Compile Data Set for Download or QSAR
maximum 50k data
Found 513 with Last Name = 'marston' and Initial = 'rw'
TargetCaspase-3(Homo sapiens (Human))
Evotec (Uk)

Curated by ChEMBL
LigandPNGBDBM50420474(CHEMBL2086889 | US9073941, 607)
Affinity DataIC50:  3nMAssay Description:Inhibition of caspase3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Evotec (Uk)

Curated by ChEMBL
LigandPNGBDBM50420459(CHEMBL2086528)
Affinity DataIC50:  10nMAssay Description:Inhibition of human recombinant TG2 by fluorescent transamidation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-glutamine gamma-glutamyltransferase E(Homo sapiens (Human))
Evotec (Uk)

Curated by ChEMBL
LigandPNGBDBM50420474(CHEMBL2086889 | US9073941, 607)
Affinity DataIC50:  11nMAssay Description:Inhibition of thrombin activated human TG3 by fluorescent transamidation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Evotec (Uk)

Curated by ChEMBL
LigandPNGBDBM50335329(2-(4-Fluorobenzyl)-4-(5-methyl-1H-pyrazol-3-ylamin...)
Affinity DataIC50:  14nMAssay Description:Inhibition of Aurora A by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Evotec (Uk)

Curated by ChEMBL
LigandPNGBDBM50400621(CHEMBL2203451)
Affinity DataIC50:  14nMAssay Description:Irreversible inhibition of transglutaminase 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Evotec (Uk)

Curated by ChEMBL
LigandPNGBDBM50420454(CHEMBL2086544)
Affinity DataIC50:  14nMAssay Description:Inhibition of human recombinant TG2 by fluorescent transamidation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Evotec (Uk)

Curated by ChEMBL
LigandPNGBDBM50420451(CHEMBL2086541)
Affinity DataIC50:  15nMAssay Description:Inhibition of human recombinant TG2 by fluorescent transamidation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Mus musculus)
Evotec (Uk)

Curated by ChEMBL
LigandPNGBDBM50420459(CHEMBL2086528)
Affinity DataIC50:  16nMAssay Description:Inhibition of mouse recombinant TG2 by fluorescent transamidation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Evotec (Uk)

Curated by ChEMBL
LigandPNGBDBM50335315(2-(Methyl-3-pyridine)-4-(5-methyl-1H-pyrazol-3-yla...)
Affinity DataIC50:  17nMAssay Description:Inhibition of Aurora A by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-glutamine gamma-glutamyltransferase K(Homo sapiens (Human))
Evotec (Uk)

Curated by ChEMBL
LigandPNGBDBM50420474(CHEMBL2086889 | US9073941, 607)
Affinity DataIC50:  18nMAssay Description:Inhibition of human recombinant TG1 by fluorescent transamidation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Evotec (Uk)

Curated by ChEMBL
LigandPNGBDBM50420515(CHEMBL2086523)
Affinity DataIC50:  20nMAssay Description:Inhibition of human recombinant TG2 by fluorescent transamidation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Evotec (Uk)

Curated by ChEMBL
LigandPNGBDBM50335332(4-(1H-Pyrazol-3-ylamino)-2-p-tolyl-2H-phthalazin-1...)
Affinity DataIC50:  23nMAssay Description:Inhibition of Aurora A by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Evotec (Uk)

Curated by ChEMBL
LigandPNGBDBM50335333(4-(5-Methyl-1H-pyrazol-3-ylamino)-2-m-tolyl-2H-pht...)
Affinity DataIC50:  24nMAssay Description:Inhibition of Aurora A by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Evotec (Uk)

Curated by ChEMBL
LigandPNGBDBM50420474(CHEMBL2086889 | US9073941, 607)
Affinity DataIC50:  25nMAssay Description:Inhibition of human recombinant TG2 by fluorescent transamidation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Evotec (Uk)

Curated by ChEMBL
LigandPNGBDBM50420471(CHEMBL2086530)
Affinity DataIC50:  25nMAssay Description:Inhibition of human recombinant TG2 by fluorescent transamidation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Evotec (Uk)

Curated by ChEMBL
LigandPNGBDBM50249453(2-(2,5-difluorobenzyl)-4-(5-methyl-1H-pyrazol-3-yl...)
Affinity DataIC50:  25nMAssay Description:Inhibition of Aurora A by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Evotec (Uk)

Curated by ChEMBL
LigandPNGBDBM50420468(CHEMBL2086524)
Affinity DataIC50:  26nMAssay Description:Inhibition of human recombinant TG2 by fluorescent transamidation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Evotec (Uk)

Curated by ChEMBL
LigandPNGBDBM50420452(CHEMBL2086542)
Affinity DataIC50:  26nMAssay Description:Inhibition of human recombinant TG2 by fluorescent transamidation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Evotec (Uk)

Curated by ChEMBL
LigandPNGBDBM50335331(2-(4-Methoxyphenyl)-4-(5-methyl-1H-pyrazol-3-ylami...)
Affinity DataIC50:  29nMAssay Description:Inhibition of Aurora A by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Evotec (Uk)

Curated by ChEMBL
LigandPNGBDBM50335330(4-(5-Methyl-2H-pyrazole-3-ylamino)phenyl-2H-phthal...)
Affinity DataIC50:  31nMAssay Description:Inhibition of Aurora A by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedMMDB

TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Evotec (Uk)

Curated by ChEMBL
LigandPNGBDBM50420463(CHEMBL2086480)
Affinity DataIC50:  32nMAssay Description:Inhibition of human recombinant TG2 by fluorescent transamidation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Evotec (Uk)

Curated by ChEMBL
LigandPNGBDBM50335327(2-(4-Methoxybenzyl)-4-(5-methyl-1H-pyrazol-3-ylami...)
Affinity DataIC50:  32nMAssay Description:Inhibition of Aurora A by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Evotec (Uk)

Curated by ChEMBL
LigandPNGBDBM50420467(CHEMBL2086521)
Affinity DataIC50:  34nMAssay Description:Inhibition of human recombinant TG2 by fluorescent transamidation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Evotec (Uk)

Curated by ChEMBL
LigandPNGBDBM50420518(CHEMBL2086531)
Affinity DataIC50:  35nMAssay Description:Inhibition of human recombinant TG2 by fluorescent transamidation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Evotec (Uk)

Curated by ChEMBL
LigandPNGBDBM50335323(2-Isopropyl-4-(5-methyl-1H-pyrazol-3-ylamino)-2H-p...)
Affinity DataIC50:  35nMAssay Description:Inhibition of Aurora A by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Evotec (Uk)

Curated by ChEMBL
LigandPNGBDBM50335322(2-(3-Methoxybenzyl)-4-(5-methyl-1H-pyrazol-3-ylami...)
Affinity DataIC50:  36nMAssay Description:Inhibition of Aurora A by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Evotec (Uk)

Curated by ChEMBL
LigandPNGBDBM50335334(2-(4-Fluorophenyl)-4-(5-methyl-1H-pyrazol-3-ylamin...)
Affinity DataIC50:  37nMAssay Description:Inhibition of Aurora A by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Evotec (Uk)

Curated by ChEMBL
LigandPNGBDBM50420469(CHEMBL2086525)
Affinity DataIC50:  37nMAssay Description:Inhibition of human recombinant TG2 by fluorescent transamidation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor XIII A chain(Homo sapiens (Human))
Evotec (Uk)

Curated by ChEMBL
LigandPNGBDBM50420503(CHEMBL2086505)
Affinity DataIC50:  39nMAssay Description:Inhibition of thrombin activated human F13a by fluorescent transamidation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Evotec (Uk)

Curated by ChEMBL
LigandPNGBDBM50420470(CHEMBL2086526)
Affinity DataIC50:  41nMAssay Description:Inhibition of human recombinant TG2 by fluorescent transamidation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Evotec (Uk)

Curated by ChEMBL
LigandPNGBDBM50420519(CHEMBL2086519)
Affinity DataIC50:  44nMAssay Description:Inhibition of human recombinant TG2 by fluorescent transamidation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Evotec (Uk)

Curated by ChEMBL
LigandPNGBDBM50420464(CHEMBL2086506)
Affinity DataIC50:  46nMAssay Description:Inhibition of human recombinant TG2 by fluorescent transamidation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Evotec (Uk)

Curated by ChEMBL
LigandPNGBDBM50335336(2-(3,5-Difluorobenzyl)-4-(5-methyl-1H-pyrazol-3-yl...)
Affinity DataIC50:  49nMAssay Description:Inhibition of Aurora A by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor XIII A chain(Homo sapiens (Human))
Evotec (Uk)

Curated by ChEMBL
LigandPNGBDBM50420457(CHEMBL2086890)
Affinity DataIC50:  51nMAssay Description:Inhibition of thrombin activated human F13a by fluorescent transamidation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Evotec (Uk)

Curated by ChEMBL
LigandPNGBDBM50420443(CHEMBL2086532)
Affinity DataIC50:  52nMAssay Description:Inhibition of human recombinant TG2 by fluorescent transamidation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Evotec (Uk)

Curated by ChEMBL
LigandPNGBDBM50420504(CHEMBL2086507)
Affinity DataIC50:  54nMAssay Description:Inhibition of human recombinant TG2 by fluorescent transamidation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Evotec (Uk)

Curated by ChEMBL
LigandPNGBDBM50420510(CHEMBL2086515)
Affinity DataIC50:  54nMAssay Description:Inhibition of human recombinant TG2 by fluorescent transamidation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Evotec (Uk)

Curated by ChEMBL
LigandPNGBDBM50400626(CHEMBL2203467)
Affinity DataIC50:  54nMAssay Description:Irreversible inhibition of transglutaminase 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Mus musculus)
Evotec (Uk)

Curated by ChEMBL
LigandPNGBDBM50392906(CHEMBL2152204)
Affinity DataIC50:  55nMAssay Description:Inhibition of mouse TGM2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Evotec (Uk)

Curated by ChEMBL
LigandPNGBDBM50420517(CHEMBL2086529)
Affinity DataIC50:  55nMAssay Description:Inhibition of human recombinant TG2 by fluorescent transamidation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Evotec (Uk)

Curated by ChEMBL
LigandPNGBDBM50400633(CHEMBL2203473)
Affinity DataIC50:  55nMAssay Description:Irreversible inhibition of transglutaminase 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Evotec (Uk)

Curated by ChEMBL
LigandPNGBDBM50335324(2-(4-Toluylsulfonate)-4-(5-methyl-1H-pyrazol-3-yla...)
Affinity DataIC50:  56nMAssay Description:Inhibition of Aurora A by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Evotec (Uk)

Curated by ChEMBL
LigandPNGBDBM50420516(CHEMBL2086527)
Affinity DataIC50:  57nMAssay Description:Inhibition of human recombinant TG2 by fluorescent transamidation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Evotec (Uk)

Curated by ChEMBL
LigandPNGBDBM50420511(CHEMBL2086516)
Affinity DataIC50:  60nMAssay Description:Inhibition of human recombinant TG2 by fluorescent transamidation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Evotec (Uk)

Curated by ChEMBL
LigandPNGBDBM50400625(CHEMBL2203469)
Affinity DataIC50:  62nMAssay Description:Irreversible inhibition of transglutaminase 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Evotec (Uk)

Curated by ChEMBL
LigandPNGBDBM50335335(2-Benzyl-4-(5-methyl-1H-pyrazol-3-ylamino)-2H-phth...)
Affinity DataIC50:  65nMAssay Description:Inhibition of Aurora A by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Evotec (Uk)

Curated by ChEMBL
LigandPNGBDBM50249210(4-(5-methyl-1H-pyrazol-3-ylamino)-2-(2,2,2-trifluo...)
Affinity DataIC50:  66nMAssay Description:Inhibition of Aurora A by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor XIII A chain(Homo sapiens (Human))
Evotec (Uk)

Curated by ChEMBL
LigandPNGBDBM50420458(CHEMBL2086891)
Affinity DataIC50:  66nMAssay Description:Inhibition of thrombin activated human F13a by fluorescent transamidation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Evotec (Uk)

Curated by ChEMBL
LigandPNGBDBM50335337(2-[2-(4-Methoxyphenyl)-2-oxoethyl]-4-(5-methyl-1H-...)
Affinity DataIC50:  67nMAssay Description:Inhibition of Aurora A by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Evotec (Uk)

Curated by ChEMBL
LigandPNGBDBM50420453(CHEMBL2086543)
Affinity DataIC50:  69nMAssay Description:Inhibition of human recombinant TG2 by fluorescent transamidation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Displayed 1 to 50 (of 513 total ) | Next | Last >>
Jump to: