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Found 917 with Last Name = 'imai' and Initial = 'm'
TargetTranslocator protein(Rattus norvegicus (rat))
National Institute Of Mental Health

Curated by ChEMBL
LigandPNGBDBM50122293(CHEMBL401000 | CHEMBL63064 | N-(2,5-Dimethoxy-benz...)
Affinity DataKi:  0.0726nMAssay Description:Displacement of [3H]PK11195 from rat PBR receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
National Institute Of Mental Health

Curated by ChEMBL
LigandPNGBDBM50122293(CHEMBL401000 | CHEMBL63064 | N-(2,5-Dimethoxy-benz...)
Affinity DataKi:  0.0726nMAssay Description:Binding affinity to PBR in Sprague-Dawley rat mitochondrial tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
National Institute Of Mental Health

Curated by ChEMBL
LigandPNGBDBM50229593(CHEMBL253596 | N-acetyl-N-(2-methoxycarbonylbenzyl...)
Affinity DataKi:  0.0978nMAssay Description:Binding affinity to PBR in Sprague-Dawley rat mitochondrial tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50360146(CHEMBL1929368)
Affinity DataKi:  0.120nMAssay Description:Displacement of [3H]DPDPE from delta opioid receptor in mouse whole brain membranes without cerebellumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50294428(CHEMBL552308 | SN-28)
Affinity DataKi:  0.140nMAssay Description:Displacement of [3H]DADLE from delta opioid receptor in rat cerebrum membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50294428(CHEMBL552308 | SN-28)
Affinity DataKi:  0.140nMAssay Description:Displacement of [3H]DADLE from delta opioid receptor in rat cerebellum membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
National Institute Of Mental Health

Curated by ChEMBL
LigandPNGBDBM50255877(CHEMBL473435 | N-Fluoroacetyl-N-(2,5-dimethoxybenz...)
Affinity DataKi:  0.180nMAssay Description:Displacement of [3H]PK11195 from rat PBR receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50294427(CHEMBL564538 | SN-23)
Affinity DataKi:  0.190nMAssay Description:Displacement of [3H]DADLE from delta opioid receptor in rat cerebrum membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50294427(CHEMBL564538 | SN-23)
Affinity DataKi:  0.190nMAssay Description:Displacement of [3H]DADLE from delta opioid receptor in rat cerebellum membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50294426(CHEMBL559518 | SN-11)
Affinity DataKi:  0.190nMAssay Description:Displacement of [3H]DADLE from delta opioid receptor in rat cerebrum membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50294426(CHEMBL559518 | SN-11)
Affinity DataKi:  0.190nMAssay Description:Displacement of [3H]DADLE from delta opioid receptor in rat cerebellum membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Homo sapiens (Human))
National Institute Of Mental Health

Curated by ChEMBL
LigandPNGBDBM50122293(CHEMBL401000 | CHEMBL63064 | N-(2,5-Dimethoxy-benz...)
Affinity DataKi:  0.242nMAssay Description:Binding affinity to PBR in human mitochondrial tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Homo sapiens (Human))
National Institute Of Mental Health

Curated by ChEMBL
LigandPNGBDBM50122293(CHEMBL401000 | CHEMBL63064 | N-(2,5-Dimethoxy-benz...)
Affinity DataKi:  0.242nMAssay Description:Displacement of [3H]PK11195 from human PBR receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50360142(CHEMBL1929365)
Affinity DataKi:  0.270nMAssay Description:Displacement of [3H]DADLE from delta opioid receptor in rat cerebrum membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Kitasato University

Curated by ChEMBL
LigandPNGBDBM21864((21R)-22-(cyclopropylmethyl)-14-oxa-11,22-diazahep...)
Affinity DataKi:  0.290nMAssay Description:Displacement of [3H]DADLE from delta opioid receptor in rat cerebrum membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50294428(CHEMBL552308 | SN-28)
Affinity DataKi:  0.290nMAssay Description:Displacement of [3H]DPDPE from delta opioid receptor in mouse whole brain membranes without cerebellumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Kitasato University

Curated by ChEMBL
LigandPNGBDBM21864((21R)-22-(cyclopropylmethyl)-14-oxa-11,22-diazahep...)
Affinity DataKi:  0.290nMAssay Description:Displacement of [3H]DADLE from delta opioid receptor in rat cerebellum membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50360147(CHEMBL1929369)
Affinity DataKi:  0.350nMAssay Description:Displacement of [3H]DPDPE from delta opioid receptor in mouse whole brain membranes without cerebellumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50294426(CHEMBL559518 | SN-11)
Affinity DataKi:  0.360nMAssay Description:Displacement of [3H]U-69,593 from kappa opioid receptor in guinea pig cerebrum membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50294426(CHEMBL559518 | SN-11)
Affinity DataKi:  0.360nMAssay Description:Displacement of [3H]U-69593 from kappa opioid receptor in guinea pig cerebellumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50360143(CHEMBL1929363)
Affinity DataKi:  0.430nMAssay Description:Displacement of [3H]DADLE from delta opioid receptor in rat cerebrum membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
National Institute Of Mental Health

Curated by ChEMBL
LigandPNGBDBM50229594(CHEMBL253597 | N-(2-methoxybenzyl)-N-(4-phenoxypyr...)
Affinity DataKi:  0.680nMAssay Description:Binding affinity to PBR in Sprague-Dawley rat mitochondrial tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
National Institute Of Mental Health

