Affinity DataKi: 100nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 200nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 300nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.00E+3nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.00E+3nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.30E+3nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.40E+3nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.50E+3nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 2.90E+3nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB1 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
Affinity DataKi: 3.00E+3nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
Affinity DataKi: 5.40E+3nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
Affinity DataKi: 7.80E+3nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB1 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
Target7-dehydrocholesterol reductase(Homo sapiens (Human))
Martin-Luther-Universit£T Halle-Wittenberg
Curated by ChEMBL
Martin-Luther-Universit£T Halle-Wittenberg
Curated by ChEMBL
Affinity DataIC50: 2.30nMAssay Description:Inhibition of 7-dehydroxycholesterol reductase-mediated cholesterol biosynthesis in human HL60 cells assessed as inhibition of 2-[13C]acetate after 2...More data for this Ligand-Target Pair
Target7-dehydrocholesterol reductase(Homo sapiens (Human))
Martin-Luther-Universit£T Halle-Wittenberg
Curated by ChEMBL
Martin-Luther-Universit£T Halle-Wittenberg
Curated by ChEMBL
Affinity DataIC50: 120nMAssay Description:Inhibition of 7-dehydroxycholesterol reductase-mediated cholesterol biosynthesis in human HL60 cells assessed as inhibition of 2-[13C]acetate after 2...More data for this Ligand-Target Pair
Target7-dehydrocholesterol reductase(Homo sapiens (Human))
Martin-Luther-Universit£T Halle-Wittenberg
Curated by ChEMBL
Martin-Luther-Universit£T Halle-Wittenberg
Curated by ChEMBL
Affinity DataIC50: 500nMAssay Description:Inhibition of 7-dehydroxycholesterol reductase-mediated cholesterol biosynthesis in human HL60 cells assessed as inhibition of 2-[13C]acetate after 2...More data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Martin-Luther-Universit£T Halle-Wittenberg
Curated by ChEMBL
Martin-Luther-Universit£T Halle-Wittenberg
Curated by ChEMBL
Affinity DataIC50: 1.32E+3nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Philipps-Universit£T
Curated by ChEMBL
Philipps-Universit£T
Curated by ChEMBL
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of TRPV1More data for this Ligand-Target Pair
Target7-dehydrocholesterol reductase(Homo sapiens (Human))
Martin-Luther-Universit£T Halle-Wittenberg
Curated by ChEMBL
Martin-Luther-Universit£T Halle-Wittenberg
Curated by ChEMBL
Affinity DataIC50: 7.30E+3nMAssay Description:Inhibition of 7-dehydroxycholesterol reductase-mediated cholesterol biosynthesis in human HL60 cells assessed as inhibition of 2-[13C]acetate after 2...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)
Martin-Luther-Universit£T Halle-Wittenberg
Curated by ChEMBL
Martin-Luther-Universit£T Halle-Wittenberg
Curated by ChEMBL
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis PknB (279 residues) expressed in Escherichia coli BL21 (DE3) pLysS assessed as reduction in PknB autophospho...More data for this Ligand-Target Pair
Affinity DataIC50: 4.20E+4nMAssay Description:Inhibition of COX-1 in C57BL/6 mouse brain homogenateMore data for this Ligand-Target Pair
Affinity DataIC50: 6.90E+4nMAssay Description:Inhibition of COX-2 in C57BL/6 mouse brain homogenateMore data for this Ligand-Target Pair
Affinity DataIC50: 1.07E+5nMAssay Description:Inhibition of cyclooxygenase 2 in human whole blood assessed as prostaglandin H2 levelMore data for this Ligand-Target Pair
Affinity DataIC50: 1.07E+5nMAssay Description:Inhibition of cyclooxygenase 2 in human whole blood assessed as prostaglandin H2 levelMore data for this Ligand-Target Pair
Affinity DataIC50: 1.15E+5nMAssay Description:Inhibition of COX-1 in C57BL/6 mouse brain homogenateMore data for this Ligand-Target Pair
Affinity DataIC50: 1.38E+5nMAssay Description:Inhibition of cyclooxygenase 2 in human whole blood assessed as prostaglandin H2 levelMore data for this Ligand-Target Pair
Affinity DataIC50: 1.38E+5nMAssay Description:Inhibition of cyclooxygenase 2 in human whole blood assessed as prostaglandin H2 levelMore data for this Ligand-Target Pair
Affinity DataIC50: 1.41E+5nMAssay Description:Inhibition of cyclooxygenase 2 in human whole blood assessed as prostaglandin H2 levelMore data for this Ligand-Target Pair
Affinity DataIC50: 1.41E+5nMAssay Description:Inhibition of cyclooxygenase 2 in human whole blood assessed as prostaglandin H2 levelMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Martin-Luther-Universit£T Halle-Wittenberg
Curated by ChEMBL
Martin-Luther-Universit£T Halle-Wittenberg
Curated by ChEMBL
Affinity DataIC50: 1.55E+5nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
Affinity DataIC50: 2.34E+5nMAssay Description:Inhibition of cyclooxygenase 1 in human whole blood assessed as thromboxane B2 levelMore data for this Ligand-Target Pair
Affinity DataIC50: 3.07E+5nMAssay Description:Inhibition of COX-2 in C57BL/6 mouse brain homogenateMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibition of COX-1 in C57BL/6 mouse brain homogenateMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibition of COX-2 in C57BL/6 mouse brain homogenateMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Philipps-Universit£T
Curated by ChEMBL
Philipps-Universit£T
Curated by ChEMBL
Affinity DataEC50: 26nMAssay Description:Agonist activity at TRPV1More data for this Ligand-Target Pair