TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universit�
Curated by ChEMBL
Universit�
Curated by ChEMBL
Affinity DataEC50: 39nMAssay Description:Transactivation of GAL4-fused human PPARgamma ligand binding domain expressed in HepG2 cells after 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universit�
Curated by ChEMBL
Universit�
Curated by ChEMBL
Affinity DataEC50: 1.00E+3nMAssay Description:Transactivation of GAL4-fused human PPARgamma ligand binding domain expressed in HepG2 cells after 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universit�
Curated by ChEMBL
Universit�
Curated by ChEMBL
Affinity DataEC50: 1.20E+3nMAssay Description:Transactivation of GAL4-fused human PPARgamma ligand binding domain expressed in HepG2 cells after 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universit�
Curated by ChEMBL
Universit�
Curated by ChEMBL
Affinity DataEC50: 2.30E+3nMAssay Description:Transactivation of GAL4-fused human PPARgamma ligand binding domain expressed in HepG2 cells after 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universit�
Curated by ChEMBL
Universit�
Curated by ChEMBL
Affinity DataEC50: 1.40E+3nMAssay Description:Transactivation of GAL4-fused human PPARgamma ligand binding domain expressed in HepG2 cells after 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universit�
Curated by ChEMBL
Universit�
Curated by ChEMBL
Affinity DataEC50: 1.00E+3nMAssay Description:Transactivation of GAL4-fused human PPARgamma ligand binding domain expressed in HepG2 cells after 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universit�
Curated by ChEMBL
Universit�
Curated by ChEMBL
Affinity DataEC50: 690nMAssay Description:Transactivation of GAL4-fused human PPARgamma ligand binding domain expressed in HepG2 cells after 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universit�
Curated by ChEMBL
Universit�
Curated by ChEMBL
Affinity DataEC50: 640nMAssay Description:Transactivation of GAL4-fused human PPARgamma ligand binding domain expressed in HepG2 cells after 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universit�
Curated by ChEMBL
Universit�
Curated by ChEMBL
Affinity DataEC50: 1.36E+3nMAssay Description:Transactivation of GAL4-fused human PPARgamma ligand binding domain expressed in HepG2 cells after 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universit�
Curated by ChEMBL
Universit�
Curated by ChEMBL
Affinity DataEC50: 460nMAssay Description:Transactivation of GAL4-fused human PPARgamma ligand binding domain expressed in HepG2 cells after 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universit�
Curated by ChEMBL
Universit�
Curated by ChEMBL
Affinity DataEC50: 590nMAssay Description:Transactivation of GAL4-fused human PPARgamma ligand binding domain expressed in HepG2 cells after 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universit�
Curated by ChEMBL
Universit�
Curated by ChEMBL
Affinity DataEC50: 2.54E+3nMAssay Description:Transactivation of GAL4-fused human PPARgamma ligand binding domain expressed in HepG2 cells after 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universit�
Curated by ChEMBL
Universit�
Curated by ChEMBL
Affinity DataEC50: 2.04E+3nMAssay Description:Transactivation of GAL4-fused human PPARgamma ligand binding domain expressed in HepG2 cells after 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universit�
Curated by ChEMBL
Universit�
Curated by ChEMBL
Affinity DataEC50: 3.10E+3nMAssay Description:Transactivation of GAL4-fused human PPARgamma ligand binding domain expressed in HepG2 cells after 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universit�
Curated by ChEMBL
Universit�
Curated by ChEMBL
Affinity DataEC50: 700nMAssay Description:Transactivation of GAL4-fused human PPARgamma ligand binding domain expressed in HepG2 cells after 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universit�
Curated by ChEMBL
Universit�
Curated by ChEMBL
Affinity DataEC50: 700nMAssay Description:Transactivation of GAL4-fused human PPARgamma ligand binding domain expressed in HepG2 cells after 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universit�
Curated by ChEMBL
Universit�
Curated by ChEMBL
Affinity DataEC50: 550nMAssay Description:Transactivation of GAL4-fused human PPARgamma ligand binding domain expressed in HepG2 cells after 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Universit�
