TargetTrifunctional purine biosynthetic protein adenosine-3(Homo sapiens (Human))
Wellcome Research Laboratories
Curated by ChEMBL
Wellcome Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 220nMAssay Description:In vitro inhibition of hog liver GAR transformylase with (6R)-10-formyl-FH4 as cofactorMore data for this Ligand-Target Pair
TargetTrifunctional purine biosynthetic protein adenosine-3(Homo sapiens (Human))
Wellcome Research Laboratories
Curated by ChEMBL
Wellcome Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 1.60E+3nMAssay Description:In vitro inhibition of hog liver GAR transformylase with (6R)-10-formyl-FH4 as cofactorMore data for this Ligand-Target Pair
TargetTrifunctional purine biosynthetic protein adenosine-3(Homo sapiens (Human))
Wellcome Research Laboratories
Curated by ChEMBL
Wellcome Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 2.60E+3nMAssay Description:In vitro inhibition of hog liver GAR transformylase with (6R)-10-formyl-FH4 as cofactorMore data for this Ligand-Target Pair
TargetTrifunctional purine biosynthetic protein adenosine-3(Homo sapiens (Human))
Wellcome Research Laboratories
Curated by ChEMBL
Wellcome Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 3.00E+3nMAssay Description:In vitro inhibition of hog liver GAR transformylase with (6R)-10-formyl-FH4 as cofactorMore data for this Ligand-Target Pair
TargetTrifunctional purine biosynthetic protein adenosine-3(Homo sapiens (Human))
Wellcome Research Laboratories
Curated by ChEMBL
Wellcome Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 3.10E+3nMAssay Description:In vitro inhibition of hog liver GAR transformylase with (6R)-10-formyl-FH4 as cofactorMore data for this Ligand-Target Pair
TargetTrifunctional purine biosynthetic protein adenosine-3(Homo sapiens (Human))
Wellcome Research Laboratories
Curated by ChEMBL
Wellcome Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 3.50E+3nMAssay Description:In vitro inhibition of hog liver GAR transformylase with (6R)-10-formyl-FH4 as cofactorMore data for this Ligand-Target Pair
TargetTrifunctional purine biosynthetic protein adenosine-3(Homo sapiens (Human))
Wellcome Research Laboratories
Curated by ChEMBL
Wellcome Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 5.30E+3nMAssay Description:In vitro inhibition of hog liver GAR transformylase with (6R)-10-formyl-FH4 as cofactorMore data for this Ligand-Target Pair
TargetTrifunctional purine biosynthetic protein adenosine-3(Homo sapiens (Human))
Wellcome Research Laboratories
Curated by ChEMBL
Wellcome Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 6.10E+3nMAssay Description:In vitro inhibition of hog liver GAR transformylase with (6R)-10-formyl-FH4 as cofactorMore data for this Ligand-Target Pair
TargetTrifunctional purine biosynthetic protein adenosine-3(Homo sapiens (Human))
Wellcome Research Laboratories
Curated by ChEMBL
Wellcome Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 6.60E+3nMAssay Description:In vitro inhibition of hog liver GAR transformylase with (6R)-10-formyl-FH4 as cofactorMore data for this Ligand-Target Pair
TargetTrifunctional purine biosynthetic protein adenosine-3(Homo sapiens (Human))
Wellcome Research Laboratories
Curated by ChEMBL
Wellcome Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 1.82E+4nMAssay Description:In vitro inhibition of hog liver GAR transformylase with (6R)-10-formyl-FH4 as cofactorMore data for this Ligand-Target Pair
TargetTrifunctional purine biosynthetic protein adenosine-3(Homo sapiens (Human))
Wellcome Research Laboratories
Curated by ChEMBL
Wellcome Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 1.87E+4nMAssay Description:In vitro inhibition of hog liver GAR transformylase with (6R)-10-formyl-FH4 as cofactorMore data for this Ligand-Target Pair
TargetTrifunctional purine biosynthetic protein adenosine-3(Homo sapiens (Human))
Wellcome Research Laboratories
Curated by ChEMBL
Wellcome Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 5.20E+4nMAssay Description:In vitro inhibition of hog liver GAR transformylase with (6R)-10-formyl-FH4 as cofactorMore data for this Ligand-Target Pair
