TargetProtein kinase C alpha type(Homo sapiens (Human))
National Cancer Institute-Bethesda
Curated by ChEMBL
National Cancer Institute-Bethesda
Curated by ChEMBL
Affinity DataKi: 78nMAssay Description:Displacement of [20-3H]phorbol12,13-dibutyrate from a recombinant PK-C alphaMore data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Homo sapiens (Human))
National Cancer Institute-Bethesda
Curated by ChEMBL
National Cancer Institute-Bethesda
Curated by ChEMBL
Affinity DataKi: 91nMAssay Description:Displacement of [20-3H]phorbol12,13-dibutyrate from a recombinant PK-C alphaMore data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Homo sapiens (Human))
National Cancer Institute-Bethesda
Curated by ChEMBL
National Cancer Institute-Bethesda
Curated by ChEMBL
Affinity DataKi: 138nMAssay Description:Displacement of [20-3H]phorbol12,13-dibutyrate from a recombinant PK-C alphaMore data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Homo sapiens (Human))
National Cancer Institute-Bethesda
Curated by ChEMBL
National Cancer Institute-Bethesda
Curated by ChEMBL
Affinity DataKi: 320nMAssay Description:Displacement of [20-3H]phorbol12,13-dibutyrate from a recombinant PK-C alphaMore data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Homo sapiens (Human))
National Cancer Institute-Bethesda
Curated by ChEMBL
National Cancer Institute-Bethesda
Curated by ChEMBL
Affinity DataKi: 823nMAssay Description:Displacement of [20-3H]phorbol12,13-dibutyrate from a recombinant PK-C alphaMore data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Homo sapiens (Human))
National Cancer Institute-Bethesda
Curated by ChEMBL
National Cancer Institute-Bethesda
Curated by ChEMBL
Affinity DataKi: 1.04E+3nMAssay Description:Displacement of [20-3H]phorbol12,13-dibutyrate from a recombinant PK-C alphaMore data for this Ligand-Target Pair
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Sungkyunkwan University
Curated by ChEMBL
Sungkyunkwan University
Curated by ChEMBL
Affinity DataIC50: 0.900nMAssay Description:Inhibition of c-Met (unknown origin) by ADP-Glo kinase assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Inhibition of PREP (unknown origin) using AMC substrate by fluorometric assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Inhibition of PREP (unknown origin) using AMC substrate by fluorometric assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Inhibition of PREP (unknown origin) using AMC substrate by fluorometric assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Inhibition of FAP (unknown origin) using AMC substrate by fluorometric assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.70nMAssay Description:Inhibition of full length human recombinant N-terminal GST-tagged HDAC6 (1 to 1215 residues) expressed in sf9 cells using RHK-K(Ac)-AMC as substrate ...More data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:Inhibition of DPP4 (unknown origin) using AMC substrate by fluorometric assayMore data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:Inhibition of FAP (unknown origin) using AMC substrate by fluorometric assayMore data for this Ligand-Target Pair
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Sungkyunkwan University
Curated by ChEMBL
Sungkyunkwan University
Curated by ChEMBL
Affinity DataIC50: 3nMAssay Description:Inhibition of c-Met (unknown origin) by ADP-Glo kinase assayMore data for this Ligand-Target Pair
Affinity DataIC50: 3.30nMAssay Description:Inhibition of FAP (unknown origin) using AMC substrate by fluorometric assayMore data for this Ligand-Target Pair
Affinity DataIC50: 4nMAssay Description:Inhibition of FAP (unknown origin) using AMC substrate by fluorometric assayMore data for this Ligand-Target Pair
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Sungkyunkwan University
Curated by ChEMBL
Sungkyunkwan University
Curated by ChEMBL
Affinity DataIC50: 4nMAssay Description:Inhibition of c-Met (unknown origin) by ADP-Glo kinase assayMore data for this Ligand-Target Pair
Affinity DataIC50: 5nMAssay Description:Inhibition of FAP (unknown origin) using AMC substrate by fluorometric assayMore data for this Ligand-Target Pair
Affinity DataIC50: 5nMAssay Description:Inhibition of PREP (unknown origin) using AMC substrate by fluorometric assayMore data for this Ligand-Target Pair
Affinity DataIC50: 5nMAssay Description:Inhibition of FAP (unknown origin) using AMC substrate by fluorometric assayMore data for this Ligand-Target Pair
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Sungkyunkwan University
Curated by ChEMBL
Sungkyunkwan University
Curated by ChEMBL
Affinity DataIC50: 5nMAssay Description:Inhibition of c-Met (unknown origin) by ADP-Glo kinase assayMore data for this Ligand-Target Pair
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Sungkyunkwan University
Curated by ChEMBL
Sungkyunkwan University
Curated by ChEMBL
Affinity DataIC50: 6nMAssay Description:Inhibition of c-Met (unknown origin) by ADP-Glo kinase assayMore data for this Ligand-Target Pair
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Sungkyunkwan University
Curated by ChEMBL
Sungkyunkwan University
Curated by ChEMBL
Affinity DataIC50: 6nMAssay Description:Inhibition of c-Met (unknown origin) by ADP-Glo kinase assayMore data for this Ligand-Target Pair
