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Found 26 with Last Name = 'inui' and Initial = 'ki'
TargetSolute carrier family 22 member 1(RAT)
Kyoto University Hospital

Curated by ChEMBL
LigandPNGBDBM81945(CAS_39484 | CHEMBL105891 | CHEMBL108926 | CHEMBL27...)
Affinity DataKi:  800nMAssay Description:TP_TRANSPORTER: inhibition of TEA uptake (basolateral to cell) in OCT1-expressing MDCK cellsMore data for this Ligand-Target Pair
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TargetSolute carrier family 22 member 2(RAT)
Kyoto University Hospital

Curated by ChEMBL
LigandPNGBDBM81945(CAS_39484 | CHEMBL105891 | CHEMBL108926 | CHEMBL27...)
Affinity DataKi:  1.80E+3nMAssay Description:TP_TRANSPORTER: inhibition of TEA uptake (basolateral to cell) in OCT2-expressing MDCK cellsMore data for this Ligand-Target Pair
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TargetSolute carrier family 22 member 6(Rattus norvegicus)
Kyoto University Hospital

Curated by ChEMBL
LigandPNGBDBM25903(3-(butylamino)-4-phenoxy-5-sulfamoylbenzoic acid |...)
Affinity DataKi:  5.50E+3nMAssay Description:TP_TRANSPORTER: inhibition of PAH uptake in Xenopus laevis oocytesMore data for this Ligand-Target Pair
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TargetSolute carrier family 22 member 1(RAT)
Kyoto University Hospital

Curated by ChEMBL
LigandPNGBDBM50403559(Brumetadina | CIMETIDINE)
Affinity DataKi:  5.70E+3nMAssay Description:TP_TRANSPORTER: inhibition of TEA uptake (basolateral to cell) in OCT1-expressing MDCK cellsMore data for this Ligand-Target Pair
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TargetSolute carrier family 22 member 2(RAT)
Kyoto University Hospital

Curated by ChEMBL
LigandPNGBDBM50403559(Brumetadina | CIMETIDINE)
Affinity DataKi:  9.40E+3nMAssay Description:TP_TRANSPORTER: inhibition of TEA uptake (basolateral to cell) in OCT2-expressing MDCK cellsMore data for this Ligand-Target Pair
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TargetSolute carrier family 22 member 6(Rattus norvegicus)
Kyoto University Hospital

Curated by ChEMBL
LigandPNGBDBM25902(4-chloro-2-[(furan-2-ylmethyl)amino]-5-sulfamoylbe...)
Affinity DataKi:  9.50E+3nMAssay Description:TP_TRANSPORTER: inhibition of PAH uptake in Xenopus laevis oocytesMore data for this Ligand-Target Pair
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TargetSolute carrier family 22 member 1(RAT)
Kyoto University Hospital

Curated by ChEMBL
LigandPNGBDBM50017681((1S,2R,4S,5R)-2-[(S)-Hydroxy-(6-methoxy-quinolin-4...)
Affinity DataKi:  1.46E+4nMAssay Description:TP_TRANSPORTER: inhibition of TEA uptake (basolateral to cell) in OCT1-expressing MDCK cellsMore data for this Ligand-Target Pair
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TargetSolute carrier family 22 member 2(RAT)
Kyoto University Hospital

Curated by ChEMBL
LigandPNGBDBM50017681((1S,2R,4S,5R)-2-[(S)-Hydroxy-(6-methoxy-quinolin-4...)
Affinity DataKi:  1.91E+4nMAssay Description:TP_TRANSPORTER: inhibition of TEA uptake (basolateral to cell) in OCT2-expressing MDCK cellsMore data for this Ligand-Target Pair
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TargetSolute carrier family 22 member 1(RAT)
Kyoto University Hospital

Curated by ChEMBL
LigandPNGBDBM50149890(CHEMBL9324 | tetraethylammonium)
Affinity DataKi:  4.66E+4nMAssay Description:TP_TRANSPORTER: inhibition of TEA uptake (basolateral to cell) in OCT1-expressing MDCK cellsMore data for this Ligand-Target Pair
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TargetSolute carrier family 22 member 2(RAT)
Kyoto University Hospital

Curated by ChEMBL
LigandPNGBDBM82070(CAS_29790-52-1 | NICOTINE-L (BASE) | Nicotine-D sa...)
Affinity DataKi:  5.05E+4nMAssay Description:TP_TRANSPORTER: inhibition of TEA uptake (basolateral to cell) in OCT2-expressing MDCK cellsMore data for this Ligand-Target Pair
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TargetSolute carrier family 22 member 2(RAT)
Kyoto University Hospital

Curated by ChEMBL
LigandPNGBDBM50149890(CHEMBL9324 | tetraethylammonium)
Affinity DataKi:  5.22E+4nMAssay Description:TP_TRANSPORTER: inhibition of TEA uptake (apical to cell) in OCT2-expressing MDCK cellsMore data for this Ligand-Target Pair
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TargetSolute carrier family 22 member 1(RAT)
Kyoto University Hospital

Curated by ChEMBL
LigandPNGBDBM82070(CAS_29790-52-1 | NICOTINE-L (BASE) | Nicotine-D sa...)
Affinity DataKi:  6.43E+4nMAssay Description:TP_TRANSPORTER: inhibition of TEA uptake (basolateral to cell) in OCT1-expressing MDCK cellsMore data for this Ligand-Target Pair
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TargetSolute carrier family 22 member 6(Rattus norvegicus)
Kyoto University Hospital

Curated by ChEMBL
LigandPNGBDBM13076(6-chloro-1,1-dioxo-3,4-dihydro-2H-1,2,4-benzothiad...)
Affinity DataKi:  1.50E+5nMAssay Description:TP_TRANSPORTER: inhibition of PAH uptake in Xenopus laevis oocytesMore data for this Ligand-Target Pair
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TargetSolute carrier family 15 member 2(Rattus norvegicus)
Kyoto University Hospital

Curated by ChEMBL
LigandPNGBDBM50162073((S)-2-((2-amino-6-oxo-3H-purin-9(6H)-yl)methoxy)et...)
Affinity DataKi:  2.20E+5nMAssay Description:TP_TRANSPORTER: inhibition of Gly-Sar uptake in PEPT2-expressing LLC-PK1 cellsMore data for this Ligand-Target Pair
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TargetSolute carrier family 15 member 2(Rattus norvegicus)
Kyoto University Hospital

Curated by ChEMBL
LigandPNGBDBM50162073((S)-2-((2-amino-6-oxo-3H-purin-9(6H)-yl)methoxy)et...)
Affinity DataKi:  2.20E+5nMAssay Description:TP_TRANSPORTER: inhibition of Gly-Sar uptake in PEPT2-expressing LLC-PK1 cellsMore data for this Ligand-Target Pair
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TargetSolute carrier family 22 member 2(RAT)
Kyoto University Hospital

Curated by ChEMBL
LigandPNGBDBM50420177(NICOTINYL METHYLAMIDE)
Affinity DataKi:  4.03E+5nMAssay Description:TP_TRANSPORTER: inhibition of TEA uptake (basolateral to cell) in OCT2-expressing MDCK cellsMore data for this Ligand-Target Pair
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TargetSolute carrier family 22 member 1(RAT)
Kyoto University Hospital

Curated by ChEMBL
LigandPNGBDBM50420177(NICOTINYL METHYLAMIDE)
Affinity DataKi:  6.69E+5nMAssay Description:TP_TRANSPORTER: inhibition of TEA uptake (basolateral to cell) in OCT1-expressing MDCK cellsMore data for this Ligand-Target Pair
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TargetSolute carrier family 22 member 2(RAT)
Kyoto University Hospital

