Affinity DataIC50: 0.260nMAssay Description:Inhibitory concentration towards melanocortin MC4 receptor by displacing radioligand [125I]-hAGRP(82-132)More data for this Ligand-Target Pair
Affinity DataIC50: 0.960nMAssay Description:Inhibitory concentration towards melanocortin MC4 receptor by displacing radioligand [125I]NDP-MSHMore data for this Ligand-Target Pair
Affinity DataIC50: 1.46nMAssay Description:Inhibitory concentration towards melanocortin MC4 receptor by displacing radioligand [125I]NDP-MSHMore data for this Ligand-Target Pair
Affinity DataIC50: 4.22nMAssay Description:Inhibitory concentration towards melanocortin MC4 receptor by displacing radioligand [125I]-NDP-MSH; ND = not determinedMore data for this Ligand-Target Pair
Affinity DataIC50: 4.45nMAssay Description:Inhibitory concentration towards melanocortin MC4 receptor by displacing radioligand [125I]-hAGRP(82-132)More data for this Ligand-Target Pair
Affinity DataIC50: 4.74nMAssay Description:Inhibitory concentration towards melanocortin MC4 receptor by displacing radioligand [125I]-hAGRP(82-132)More data for this Ligand-Target Pair
Affinity DataIC50: 5.48nMAssay Description:Inhibitory concentration towards melanocortin MC4 receptor by displacing radioligand [125I]-hAGRP(82-132)More data for this Ligand-Target Pair
Affinity DataIC50: 29.8nMAssay Description:Inhibitory concentration towards melanocortin MC4 receptor by displacing radioligand [125I]NDP-MSHMore data for this Ligand-Target Pair
Affinity DataIC50: 290nMAssay Description:Inhibitory concentration towards melanocortin MC4 receptor by displacing radioligand [125I]-hAGRP(82-132)More data for this Ligand-Target Pair
Affinity DataIC50: 540nMAssay Description:Inhibitory concentration towards melanocortin MC4 receptor by displacing radioligand [125I]NDP-MSHMore data for this Ligand-Target Pair
Affinity DataIC50: 3.10E+3nMAssay Description:Inhibitory concentration towards melanocortin MC4 receptor by displacing radioligand [125I]-hAGRP(82-132)More data for this Ligand-Target Pair
Affinity DataIC50: 3.20E+3nMAssay Description:Inhibitory concentration towards melanocortin MC4 receptor by displacing radioligand [125I]-hAGRP(82-132)More data for this Ligand-Target Pair
Affinity DataIC50: 4.10E+3nMAssay Description:Inhibitory concentration towards melanocortin MC4 receptor by displacing radioligand [125I]-hAGRP(82-132)More data for this Ligand-Target Pair
Affinity DataIC50: 4.80E+3nMAssay Description:Inhibitory concentration towards melanocortin MC4 receptor by displacing radioligand [125I]NDP-MSHMore data for this Ligand-Target Pair
Affinity DataIC50: 6.80E+3nMAssay Description:Inhibitory concentration towards melanocortin MC4 receptor by displacing radioligand [125I]NDP-MSHMore data for this Ligand-Target Pair
Affinity DataIC50: 7.30E+3nMAssay Description:Inhibitory concentration towards melanocortin MC4 receptor by displacing radioligand [125I]-hAGRP(82-132)More data for this Ligand-Target Pair
Affinity DataIC50: 9.20E+3nMAssay Description:Inhibitory concentration towards melanocortin MC4 receptor by displacing radioligand [125I]NDP-MSHMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibitory concentration towards melanocortin MC4 receptor by displacing radioligand [125I]-hAGRP(82-132)More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibitory concentration towards melanocortin MC4 receptor by displacing radioligand [125I]NDP-MSHMore data for this Ligand-Target Pair
Affinity DataIC50: 1.03E+4nMAssay Description:Inhibitory concentration towards melanocortin MC4 receptor by displacing radioligand [125I]NDP-MSHMore data for this Ligand-Target Pair
Affinity DataEC50: 6.20nMAssay Description:Displacement of MT2 from mouse MC3R expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 8.30E+3nMAssay Description:Agonist activity at mouse MC4R expressed in HEK293 cells by beta-galactosidase assayMore data for this Ligand-Target Pair
Affinity DataEC50: 6.24E+3nMAssay Description:Agonist activity at mouse MC4R expressed in HEK293 cells by beta-galactosidase assayMore data for this Ligand-Target Pair
Affinity DataEC50: 1.75E+3nMAssay Description:Agonist activity at mouse MC1R expressed in HEK293 cells by beta-galactosidase assayMore data for this Ligand-Target Pair
