Affinity DataKi: 0.140nMAssay Description:Inhibition of human recombinant melanocortin 4 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
The University Of Newcastle
Curated by ChEMBL
The University Of Newcastle
Curated by ChEMBL
Affinity DataKi: 0.170nMAssay Description:Displacement of [3H]LSD from human recombinant 5-HT7 receptor expressed in CHO cells after 120 mins by scintillation countingMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
The University Of Newcastle
Curated by ChEMBL
The University Of Newcastle
Curated by ChEMBL
Affinity DataKi: 0.220nMAssay Description:Displacement of [3H]4-DAMP from human recombinant Muscarinic acetylcholine receptor M3 expressed in CHO cells after 60 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 0.270nMAssay Description:Displacement of [3H]methyl-spiperone from human recombinant D2S receptor in HEK293 cells after 60 mins by scintillation countingMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
The University Of Newcastle
Curated by ChEMBL
The University Of Newcastle
Curated by ChEMBL
Affinity DataKi: 0.280nMAssay Description:Displacement of [3H]ketanserin from human recombinant 5-HT2A receptor in HEK293 cells after 60 mins by scintillation countingMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Rattus norvegicus (rat))
The University Of Newcastle
Curated by ChEMBL
The University Of Newcastle
Curated by ChEMBL
Affinity DataKi: 0.450nMAssay Description:Displacement of [3H]U 69593 from rat recombinant kappa opioid receptor expressed in CHO cells after 60 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 0.710nMAssay Description:Displacement of [3H]pyrilamine from human recombinant histamine H1 receptor in HEK293 cells after 60 mins by scintillation countingMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
The University Of Newcastle
Curated by ChEMBL
The University Of Newcastle
Curated by ChEMBL
Affinity DataKi: 1.60nMAssay Description:Displacement of [125I](+/-)DOI from human recombinant 5-HT2B receptor expressed in CHO cells after 60 mins by scintillation countingMore data for this Ligand-Target Pair
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
The University Of Wollongong
Curated by ChEMBL
The University Of Wollongong
Curated by ChEMBL
Affinity DataKi: 1.70nMAssay Description:Inhibition of [125I]-CRH binding to human Corticotropin releasing factor receptor 1.More data for this Ligand-Target Pair
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
The University Of Wollongong
Curated by ChEMBL
The University Of Wollongong
Curated by ChEMBL
Affinity DataKi: 2nMAssay Description:Ability to inhibit [125I]-CRH binding to human Corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Displacement of [125I]NKA from human recombinant tachykinin NK2 receptor expressed in CHO cells after 60 mins by scintillation countingMore data for this Ligand-Target Pair
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
The University Of Newcastle
Curated by ChEMBL
The University Of Newcastle
Curated by ChEMBL
Affinity DataKi: 2.10nMAssay Description:Displacement of [3H]nisoxetine from human recombinant norepinephrine transporter expressed in CHO cells after 120 mins by scintillation countingMore data for this Ligand-Target Pair
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
The University Of Wollongong
Curated by ChEMBL
The University Of Wollongong
Curated by ChEMBL
Affinity DataKi: 2.30nMAssay Description:Inhibition of [125I]-CRH binding to human Corticotropin releasing factor receptor 1.More data for this Ligand-Target Pair
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
The University Of Wollongong
Curated by ChEMBL
The University Of Wollongong
Curated by ChEMBL
Affinity DataKi: 2.5nMAssay Description:Inhibition of [125I]-CRH binding to human Corticotropin releasing factor receptor 1.More data for this Ligand-Target Pair
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
The University Of Wollongong
Curated by ChEMBL
The University Of Wollongong
Curated by ChEMBL
Affinity DataKi: 3.80nMAssay Description:Inhibition of [125I]-CRH binding to human Corticotropin releasing factor receptor 1.More data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
The University Of Newcastle
Curated by ChEMBL
The University Of Newcastle
Curated by ChEMBL
Affinity DataKi: 6.20nMAssay Description:Displacement of [3H]BTCP from human recombinant dopamine transporter expressed in CHO cells after 120 mins by scintillation countingMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
The University Of Newcastle
Curated by ChEMBL
The University Of Newcastle
Curated by ChEMBL
Affinity DataKi: 24nMAssay Description:Displacement of [3H]pirenzepine from human recombinant Muscarinic acetylcholine receptor M1 expressed in CHO cells after 60 mins by scintillation cou...More data for this Ligand-Target Pair
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
The University Of Wollongong
Curated by ChEMBL
The University Of Wollongong
Curated by ChEMBL
Affinity DataKi: 57nMAssay Description:Inhibition of [125I]-CRH binding to human Corticotropin releasing factor receptor 1.More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
The University Of Newcastle
Curated by ChEMBL
The University Of Newcastle
Curated by ChEMBL
Affinity DataKi: 61nMAssay Description:Displacement of [3H]LSD from human recombinant 5-HT6 receptor expressed in CHO cells after 120 mins by scintillation countingMore data for this Ligand-Target Pair
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
The University Of Wollongong
Curated by ChEMBL
The University Of Wollongong
Curated by ChEMBL
Affinity DataKi: 115nMAssay Description:Inhibition of [125I]-CRH binding to human Corticotropin releasing factor receptor 1.More data for this Ligand-Target Pair
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
The University Of Wollongong
Curated by ChEMBL
The University Of Wollongong
Curated by ChEMBL
Affinity DataKi: 130nMAssay Description:Inhibition of [125I]-CRH binding to human Corticotropin releasing factor receptor 1.More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 5A(Homo sapiens (Human))
The University Of Newcastle
Curated by ChEMBL
The University Of Newcastle
Curated by ChEMBL
Affinity DataKi: 130nMAssay Description:Displacement of [3H]LSD from human recombinant 5-HT5a receptor in HEK293 cells after 120 mins by scintillation countingMore data for this Ligand-Target Pair
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
The University Of Wollongong
Curated by ChEMBL
The University Of Wollongong
Curated by ChEMBL
Affinity DataKi: 253nMAssay Description:Inhibition of [125I]-CRH binding to human Corticotropin releasing factor receptor 1.More data for this Ligand-Target Pair
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
The University Of Wollongong
Curated by ChEMBL
The University Of Wollongong
Curated by ChEMBL
Affinity DataKi: 253nMAssay Description:Inhibition of [125I]-CRH binding to human Corticotropin releasing factor receptor 1.More data for this Ligand-Target Pair
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
The University Of Wollongong
Curated by ChEMBL
The University Of Wollongong
Curated by ChEMBL
Affinity DataKi: 490nMAssay Description:Inhibition of [125I]-CRH binding to human Corticotropin releasing factor receptor 1.More data for this Ligand-Target Pair
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
The University Of Wollongong
Curated by ChEMBL
The University Of Wollongong
Curated by ChEMBL
Affinity DataKi: 490nMAssay Description:Inhibition of [125I]-CRH binding to human Corticotropin releasing factor receptor 1.More data for this Ligand-Target Pair
Affinity DataKi: 490nMAssay Description:Displacement of [125I]APT from human recombinant histamine H2 receptor expressed in CHO cells after 120 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 620nMAssay Description:Binding affinity for rat brain Adenosine A1 receptorMore data for this Ligand-Target Pair
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
The University Of Wollongong
Curated by ChEMBL
The University Of Wollongong
Curated by ChEMBL
Affinity DataKi: 1.05E+3nMAssay Description:Inhibition of [125I]-CRH binding to human Corticotropin releasing factor receptor 1.More data for this Ligand-Target Pair
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
The University Of Wollongong
Curated by ChEMBL
The University Of Wollongong
Curated by ChEMBL
Affinity DataKi: 1.05E+3nMAssay Description:Inhibition of [125I]-CRH binding to human Corticotropin releasing factor receptor 1.More data for this Ligand-Target Pair
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
The University Of Wollongong
Curated by ChEMBL
The University Of Wollongong
Curated by ChEMBL
Affinity DataKi: 1.39E+3nMAssay Description:Inhibition of [125I]-CRH binding to human Corticotropin releasing factor receptor 1.More data for this Ligand-Target Pair
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
The University Of Wollongong
Curated by ChEMBL
The University Of Wollongong
Curated by ChEMBL
Affinity DataKi: 1.47E+3nMAssay Description:Inhibition of [125I]-CRH binding to human Corticotropin releasing factor receptor 1.More data for this Ligand-Target Pair
Affinity DataKi: 1.60E+3nMAssay Description:Binding affinity against Adenosine A2a receptor from rat striataMore data for this Ligand-Target Pair
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
The University Of Wollongong
Curated by ChEMBL
The University Of Wollongong
Curated by ChEMBL
Affinity DataKi: 1.69E+3nMAssay Description:Inhibition of [125I]-CRH binding to human Corticotropin releasing factor receptor 1.More data for this Ligand-Target Pair
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
The University Of Wollongong
Curated by ChEMBL
The University Of Wollongong
Curated by ChEMBL
Affinity DataKi: 2.10E+3nMAssay Description:Inhibition of [125I]-CRH binding to human Corticotropin releasing factor receptor 1.More data for this Ligand-Target Pair
Affinity DataKi: 2.23E+3nMAssay Description:Binding affinity for rat brain Adenosine A1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 2.99E+3nMAssay Description:Binding affinity for rat brain Adenosine A1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 3.20E+3nMAssay Description:Binding affinity for rat brain Adenosine A1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 3.30E+3nMAssay Description:Binding affinity against Adenosine A2a receptor from rat striataMore data for this Ligand-Target Pair
Affinity DataKi: 3.82E+3nMAssay Description:Binding affinity for rat brain Adenosine A1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 4.54E+3nMAssay Description:Binding affinity for rat brain Adenosine A1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 7.40E+3nMAssay Description:Binding affinity for rat brain Adenosine A1 receptorMore data for this Ligand-Target Pair
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
The University Of Wollongong
Curated by ChEMBL
The University Of Wollongong
Curated by ChEMBL
Affinity DataKi: 8.00E+3nMAssay Description:Inhibition of [125I]-CRH binding to human Corticotropin releasing factor receptor 1.More data for this Ligand-Target Pair
Affinity DataKi: 9.00E+3nMAssay Description:Binding affinity for rat brain Adenosine A1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 9.40E+3nMAssay Description:Binding affinity for rat brain Adenosine A1 receptorMore data for this Ligand-Target Pair
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
The University Of Wollongong
Curated by ChEMBL
The University Of Wollongong
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of [125I]-CRH binding to human Corticotropin releasing factor receptor 1.More data for this Ligand-Target Pair
Affinity DataKi: 1.10E+4nMAssay Description:Binding affinity against Adenosine A2a receptor from rat striataMore data for this Ligand-Target Pair
Affinity DataKi: 1.12E+4nMAssay Description:Binding affinity for rat brain Adenosine A1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.26E+4nMAssay Description:Binding affinity for rat brain Adenosine A1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.35E+4nMAssay Description:Binding affinity against Adenosine A2a receptor from rat striataMore data for this Ligand-Target Pair