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Found 55 with Last Name = 'kettmann' and Initial = 'v'
TargetEndothelin-1 receptor(RAT)
University Of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50061096((2R,3R,4S)-4-Benzo[1,3]dioxol-5-yl-1-{2-[(butane-1...)
Affinity DataIC50:  0.0400nMAssay Description:Ability to displace [125I]-ET-1 from the rat endothelin A receptor expressed in rat aorta smooth muscle cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(RAT)
University Of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50146613(5-{5-[(Z)-3-Benzo[1,3]dioxol-5-yl-3-carboxy-2-(4-m...)
Affinity DataIC50:  0.0500nMAssay Description:Ability to displace [125I]-ET-1 from the rat endothelin A receptor expressed in rat aorta smooth muscle cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(RAT)
University Of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50146606((Z)-2-Benzo[1,3]dioxol-5-yl-4-(4-methoxy-phenyl)-4...)
Affinity DataIC50:  0.120nMAssay Description:Ability to displace [125I]-ET-1 from the rat endothelin A receptor expressed in rat aorta smooth muscle cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(RAT)
University Of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50112678((R)-2-Benzo[1,3]dioxol-5-yl-6-isopropoxy-4-(4-meth...)
Affinity DataIC50:  0.190nMAssay Description:Ability to displace [125I]-ET-1 from the rat endothelin A receptor expressed in rat aorta smooth muscle cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(RAT)
University Of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50146619((2S,3R,4S)-4-Benzo[1,3]dioxol-5-yl-1-dibutylcarbam...)
Affinity DataIC50:  0.290nMAssay Description:Ability to displace [125I]-ET-1 from the rat endothelin A receptor expressed in rat aorta smooth muscle cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(RAT)
University Of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50051007((2R,3R,4S)-4-Benzo[1,3]dioxol-5-yl-1-dibutylcarbam...)
Affinity DataIC50:  0.310nMAssay Description:Ability to displace [125I]-ET-1 from the rat endothelin A receptor expressed in rat aorta smooth muscle cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(RAT)
University Of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50112748((R)-2-Benzo[1,3]dioxol-5-yl-4-butyl-6-isopropoxy-2...)
Affinity DataIC50:  0.420nMAssay Description:Ability to displace [125I]-ET-1 from the rat endothelin A receptor expressed in rat aorta smooth muscle cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(RAT)
University Of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50146610(CHEMBL368558 | [(2R,3R,4S)-4-Benzo[1,3]dioxol-5-yl...)
Affinity DataIC50:  0.5nMAssay Description:Ability to displace [125I]-ET-1 from the rat endothelin A receptor expressed in rat aorta smooth muscle cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(RAT)
University Of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50056071((2R,3R,4S)-4-Benzofuran-5-yl-1-dibutylcarbamoylmet...)
Affinity DataIC50:  0.5nMAssay Description:Ability to displace [125I]-ET-1 from the rat endothelin A receptor expressed in rat aorta smooth muscle cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(RAT)
University Of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50146622((Z)-2-(7-Methoxy-benzo[1,3]dioxol-5-yl)-4-(4-metho...)
Affinity DataIC50:  0.5nMAssay Description:Ability to displace [125I]-ET-1 from the rat endothelin A receptor expressed in rat aorta smooth muscle cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(RAT)
University Of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50080622((2R,3R,4S)-4-Benzo[1,3]dioxol-5-yl-2-(4-methoxy-ph...)
Affinity DataIC50:  0.700nMAssay Description:Ability to displace [125I]-ET-1 from the rat endothelin A receptor expressed in rat aorta smooth muscle cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(RAT)
University Of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50066408((2S,3R,4S)-4-Benzo[1,3]dioxol-5-yl-1-dibutylcarbam...)
Affinity DataIC50:  0.780nMAssay Description:Ability to displace [125I]-ET-1 from the rat endothelin A receptor expressed in rat aorta smooth muscle cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(RAT)
University Of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50112661((2S,3S,4R)-2-Benzo[1,3]dioxol-5-yl-6-isopropoxy-4-...)