Curated by ChEMBL
Universit�
Curated by ChEMBL
Affinity DataEC50: 1.56E+3nMAssay Description:Transactivation of GAL4-fused human PPARalpha ligand binding domain expressed in HepG2 cells after 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Universit�
Curated by ChEMBL
Universit�
Curated by ChEMBL
Affinity DataEC50: 280nMAssay Description:Transactivation of GAL4-fused human PPARalpha ligand binding domain expressed in HepG2 cells after 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Universit�
Curated by ChEMBL
Universit�
Curated by ChEMBL
Affinity DataEC50: 500nMAssay Description:Transactivation of GAL4-fused human PPARalpha ligand binding domain expressed in HepG2 cells after 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Universit�
Curated by ChEMBL
Universit�
Curated by ChEMBL
Affinity DataEC50: 240nMAssay Description:Transactivation of GAL4-fused human PPARalpha ligand binding domain expressed in HepG2 cells after 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Universit�
Curated by ChEMBL
Universit�
Curated by ChEMBL
Affinity DataEC50: 100nMAssay Description:Transactivation of GAL4-fused human PPARalpha ligand binding domain expressed in HepG2 cells after 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Universit�
Curated by ChEMBL
Universit�
Curated by ChEMBL
Affinity DataEC50: 12nMAssay Description:Transactivation of GAL4-fused human PPARalpha ligand binding domain expressed in HepG2 cells after 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Universit�
Curated by ChEMBL
Universit�
Curated by ChEMBL
Affinity DataEC50: 12nMAssay Description:Transactivation of GAL4-fused human PPARalpha ligand binding domain expressed in HepG2 cells after 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Universit�
Curated by ChEMBL
Universit�
Curated by ChEMBL
Affinity DataEC50: 130nMAssay Description:Transactivation of GAL4-fused human PPARalpha ligand binding domain expressed in HepG2 cells after 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Universit�
Curated by ChEMBL
Universit�
Curated by ChEMBL
Affinity DataEC50: 44nMAssay Description:Transactivation of GAL4-fused human PPARalpha ligand binding domain expressed in HepG2 cells after 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Universit�
Curated by ChEMBL
Universit�
Curated by ChEMBL
Affinity DataEC50: 22nMAssay Description:Transactivation of GAL4-fused human PPARalpha ligand binding domain expressed in HepG2 cells after 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Universit�
Curated by ChEMBL
Universit�
Curated by ChEMBL
Affinity DataEC50: 120nMAssay Description:Transactivation of GAL4-fused human PPARalpha ligand binding domain expressed in HepG2 cells after 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Universit�
Curated by ChEMBL
Universit�
Curated by ChEMBL
Affinity DataEC50: 31nMAssay Description:Transactivation of GAL4-fused human PPARalpha ligand binding domain expressed in HepG2 cells after 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Universit�
Curated by ChEMBL
Universit�
Curated by ChEMBL
Affinity DataEC50: 67nMAssay Description:Transactivation of GAL4-fused human PPARalpha ligand binding domain expressed in HepG2 cells after 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Universit�
Curated by ChEMBL
Universit�
Curated by ChEMBL
Affinity DataEC50: 220nMAssay Description:Transactivation of GAL4-fused human PPARalpha ligand binding domain expressed in HepG2 cells after 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Universit�
Curated by ChEMBL
Universit�
Curated by ChEMBL
Affinity DataEC50: 210nMAssay Description:Transactivation of GAL4-fused human PPARalpha ligand binding domain expressed in HepG2 cells after 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Universit�
Curated by ChEMBL
Universit�
Curated by ChEMBL
Affinity DataEC50: 230nMAssay Description:Transactivation of GAL4-fused human PPARalpha ligand binding domain expressed in HepG2 cells after 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Universit�
Curated by ChEMBL
Universit�
Curated by ChEMBL
Affinity DataEC50: 2.10E+3nMAssay Description:Transactivation of GAL4-fused human PPARalpha ligand binding domain expressed in HepG2 cells after 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Universit�
Curated by ChEMBL
Universit�
Curated by ChEMBL
