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Found 87 with Last Name = 'klimko' and Initial = 'pg'
TargetProstaglandin F2-alpha receptor(Homo sapiens (Human))
Alcon Laboratories

Curated by ChEMBL
LigandPNGBDBM50085910((Z)-7-{(1R,2R,3R,5S)-2-[(E)-(R)-4-(3-Chloro-phenox...)
Affinity DataKi:  31nMAssay Description:Inhibitory Binding constant (n=2) to Prostanoid FP receptor expressed in bovine corpus luteumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin F2-alpha receptor(BOVINE)
Alcon Research

Curated by ChEMBL
LigandPNGBDBM50150906((E)-7-{(1R,2R,3R,5S)-3,5-Dihydroxy-2-[(E)-3-hydrox...)
Affinity DataKi:  52nMAssay Description:Binding affinity for Prostanoid FP receptor of bovine corpus luteumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin F2-alpha receptor(BOVINE)
Alcon Research

Curated by ChEMBL
LigandPNGBDBM50150899((E)-7-[(1R,2R,3R,5S)-3,5-Dihydroxy-2-((R)-3-hydrox...)
Affinity DataKi:  92nMAssay Description:Binding affinity for Prostanoid FP receptor of bovine corpus luteumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin F2-alpha receptor(Homo sapiens (Human))
Alcon Laboratories

Curated by ChEMBL
LigandPNGBDBM50035622((5Z,13E,15S)-9alpha,11alpha,15-trihydroxyprosta-5,...)
Affinity DataKi:  119nMAssay Description:Inhibitory Binding constant (n=2) to Prostanoid FP receptor expressed in bovine corpus luteumMore data for this Ligand-Target Pair
TargetProstaglandin F2-alpha receptor(BOVINE)
Alcon Research

Curated by ChEMBL
LigandPNGBDBM50035622((5Z,13E,15S)-9alpha,11alpha,15-trihydroxyprosta-5,...)
Affinity DataKi:  129nMAssay Description:Binding affinity for Prostanoid FP receptor of bovine corpus luteumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin F2-alpha receptor(BOVINE)
Alcon Research

Curated by ChEMBL
LigandPNGBDBM50150898((Z)-8-{(2R,3S,4R)-2-[(E)-(R)-4-(3-Chloro-phenoxy)-...)
Affinity DataKi:  147nMAssay Description:Binding affinity for Prostanoid FP receptor of bovine corpus luteumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin F2-alpha receptor(BOVINE)
Alcon Research

Curated by ChEMBL
LigandPNGBDBM50150904((Z)-8-[(2R,3S,4R)-4-Hydroxy-2-((E)-(R)-3-hydroxy-4...)
Affinity DataKi:  330nMAssay Description:Binding affinity for Prostanoid FP receptor of bovine corpus luteumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin F2-alpha receptor(BOVINE)
Alcon Research

Curated by ChEMBL
LigandPNGBDBM50150892((Z)-8-{(2R,3S,4R)-4-Hydroxy-2-[(E)-(R)-3-hydroxy-4...)
Affinity DataKi:  350nMAssay Description:Binding affinity for Prostanoid FP receptor of bovine corpus luteumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin F2-alpha receptor(BOVINE)
Alcon Research

Curated by ChEMBL
LigandPNGBDBM50150902((Z)-8-[(2R,3S,4R)-4-Hydroxy-2-((E)-(R)-3-hydroxy-4...)
Affinity DataKi:  640nMAssay Description:Binding affinity for Prostanoid FP receptor of bovine corpus luteumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin F2-alpha receptor(BOVINE)
Alcon Research

Curated by ChEMBL
LigandPNGBDBM50150896((Z)-8-{(2R,3S,4R)-2-[(E)-(S)-4-(3-Chloro-phenoxy)-...)
Affinity DataKi:  820nMAssay Description:Binding affinity for Prostanoid FP receptor of bovine corpus luteumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin F2-alpha receptor(BOVINE)
Alcon Research

Curated by ChEMBL
LigandPNGBDBM50150900((Z)-8-{(2R,3S,4R)-2-[(E)-(R)-4-(3-Chloro-phenoxy)-...)
Affinity DataKi:  890nMAssay Description:Binding affinity for Prostanoid FP receptor of bovine corpus luteumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin F2-alpha receptor(Homo sapiens (Human))
Alcon Laboratories

Curated by ChEMBL
LigandPNGBDBM50091623(7-{2-[4-(3-Chloro-phenoxy)-3-hydroxy-but-1-enyl]-3...)
Affinity DataKi:  1.90E+3nMAssay Description:Inhibitory Binding constant (n=2) to Prostanoid FP receptor expressed in bovine corpus luteumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin F2-alpha receptor(BOVINE)
Alcon Research

Curated by ChEMBL
LigandPNGBDBM50150891((Z)-8-[(R)-4-Hydroxy-2-((1R,2S,4S)-3-hydroxy-4-phe...)
Affinity DataKi:  2.80E+3nMAssay Description:Binding affinity for Prostanoid FP receptor of bovine corpus luteumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin F2-alpha receptor(BOVINE)
Alcon Research

Curated by ChEMBL
LigandPNGBDBM50150894((Z)-8-{(2R,3S,4R)-4-Hydroxy-2-[(E)-(R)-3-hydroxy-4...)
Affinity DataKi:  3.10E+3nMAssay Description:Binding affinity for Prostanoid FP receptor of bovine corpus luteumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin F2-alpha receptor(BOVINE)
Alcon Research

Curated by ChEMBL
LigandPNGBDBM50150897((Z)-8-[(2R,3S,4R)-4-Hydroxy-2-((E)-(S)-3-hydroxy-4...)
Affinity DataKi:  5.10E+3nMAssay Description:Binding affinity for Prostanoid FP receptor of bovine corpus luteumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin F2-alpha receptor(BOVINE)
Alcon Research

Curated by ChEMBL
LigandPNGBDBM50150903((Z)-7-[(2R,3S,4R)-4-Hydroxy-2-((E)-(S)-3-hydroxy-o...)
Affinity DataKi:  6.70E+3nMAssay Description:Binding affinity for Prostanoid FP receptor of bovine corpus luteumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin F2-alpha receptor(BOVINE)
Alcon Research

Curated by ChEMBL
LigandPNGBDBM50150901((Z)-8-{(2R,3S,4R)-2-[(E)-(S)-4-(3-Chloro-phenoxy)-...)
Affinity DataKi:  7.30E+3nMAssay Description:Binding affinity for Prostanoid FP receptor of bovine corpus luteumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin F2-alpha receptor(BOVINE)
Alcon Research

Curated by ChEMBL
LigandPNGBDBM50150893((Z)-8-{(2R,3S,4R)-4-Hydroxy-2-[(E)-(S)-3-hydroxy-4...)
Affinity DataKi:  9.90E+3nMAssay Description:Binding affinity for Prostanoid FP receptor of bovine corpus luteumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin F2-alpha receptor(BOVINE)
Alcon Research

Curated by ChEMBL
LigandPNGBDBM50150905((Z)-8-{(2R,3S,4R)-4-Hydroxy-2-[(E)-(S)-3-hydroxy-4...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity for Prostanoid FP receptor of bovine corpus luteumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin F2-alpha receptor(BOVINE)
Alcon Research

Curated by ChEMBL
LigandPNGBDBM50150895((Z)-7-[(2R,3S,4R)-4-Hydroxy-2-((E)-(R)-3-hydroxy-o...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity for Prostanoid FP receptor of bovine corpus luteumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin F2-alpha receptor(Homo sapiens (Human))
Alcon Laboratories

Curated by ChEMBL
LigandPNGBDBM50091622(7-{2-[4-(3-Chloro-phenoxy)-3-hydroxy-but-1-enyl]-3...)
Affinity DataKi:  5.60E+4nMAssay Description:Inhibitory Binding constant (n=2) to Prostanoid FP receptor expressed in bovine corpus luteumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Alcon Research

Curated by ChEMBL
LigandPNGBDBM50210089((R)-2-(8-methoxymethyl-benzo[1,2-b;4,5-b']difuran-...)
Affinity DataIC50:  0.110nMAssay Description:Displacement of [125I]DOI from 5HT2A receptor in rat cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Alcon Research

Curated by ChEMBL
LigandPNGBDBM50210078((R)-2-(8-methoxymethyl-2,3,6,7-tetrahydro-benzo[1,...)
Affinity DataIC50:  0.280nMAssay Description:Displacement of [125I]DOI from 5HT2A receptor in rat cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Alcon Research

Curated by ChEMBL
LigandPNGBDBM50210083(CHEMBL232995 | [8-((R)-2-amino-propyl)-2,3,6,7-tet...)
Affinity DataIC50:  0.290nMAssay Description:Displacement of [125I]DOI from 5HT2A receptor in rat cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Alcon Research

Curated by ChEMBL
LigandPNGBDBM50052337(2-(8-bromo-2,3,6,7-tetrahydro-benzo[1,2-b;4,5-b']d...)
Affinity DataIC50:  0.300nMAssay Description:Displacement of [125I]DOI from 5HT2A receptor in rat cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Alcon Research

Curated by ChEMBL
LigandPNGBDBM50210093(CHEMBL393077 | [8-((R)-2-amino-propyl)-benzo[1,2-b...)
Affinity DataIC50:  0.310nMAssay Description:Displacement of [125I]DOI from 5HT2A receptor in rat cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Alcon Research

Curated by ChEMBL
LigandPNGBDBM50210084((R)-1-methyl-2-[8-(3-methyl-[1,2,4]oxadiazol-5-ylm...)
Affinity DataIC50:  0.380nMAssay Description:Displacement of [125I]DOI from 5HT2A receptor in rat cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Alcon Research

Curated by ChEMBL
LigandPNGBDBM50133231((R)-1-(4-iodo-2,5-dimethoxyphenyl)propan-2-amine |...)
Affinity DataIC50:  0.460nMAssay Description:Displacement of [125I]DOI from 5HT2A receptor in rat cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Alcon Research

Curated by ChEMBL
LigandPNGBDBM50210081((1R,2R)-2-amino-1-(8-bromo-2,3,6,7-tetrahydro-benz...)
Affinity DataIC50:  0.700nMAssay Description:Displacement of [125I]DOI from 5HT2A receptor in rat cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Alcon Research

Curated by ChEMBL
LigandPNGBDBM50210092(3-[8-((R)-2-amino-propyl)-2,3,6,7-tetrahydro-benzo...)
Affinity DataIC50:  0.860nMAssay Description:Displacement of [125I]DOI from 5HT2A receptor in rat cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Alcon Research

Curated by ChEMBL
LigandPNGBDBM50210079((R)-2-[8-(2-methoxy-ethoxymethyl)-2,3,6,7-tetrahyd...)
Affinity DataIC50:  0.880nMAssay Description:Displacement of [125I]DOI from 5HT2A receptor in rat cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Alcon Research

Curated by ChEMBL
LigandPNGBDBM50210087(CHEMBL394664 | [8-((R)-2-amino-propyl)-2,3,6,7-tet...)
Affinity DataIC50:  1nMAssay Description:Displacement of [125I]DOI from 5HT2A receptor in rat cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Alcon Research

Curated by ChEMBL
LigandPNGBDBM50210088((R)-1-methyl-2-{8-[2-(3-methyl-[1,2,4]oxadiazol-5-...)
Affinity DataIC50:  1nMAssay Description:Displacement of [125I]DOI from 5HT2A receptor in rat cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Alcon Research

Curated by ChEMBL
LigandPNGBDBM50210085((R)-1-methyl-2-[8-(3-methyl-[1,2,4]oxadiazol-5-ylm...)
Affinity DataIC50:  1.60nMAssay Description:Displacement of [125I]DOI from 5HT2A receptor in rat cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Alcon Research

Curated by ChEMBL
LigandPNGBDBM50210091((1S,2R)-2-amino-1-(8-bromo-2,3,6,7-tetrahydro-benz...)
Affinity DataIC50:  2.60nMAssay Description:Displacement of [125I]DOI from 5HT2A receptor in rat cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Alcon Research

Curated by ChEMBL
LigandPNGBDBM50210080(8-((R)-2-amino-propyl)-2,3,6,7-tetrahydro-benzo[1,...)
Affinity DataIC50:  14nMAssay Description:Displacement of [125I]DOI from 5HT2A receptor in rat cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Alcon Research

Curated by ChEMBL
LigandPNGBDBM50210090(CHEMBL232997 | [8-((R)-2-amino-propyl)-2,3,6,7-tet...)
Affinity DataIC50:  104nMAssay Description:Displacement of [125I]DOI from 5HT2A receptor in rat cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Alcon Research

Curated by ChEMBL
LigandPNGBDBM50210086((R)-1-methyl-2-[8-(3-methyl-[1,2,4]oxadiazol-5-yl)...)
Affinity DataIC50:  910nMAssay Description:Displacement of [125I]DOI from 5HT2A receptor in rat cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Alcon Research

Curated by ChEMBL
LigandPNGBDBM50210082(3-[8-((R)-2-amino-propyl)-2,3,6,7-tetrahydro-benzo...)
Affinity DataIC50:  4.70E+3nMAssay Description:Displacement of [125I]DOI from 5HT2A receptor in rat cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2B(RAT)
Alcon Research

Curated by ChEMBL
LigandPNGBDBM50210079((R)-2-[8-(2-methoxy-ethoxymethyl)-2,3,6,7-tetrahyd...)
Affinity DataEC50:  5.80nMAssay Description:Agonist activity at 5HT2B receptor in rat stomach fundus assessed as intracellular calcium mobilization relative to 5HTMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Alcon Research

Curated by ChEMBL
LigandPNGBDBM50210080(8-((R)-2-amino-propyl)-2,3,6,7-tetrahydro-benzo[1,...)
Affinity DataEC50:  880nMAssay Description:Agonist activity at 5HT2A receptor in rat A7r5 cells assessed as intracellular calcium mobilization relative to 5HTMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Alcon Research

Curated by ChEMBL
LigandPNGBDBM50210081((1R,2R)-2-amino-1-(8-bromo-2,3,6,7-tetrahydro-benz...)
Affinity DataEC50:  32.7nMAssay Description:Agonist activity at 5HT2A receptor in rat A7r5 cells assessed as intracellular calcium mobilization relative to 5HTMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Alcon Research

Curated by ChEMBL
LigandPNGBDBM50210079((R)-2-[8-(2-methoxy-ethoxymethyl)-2,3,6,7-tetrahyd...)
Affinity DataEC50:  71nMAssay Description:Agonist activity at 5HT2A receptor in rat A7r5 cells assessed as intracellular calcium mobilization relative to 5HTMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2B(RAT)
Alcon Research

Curated by ChEMBL
LigandPNGBDBM50210081((1R,2R)-2-amino-1-(8-bromo-2,3,6,7-tetrahydro-benz...)
Affinity DataEC50:  6.20nMAssay Description:Agonist activity at 5HT2B receptor in rat stomach fundus assessed as intracellular calcium mobilization relative to 5HTMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Alcon Research

Curated by ChEMBL
LigandPNGBDBM50210083(CHEMBL232995 | [8-((R)-2-amino-propyl)-2,3,6,7-tet...)
Affinity DataEC50:  6.20nMAssay Description:Agonist activity at 5HT2A receptor in rat A7r5 cells assessed as intracellular calcium mobilization relative to 5HTMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2B(RAT)
Alcon Research

Curated by ChEMBL
LigandPNGBDBM50210083(CHEMBL232995 | [8-((R)-2-amino-propyl)-2,3,6,7-tet...)
Affinity DataEC50:  59nMAssay Description:Agonist activity at 5HT2B receptor in rat stomach fundus assessed as intracellular calcium mobilization relative to 5HTMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Alcon Research

Curated by ChEMBL
LigandPNGBDBM50210078((R)-2-(8-methoxymethyl-2,3,6,7-tetrahydro-benzo[1,...)
Affinity DataEC50:  12nMAssay Description:Agonist activity at 5HT2A receptor in rat A7r5 cells assessed as intracellular calcium mobilization relative to 5HTMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Alcon Research

Curated by ChEMBL
LigandPNGBDBM50052337(2-(8-bromo-2,3,6,7-tetrahydro-benzo[1,2-b;4,5-b']d...)
Affinity DataEC50:  13nMAssay Description:Agonist activity at 5HT2A receptor in rat A7r5 cells assessed as intracellular calcium mobilization relative to 5HTMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Alcon Research

Curated by ChEMBL
LigandPNGBDBM50210084((R)-1-methyl-2-[8-(3-methyl-[1,2,4]oxadiazol-5-ylm...)
Affinity DataEC50:  16.9nMAssay Description:Agonist activity at 5HT2A receptor in rat A7r5 cells assessed as intracellular calcium mobilization relative to 5HTMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Alcon Research

Curated by ChEMBL
LigandPNGBDBM50210089((R)-2-(8-methoxymethyl-benzo[1,2-b;4,5-b']difuran-...)
Affinity DataEC50:  3.60nMAssay Description:Agonist activity at 5HT2A receptor in rat A7r5 cells assessed as intracellular calcium mobilization relative to 5HTMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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