Affinity DataKi: 0.574nMAssay Description:Displacement of [33P]-S1P from human S1P5 receptor expressed in CHO-K1 cells after 60 mins by scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 0.626nMAssay Description:Agonist activity at human S1P5 receptor expressed in CHO-K1 cells assessed as inhibition of forskolin-stimulated cAMP accumulation after 30 mins by E...More data for this Ligand-Target Pair
Affinity DataKi: 0.772nMAssay Description:Displacement of [33P]-S1P from human S1P2 receptor expressed in CHO-K1 cells after 60 mins by scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 29nMAssay Description:Displacement of [33P]-S1P from human S1P4 receptor expressed in CHO-K1 cells after 60 mins by scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: >5.45E+3nMAssay Description:Displacement of [33P]-S1P from rat S1P1 receptor after 60 mins by scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: >5.63E+3nMAssay Description:Displacement of [33P]-S1P from human S1P3 receptor expressed in CHO-K1 cells after 60 mins by scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataIC50: 0.270nMAssay Description:In vitro inhibitory activity against enkephalinase enzyme from rat.More data for this Ligand-Target Pair
Affinity DataIC50: 0.820nMAssay Description:In vitro inhibitory activity against enkephalinase enzyme from rat.More data for this Ligand-Target Pair
Affinity DataIC50: 0.900nMAssay Description:In vitro inhibitory activity against enkephalinase enzyme from rat.More data for this Ligand-Target Pair
Affinity DataIC50: 1.10nMAssay Description:In vitro inhibitory activity against enkephalinase enzyme from rat.More data for this Ligand-Target Pair
Affinity DataIC50: 1.5nMAssay Description:In vitro inhibitory activity against enkephalinase enzyme from rat.More data for this Ligand-Target Pair
Affinity DataIC50: 1.70nMAssay Description:In vitro inhibitory activity against enkephalinase enzyme from rat.More data for this Ligand-Target Pair
Affinity DataIC50: 2.20nMAssay Description:In vitro inhibitory activity against enkephalinase enzyme from rat.More data for this Ligand-Target Pair
Affinity DataIC50: 2.40nMAssay Description:In vitro inhibitory activity against enkephalinase enzyme from rat.More data for this Ligand-Target Pair
Affinity DataIC50: 2.5nMAssay Description:In vitro inhibitory activity against enkephalinase enzyme from rat.More data for this Ligand-Target Pair
Affinity DataIC50: 2.60nMAssay Description:The compound was tested in vitro for its inhibitory activity against Enkephalinase enzymeMore data for this Ligand-Target Pair
Affinity DataIC50: 3.10nMAssay Description:In vitro inhibitory activity against enkephalinase enzyme from rat.More data for this Ligand-Target Pair
Affinity DataIC50: 3.20nMAssay Description:In vitro inhibitory activity against enkephalinase enzyme from rat.More data for this Ligand-Target Pair
Affinity DataIC50: 3.5nMAssay Description:In vitro inhibitory activity against enkephalinase enzyme from rat.More data for this Ligand-Target Pair
Affinity DataIC50: 4.40nMAssay Description:In vitro inhibitory activity against enkephalinase enzyme from rat.More data for this Ligand-Target Pair
Affinity DataIC50: 4.40nMAssay Description:In vitro inhibitory activity against enkephalinase enzyme from rat.More data for this Ligand-Target Pair
Affinity DataIC50: 5nMAssay Description:In vitro inhibitory activity against enkephalinase enzyme from rat.More data for this Ligand-Target Pair
Affinity DataIC50: 5.20nMAssay Description:The compound was tested in vitro for its inhibitory activity against Enkephalinase enzymeMore data for this Ligand-Target Pair
Affinity DataIC50: 5.40nMAssay Description:In vitro inhibitory activity against enkephalinase enzyme from rat.More data for this Ligand-Target Pair
Affinity DataIC50: 7.40nMAssay Description:The compound was tested in vitro for its inhibitory activity against Enkephalinase enzymeMore data for this Ligand-Target Pair
Affinity DataIC50: 8.40nMAssay Description:In vitro inhibitory activity against enkephalinase enzyme from rat.More data for this Ligand-Target Pair