Affinity DataIC50:  1.30nMAssay Description:Ability to displace [125I]-ET-1 from the rat endothelin A receptor expressed in rat aorta smooth muscle cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(RAT)
University Of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50146605((Z)-2-Benzo[1,3]dioxol-5-yl-3-(4-methoxy-benzyl)-4...)
Affinity DataIC50:  1.80nMAssay Description:Ability to displace [125I]-ET-1 from the rat endothelin A receptor expressed in rat aorta smooth muscle cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(RAT)
University Of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50146608((Z)-2-Benzo[1,3]dioxol-5-yl-3-(3-methoxy-benzyl)-4...)
Affinity DataIC50:  3nMAssay Description:Ability to displace [125I]-ET-1 from the rat endothelin A receptor expressed in rat aorta smooth muscle cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(RAT)
University Of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50146627((Z)-3-Cyclohexylmethyl-4-(2,3-dihydro-benzo[1,4]di...)
Affinity DataIC50:  3.5nMAssay Description:Ability to displace [125I]-ET-1 from the rat endothelin A receptor expressed in rat aorta smooth muscle cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(RAT)
University Of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50112692(2-Benzo[1,3]dioxol-5-yl-6-ethoxy-4-(4-methoxy-phen...)
Affinity DataIC50:  3.80nMAssay Description:Ability to displace [125I]-ET-1 from the rat endothelin A receptor expressed in rat aorta smooth muscle cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(RAT)
University Of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50080630((2R,3R,4S)-4-Benzo[1,3]dioxol-5-yl-1-[(1,2-dipheny...)
Affinity DataIC50:  3.90nMAssay Description:Ability to displace [125I]-ET-1 from the rat endothelin A receptor expressed in rat aorta smooth muscle cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(RAT)
University Of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50050996((2S,3R,4S)-4-Benzo[1,3]dioxol-5-yl-1-dibutylcarbam...)
Affinity DataIC50:  4.60nMAssay Description:Ability to displace [125I]-ET-1 from the rat endothelin A receptor expressed in rat aorta smooth muscle cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(RAT)
University Of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50146616((S)-2-Benzo[1,3]dioxol-5-yl-6-isopropoxy-4-methoxy...)
Affinity DataIC50:  5.20nMAssay Description:Ability to displace [125I]-ET-1 from the rat endothelin A receptor expressed in rat aorta smooth muscle cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(RAT)
University Of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50101258(CHEMBL295440 | [(1R,3S)-1-Benzo[1,3]dioxol-5-yl-3-...)
Affinity DataIC50:  5.40nMAssay Description:Ability to displace [125I]-ET-1 from the rat endothelin A receptor expressed in rat aorta smooth muscle cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(Homo sapiens (Human))
University Of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50146614(2-Methyl-5-(3-oxazol-5-yl-phenylsulfamoyl)-furan-3...)
Affinity DataIC50:  6.20nMAssay Description:Inhibition of [125]ET-1 binding to human Endothelin A receptor expressed in vero cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(RAT)
University Of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50146609((Z)-3-Benzyl-2-(7-methoxy-benzo[1,3]dioxol-5-yl)-4...)
Affinity DataIC50:  6.70nMAssay Description:Ability to displace [125I]-ET-1 from the rat endothelin A receptor expressed in rat aorta smooth muscle cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(RAT)
University Of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50146623((Z)-2-Benzo[1,3]dioxol-5-yl-3-benzyl-4-(3,4-dimeth...)
Affinity DataIC50:  11nMAssay Description:Ability to displace [125I]-ET-1 from the rat endothelin A receptor expressed in rat aorta smooth muscle cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(RAT)
University Of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50146620((Z)-2-Benzo[1,3]dioxol-5-yl-4-(4-methoxy-phenyl)-3...)
Affinity DataIC50:  14nMAssay Description:Ability to displace [125I]-ET-1 from the rat endothelin A receptor expressed in rat aorta smooth muscle cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(RAT)
University Of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50056065((2R,3R,4S)-1-Dibutylcarbamoylmethyl-4-(4-fluoro-ph...)
Affinity DataIC50:  14nMAssay Description:Ability to displace [125I]-ET-1 from the rat endothelin A receptor expressed in rat aorta smooth muscle cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(RAT)
University Of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50112697((S)-2-Benzo[1,3]dioxol-5-yl-6-isopropoxy-4-(4-meth...)
Affinity DataIC50:  15nMAssay Description:Ability to displace [125I]-ET-1 from the rat endothelin A receptor expressed in rat aorta smooth muscle cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(RAT)
University Of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50080604((2R,3R,4S)-4-Benzo[1,3]dioxol-5-yl-1-[(2,3-dimethy...)
Affinity DataIC50:  16nMAssay Description:Ability to displace [125I]-ET-1 from the rat endothelin A receptor expressed in rat aorta smooth muscle cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(RAT)
University Of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50075412(1-(2,5-Dimethoxy-benzyl)-4-(4-methoxy-phenyl)-2-ox...)
Affinity DataIC50:  21nMAssay Description:Ability to displace [125I]-ET-1 from the rat endothelin A receptor expressed in rat aorta smooth muscle cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(RAT)
University Of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50112679(2-Benzo[1,3]dioxol-5-yl-4-pentyloxy-2H-chromene-3-...)
Affinity DataIC50:  29nMAssay Description:Ability to displace [125I]-ET-1 from the rat endothelin A receptor expressed in rat aorta smooth muscle cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(RAT)
University Of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50112726(6-Isopropoxy-2,4-bis-(4-methoxy-phenyl)-2H-chromen...)
Affinity DataIC50:  35nMAssay Description:Ability to displace [125I]-ET-1 from the rat endothelin A receptor expressed in rat aorta smooth muscle cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(RAT)
University Of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50050979((2S,3S,4R)-4-Benzo[1,3]dioxol-5-yl-2-(4-methoxy-ph...)
Affinity DataIC50:  45nMAssay Description:Ability to displace [125I]-ET-1 from the rat endothelin A receptor expressed in rat aorta smooth muscle cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(RAT)
University Of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50146617((Z)-3-Benzyl-2-(3,5-dimethoxy-phenyl)-4-(4-methoxy...)
Affinity DataIC50:  46nMAssay Description:Ability to displace [125I]-ET-1 from the rat endothelin A receptor expressed in rat aorta smooth muscle cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(RAT)
University Of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50112703(2-Benzo[1,3]dioxol-5-yl-6-methoxy-4-(4-methoxy-phe...)
Affinity DataIC50:  74nMAssay Description:Ability to displace [125I]-ET-1 from the rat endothelin A receptor expressed in rat aorta smooth muscle cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(RAT)
University Of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50112716((2S,3S,4S)-2-Benzo[1,3]dioxol-5-yl-4-butyl-6-isopr...)
Affinity DataIC50:  77nMAssay Description:Ability to displace [125I]-ET-1 from the rat endothelin A receptor expressed in rat aorta smooth muscle cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(RAT)
University Of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50112723(2-Benzo[1,3]dioxol-5-yl-4-(4-methoxy-phenyl)-2H-ch...)
Affinity DataIC50:  86nMAssay Description:Ability to displace [125I]-ET-1 from the rat endothelin A receptor expressed in rat aorta smooth muscle cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(RAT)
University Of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50101263(CHEMBL49040 | [(1R,3R)-1-Benzo[1,3]dioxol-5-yl-5-e...)
Affinity DataIC50:  96nMAssay Description:Ability to displace [125I]-ET-1 from the rat endothelin A receptor expressed in rat aorta smooth muscle cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(RAT)
University Of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50146615((Z)-2-Benzo[1,3]dioxol-5-yl-3-(4-chloro-benzyl)-4-...)
