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Found 21 with Last Name = 'macritchie' and Initial = 'n'
TargetSphingosine kinase 1(Homo sapiens (Human))
The City University Of New York

Curated by ChEMBL
LigandPNGBDBM50443388(CHEMBL3086782 | US9688668, SLR080811)
Affinity DataKi:  1.00E+3nMAssay Description:Inhibition of sphingosine kinase 1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine kinase 1(Homo sapiens (Human))
The City University Of New York

Curated by ChEMBL
LigandPNGBDBM50443385(SPC-100270 | Safingol | Safingol HCl)
Affinity DataKi:  5.00E+3nMAssay Description:Inhibition of sphingosine kinase 1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine kinase 2(Homo sapiens (Human))
The City University Of New York

Curated by ChEMBL
LigandPNGBDBM50393642(CHEMBL2158685)
Affinity DataKi:  1.00E+4nMAssay Description:Inhibition of SK2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine kinase 1(Homo sapiens (Human))
The City University Of New York

Curated by ChEMBL
LigandPNGBDBM50443389(CHEMBL2376441)
Affinity DataKi:  1.00E+4nMAssay Description:Inhibition of sphingosine kinase 1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine kinase 1(Homo sapiens (Human))
The City University Of New York

Curated by ChEMBL
LigandPNGBDBM50004888((S)-Fingolimod Vinylphosphonate | CHEMBL1773676)
Affinity DataKi:  1.00E+4nMAssay Description:Competitive inhibition of SK1 (unknown origin) in presence of ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine kinase 2(Homo sapiens (Human))
The City University Of New York

Curated by ChEMBL
LigandPNGBDBM50393641(CHEMBL2158686)
Affinity DataKi:  1.65E+4nMAssay Description:Inhibition of SK2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine kinase 1(Homo sapiens (Human))
The City University Of New York

Curated by ChEMBL
LigandPNGBDBM50041978(CHEMBL3134157)
Affinity DataIC50:  28nMAssay Description:Inhibition of recombinant SK1 (unknown origin) using sphingosine and [gamma-32P]ATP as substrate after 30 minsMore data for this Ligand-Target Pair
TargetSphingosine kinase 1(Homo sapiens (Human))
The City University Of New York

Curated by ChEMBL
LigandPNGBDBM50443384(CHEMBL3086799)
Affinity DataIC50:  2.20E+3nMAssay Description:Inhibition of recombinant sphingosine kinase 1 (unknown origin) expressed in HEK293 cells using sphingosine as substrate after 30 mins in presence of...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine kinase 1(Homo sapiens (Human))
The City University Of New York

Curated by ChEMBL
LigandPNGBDBM50443387(CHEMBL3086811)
Affinity DataIC50:  3.60E+3nMAssay Description:Inhibition of recombinant sphingosine kinase 1 (unknown origin) expressed in HEK293 cells using sphingosine as substrate after 30 mins in presence of...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine kinase 2(Homo sapiens (Human))
The City University Of New York

Curated by ChEMBL
LigandPNGBDBM50443383(CHEMBL3086796)
Affinity DataIC50:  5.00E+3nMAssay Description:Inhibition of sphingosine kinase 2 (unknown origin) using sphingosine as substrate after 30 mins in presence of [gamma32P]-ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine kinase 2(Homo sapiens (Human))
The City University Of New York

Curated by ChEMBL
LigandPNGBDBM50443384(CHEMBL3086799)
Affinity DataIC50:  5.20E+3nMAssay Description:Inhibition of sphingosine kinase 2 (unknown origin) using sphingosine as substrate after 30 mins in presence of [gamma32P]-ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine kinase 1(Homo sapiens (Human))
The City University Of New York

Curated by ChEMBL
LigandPNGBDBM50443383(CHEMBL3086796)
Affinity DataIC50:  5.30E+3nMAssay Description:Inhibition of recombinant sphingosine kinase 1 (unknown origin) expressed in HEK293 cells using sphingosine as substrate after 30 mins in presence of...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine kinase 1(Homo sapiens (Human))
The City University Of New York

Curated by ChEMBL
LigandPNGBDBM50496601((2S,3R)-Sphingosine | CHEBI:67106 | CHEMBL1835439)
Affinity DataIC50:  7.10E+3nMAssay Description:Inhibition of recombinant SK1 (unknown origin) using sphingosine and [gamma-32P]ATP as substrate after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine kinase 1(Homo sapiens (Human))
The City University Of New York

Curated by ChEMBL
LigandPNGBDBM50443386(CHEMBL3086806)
Affinity DataIC50:  1.69E+4nMAssay Description:Inhibition of recombinant sphingosine kinase 1 (unknown origin) expressed in HEK293 cells using sphingosine as substrate after 30 mins in presence of...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine kinase 2(Homo sapiens (Human))
The City University Of New York

Curated by ChEMBL
LigandPNGBDBM50496602(CHEMBL3134155)
Affinity DataIC50:  2.18E+4nMAssay Description:Inhibition of purified SK2 (unknown origin) using sphingosine and [gamma-32P]ATP as substrate after 30 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSphingosine kinase 1(Homo sapiens (Human))
The City University Of New York

Curated by ChEMBL
LigandPNGBDBM50496603(CHEMBL3134156)
Affinity DataIC50:  2.78E+4nMAssay Description:Inhibition of recombinant SK1 (unknown origin) using sphingosine and [gamma-32P]ATP as substrate after 30 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSphingosine kinase 1(Homo sapiens (Human))
The City University Of New York

Curated by ChEMBL
LigandPNGBDBM50496602(CHEMBL3134155)
Affinity DataIC50:  6.90E+4nMAssay Description:Inhibition of recombinant SK1 (unknown origin) using sphingosine and [gamma-32P]ATP as substrate after 30 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSphingosine kinase 2(Homo sapiens (Human))
The City University Of New York

Curated by ChEMBL
LigandPNGBDBM50496603(CHEMBL3134156)
Affinity DataIC50:  3.00E+5nMAssay Description:Inhibition of purified SK2 (unknown origin) using sphingosine and [gamma-32P]ATP as substrate after 30 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSphingosine kinase 2(Homo sapiens (Human))
The City University Of New York

Curated by ChEMBL
LigandPNGBDBM50496601((2S,3R)-Sphingosine | CHEBI:67106 | CHEMBL1835439)
Affinity DataIC50:  7.66E+5nMAssay Description:Inhibition of purified SK2 (unknown origin) using sphingosine and [gamma-32P]ATP as substrate after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine kinase 1(Homo sapiens (Human))
The City University Of New York

Curated by ChEMBL
LigandPNGBDBM50433311(CHEMBL2376444)
Affinity DataEC50:  8.30E+3nMAssay Description:Activation of recombinant GFP-tagged SK1 (unknown origin) expressed in HEK293 cells using sphingosine as substrate after 30 mins by Cerenkov counting...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine kinase 1(Homo sapiens (Human))
The City University Of New York

Curated by ChEMBL
LigandPNGBDBM50433312(CHEMBL2376443)
Affinity DataEC50:  5.70E+3nMAssay Description:Activation of recombinant GFP-tagged SK1 (unknown origin) expressed in HEK293 cells using sphingosine as substrate after 30 mins by Cerenkov counting...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed