Affinity DataKi: 0.100nMAssay Description:Antagonist activity at human Adenosine receptor A2a assessed as inhibition of cAMP productionMore data for this Ligand-Target Pair
Affinity DataKi: 0.300nMAssay Description:Antagonist activity at human Adenosine receptor A2a assessed as inhibition of cAMP productionMore data for this Ligand-Target Pair
Affinity DataKi: 0.5nMAssay Description:Antagonist activity at human Adenosine receptor A1 assessed as inhibition of cAMP productionMore data for this Ligand-Target Pair
Affinity DataKi: 0.5nMAssay Description:Antagonist activity at human Adenosine receptor A2a assessed as inhibition of cAMP productionMore data for this Ligand-Target Pair
Affinity DataKi: 0.700nMAssay Description:Antagonist activity at human Adenosine receptor A2a assessed as inhibition of cAMP productionMore data for this Ligand-Target Pair
Affinity DataKi: 1.30nMAssay Description:Antagonist activity at human Adenosine receptor A2a assessed as inhibition of cAMP productionMore data for this Ligand-Target Pair
Affinity DataKi: 1.40nMAssay Description:Antagonist activity at human Adenosine receptor A2a assessed as inhibition of cAMP productionMore data for this Ligand-Target Pair
Affinity DataKi: 1.60nMAssay Description:Antagonist activity at human Adenosine receptor A2a assessed as inhibition of cAMP productionMore data for this Ligand-Target Pair
Affinity DataKi: 1.80nMAssay Description:Antagonist activity at human Adenosine receptor A1 assessed as inhibition of cAMP productionMore data for this Ligand-Target Pair
Affinity DataKi: 1.80nMAssay Description:Antagonist activity at human Adenosine receptor A2a assessed as inhibition of cAMP productionMore data for this Ligand-Target Pair
Affinity DataKi: 2.40nMAssay Description:Antagonist activity at human Adenosine receptor A1 assessed as inhibition of cAMP productionMore data for this Ligand-Target Pair
Affinity DataKi: 2.5nMAssay Description:Antagonist activity at human Adenosine receptor A1 assessed as inhibition of cAMP productionMore data for this Ligand-Target Pair
Affinity DataKi: 3.10nMAssay Description:Antagonist activity at human Adenosine receptor A2a assessed as inhibition of cAMP productionMore data for this Ligand-Target Pair
Affinity DataKi: 4.10nMAssay Description:Antagonist activity at human Adenosine receptor A2a assessed as inhibition of cAMP productionMore data for this Ligand-Target Pair
Affinity DataKi: 5.20nMAssay Description:Antagonist activity at human Adenosine receptor A1 assessed as inhibition of cAMP productionMore data for this Ligand-Target Pair
Affinity DataKi: 6nMAssay Description:Antagonist activity at human Adenosine receptor A1 assessed as inhibition of cAMP productionMore data for this Ligand-Target Pair
Affinity DataKi: 6.5nMAssay Description:Antagonist activity at human Adenosine receptor A2a assessed as inhibition of cAMP productionMore data for this Ligand-Target Pair
Affinity DataKi: 8.20nMAssay Description:Antagonist activity at human Adenosine receptor A2a assessed as inhibition of cAMP productionMore data for this Ligand-Target Pair
Affinity DataKi: 8.40nMAssay Description:Binding affinity to wild-type androgen receptor in human LNCaP cells assessed as inhibition constant incubated for 24 hrs by Cheng-Prusoff equation a...More data for this Ligand-Target Pair
Affinity DataKi: 9nMAssay Description:Antagonist activity at human Adenosine receptor A1 assessed as inhibition of cAMP productionMore data for this Ligand-Target Pair
Affinity DataKi: 13.1nMAssay Description:Antagonist activity at human Adenosine receptor A2a assessed as inhibition of cAMP productionMore data for this Ligand-Target Pair
Affinity DataKi: 17nMAssay Description:Binding affinity to wild-type androgen receptor in human LNCaP cells assessed as inhibition constant incubated for 24 hrs by Cheng-Prusoff equation a...More data for this Ligand-Target Pair