Affinity DataIC50: 6.60nMAssay Description:Inhibition of full length human recombinant C-terminal FLAG-His-tagged HDAC1 (1 to 482 residues) expressed in Sf21 cells using RHK-K(Ac)-AMC as subst...More data for this Ligand-Target Pair
Affinity DataIC50: 7nMAssay Description:Inhibition of FAP (unknown origin) using AMC substrate by fluorometric assayMore data for this Ligand-Target Pair
Affinity DataIC50: 9nMAssay Description:Inhibition of PREP (unknown origin) using AMC substrate by fluorometric assayMore data for this Ligand-Target Pair
Affinity DataIC50: 9nMAssay Description:Inhibition of FAP (unknown origin) using AMC substrate by fluorometric assayMore data for this Ligand-Target Pair
Affinity DataIC50: 10.5nMAssay Description:Inhibition of full length human recombinant C-terminal GST-tagged HDAC2 (1 to 488 residues) expressed in insect cells using RHK-K(Ac)-AMC as substrat...More data for this Ligand-Target Pair
Affinity DataIC50: 11nMAssay Description:Inhibition of FAP (unknown origin) using AMC substrate by fluorometric assayMore data for this Ligand-Target Pair
TargetHistone deacetylase 3/Nuclear receptor corepressor 2 (HDAC3/NCoR2)(Homo sapiens (Human))
Sungkyunkwan University
Curated by ChEMBL
Sungkyunkwan University
Curated by ChEMBL
Affinity DataIC50: 11.1nMAssay Description:Inhibition of full length human recombinant C-terminal His-tagged HDAC3 (1 to 428 residues)/human recombinant N-terminal GST-tagged NCOR2 expressed i...More data for this Ligand-Target Pair
Affinity DataIC50: 11.4nMAssay Description:Inhibition of human recombinant N-terminal His-tagged HDAC11 (1 to 347 residues) expressed in insect cells/baculovirus expression system using RHK-K(...More data for this Ligand-Target Pair
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Sungkyunkwan University
Curated by ChEMBL
Sungkyunkwan University
Curated by ChEMBL
Affinity DataIC50: 12nMAssay Description:Inhibition of c-Met (unknown origin) by ADP-Glo kinase assayMore data for this Ligand-Target Pair
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Sungkyunkwan University
Curated by ChEMBL
Sungkyunkwan University
Curated by ChEMBL
Affinity DataIC50: 12nMAssay Description:Inhibition of c-Met (unknown origin) by ADP-Glo kinase assayMore data for this Ligand-Target Pair
Affinity DataIC50: 12nMAssay Description:Inhibition of FAP (unknown origin) using AMC substrate by fluorometric assayMore data for this Ligand-Target Pair
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Sungkyunkwan University
Curated by ChEMBL
Sungkyunkwan University
Curated by ChEMBL
Affinity DataIC50: 14nMAssay Description:Inhibition of c-Met (unknown origin) by ADP-Glo kinase assayMore data for this Ligand-Target Pair
Affinity DataIC50: 14nMAssay Description:Inhibition of FAP (unknown origin) using AMC substrate by fluorometric assayMore data for this Ligand-Target Pair
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Sungkyunkwan University
Curated by ChEMBL
Sungkyunkwan University
Curated by ChEMBL
Affinity DataIC50: 14nMAssay Description:Inhibition of c-Met (unknown origin) by ADP-Glo kinase assayMore data for this Ligand-Target Pair
Affinity DataIC50: 16nMAssay Description:Inhibition of PREP (unknown origin) using AMC substrate by fluorometric assayMore data for this Ligand-Target Pair
Affinity DataIC50: 16nMAssay Description:Inhibition of FAP (unknown origin) using AMC substrate by fluorometric assayMore data for this Ligand-Target Pair
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Sungkyunkwan University
Curated by ChEMBL
Sungkyunkwan University
Curated by ChEMBL
Affinity DataIC50: 17nMAssay Description:Inhibition of c-Met (unknown origin) by ADP-Glo kinase assayMore data for this Ligand-Target Pair
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Sungkyunkwan University
Curated by ChEMBL
Sungkyunkwan University
Curated by ChEMBL
Affinity DataIC50: 18nMAssay Description:Inhibition of c-Met (unknown origin) by ADP-Glo kinase assayMore data for this Ligand-Target Pair
Affinity DataIC50: 19nMAssay Description:Inhibition of FAP (unknown origin) using AMC substrate by fluorometric assayMore data for this Ligand-Target Pair
Affinity DataIC50: 20nMAssay Description:Inhibition of FAP (unknown origin) using AMC substrate by fluorometric assayMore data for this Ligand-Target Pair
Affinity DataIC50: 20nMAssay Description:Inhibition of FAP (unknown origin) using AMC substrate by fluorometric assayMore data for this Ligand-Target Pair
Affinity DataIC50: 21nMAssay Description:Inhibition of FAP (unknown origin) using AMC substrate by fluorometric assayMore data for this Ligand-Target Pair
Affinity DataIC50: 21nMAssay Description:Inhibition of FAP (unknown origin) using AMC substrate by fluorometric assayMore data for this Ligand-Target Pair
Affinity DataIC50: 22nMAssay Description:Inhibition of DPP4 (unknown origin) using AMC substrate by fluorometric assayMore data for this Ligand-Target Pair
Affinity DataIC50: 22nMAssay Description:Inhibition of FAP (unknown origin) using AMC substrate by fluorometric assayMore data for this Ligand-Target Pair
Affinity DataIC50: 23nMAssay Description:Inhibition of FAP (unknown origin) using AMC substrate by fluorometric assayMore data for this Ligand-Target Pair