TargetBifunctional purine biosynthesis protein ATIC(Homo sapiens (Human))
Wellcome Research Laboratories
Curated by ChEMBL
Wellcome Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 9.40E+4nMAssay Description:In vitro inhibitory activity of the compound against MOLT-4 T-cell leukemia cell AICAR transformylaseMore data for this Ligand-Target Pair
TargetTrifunctional purine biosynthetic protein adenosine-3(Homo sapiens (Human))
Wellcome Research Laboratories
Curated by ChEMBL
Wellcome Research Laboratories
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:In vitro inhibition of hog liver GAR transformylase with (6R)-10-formyl-FH4 as cofactorMore data for this Ligand-Target Pair
TargetBifunctional purine biosynthesis protein ATIC(Homo sapiens (Human))
Wellcome Research Laboratories
Curated by ChEMBL
Wellcome Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 1.30E+5nMAssay Description:In vitro inhibitory activity of the compound against MOLT-4 T-cell leukemia cell AICAR transformylaseMore data for this Ligand-Target Pair
Affinity DataIC50: 2.20E+5nMAssay Description:Inhibitory activity against Arabinose-5-phosphate isomeraseMore data for this Ligand-Target Pair
Affinity DataIC50: 5.30E+5nMAssay Description:Inhibitory activity against Arabinose-5-phosphate isomeraseMore data for this Ligand-Target Pair
Affinity DataIC50: 5.30E+5nMAssay Description:Inhibitory activity against Arabinose-5-phosphate isomeraseMore data for this Ligand-Target Pair
Affinity DataIC50: 7.00E+5nMAssay Description:Inhibitory activity against Arabinose-5-phosphate isomeraseMore data for this Ligand-Target Pair
Affinity DataIC50: 4.70E+6nMAssay Description:Inhibitory activity against Arabinose-5-phosphate isomeraseMore data for this Ligand-Target Pair
Affinity DataIC50: 5.30E+6nMAssay Description:Inhibitory activity against Arabinose-5-phosphate isomeraseMore data for this Ligand-Target Pair
Affinity DataIC50: 8.40E+6nMAssay Description:Inhibitory activity against Arabinose-5-phosphate isomeraseMore data for this Ligand-Target Pair
Affinity DataIC50: 8.40E+6nMAssay Description:Inhibitory activity against Arabinose-5-phosphate isomeraseMore data for this Ligand-Target Pair
Affinity DataIC50: 8.70E+6nMAssay Description:Inhibitory activity against Arabinose-5-phosphate isomeraseMore data for this Ligand-Target Pair
Affinity DataIC50: 1.92E+7nMAssay Description:Inhibitory activity against Arabinose-5-phosphate isomeraseMore data for this Ligand-Target Pair
Affinity DataIC50: 1.92E+7nMAssay Description:Inhibitory activity against Arabinose-5-phosphate isomeraseMore data for this Ligand-Target Pair
Affinity DataIC50: 2.00E+7nMAssay Description:Inhibitory activity against Arabinose-5-phosphate isomeraseMore data for this Ligand-Target Pair
Affinity DataIC50: 2.69E+7nMAssay Description:Inhibitory activity against Arabinose-5-phosphate isomeraseMore data for this Ligand-Target Pair
Affinity DataIC50: 3.59E+7nMAssay Description:Inhibitory activity against Arabinose-5-phosphate isomeraseMore data for this Ligand-Target Pair
Affinity DataIC50: 6.13E+7nMAssay Description:Inhibitory activity against Arabinose-5-phosphate isomeraseMore data for this Ligand-Target Pair
Affinity DataIC50: 6.20E+7nMAssay Description:Inhibitory activity against Arabinose-5-phosphate isomeraseMore data for this Ligand-Target Pair
Affinity DataIC50: 6.67E+7nMAssay Description:Inhibitory activity against Arabinose-5-phosphate isomeraseMore data for this Ligand-Target Pair
Affinity DataIC50: 8.00E+7nMAssay Description:Inhibitory activity against Arabinose-5-phosphate isomeraseMore data for this Ligand-Target Pair
Affinity DataIC50: 8.67E+7nMAssay Description:Inhibitory activity against Arabinose-5-phosphate isomeraseMore data for this Ligand-Target Pair
Affinity DataIC50: 9.13E+7nMAssay Description:Inhibitory activity against Arabinose-5-phosphate isomeraseMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+8nMAssay Description:Inhibitory activity against Arabinose-5-phosphate isomeraseMore data for this Ligand-Target Pair
Affinity DataIC50: 2.33E+8nMAssay Description:Inhibitory activity against Arabinose-5-phosphate isomeraseMore data for this Ligand-Target Pair