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Found 4 Enz. Inhib. hit(s) with Target = 'Solute carrier family 22 member 2' and Ligand = 'BDBM50420177'
TargetSolute carrier family 22 member 2(Homo sapiens (Human))
Anatomisches Institut Der Bayerischen Julius-Maximilians-Universit£T

Curated by ChEMBL
LigandPNGBDBM50420177(NICOTINYL METHYLAMIDE)
Affinity DataKi:  2.66E+5nMAssay Description:TP_TRANSPORTER: inhibition of TEA uptake in Xenopus laevis oocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 22 member 2(RAT)
Kyoto University Hospital

Curated by ChEMBL
LigandPNGBDBM50420177(NICOTINYL METHYLAMIDE)
Affinity DataKi:  4.03E+5nMAssay Description:TP_TRANSPORTER: inhibition of TEA uptake (basolateral to cell) in OCT2-expressing MDCK cellsMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSolute carrier family 22 member 2(RAT)
Kyoto University Hospital

Curated by ChEMBL
LigandPNGBDBM50420177(NICOTINYL METHYLAMIDE)
Affinity DataIC50:  1.56E+6nMAssay Description:TP_TRANSPORTER: inhibition of TEA uptake (TEA: 100 uM) in Xenopus laevis oocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 22 member 2(Mus musculus)
Kyushu University

Curated by ChEMBL
LigandPNGBDBM50420177(NICOTINYL METHYLAMIDE)
Affinity DataIC50:  1.37E+7nMAssay Description:TP_TRANSPORTER: inhibition of MPP+ uptake (MPP+: 1 uM) in Xenopus laevis oocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed