Affinity DataKi: 0.390nMAssay Description:Inhibition of binding to human D1 receptor expressed in HEK 293 cells by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 1.5nMAssay Description:Inhibition of binding to human D5 receptor expressed in HEK 293 cells by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 1.69nMAssay Description:Inhibition of binding to human D5 receptor expressed in HEK 293 cells by functional calcium assayMore data for this Ligand-Target Pair
Affinity DataKi: 2.32nMAssay Description:Inhibition of binding to human D5 receptor expressed in HEK 293 cells by functional calcium assayMore data for this Ligand-Target Pair
Affinity DataKi: 3.09nMAssay Description:Inhibition of binding to human D5 receptor expressed in HEK 293 cells by functional calcium assayMore data for this Ligand-Target Pair
Affinity DataKi: 4.5nMAssay Description:Inhibition of binding to human D1 receptor expressed in HEK 293 cells by radioligand binding assayMore data for this Ligand-Target Pair
TargetHistone deacetylase 3/Nuclear receptor corepressor 2 (HDAC3/NCoR2)(Homo sapiens (Human))
Heinrich-Heine-Universit£T D£Sseldorf
Curated by ChEMBL
Heinrich-Heine-Universit£T D£Sseldorf
Curated by ChEMBL
Affinity DataKi: 5nMAssay Description:Inhibition of recombinant HDAC3 (unknown origin)/NCOR2 (unknown origin) using acetyl-Lys(Ac)-AMC as substrate preincubated for up to 3 hrs followed b...More data for this Ligand-Target Pair
Affinity DataKi: 6.93nMAssay Description:Inhibition of binding to human D1 receptor expressed in HEK 293 cells by functional calcium assayMore data for this Ligand-Target Pair
TargetHistone deacetylase 9(Homo sapiens (Human))
Heinrich-Heine-Universit£T D£Sseldorf
Curated by ChEMBL
Heinrich-Heine-Universit£T D£Sseldorf
Curated by ChEMBL
Affinity DataKi: 8nMAssay Description:Inhibition of HDAC9 (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 8.47nMAssay Description:Inhibition of binding to human D2L receptor expressed in HEK 293 cells by functional calcium assayMore data for this Ligand-Target Pair
TargetHistone deacetylase 6(Homo sapiens (Human))
Heinrich-Heine-University D£Sseldorf
Curated by ChEMBL
Heinrich-Heine-University D£Sseldorf
Curated by ChEMBL
Affinity DataKi: 10nMAssay Description:Inhibition of N-terminal GST-tagged recombinant human HDAC6 (1 to 1215 residues) expressed in Baculovirus infected insect cells using Boc-Lys(Ac)-AMC...More data for this Ligand-Target Pair
Affinity DataKi: 10.7nMAssay Description:Inhibition of binding to human D1 receptor expressed in HEK 293 cells by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 11.2nMAssay Description:Inhibition of binding to human D5 receptor expressed in HEK 293 cells by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 11.3nMAssay Description:Inhibition of binding to human D4 receptor expressed in HEK 293 cells by radioligand binding assayMore data for this Ligand-Target Pair
TargetHistone deacetylase 2(Homo sapiens (Human))
Heinrich-Heine-University D£Sseldorf
Curated by ChEMBL
Heinrich-Heine-University D£Sseldorf
Curated by ChEMBL
Affinity DataKi: 13nMAssay Description:Inhibition of C-terminal GST-tagged recombinant human HDAC2 (1 to 488 residues) expressed in Baculovirus infected insect cells using Boc-Lys(Ac)-AMC ...More data for this Ligand-Target Pair
Affinity DataKi: 14.7nMAssay Description:Inhibition of binding to human D5 receptor expressed in HEK 293 cells by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 16.4nMAssay Description:Inhibition of binding to human D1 receptor expressed in HEK 293 cells by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 17.5nMAssay Description:Inhibition of binding to human D2L receptor expressed in HEK 293 cells by radioligand binding assayMore data for this Ligand-Target Pair
TargetHistone deacetylase 6(Homo sapiens (Human))
Heinrich-Heine-University D£Sseldorf
Curated by ChEMBL
Heinrich-Heine-University D£Sseldorf
Curated by ChEMBL
Affinity DataKi: 20nMAssay Description:Inhibition of recombinant human HDAC6More data for this Ligand-Target Pair
Affinity DataKi: 20.7nMAssay Description:Inhibition of binding to human D1 receptor expressed in HEK 293 cells by functional calcium assayMore data for this Ligand-Target Pair
Affinity DataKi: 22.3nMAssay Description:Inhibition of binding to human D5 receptor expressed in HEK 293 cells by functional calcium assayMore data for this Ligand-Target Pair
TargetHistone deacetylase 6(Homo sapiens (Human))
Heinrich-Heine-University D£Sseldorf
Curated by ChEMBL
Heinrich-Heine-University D£Sseldorf
Curated by ChEMBL
Affinity DataKi: 30nMAssay Description:Inhibition of N-terminal GST-tagged recombinant human HDAC6 (1 to 1215 residues) expressed in Baculovirus infected insect cells using Boc-Lys(Ac)-AMC...More data for this Ligand-Target Pair
TargetHistone deacetylase 6(Homo sapiens (Human))
Heinrich-Heine-University D£Sseldorf
Curated by ChEMBL
Heinrich-Heine-University D£Sseldorf
Curated by ChEMBL
Affinity DataKi: 30nMAssay Description:Inhibition of N-terminal GST-tagged recombinant human HDAC6 (1 to 1215 residues) expressed in Baculovirus infected insect cells using Boc-Lys(Ac)-AMC...More data for this Ligand-Target Pair
TargetHistone deacetylase 6(Homo sapiens (Human))
Heinrich-Heine-University D£Sseldorf
Curated by ChEMBL
Heinrich-Heine-University D£Sseldorf
Curated by ChEMBL
Affinity DataKi: 30nMAssay Description:Inhibition of recombinant human HDAC6More data for this Ligand-Target Pair
TargetHistone deacetylase 1(Homo sapiens (Human))
Heinrich-Heine-Universit£T D£Sseldorf
Curated by ChEMBL
Heinrich-Heine-Universit£T D£Sseldorf
Curated by ChEMBL
Affinity DataKi: 32nMAssay Description:Inhibition of recombinant HDAC1 (unknown origin) using acetyl-Lys(Ac)-AMC as substrate preincubated for up to 3 hrs followed by substrate addition an...More data for this Ligand-Target Pair
Affinity DataKi: 33.5nMAssay Description:Inhibition of binding to human D2L receptor expressed in HEK 293 cells by functional calcium assayMore data for this Ligand-Target Pair
Affinity DataKi: 33.7nMAssay Description:Inhibition of binding to human D5 receptor expressed in HEK 293 cells by functional calcium assayMore data for this Ligand-Target Pair
TargetHistone deacetylase 7(Homo sapiens (Human))
Heinrich-Heine-Universit£T D£Sseldorf
Curated by ChEMBL
Heinrich-Heine-Universit£T D£Sseldorf
Curated by ChEMBL
Affinity DataKi: 39nMAssay Description:Inhibition of HDAC7 (unknown origin)More data for this Ligand-Target Pair
TargetHistone deacetylase 6(Homo sapiens (Human))
Heinrich-Heine-University D£Sseldorf
Curated by ChEMBL
Heinrich-Heine-University D£Sseldorf
Curated by ChEMBL
Affinity DataKi: 40nMAssay Description:Inhibition of N-terminal GST-tagged recombinant human HDAC6 (1 to 1215 residues) expressed in Baculovirus infected insect cells using Boc-Lys(Ac)-AMC...More data for this Ligand-Target Pair
Affinity DataKi: 40.4nMAssay Description:Inhibition of binding to human D1 receptor expressed in HEK 293 cells by functional calcium assayMore data for this Ligand-Target Pair
Affinity DataKi: 47.5nMAssay Description:Inhibition of binding to human D3 receptor expressed in HEK 293 cells by radioligand binding assayMore data for this Ligand-Target Pair
TargetHistone deacetylase 6(Homo sapiens (Human))
Heinrich-Heine-University D£Sseldorf
Curated by ChEMBL
Heinrich-Heine-University D£Sseldorf
Curated by ChEMBL
Affinity DataKi: 50nMAssay Description:Inhibition of recombinant human HDAC6More data for this Ligand-Target Pair
Affinity DataKi: 52.5nMAssay Description:Inhibition of binding to human D3 receptor expressed in HEK 293 cells by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 56.5nMAssay Description:Inhibition of binding to human D2L receptor expressed in HEK 293 cells by radioligand binding assayMore data for this Ligand-Target Pair
TargetHistone deacetylase 2(Homo sapiens (Human))
Heinrich-Heine-University D£Sseldorf
Curated by ChEMBL
Heinrich-Heine-University D£Sseldorf
Curated by ChEMBL
Affinity DataKi: 60nMAssay Description:Inhibition of recombinant human HDAC2More data for this Ligand-Target Pair
TargetHistone deacetylase 6(Homo sapiens (Human))
Heinrich-Heine-University D£Sseldorf
Curated by ChEMBL
Heinrich-Heine-University D£Sseldorf
Curated by ChEMBL
Affinity DataKi: 60nMAssay Description:Inhibition of recombinant human HDAC6More data for this Ligand-Target Pair
Affinity DataKi: 61nMAssay Description:Inhibition of binding to human D1 receptor expressed in HEK 293 cells by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 65.7nMAssay Description:Inhibition of binding to human D2L receptor expressed in HEK 293 cells by functional calcium assayMore data for this Ligand-Target Pair
TargetHistone deacetylase 2(Homo sapiens (Human))
Heinrich-Heine-University D£Sseldorf
Curated by ChEMBL
Heinrich-Heine-University D£Sseldorf
Curated by ChEMBL
Affinity DataKi: 70nMAssay Description:Inhibition of C-terminal GST-tagged recombinant human HDAC2 (1 to 488 residues) expressed in Baculovirus infected insect cells using Boc-Lys(Ac)-AMC ...More data for this Ligand-Target Pair
TargetHistone deacetylase 4(Homo sapiens (Human))
Heinrich-Heine-Universit£T D£Sseldorf
Curated by ChEMBL
Heinrich-Heine-Universit£T D£Sseldorf
Curated by ChEMBL
Affinity DataKi: 75nMAssay Description:Inhibition of HDAC4 (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 79.1nMAssay Description:Inhibition of binding to human D5 receptor expressed in HEK 293 cells by radioligand binding assayMore data for this Ligand-Target Pair
TargetHistone deacetylase 2(Homo sapiens (Human))
Heinrich-Heine-University D£Sseldorf
Curated by ChEMBL
Heinrich-Heine-University D£Sseldorf
Curated by ChEMBL
Affinity DataKi: 80nMAssay Description:Inhibition of recombinant human HDAC2More data for this Ligand-Target Pair
Affinity DataKi: 82.6nMAssay Description:Inhibition of binding to human D2L receptor expressed in HEK 293 cells by functional calcium assayMore data for this Ligand-Target Pair
TargetHistone deacetylase 2(Homo sapiens (Human))
Heinrich-Heine-University D£Sseldorf
Curated by ChEMBL
Heinrich-Heine-University D£Sseldorf
Curated by ChEMBL
Affinity DataKi: 90nMAssay Description:Inhibition of recombinant human HDAC2More data for this Ligand-Target Pair
TargetHistone deacetylase 2(Homo sapiens (Human))
Heinrich-Heine-University D£Sseldorf
Curated by ChEMBL
Heinrich-Heine-University D£Sseldorf
Curated by ChEMBL
Affinity DataKi: 90nMAssay Description:Inhibition of recombinant human HDAC2More data for this Ligand-Target Pair
Affinity DataKi: 92nMAssay Description:Inhibition of binding to human D2L receptor expressed in HEK 293 cells by functional calcium assayMore data for this Ligand-Target Pair
TargetHistone deacetylase 6(Homo sapiens (Human))
Heinrich-Heine-University D£Sseldorf
Curated by ChEMBL
Heinrich-Heine-University D£Sseldorf
Curated by ChEMBL
Affinity DataKi: 100nMAssay Description:Inhibition of N-terminal GST-tagged recombinant human HDAC6 (1 to 1215 residues) expressed in Baculovirus infected insect cells using Boc-Lys(Ac)-AMC...More data for this Ligand-Target Pair
TargetHistone deacetylase 6(Homo sapiens (Human))
Heinrich-Heine-University D£Sseldorf
Curated by ChEMBL
Heinrich-Heine-University D£Sseldorf
Curated by ChEMBL
Affinity DataKi: 100nMAssay Description:Inhibition of recombinant human HDAC6More data for this Ligand-Target Pair
TargetHistone deacetylase 2(Homo sapiens (Human))
Heinrich-Heine-University D£Sseldorf
Curated by ChEMBL
Heinrich-Heine-University D£Sseldorf
Curated by ChEMBL
Affinity DataKi: 100nMAssay Description:Inhibition of C-terminal GST-tagged recombinant human HDAC2 (1 to 488 residues) expressed in Baculovirus infected insect cells using Boc-Lys(Ac)-AMC ...More data for this Ligand-Target Pair
Affinity DataKi: 112nMAssay Description:Inhibition of binding to human D5 receptor expressed in HEK 293 cells by functional calcium assayMore data for this Ligand-Target Pair