Affinity DataIC50: 11nMAssay Description:In vitro inhibitory activity against enkephalinase enzyme from rat.More data for this Ligand-Target Pair
Affinity DataIC50: 11nMAssay Description:In vitro inhibitory activity against enkephalinase enzyme from rat.More data for this Ligand-Target Pair
Affinity DataIC50: 12nMAssay Description:In vitro inhibitory activity against enkephalinase enzyme from rat.More data for this Ligand-Target Pair
Affinity DataIC50: 14nMAssay Description:The compound was tested in vitro for its inhibitory activity against Enkephalinase enzymeMore data for this Ligand-Target Pair
Affinity DataIC50: 14nMAssay Description:In vitro inhibitory activity against enkephalinase enzyme from rat.More data for this Ligand-Target Pair
Affinity DataIC50: 17nMAssay Description:The compound was tested in vitro for its inhibitory activity against Enkephalinase enzymeMore data for this Ligand-Target Pair
Affinity DataIC50: 31nMAssay Description:In vitro inhibitory activity against enkephalinase enzyme from rat.More data for this Ligand-Target Pair
Affinity DataIC50: 33nMAssay Description:In vitro inhibitory activity against enkephalinase enzyme from rat.More data for this Ligand-Target Pair
Affinity DataIC50: 34nMAssay Description:In vitro inhibitory activity against enkephalinase enzyme from rat.More data for this Ligand-Target Pair
Affinity DataIC50: 37nMAssay Description:In vitro inhibitory activity against enkephalinase enzyme from rat.More data for this Ligand-Target Pair
Affinity DataIC50: 52nMAssay Description:In vitro inhibitory activity against enkephalinase enzyme from rat.More data for this Ligand-Target Pair
Affinity DataIC50: 110nMAssay Description:In vitro inhibitory activity against enkephalinase enzyme from rat.More data for this Ligand-Target Pair
Affinity DataIC50: 140nMAssay Description:In vitro inhibitory activity against enkephalinase enzyme from rat.More data for this Ligand-Target Pair
Affinity DataIC50: 150nMAssay Description:In vitro inhibitory activity against enkephalinase enzyme from rat.More data for this Ligand-Target Pair
Affinity DataIC50: 250nMAssay Description:In vitro inhibitory activity against enkephalinase enzyme from rat.More data for this Ligand-Target Pair
Affinity DataIC50: 420nMAssay Description:In vitro inhibitory activity against angiotensin I converting enzyme (ACE) from rabbit lungMore data for this Ligand-Target Pair
Affinity DataIC50: 490nMAssay Description:In vitro inhibitory activity against enkephalinase enzyme from rat.More data for this Ligand-Target Pair
Affinity DataIC50: 4.20E+3nMAssay Description:In vitro inhibitory activity against enkephalinase enzyme from rat.More data for this Ligand-Target Pair
Target1,3-beta-D-glucan synthase catalytic subunit(Candida albicans)
Inner Mongolia University
Curated by ChEMBL
Inner Mongolia University
Curated by ChEMBL
Affinity DataIC50: 8.00E+3nMAssay Description:Inhibition of Candida albicans 1,3 beta-D-glucan synthaseMore data for this Ligand-Target Pair
Affinity DataIC50: 1.20E+4nMAssay Description:In vitro inhibitory activity against Angiotensin I converting enzyme from rabbit lungMore data for this Ligand-Target Pair
Target1,3-beta-D-glucan synthase catalytic subunit(Candida albicans)
Inner Mongolia University
Curated by ChEMBL
Inner Mongolia University
Curated by ChEMBL
Affinity DataIC50: 1.50E+4nMAssay Description:Inhibition of Candida albicans 1,3 beta-D-glucan synthaseMore data for this Ligand-Target Pair
Target1,3-beta-D-glucan synthase catalytic subunit(Candida albicans)
Inner Mongolia University
Curated by ChEMBL
Inner Mongolia University
Curated by ChEMBL
Affinity DataIC50: 2.20E+4nMAssay Description:Inhibition of Candida albicans 1,3 beta-D-glucan synthaseMore data for this Ligand-Target Pair
Affinity DataIC50: 3.70E+4nMAssay Description:In vitro inhibitory activity against angiotensin I converting enzyme (ACE) from rabbit lungMore data for this Ligand-Target Pair
Target1,3-beta-D-glucan synthase catalytic subunit(Candida albicans)
Inner Mongolia University
Curated by ChEMBL
Inner Mongolia University
Curated by ChEMBL
Affinity DataIC50: 3.70E+4nMAssay Description:Inhibition of Candida albicans 1,3 beta-D-glucan synthaseMore data for this Ligand-Target Pair