Affinity DataEC50: 1.13E+3nMAssay Description:Transactivation of GAL4-fused human PPARalpha ligand binding domain expressed in HepG2 cells after 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Universit�
Curated by ChEMBL
Universit�
Curated by ChEMBL
Affinity DataEC50: 80nMAssay Description:Transactivation of GAL4-fused human PPARalpha ligand binding domain expressed in HepG2 cells after 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Universit�
Curated by ChEMBL
Universit�
Curated by ChEMBL
Affinity DataEC50: 990nMAssay Description:Transactivation of GAL4-fused human PPARalpha ligand binding domain expressed in HepG2 cells after 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Universit�
Curated by ChEMBL
Universit�
Curated by ChEMBL
Affinity DataEC50: 190nMAssay Description:Transactivation of GAL4-fused human PPARalpha ligand binding domain expressed in HepG2 cells after 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Universit£
Curated by ChEMBL
Universit£
Curated by ChEMBL
Affinity DataKon: 0.430M-1s-1Assay Description:Binding affinity to PPARdelta (unknown origin) assessed as kinetic dissociation constant by SPR assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Universit�
Curated by ChEMBL
Universit�
Curated by ChEMBL
Affinity DataEC50: 39nMAssay Description:Inhibition of FTase-catalyzed incorporation of [3H]- FPP radioligand into recombinant Ha-Ras by 50% at an enzyme concentration of 1 nM.More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Universit�
Curated by ChEMBL
Universit�
Curated by ChEMBL
Affinity DataEC50: 46nMAssay Description:Inhibition of FTase-catalyzed incorporation of [3H]- FPP radioligand into recombinant Ha-Ras by 50% at an enzyme concentration of 1 nM.More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Universit�
Curated by ChEMBL
Universit�
Curated by ChEMBL
Affinity DataEC50: 42nMAssay Description:Inhibition of FTase-catalyzed incorporation of [3H]- FPP radioligand into recombinant Ha-Ras by 50% at an enzyme concentration of 1 nM.More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Universit£
Curated by ChEMBL
Universit£
Curated by ChEMBL
Affinity DataEC50: 20nMAssay Description:Inhibition of FTase-catalyzed incorporation of [3H]- FPP radioligand into recombinant Ha-Ras by 50% at an enzyme concentration of 1 nM.More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Universit�
Curated by ChEMBL
Universit�
Curated by ChEMBL
Affinity DataKon: 0.0160M-1s-1Assay Description:Inhibition of FTase-catalyzed incorporation of [3H]- FPP radioligand into recombinant Ha-Ras by 50% at an enzyme concentration of 1 nM.More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Universit�
Curated by ChEMBL
Universit�
Curated by ChEMBL
Affinity DataKon: 0.0250M-1s-1Assay Description:Inhibition of FTase-catalyzed incorporation of [3H]- FPP radioligand into recombinant Ha-Ras by 50% at an enzyme concentration of 1 nM.More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Universit�
Curated by ChEMBL
Universit�
Curated by ChEMBL
Affinity DataKon: 0.360M-1s-1Assay Description:Inhibition of FTase-catalyzed incorporation of [3H]- FPP radioligand into recombinant Ha-Ras by 50% at an enzyme concentration of 1 nM.More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universit�
Curated by ChEMBL
Universit�
Curated by ChEMBL
Affinity DataKon: 0.0950M-1s-1Assay Description:Inhibition of FTase-catalyzed incorporation of [3H]- FPP radioligand into recombinant Ha-Ras by 50% at an enzyme concentration of 1 nM.More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universit�
Curated by ChEMBL
Universit�
Curated by ChEMBL
Affinity DataKon: 2.30M-1s-1Assay Description:Inhibition of FTase-catalyzed incorporation of [3H]- FPP radioligand into recombinant Ha-Ras by 50% at an enzyme concentration of 1 nM.More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universit�
Curated by ChEMBL
Universit�
Curated by ChEMBL
Affinity DataKon: 0.0990M-1s-1Assay Description:Inhibition of FTase-catalyzed incorporation of [3H]- FPP radioligand into recombinant Ha-Ras by 50% at an enzyme concentration of 1 nM.More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universit�
Curated by ChEMBL
Universit�
Curated by ChEMBL
Affinity DataEC50: 290nMAssay Description:Inhibition of FTase-catalyzed incorporation of [3H]- FPP radioligand into recombinant Ha-Ras by 50% at an enzyme concentration of 1 nM.More data for this Ligand-Target Pair