Curated by ChEMBL
LigandPNGBDBM50420178(GUANIDINE)
Affinity DataKi:  7.14E+5nMAssay Description:TP_TRANSPORTER: inhibition of TEA uptake (basolateral to cell) in OCT2-expressing MDCK cellsMore data for this Ligand-Target Pair
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TargetSolute carrier family 22 member 1(RAT)
Kyoto University Hospital

Curated by ChEMBL
LigandPNGBDBM50420178(GUANIDINE)
Affinity DataKi:  7.24E+5nMAssay Description:TP_TRANSPORTER: inhibition of TEA uptake (basolateral to cell) in OCT1-expressing MDCK cellsMore data for this Ligand-Target Pair
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TargetSolute carrier family 15 member 2(Rattus norvegicus)
Kyoto University Hospital

Curated by ChEMBL
LigandPNGBDBM50485607(CHEMBL1209949 | L-Valine Methyl Ester)
Affinity DataKi:  8.30E+5nMAssay Description:TP_TRANSPORTER: inhibition of Gly-Sar uptake in PEPT2-expressing LLC-PK1 cellsMore data for this Ligand-Target Pair
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TargetSolute carrier organic anion transporter family member 1A3(Rattus norvegicus)
Kyoto University Hospital

Curated by ChEMBL
LigandPNGBDBM17638(2-{1-[(4-chlorophenyl)carbonyl]-5-methoxy-2-methyl...)
Affinity DataKi:  1.00E+6nMAssay Description:TP_TRANSPORTER: inhibition of MTX uptake in OAT-K1-expressing LLC-PK1 cellsMore data for this Ligand-Target Pair
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TargetSolute carrier family 22 member 6(Rattus norvegicus)
Kyoto University Hospital

Curated by ChEMBL
LigandPNGBDBM10880(AZA | AZA2 | AZM acetazolamide | Acerazolamide, AA...)
Affinity DataKi:  1.10E+6nMAssay Description:TP_TRANSPORTER: inhibition of PAH uptake in Xenopus laevis oocytesMore data for this Ligand-Target Pair
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TargetSolute carrier organic anion transporter family member 1A3(Rattus norvegicus)
Kyoto University Hospital

Curated by ChEMBL
LigandPNGBDBM50022271(2-(3-Benzoylphenyl)propionic acid | 2-(3-benzoylph...)
Affinity DataKi:  1.90E+6nMAssay Description:TP_TRANSPORTER: inhibition of MTX uptake in OAT-K1-expressing LLC-PK1 cellsMore data for this Ligand-Target Pair
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TargetSolute carrier family 15 member 1(Rattus norvegicus)
Kyoto University Hospital

Curated by ChEMBL
LigandPNGBDBM50162073((S)-2-((2-amino-6-oxo-3H-purin-9(6H)-yl)methoxy)et...)
Affinity DataKi:  2.50E+6nMAssay Description:TP_TRANSPORTER: inhibition of Gly-Sar uptake in PEPT1-expressing LLC-PK1 cellsMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSolute carrier family 15 member 1(Rattus norvegicus)
Kyoto University Hospital

Curated by ChEMBL
LigandPNGBDBM50162073((S)-2-((2-amino-6-oxo-3H-purin-9(6H)-yl)methoxy)et...)
Affinity DataKi:  2.70E+6nMAssay Description:TP_TRANSPORTER: inhibition of Gly-Sar uptake in PEPT1-expressing LLC-PK1 cellsMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSolute carrier family 15 member 1(Rattus norvegicus)
Kyoto University Hospital

Curated by ChEMBL
LigandPNGBDBM50485607(CHEMBL1209949 | L-Valine Methyl Ester)
Affinity DataKi:  3.60E+6nMAssay Description:TP_TRANSPORTER: inhibition of Gly-Sar uptake in PEPT1-expressing LLC-PK1 cellsMore data for this Ligand-Target Pair
In DepthDetails PubMed