Affinity DataKi: 0.447nMAssay Description:Inhibition of N/OFQ binding to human Orphanin FQ receptor (Nociceptin/Orphanin)More data for this Ligand-Target Pair
Affinity DataKi: 0.525nMAssay Description:Inhibition of N/OFQ binding to human Orphanin FQ receptor (Nociceptin/Orphanin)More data for this Ligand-Target Pair
Affinity DataKi: 0.646nMAssay Description:Inhibition of N/OFQ binding to human Orphanin FQ receptor (Nociceptin/Orphanin)More data for this Ligand-Target Pair
Affinity DataKi: 0.661nMAssay Description:Inhibition of N/OFQ binding to human Orphanin FQ receptor (Nociceptin/Orphanin)More data for this Ligand-Target Pair
Affinity DataKi: 0.776nMAssay Description:Inhibition of N/OFQ binding to human Orphanin FQ receptor (Nociceptin/Orphanin)More data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Displacement of [3H]MPEP from recombinant human mGlu5 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Displacement of [3H]LSD from human recombinant 5HT7 receptor expressed in HEK293-EBNA cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.20nMAssay Description:Inhibition of N/OFQ binding to human Orphanin FQ receptor (Nociceptin/Orphanin)More data for this Ligand-Target Pair
Affinity DataKi: 1.20nMAssay Description:Inhibition of N/OFQ binding to human Orphanin FQ receptor (Nociceptin/Orphanin)More data for this Ligand-Target Pair
Affinity DataKi: 1.30nMAssay Description:Binding affinity to rat 5HT5A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.60nMAssay Description:Binding affinity to human 5HT5A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.70nMAssay Description:Inhibition of N/OFQ binding to human Orphanin FQ receptor (Nociceptin/Orphanin)More data for this Ligand-Target Pair
Affinity DataKi: 1.70nMAssay Description:Inhibition of N/OFQ binding to human Orphanin FQ receptor (Nociceptin/Orphanin)More data for this Ligand-Target Pair
Affinity DataKi: 1.80nMAssay Description:Binding affinity to human 5HT5A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Displacement of [3H]LSD from human recombinant 5HT5A receptor expressed in HEK293-EBNA cellsMore data for this Ligand-Target Pair
Affinity DataKi: 2.10nMAssay Description:Inhibition of N/OFQ binding to human Orphanin FQ receptor (Nociceptin/Orphanin)More data for this Ligand-Target Pair
Affinity DataKi: 2.10nMAssay Description:Inhibition of N/OFQ binding to human Orphanin FQ receptor (Nociceptin/Orphanin)More data for this Ligand-Target Pair
Affinity DataKi: 2.20nMAssay Description:Inhibition of N/OFQ binding to human Orphanin FQ receptor (Nociceptin/Orphanin)More data for this Ligand-Target Pair
Affinity DataKi: 2.40nMAssay Description:Displacement of [3H]LSD from human recombinant 5HT7 receptor expressed in HEK293-EBNA cellsMore data for this Ligand-Target Pair
Affinity DataKi: 2.40nMAssay Description:Displacement of [3H]LSD from human recombinant 5HT7 receptor expressed in HEK293-EBNA cellsMore data for this Ligand-Target Pair
Affinity DataKi: 2.5nMAssay Description:Displacement of [3H]LSD from human recombinant 5HT7 receptor expressed in HEK293-EBNA cellsMore data for this Ligand-Target Pair
Affinity DataKi: 2.60nMAssay Description:Binding affinity to histamine H1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 2.90nMAssay Description:Binding affinity to rat 5HT5A receptorMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 5(Rattus norvegicus (Rat))
F. Hoffmann-La Roche
Curated by PDSP Ki Database
F. Hoffmann-La Roche
Curated by PDSP Ki Database
Affinity DataKi: 4.20nMAssay Description:Binding affinity to human 5HT7 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 4.70nMAssay Description:Displacement of [3H]LSD from human recombinant 5HT5A receptor expressed in HEK293-EBNA cellsMore data for this Ligand-Target Pair
Affinity DataKi: 4.70nMAssay Description:Displacement of [3H]MPEP from recombinant human mGlu5 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 5nMAssay Description:Displacement of [3H]MPEP from recombinant human mGlu5 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 5.10nMAssay Description:Displacement of [3H]LSD from human recombinant 5HT5A receptor expressed in HEK293-EBNA cellsMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 5(Rattus norvegicus (Rat))
F. Hoffmann-La Roche
Curated by PDSP Ki Database
F. Hoffmann-La Roche
Curated by PDSP Ki Database
Affinity DataKi: 5.70nMAssay Description:Binding affinity to human 5HT5A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 6nMAssay Description:Displacement of [3H]MPEP from recombinant human mGlu5 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 6nMAssay Description:Binding affinity to human 5HT7 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 6.30nMAssay Description:Displacement of [3H]LSD from human recombinant 5HT5A receptor expressed in HEK293-EBNA cellsMore data for this Ligand-Target Pair
Affinity DataKi: 6.30nMAssay Description:Displacement of [3H]LSD from human recombinant 5HT5A receptor expressed in HEK293-EBNA cellsMore data for this Ligand-Target Pair
Affinity DataKi: 6.5nMAssay Description:Displacement of [3H]LSD from human recombinant 5HT5A receptor expressed in HEK293-EBNA cellsMore data for this Ligand-Target Pair
Affinity DataKi: 6.80nMAssay Description:Binding affinity to human 5HT5A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 7.70nMAssay Description:Binding affinity to human 5HT7 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 8nMAssay Description:Binding affinity to histamine H1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 8.20nMAssay Description:Displacement of [3H]LSD from human recombinant 5HT7 receptor expressed in HEK293-EBNA cellsMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 5(Rattus norvegicus (Rat))
F. Hoffmann-La Roche
Curated by PDSP Ki Database
F. Hoffmann-La Roche
Curated by PDSP Ki Database
Affinity DataKi: 8.70nMAssay Description:Displacement of [3H]LSD from human recombinant 5HT7 receptor expressed in HEK293-EBNA cellsMore data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Displacement of [3H]MPEP from recombinant human mGlu5 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Displacement of [3H]LSD from human recombinant 5HT5A receptor expressed in HEK293-EBNA cellsMore data for this Ligand-Target Pair
Affinity DataKi: 10.1nMAssay Description:Binding affinity to human 5HT5A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 10.8nMAssay Description:Displacement of [3H]LSD from human recombinant 5HT5A receptor expressed in HEK293-EBNA cellsMore data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:Displacement of [3H]MPEP from recombinant human mGlu5 receptorMore data for this Ligand-Target Pair