Pair
Affinity DataIC50: 5.30nMAssay Description:Inhibition of acetylcholinesterase activityMore data for this Ligand-Target Pair
Affinity DataIC50: 5.30nMAssay Description:Inhibition of acetylcholinesterase activityMore data for this Ligand-Target Pair
Affinity DataIC50: 5.30nMAssay Description:In vitro inhibitory activity of the compound against acetylcholinesteraseMore data for this Ligand-Target Pair
Affinity DataIC50: 5.40nMAssay Description:In vitro inhibitory concentration against acetylcholinesterase (AChE) obtained from mouse brain homogenate.More data for this Ligand-Target Pair
Affinity DataIC50: 5.70nMAssay Description:Inhibitory activity against acetylcholinesteraseMore data for this Ligand-Target Pair