Affinity DataKi: 15nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 1.10E+7nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in rat membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 1.5nMAssay Description:Inhibition of wild type EGFR (unknown origin) by bioluminescent ADP-glo kinase assayMore data for this Ligand-Target Pair
Affinity DataIC50: 2.5nMAssay Description:Inhibition of wild type EGFR (unknown origin) by bioluminescent ADP-glo kinase assayMore data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:Inhibition of EGFR (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Inhibition of wild type EGFR (unknown origin) by bioluminescent ADP-glo kinase assayMore data for this Ligand-Target Pair
Affinity DataIC50: 23nMAssay Description:Inhibition of wild type EGFR (unknown origin) by bioluminescent ADP-glo kinase assayMore data for this Ligand-Target Pair
Affinity DataIC50: 30nMAssay Description:Inhibition of wild type EGFR (unknown origin) by bioluminescent ADP-glo kinase assayMore data for this Ligand-Target Pair
Affinity DataIC50: 52nMAssay Description:Inhibition of wild type EGFR (unknown origin) by bioluminescent ADP-glo kinase assayMore data for this Ligand-Target Pair
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Universit£
Curated by ChEMBL
Universit£
Curated by ChEMBL
Affinity DataIC50: 80nMAssay Description:Inhibition of VEGFR2 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 100nMAssay Description:Inhibition of EGFR (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 140nMAssay Description:Inhibition of wild type EGFR (unknown origin) by bioluminescent ADP-glo kinase assayMore data for this Ligand-Target Pair
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Universit£
Curated by ChEMBL
Universit£
Curated by ChEMBL
Affinity DataIC50: 140nMAssay Description:Inhibition of VEGFR2 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 273nMAssay Description:Inhibition of wild type EGFR (unknown origin) by bioluminescent ADP-glo kinase assayMore data for this Ligand-Target Pair
Affinity DataIC50: 326nMAssay Description:Inhibition of wild type EGFR (unknown origin) by bioluminescent ADP-glo kinase assayMore data for this Ligand-Target Pair
Affinity DataIC50: 710nMAssay Description:Inhibition of bovine brain tubulin polymerization after 20 minsMore data for this Ligand-Target Pair
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Universit£
Curated by ChEMBL
Universit£
Curated by ChEMBL
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of wild type VEGFR2 (unknown origin) by bioluminescent ADP-glo kinase assayMore data for this Ligand-Target Pair
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Universit£
Curated by ChEMBL
Universit£
Curated by ChEMBL
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of wild type VEGFR2 (unknown origin) by bioluminescent ADP-glo kinase assayMore data for this Ligand-Target Pair
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Universit£
Curated by ChEMBL
Universit£
Curated by ChEMBL
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of wild type VEGFR2 (unknown origin) by bioluminescent ADP-glo kinase assayMore data for this Ligand-Target Pair
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Universit£
Curated by ChEMBL
Universit£
Curated by ChEMBL
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of wild type VEGFR2 (unknown origin) by bioluminescent ADP-glo kinase assayMore data for this Ligand-Target Pair
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Universit£
Curated by ChEMBL
Universit£
Curated by ChEMBL
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of wild type VEGFR2 (unknown origin) by bioluminescent ADP-glo kinase assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of bovine brain tubulin polymerization after 20 minsMore data for this Ligand-Target Pair
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibition of bovine brain tubulin polymerization after 20 minsMore data for this Ligand-Target Pair
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibition of bovine brain tubulin polymerization after 20 minsMore data for this Ligand-Target Pair
Affinity DataIC50: 2.80E+3nMAssay Description:Inhibition of bovine brain tubulin polymerization after 20 minsMore data for this Ligand-Target Pair
Affinity DataIC50: 3.30E+3nMAssay Description:Inhibition of bovine brain tubulin polymerization after 20 minsMore data for this Ligand-Target Pair
TargetCholine kinase alpha(Homo sapiens (Human))
Campus Cartuja S/N. University Of Granada
Curated by ChEMBL
Campus Cartuja S/N. University Of Granada
Curated by ChEMBL
Affinity DataIC50: 6.74E+3nMAssay Description:Inhibition of human CKalpha1 assessed as reduction in 14C incorporation from [methyl-14C]choline to phosphatidylcholine using [methyl-14C]choline as ...More data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of bovine brain tubulin polymerization after 20 minsMore data for this Ligand-Target Pair
TargetCholine kinase alpha(Homo sapiens (Human))
Campus Cartuja S/N. University Of Granada
Curated by ChEMBL
Campus Cartuja S/N. University Of Granada
Curated by ChEMBL
Affinity DataIC50: 1.26E+4nMAssay Description:Inhibition of human CKalpha1 assessed as reduction in 14C incorporation from [methyl-14C]choline to phosphatidylcholine using [methyl-14C]choline as ...More data for this Ligand-Target Pair
Affinity DataIC50: 1.80E+4nMAssay Description:Inhibition of bovine brain tubulin polymerization after 20 minsMore data for this Ligand-Target Pair
TargetCholine kinase alpha(Homo sapiens (Human))
Campus Cartuja S/N. University Of Granada
Curated by ChEMBL
Campus Cartuja S/N. University Of Granada
Curated by ChEMBL
Affinity DataKd: 2.40E+4nMAssay Description:Binding affinity to human CKalpha1 assessed as dissociation constant by spectroflurometryMore data for this Ligand-Target Pair
TargetCholine kinase alpha(Homo sapiens (Human))
Campus Cartuja S/N. University Of Granada
Curated by ChEMBL
Campus Cartuja S/N. University Of Granada
Curated by ChEMBL
Affinity DataKd: 400nMAssay Description:Binding affinity to human CKalpha1 assessed as dissociation constant by spectroflurometryMore data for this Ligand-Target Pair
TargetCholine kinase alpha(Homo sapiens (Human))
Campus Cartuja S/N. University Of Granada
Curated by ChEMBL
Campus Cartuja S/N. University Of Granada
Curated by ChEMBL
Affinity DataKd: 890nMAssay Description:Binding affinity to human CKalpha1 assessed as dissociation constant by spectroflurometryMore data for this Ligand-Target Pair
TargetCholine kinase alpha(Homo sapiens (Human))
Campus Cartuja S/N. University Of Granada
Curated by ChEMBL
Campus Cartuja S/N. University Of Granada
Curated by ChEMBL
Affinity DataKd: 1.70E+3nMAssay Description:Binding affinity to human CKalpha1 assessed as dissociation constant by spectroflurometryMore data for this Ligand-Target Pair
TargetCholine kinase alpha(Homo sapiens (Human))
Campus Cartuja S/N. University Of Granada
Curated by ChEMBL
Campus Cartuja S/N. University Of Granada
Curated by ChEMBL
Affinity DataKd: 670nMAssay Description:Binding affinity to human CKalpha1 assessed as dissociation constant by spectroflurometryMore data for this Ligand-Target Pair
TargetCholine kinase alpha(Homo sapiens (Human))
Campus Cartuja S/N. University Of Granada
Curated by ChEMBL
Campus Cartuja S/N. University Of Granada
Curated by ChEMBL
Affinity DataKd: 370nMAssay Description:Binding affinity to human CKalpha1 assessed as dissociation constant by spectroflurometryMore data for this Ligand-Target Pair
TargetCholine kinase alpha(Homo sapiens (Human))
Campus Cartuja S/N. University Of Granada
Curated by ChEMBL
Campus Cartuja S/N. University Of Granada
Curated by ChEMBL
Affinity DataKd: 185nMAssay Description:Binding affinity to human CKalpha1 assessed as dissociation constant by spectroflurometryMore data for this Ligand-Target Pair
TargetCholine kinase alpha(Homo sapiens (Human))
Campus Cartuja S/N. University Of Granada
Curated by ChEMBL
Campus Cartuja S/N. University Of Granada
Curated by ChEMBL
Affinity DataKd: 3.50E+4nMAssay Description:Binding affinity to human CKalpha1 assessed as dissociation constant by spectroflurometryMore data for this Ligand-Target Pair
TargetCholine kinase alpha(Homo sapiens (Human))
Campus Cartuja S/N. University Of Granada
Curated by ChEMBL
Campus Cartuja S/N. University Of Granada
Curated by ChEMBL
Affinity DataKd: 4.90E+4nMAssay Description:Binding affinity to human CKalpha1 assessed as dissociation constant by spectroflurometryMore data for this Ligand-Target Pair
TargetCholine kinase alpha(Homo sapiens (Human))
Campus Cartuja S/N. University Of Granada
Curated by ChEMBL
Campus Cartuja S/N. University Of Granada
Curated by ChEMBL
Affinity DataKd: 4.50E+4nMAssay Description:Binding affinity to human CKalpha1 assessed as dissociation constant by spectroflurometryMore data for this Ligand-Target Pair
TargetCholine kinase alpha(Homo sapiens (Human))
Campus Cartuja S/N. University Of Granada
Curated by ChEMBL
Campus Cartuja S/N. University Of Granada
Curated by ChEMBL
Affinity DataKd: 8.20E+4nMAssay Description:Binding affinity to human CKalpha1 assessed as dissociation constant by spectroflurometryMore data for this Ligand-Target Pair
TargetCholine/ethanolamine kinase(Homo sapiens (Human))
Campus Cartuja S/N. University Of Granada
Curated by ChEMBL
Campus Cartuja S/N. University Of Granada
Curated by ChEMBL
Affinity DataKd: 3.30E+4nMAssay Description:Binding affinity to human CKbeta assessed as dissociation constant by spectroflurometryMore data for this Ligand-Target Pair
TargetCholine/ethanolamine kinase(Homo sapiens (Human))
Campus Cartuja S/N. University Of Granada
Curated by ChEMBL
Campus Cartuja S/N. University Of Granada
Curated by ChEMBL
Affinity DataKd: 3.60E+4nMAssay Description:Binding affinity to human CKbeta assessed as dissociation constant by spectroflurometryMore data for this Ligand-Target Pair
TargetCholine/ethanolamine kinase(Homo sapiens (Human))
Campus Cartuja S/N. University Of Granada
Curated by ChEMBL
Campus Cartuja S/N. University Of Granada
Curated by ChEMBL
Affinity DataKd: 6.30E+4nMAssay Description:Binding affinity to human CKbeta assessed as dissociation constant by spectroflurometryMore data for this Ligand-Target Pair
TargetCholine/ethanolamine kinase(Homo sapiens (Human))
Campus Cartuja S/N. University Of Granada
Curated by ChEMBL
Campus Cartuja S/N. University Of Granada
Curated by ChEMBL
Affinity DataKd: 2.00E+4nMAssay Description:Binding affinity to human CKbeta assessed as dissociation constant by spectroflurometryMore data for this Ligand-Target Pair
TargetCholine kinase alpha(Homo sapiens (Human))
Campus Cartuja S/N. University Of Granada
Curated by ChEMBL
Campus Cartuja S/N. University Of Granada
Curated by ChEMBL
Affinity DataKd: 1.40E+4nMAssay Description:Binding affinity to human CKalpha1 assessed as dissociation constant by spectroflurometryMore data for this Ligand-Target Pair
Affinity DataKd: 0.75nMAssay Description:Allosteric enhancer activity at human adenosine A1 receptor expressed in CHO cell membranes assessed as [3H]NECA affinity constant at 1 uM (Kd = 0.87...More data for this Ligand-Target Pair
Affinity DataKd: 0.460nMAssay Description:Allosteric enhancer activity at human adenosine A1 receptor expressed in CHO cell membranes assessed as [3H]NECA affinity constant at 1 uM (Kd = 0.87...More data for this Ligand-Target Pair