Affinity DataIC50:  110nMAssay Description:Ability to displace [125I]-ET-1 from the rat endothelin A receptor expressed in rat aorta smooth muscle cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(RAT)
University Of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50112701(2-Benzo[1,3]dioxol-5-yl-6-isopropyl-4-(4-methoxy-p...)
Affinity DataIC50:  110nMAssay Description:Ability to displace [125I]-ET-1 from the rat endothelin A receptor expressed in rat aorta smooth muscle cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(RAT)
University Of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50146625((Z)-2-Benzo[1,3]dioxol-5-yl-3-biphenyl-4-ylmethyl-...)
Affinity DataIC50:  200nMAssay Description:Ability to displace [125I]-ET-1 from the rat endothelin A receptor expressed in rat aorta smooth muscle cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(Homo sapiens (Human))
University Of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50146607(2-(2-Benzyloxycarbonylamino-3-methyl-butyrylamino)...)
Affinity DataIC50:  220nMAssay Description:Inhibition of [125]ET-1 binding to human Endothelin A receptor expressed in vero cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(RAT)
University Of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50112711((R)-2-Benzo[1,3]dioxol-5-yl-6-isopropoxy-2H-chrome...)
Affinity DataIC50:  240nMAssay Description:Ability to displace [125I]-ET-1 from the rat endothelin A receptor expressed in rat aorta smooth muscle cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin receptor type B(Homo sapiens (Human))
University Of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50146608((Z)-2-Benzo[1,3]dioxol-5-yl-3-(3-methoxy-benzyl)-4...)
Affinity DataIC50:  260nMAssay Description:Inhibitory concentration of the compound against Endothelin B receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(RAT)
University Of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50146604((Z)-3-Benzyl-2-(2,4-dimethoxy-phenyl)-4-(4-methoxy...)
Affinity DataIC50:  300nMAssay Description:Ability to displace [125I]-ET-1 from the rat endothelin A receptor expressed in rat aorta smooth muscle cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin receptor type B(Homo sapiens (Human))
University Of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50112748((R)-2-Benzo[1,3]dioxol-5-yl-4-butyl-6-isopropoxy-2...)
Affinity DataIC50:  400nMAssay Description:Inhibitory concentration of the compound against Endothelin B receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(RAT)
University Of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50112691(2-Benzo[1,3]dioxol-5-yl-4-butyl-6-isopropoxy-2H-ch...)
Affinity DataIC50:  410nMAssay Description:Ability to displace [125I]-ET-1 from the rat endothelin A receptor expressed in rat aorta smooth muscle cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(RAT)
University Of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50146621((Z)-2-Benzo[1,3]dioxol-5-yl-3-benzyl-4-(3-methoxy-...)
Affinity DataIC50:  500nMAssay Description:Ability to displace [125I]-ET-1 from the rat endothelin A receptor expressed in rat aorta smooth muscle cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(RAT)
University Of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50146612((Z)-3-(4-Methoxy-benzyl)-4-(4-methoxy-phenyl)-4-ox...)
Affinity DataIC50:  570nMAssay Description:Ability to displace [125I]-ET-1 from the rat endothelin A receptor expressed in rat aorta smooth muscle cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(RAT)
University Of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50146626((Z)-2-Benzo[1,3]dioxol-5-yl-3-benzyl-4-(4-ethyl-ph...)
Affinity DataIC50:  630nMAssay Description:Ability to displace [125I]-ET-1 from the rat endothelin A receptor expressed in rat aorta smooth muscle cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(RAT)
University Of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50112674(2-Benzo[1,3]dioxol-5-yl-4-phenyl-2H-chromene-3-car...)
Affinity DataIC50:  780nMAssay Description:Ability to displace [125I]-ET-1 from the rat endothelin A receptor expressed in rat aorta smooth muscle cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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