Found 4 Enz. Inhib. hit(s) with Target = 'Transient receptor potential cation channel subfamily V member 1' and Ligand = 'BDBM50054471' TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Universidad Complutense
Curated by ChEMBL
Universidad Complutense
Curated by ChEMBL
Affinity DataKi: >5.00E+3nMAssay Description:Binding affinity to vanilloid VR1 receptor using [3H]resiniferatoxin ([3H]-RTX) in rat spinal cord membranesMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Universidad Complutense
Curated by ChEMBL
Universidad Complutense
Curated by ChEMBL
Affinity DataKi: >5.00E+3nMAssay Description:Binding affinity against vanilloid receptor 1 (VR1) using [3H]RTX in rat spinal cord membranesMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Universidad Complutense
Curated by ChEMBL
Universidad Complutense
Curated by ChEMBL
Affinity DataEC50: 50nMAssay Description:Agonist activity at TRPV1 in rat isolated mesenteric arteries assessed as vasorelaxation of phenylephrine-induced contractionMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Philipps-Universit£T
Curated by ChEMBL
Philipps-Universit£T
Curated by ChEMBL
Affinity DataEC50: 26nMAssay Description:Agonist activity at TRPV1More data for this Ligand-Target Pair