Curated by ChEMBL
LigandPNGBDBM50229596(1-(2-chlorophenyl)-N-methyl-N-[(1S)-1-methylpropyl...)
Affinity DataKi:  0.730nMAssay Description:Binding affinity to PBR in Sprague-Dawley rat mitochondrial tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50294426(CHEMBL559518 | SN-11)
Affinity DataKi:  0.770nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat cerebrum membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50294426(CHEMBL559518 | SN-11)
Affinity DataKi:  0.770nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat cerebellum membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Homo sapiens (Human))
National Institute Of Mental Health

Curated by ChEMBL
LigandPNGBDBM50255877(CHEMBL473435 | N-Fluoroacetyl-N-(2,5-dimethoxybenz...)
Affinity DataKi:  0.997nMAssay Description:Displacement of [3H]PK11195 from human PBR receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50360141(CHEMBL1929364)
Affinity DataKi:  1nMAssay Description:Displacement of [3H]DADLE from delta opioid receptor in rat cerebrum membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50360146(CHEMBL1929368)
Affinity DataKi:  1.10nMAssay Description:Displacement of [3H]U-69,593 from kappa opioid receptor in guinea pig cerebrum membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50360140(CHEMBL1929362)
Affinity DataKi:  1.20nMAssay Description:Displacement of [3H]DADLE from delta opioid receptor in rat cerebrum membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50290872((-)-rel-3-((4aR,12aS)-2-methyl-1,2,3,4,4a,5,12,12a...)
Affinity DataKi:  1.40nMAssay Description:Displacement of [3H]DADLE from delta opioid receptor in rat cerebrum membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Homo sapiens (Human))
National Institute Of Mental Health

Curated by ChEMBL
LigandPNGBDBM50229593(CHEMBL253596 | N-acetyl-N-(2-methoxycarbonylbenzyl...)
Affinity DataKi:  1.40nMAssay Description:Binding affinity to PBR in human mitochondrial tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50290872((-)-rel-3-((4aR,12aS)-2-methyl-1,2,3,4,4a,5,12,12a...)
Affinity DataKi:  1.40nMAssay Description:Displacement of [3H]DADLE from delta opioid receptor in rat cerebellum membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Homo sapiens (Human))
National Institute Of Mental Health

Curated by ChEMBL
LigandPNGBDBM50229594(CHEMBL253597 | N-(2-methoxybenzyl)-N-(4-phenoxypyr...)
Affinity DataKi:  2.5nMAssay Description:Binding affinity to PBR in human mitochondrial tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50360147(CHEMBL1929369)
Affinity DataKi:  3.5nMAssay Description:Displacement of [3H]U-69,593 from kappa opioid receptor in guinea pig cerebrum membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50294427(CHEMBL564538 | SN-23)
Affinity DataKi:  4.40nMAssay Description:Displacement of [3H]U-69,593 from kappa opioid receptor in guinea pig cerebrum membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50294427(CHEMBL564538 | SN-23)
Affinity DataKi:  4.40nMAssay Description:Displacement of [3H]U-69593 from kappa opioid receptor in guinea pig cerebellumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Homo sapiens (Human))
National Institute Of Mental Health

Curated by ChEMBL
LigandPNGBDBM50229596(1-(2-chlorophenyl)-N-methyl-N-[(1S)-1-methylpropyl...)
Affinity DataKi:  4.5nMAssay Description:Binding affinity to PBR in human mitochondrial tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50360145(CHEMBL1929367)
Affinity DataKi:  4.70nMAssay Description:Displacement of [3H]DPDPE from delta opioid receptor in mouse whole brain membranes without cerebellumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(MOUSE)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50360146(CHEMBL1929368)
Affinity DataKi:  6.30nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in mouse whole brain membranes without cerebellumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50294428(CHEMBL552308 | SN-28)
Affinity DataKi:  10nMAssay Description:Displacement of [3H]U-69,593 from kappa opioid receptor in guinea pig cerebrum membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50294428(CHEMBL552308 | SN-28)
Affinity DataKi:  10nMAssay Description:Displacement of [3H]U-69593 from kappa opioid receptor in guinea pig cerebellumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50294428(CHEMBL552308 | SN-28)
Affinity DataKi:  12nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat cerebellum membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50294428(CHEMBL552308 | SN-28)
Affinity DataKi:  12nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat cerebrum membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50360144(CHEMBL1929366)
Affinity DataKi:  12nMAssay Description:Displacement of [3H]DPDPE from delta opioid receptor in mouse whole brain membranes without cerebellumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50360143(CHEMBL1929363)
Affinity DataKi:  13nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat cerebrum membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(MOUSE)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50360145(CHEMBL1929367)
Affinity DataKi:  13nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in mouse whole brain membranes without cerebellumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50294428(CHEMBL552308 | SN-28)
Affinity DataKi:  14nMAssay Description:Displacement of [3H]U-69,593 from kappa opioid receptor in guinea pig cerebrum membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Kitasato University

Curated by ChEMBL
LigandPNGBDBM21864((21R)-22-(cyclopropylmethyl)-14-oxa-11,22-diazahep...)
Affinity DataKi:  14nMAssay Description:Displacement of [3H]U-69593 from kappa opioid receptor in guinea pig cerebellumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Kitasato University

Curated by ChEMBL
LigandPNGBDBM21864((21R)-22-(cyclopropylmethyl)-14-oxa-11,22-diazahep...)
Affinity DataKi:  14nMAssay Description:Displacement of [3H]U-69,593 from kappa opioid receptor in guinea pig cerebrum membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50360143(CHEMBL1929363)
Affinity DataKi:  15nMAssay Description:Displacement of [3H]U-69,593 from kappa opioid receptor in guinea pig cerebrum membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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