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Found 361 with Last Name = 'lin' and Initial = 'yl'
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
National Research Institute Of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50208945(CHEMBL224024 | N6-(4-hydroxybenzyl)adenine ribosid...)
Affinity DataKi:  2.62E+3nMAssay Description:Binding affinity to adenosine A2A receptor in rat brain striatumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
National Research Institute Of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50208946(CHEMBL224380 | bis(4-hydroxybenzyl)sulfide)
Affinity DataKi:  2.41E+4nMAssay Description:Binding affinity to adenosine A2A receptor in rat brain striatumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
Medical And Pharmaceutical Industry Technology And Development Center

Curated by ChEMBL
LigandPNGBDBM35229(3-(10,11-dihydro-5H-dibenzo[b,f]azepin-5-yl)-N-met...)
Affinity DataIC50:  0.930nMAssay Description:Displacement of [125I]RTI-55 from human NET expressed in MDCK cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetPeptidyl-prolyl cis-trans isomerase A(Homo sapiens (Human))
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50181474(1-(3-benzyloxy-pyridin-2-yl)-3-(4-nitro-phenyl)-ur...)
Affinity DataIC50:  14nMAssay Description:Inhibition of isomerase activity of Cyclophilin AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase A(Homo sapiens (Human))
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50181489(4-[3-(3-benzyloxy-pyridin-2-yl)-ureido]-benzoic ac...)
Affinity DataIC50:  20nMAssay Description:Inhibition of isomerase activity of Cyclophilin AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target4-hydroxyphenylpyruvate dioxygenase(Sus scrofa)
Tunghai Christian University

Curated by ChEMBL
LigandPNGBDBM50089165(CHEMBL23622 | Cyclopropanecarboxylic acid 3-oxo-cy...)
Affinity DataIC50:  30nMAssay Description:In vitro inhibitory activity of the compound against HPPD(4-hydroxyphenylpyruvate Dioxygenase) from pig liver using enol borate assay methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target4-hydroxyphenylpyruvate dioxygenase(Sus scrofa)
Tunghai Christian University

Curated by ChEMBL
LigandPNGBDBM50075319(2-{HYDROXY[2-NITRO-4-(TRIFLUOROMETHYL)PHENYL]METHY...)
Affinity DataIC50:  40nMAssay Description:In vitro inhibitory activity of the compound against HPPD(4-hydroxyphenylpyruvate Dioxygenase) from pig liver using enol borate assay methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target4-hydroxyphenylpyruvate dioxygenase(Sus scrofa)
Tunghai Christian University

Curated by ChEMBL
LigandPNGBDBM50088804(1,3-Cyclohexanedione, 2-(2-nitro-4-(trifluoromethy...)
Affinity DataIC50:  40nMAssay Description:Inhibition of 4-hydroxyphenylpyruvate dioxygenase of purified pig liver by enol-borate methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase A(Homo sapiens (Human))
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50181493(4-[3-(3-benzyloxy-pyridin-2-yl)-ureido]-benzenesul...)
Affinity DataIC50:  60nMAssay Description:Inhibition of isomerase activity of Cyclophilin AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase p300(Homo sapiens (Human))
Avera Institute For Human Genetics

Curated by ChEMBL
LigandPNGBDBM50467836(CHEMBL4282264)
Affinity DataIC50:  60nMAssay Description:Inhibition of p300 HAT domain (unknown origin) using Biotin-C6-GRGKGGKGLGKGGAK as substrate pretreated with enzyme for 30 mins followed by incubation...More data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase A(Homo sapiens (Human))
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50181475(1-(3-benzyloxy-pyridin-2-yl)-3-(3-nitro-phenyl)-ur...)
Affinity DataIC50:  60nMAssay Description:Inhibition of isomerase activity of Cyclophilin AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase A(Homo sapiens (Human))
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50181496(3-[3-(3-benzyloxy-pyridin-2-yl)-ureido]-benzoic ac...)
Affinity DataIC50:  71nMAssay Description:Inhibition of isomerase activity of Cyclophilin AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target4-hydroxyphenylpyruvate dioxygenase(Sus scrofa)
Tunghai Christian University

Curated by ChEMBL
LigandPNGBDBM50089168(CHEMBL26162 | Propionic acid 3-oxo-cyclohex-1-enyl...)
Affinity DataIC50:  110nMAssay Description:In vitro inhibitory activity of the compound against HPPD(4-hydroxyphenylpyruvate Dioxygenase) from pig liver using enol borate assay methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(West Nile virus)
Baylor College Of Medicine

Curated by ChEMBL
LigandPNGBDBM50567466(CHEMBL4862682)
Affinity DataIC50:  120nMAssay Description:Inhibition West Nile virus NS3B/NS3 protease using 7-amino-4-methylcoumarin as substrate by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetNonstructural protein 3(Zika virus)
Baylor College Of Medicine

Curated by ChEMBL
LigandPNGBDBM50567473(CHEMBL4872757)
Affinity DataIC50:  130nMAssay Description:Inhibition Zika virus NS3B (47 to 95 residues)/NS3 (1 to 170 residues) protease expressed in Escherichia coli BL21 using 7-amino-4-methylcoumarin as ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase A(Homo sapiens (Human))
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50181491(4-[3-(3-benzyloxy-pyridin-2-yl)-ureido]-benzoic ac...)
Affinity DataIC50:  140nMAssay Description:Inhibition of isomerase activity of Cyclophilin AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target4-hydroxyphenylpyruvate dioxygenase(Sus scrofa)
Tunghai Christian University

Curated by ChEMBL
LigandPNGBDBM50088793(2-(2-Nitro-benzoyl)-cyclohexane-1,3-dione | CHEMBL...)
Affinity DataIC50:  160nMAssay Description:Inhibition of 4-hydroxyphenylpyruvate dioxygenase of purified pig liver by enol-borate methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNonstructural protein 3(Zika virus)
Baylor College Of Medicine

Curated by ChEMBL
LigandPNGBDBM50567516(CHEMBL4865964)
Affinity DataIC50:  200nMAssay Description:Inhibition Zika virus NS3B (47 to 95 residues)/NS3 (1 to 170 residues) protease expressed in Escherichia coli BL21 using 7-amino-4-methylcoumarin as ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Dengue virus 2)
Baylor College Of Medicine

Curated by ChEMBL
LigandPNGBDBM50567466(CHEMBL4862682)
Affinity DataIC50:  210nMAssay Description:Inhibition Dengue serotype-2 NS3B/NS3 protease using 7-amino-4-methylcoumarin as substrate by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetNonstructural protein 3(Zika virus)
Baylor College Of Medicine

Curated by ChEMBL
LigandPNGBDBM50567535(CHEMBL4861948)
Affinity DataIC50:  240nMAssay Description:Inhibition Zika virus NS3B (47 to 95 residues)/NS3 (1 to 170 residues) protease expressed in Escherichia coli BL21 using 7-amino-4-methylcoumarin as ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target4-hydroxyphenylpyruvate dioxygenase(Sus scrofa)
Tunghai Christian University

Curated by ChEMBL
LigandPNGBDBM50088799(2-(2-Trifluoromethyl-benzoyl)-cyclohexane-1,3-dion...)
Affinity DataIC50:  250nMAssay Description:Inhibition of 4-hydroxyphenylpyruvate dioxygenase of purified pig liver by enol-borate methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Dengue virus 2)
Baylor College Of Medicine

Curated by ChEMBL
LigandPNGBDBM50567470(CHEMBL4862353)
Affinity DataIC50:  290nMAssay Description:Inhibition Dengue serotype-2 NS3B/NS3 protease using 7-amino-4-methylcoumarin as substrate by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetPeptidyl-prolyl cis-trans isomerase A(Homo sapiens (Human))
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50181483(1-(3-benzyloxypyridin-2-yl)-3-(3-trifluoromethylph...)
Affinity DataIC50:  303nMAssay Description:Inhibition of isomerase activity of Cyclophilin AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase A(Homo sapiens (Human))
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50181495(1-(3-benzyloxypyridin-2-yl)-3-(3-chlorophenyl)-ure...)
Affinity DataIC50:  316nMAssay Description:Inhibition of isomerase activity of Cyclophilin AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNonstructural protein 3(Zika virus)
Baylor College Of Medicine

Curated by ChEMBL
LigandPNGBDBM50579310(CHEMBL4862793)
Affinity DataIC50:  320nMAssay Description:Inhibition of Zika virus recombinant NS2B (47 to 95 residues)/NS3 (1 to 177 residues) protease expressed in Escherichia coli BL21 using Bz-Nle-Lys-Ly...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase A(Homo sapiens (Human))
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50181492(4-[3-(3-benzyloxy-pyridin-2-yl)-ureido]-N-methyl-b...)
Affinity DataIC50:  320nMAssay Description:Inhibition of isomerase activity of Cyclophilin AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNonstructural protein 3(Zika virus)
Baylor College Of Medicine