Affinity DataEC50: 6.10nMAssay Description:Displacement of MT2 from mouse MC3R expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 93nMAssay Description:Agonist activity at mouse MC1R expressed in HEK293 cells by beta-galactosidase assayMore data for this Ligand-Target Pair
Affinity DataEC50: 3.77E+4nMAssay Description:Agonist activity at mouse MC4R expressed in HEK293 cells by beta-galactosidase assayMore data for this Ligand-Target Pair
Affinity DataEC50: 1.14E+4nMAssay Description:Agonist activity at mouse MC5R expressed in HEK293 cells by beta-galactosidase assayMore data for this Ligand-Target Pair
Affinity DataEC50: 1.41E+3nMAssay Description:Agonist activity at mouse MC5R expressed in HEK293 cells by beta-galactosidase assayMore data for this Ligand-Target Pair
Affinity DataEC50: >100nMAssay Description:Agonist activity at mouse MC5R expressed in HEK293 cells by beta-galactosidase assayMore data for this Ligand-Target Pair
Affinity DataEC50: 120nMAssay Description:Agonist activity at mouse MC1R expressed in HEK293 cells by beta-galactosidase assayMore data for this Ligand-Target Pair
Affinity DataEC50: 6.90nMAssay Description:Displacement of MT2 from mouse MC4R expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 5.27E+3nMAssay Description:Agonist activity at mouse MC1R expressed in HEK293 cells by beta-galactosidase assayMore data for this Ligand-Target Pair
Affinity DataEC50: 1.98E+4nMAssay Description:Agonist activity at mouse MC5R expressed in HEK293 cells by beta-galactosidase assayMore data for this Ligand-Target Pair
Affinity DataEC50: 93nMAssay Description:Agonist activity at mouse MC1R expressed in HEK293 cells by beta-galactosidase assayMore data for this Ligand-Target Pair
Affinity DataEC50: 8.33E+3nMAssay Description:Agonist activity at mouse MC4R expressed in HEK293 cells by beta-galactosidase assayMore data for this Ligand-Target Pair
Affinity DataEC50: 4.60E+3nMAssay Description:Agonist activity at mouse MC5R expressed in HEK293 cells by beta-galactosidase assayMore data for this Ligand-Target Pair
Affinity DataEC50: 2.26E+4nMAssay Description:Agonist activity at mouse MC3R expressed in HEK293 cells by beta-galactosidase assayMore data for this Ligand-Target Pair
Affinity DataEC50: 6.33E+3nMAssay Description:Agonist activity at mouse MC1R expressed in HEK293 cells by beta-galactosidase assayMore data for this Ligand-Target Pair
Affinity DataEC50: 3.70E+3nMAssay Description:Agonist activity at mouse MC4R expressed in HEK293 cells by beta-galactosidase assayMore data for this Ligand-Target Pair
Affinity DataEC50: 6.33E+4nMAssay Description:Agonist activity at mouse MC3R expressed in HEK293 cells by beta-galactosidase assayMore data for this Ligand-Target Pair
Affinity DataEC50: 1.83E+4nMAssay Description:Agonist activity at mouse MC5R expressed in HEK293 cells by beta-galactosidase assayMore data for this Ligand-Target Pair
Affinity DataEC50: 2.22E+3nMAssay Description:Agonist activity at mouse MC5R expressed in HEK293 cells by beta-galactosidase assayMore data for this Ligand-Target Pair
Affinity DataEC50: 6.60nMAssay Description:Displacement of MT2 from mouse MC4R expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 5.27E+3nMAssay Description:Agonist activity at mouse MC1R expressed in HEK293 cells by beta-galactosidase assayMore data for this Ligand-Target Pair
Affinity DataEC50: 1.98E+4nMAssay Description:Agonist activity at mouse MC5R expressed in HEK293 cells by beta-galactosidase assayMore data for this Ligand-Target Pair
Affinity DataEC50: 8.33E+3nMAssay Description:Agonist activity at mouse MC4R expressed in HEK293 cells by beta-galactosidase assayMore data for this Ligand-Target Pair
Affinity DataEC50: 1.37E+4nMAssay Description:Agonist activity at mouse MC3R expressed in HEK293 cells by beta-galactosidase assayMore data for this Ligand-Target Pair
Affinity DataEC50: 64nMAssay Description:Agonist activity at mouse MC1R expressed in HEK293 cells by beta-galactosidase assayMore data for this Ligand-Target Pair
Affinity DataEC50: 5.51E+3nMAssay Description:Agonist activity at mouse MC3R expressed in HEK293 cells by beta-galactosidase assayMore data for this Ligand-Target Pair