Affinity DataKi: 17nMAssay Description:Antagonist activity at human Adenosine receptor A1 assessed as inhibition of cAMP productionMore data for this Ligand-Target Pair
Affinity DataKi: 29.3nMAssay Description:Antagonist activity at human Adenosine receptor A1 assessed as inhibition of cAMP productionMore data for this Ligand-Target Pair
Affinity DataKi: 32nMAssay Description:In vitro inhibitory activity against tryptaseMore data for this Ligand-Target Pair
Affinity DataKi: 37.3nMAssay Description:Antagonist activity at human Adenosine receptor A1 assessed as inhibition of cAMP productionMore data for this Ligand-Target Pair
Affinity DataKi: 41nMAssay Description:In vitro inhibitory activity against tryptaseMore data for this Ligand-Target Pair
Affinity DataKi: 41nMAssay Description:In vitro inhibitory activity against tryptaseMore data for this Ligand-Target Pair
Affinity DataKi: 48.2nMAssay Description:Antagonist activity at human Adenosine receptor A1 assessed as inhibition of cAMP productionMore data for this Ligand-Target Pair
Affinity DataKi: 49nMAssay Description:In vitro inhibitory activity against tryptaseMore data for this Ligand-Target Pair
Affinity DataKi: 57nMAssay Description:In vitro inhibitory activity against tryptaseMore data for this Ligand-Target Pair
Affinity DataKi: 58.4nMAssay Description:Antagonist activity at human Adenosine receptor A1 assessed as inhibition of cAMP productionMore data for this Ligand-Target Pair
Affinity DataKi: 61nMAssay Description:In vitro inhibitory activity against tryptaseMore data for this Ligand-Target Pair
Affinity DataKi: 68nMAssay Description:Binding affinity of compound towards Factor XaMore data for this Ligand-Target Pair
Affinity DataKi: 101nMAssay Description:In vitro inhibitory activity against tryptaseMore data for this Ligand-Target Pair
Affinity DataKi: 116nMAssay Description:In vitro inhibitory activity against tryptaseMore data for this Ligand-Target Pair
Affinity DataKi: 124nMAssay Description:In vitro inhibitory activity against tryptaseMore data for this Ligand-Target Pair
Affinity DataKi: 125nMAssay Description:In vitro inhibitory activity against tryptaseMore data for this Ligand-Target Pair
Affinity DataKi: 128nMAssay Description:In vitro inhibitory activity against tryptaseMore data for this Ligand-Target Pair
Affinity DataKi: 140nMAssay Description:In vitro inhibitory activity against tryptaseMore data for this Ligand-Target Pair
Affinity DataKi: 141nMAssay Description:In vitro inhibitory activity against tryptaseMore data for this Ligand-Target Pair
Affinity DataKi: 155nMAssay Description:In vitro inhibitory activity against tryptaseMore data for this Ligand-Target Pair
Affinity DataKi: 162nMAssay Description:In vitro inhibitory activity against tryptaseMore data for this Ligand-Target Pair
Affinity DataKi: 185nMAssay Description:In vitro inhibitory activity against tryptaseMore data for this Ligand-Target Pair
Affinity DataKi: 197nMAssay Description:In vitro inhibitory activity against tryptaseMore data for this Ligand-Target Pair
Affinity DataKi: 223nMAssay Description:Antagonist activity at human Adenosine receptor A1 assessed as inhibition of cAMP productionMore data for this Ligand-Target Pair
Affinity DataKi: 240nMAssay Description:In vitro inhibitory activity against tryptaseMore data for this Ligand-Target Pair
Affinity DataKi: 246nMAssay Description:In vitro inhibitory activity against tryptaseMore data for this Ligand-Target Pair
Affinity DataKi: 290nMAssay Description:In vitro inhibitory activity against tryptaseMore data for this Ligand-Target Pair
Affinity DataKi: 310nMAssay Description:In vitro inhibitory activity against tryptaseMore data for this Ligand-Target Pair