Curated by ChEMBL
LigandPNGBDBM50567493(CHEMBL4872312)
Affinity DataIC50:  320nMAssay Description:Inhibition Zika virus NS3B (47 to 95 residues)/NS3 (1 to 170 residues) protease expressed in Escherichia coli BL21 using 7-amino-4-methylcoumarin as ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase A(Homo sapiens (Human))
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50181479(3-[3-(3-benzyloxy-pyridin-2-yl)-ureido]-benzamide ...)
Affinity DataIC50:  361nMAssay Description:Inhibition of isomerase activity of Cyclophilin AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNonstructural protein 3(Zika virus)
Baylor College Of Medicine

Curated by ChEMBL
LigandPNGBDBM50579311(CHEMBL4865004)
Affinity DataIC50:  370nMAssay Description:Inhibition of Zika virus recombinant NS2B (47 to 95 residues)/NS3 (1 to 177 residues) protease expressed in Escherichia coli BL21 using Bz-Nle-Lys-Ly...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNonstructural protein 3(Zika virus)
Baylor College Of Medicine

Curated by ChEMBL
LigandPNGBDBM50567484(CHEMBL4861102)
Affinity DataIC50:  390nMAssay Description:Inhibition Zika virus NS3B (47 to 95 residues)/NS3 (1 to 170 residues) protease expressed in Escherichia coli BL21 using 7-amino-4-methylcoumarin as ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNonstructural protein 3(Zika virus)
Baylor College Of Medicine

Curated by ChEMBL
LigandPNGBDBM50579273(CHEMBL4858884)
Affinity DataIC50:  390nMAssay Description:Inhibition of Zika virus recombinant NS2B (47 to 95 residues)/NS3 (1 to 177 residues) protease expressed in Escherichia coli BL21 using Bz-Nle-Lys-Ly...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNonstructural protein 3(Zika virus)
Baylor College Of Medicine

Curated by ChEMBL
LigandPNGBDBM50567470(CHEMBL4862353)
Affinity DataIC50:  400nMAssay Description:Inhibition Zika virus NS3B (47 to 95 residues)/NS3 (1 to 170 residues) protease expressed in Escherichia coli BL21 using 7-amino-4-methylcoumarin as ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetNonstructural protein 3(Zika virus)
Baylor College Of Medicine

Curated by ChEMBL
LigandPNGBDBM50579316(CHEMBL4852919)
Affinity DataIC50:  450nMAssay Description:Inhibition of Zika virus recombinant NS2B (47 to 95 residues)/NS3 (1 to 177 residues) protease expressed in Escherichia coli BL21 using Bz-Nle-Lys-Ly...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase A(Homo sapiens (Human))
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50181494(1-(3-benzyloxy-pyridin-2-yl)-3-(2,4-difluoro-pheny...)
Affinity DataIC50:  458nMAssay Description:Inhibition of isomerase activity of Cyclophilin AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase A(Homo sapiens (Human))
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50181487(1-(3-benzyloxy-pyridin-2-yl)-3-(4-trifluoromethyl-...)
Affinity DataIC50:  499nMAssay Description:Inhibition of isomerase activity of Cyclophilin AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target4-hydroxyphenylpyruvate dioxygenase(Sus scrofa)
Tunghai Christian University

Curated by ChEMBL
LigandPNGBDBM50088803(2-(2-Chloro-benzoyl)-cyclohexane-1,3-dione | CHEMB...)
Affinity DataIC50:  500nMAssay Description:Inhibition of 4-hydroxyphenylpyruvate dioxygenase of purified pig liver by enol-borate methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase p300(Homo sapiens (Human))
Avera Institute For Human Genetics

Curated by ChEMBL
LigandPNGBDBM50255529(Ac-Lys(CoA)-NH2 | CHEMBL505121)
Affinity DataIC50:  500nMAssay Description:Inhibition of N-terminal His-tagged human recombinant p300 catalytic domain (1284-1673 residues) using histone H4-8 peptide and [14C]acetyl CoA as su...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target4-hydroxyphenylpyruvate dioxygenase(Sus scrofa)
Tunghai Christian University

Curated by ChEMBL
LigandPNGBDBM50114880(3-Hydroxy-4-phenyl-5H-furan-2-one | CHEMBL295478)
Affinity DataIC50:  500nMAssay Description:In vitro inhibition against of 4-Hydroxyphenylpyruvate dioxygenase (4-HPPD) from pig liver by the enol borate methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNonstructural protein 3(Zika virus)
Baylor College Of Medicine

Curated by ChEMBL
LigandPNGBDBM50567477(CHEMBL4852716)
Affinity DataIC50:  510nMAssay Description:Inhibition Zika virus NS3B (47 to 95 residues)/NS3 (1 to 170 residues) protease expressed in Escherichia coli BL21 using 7-amino-4-methylcoumarin as ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGenome polyprotein(West Nile virus)
Baylor College Of Medicine

Curated by ChEMBL
LigandPNGBDBM50567470(CHEMBL4862353)
Affinity DataIC50:  510nMAssay Description:Inhibition West Nile virus NS3B/NS3 protease using 7-amino-4-methylcoumarin as substrate by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetNonstructural protein 3(Zika virus)
Baylor College Of Medicine

Curated by ChEMBL
LigandPNGBDBM50567474(CHEMBL4867031)
Affinity DataIC50:  520nMAssay Description:Inhibition Zika virus NS3B (47 to 95 residues)/NS3 (1 to 170 residues) protease expressed in Escherichia coli BL21 using 7-amino-4-methylcoumarin as ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase A(Homo sapiens (Human))
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50181481(CHEMBL199550 | {3-[3-(3-benzyloxy-pyridin-2-yl)-ur...)
Affinity DataIC50:  528nMAssay Description:Inhibition of isomerase activity of Cyclophilin AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target4-hydroxyphenylpyruvate dioxygenase(Sus scrofa)
Tunghai Christian University

Curated by ChEMBL
LigandPNGBDBM50088795(2-(2-Bromo-benzoyl)-cyclohexane-1,3-dione | CHEMBL...)
Affinity DataIC50:  560nMAssay Description:Inhibition of 4-hydroxyphenylpyruvate dioxygenase of purified pig liver by enol-borate methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNonstructural protein 3(Zika virus)
Baylor College Of Medicine

Curated by ChEMBL
LigandPNGBDBM50567550(CHEMBL4849574)
Affinity DataIC50:  590nMAssay Description:Inhibition Zika virus NS3B (47 to 95 residues)/NS3 (1 to 170 residues) protease expressed in Escherichia coli BL21 using 7-amino-4-methylcoumarin as ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Dengue virus 2)
Baylor College Of Medicine

Curated by ChEMBL
LigandPNGBDBM50567467(CHEMBL4850391)
Affinity DataIC50:  590nMAssay Description:Inhibition Dengue serotype-2 NS3B/NS3 protease using 7-amino-4-methylcoumarin as substrate by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetPeptidyl-prolyl cis-trans isomerase A(Homo sapiens (Human))
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50181478(1-(3-benzyloxy-pyridin-2-yl)-3-(2-chloro-phenyl)-u...)
Affinity DataIC50:  592nMAssay Description:Inhibition of isomerase activity of Cyclophilin AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNonstructural protein 3(Zika virus)
Baylor College Of Medicine

Curated by ChEMBL
LigandPNGBDBM50579317(CHEMBL4868723)
Affinity DataIC50:  600nMAssay Description:Inhibition of Zika virus recombinant NS2B (47 to 95 residues)/NS3 (1 to 177 residues) protease expressed in Escherichia coli BL21 using Bz-Nle-Lys-Ly...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNonstructural protein 3(Zika virus)
Baylor College Of Medicine

Curated by ChEMBL
LigandPNGBDBM50567480(CHEMBL4862454)
Affinity DataIC50:  620nMAssay Description:Inhibition Zika virus NS3B (47 to 95 residues)/NS3 (1 to 170 residues) protease expressed in Escherichia coli BL21 using 7-amino-4-methylcoumarin as ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase p300(Homo sapiens (Human))
Avera Institute For Human Genetics

Curated by ChEMBL
LigandPNGBDBM50511789(CHEMBL4474132)
Affinity DataIC50:  620nMAssay Description:Inhibition of recombinant human GST-tagged p300 HAT domain (1195 to 1673 residues) expressed in Escherichia coli BL21 codon plus cells using Histone ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNonstructural protein 3(Zika virus)
Baylor College Of Medicine

Curated by ChEMBL
LigandPNGBDBM50579275(CHEMBL4870701)
Affinity DataIC50:  630nMAssay Description:Inhibition of Zika virus recombinant NS2B (47 to 95 residues)/NS3 (1 to 177 residues) protease expressed in Escherichia coli BL21 using Bz-Nle-Lys-Ly...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
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