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Found 64 with Last Name = 'meadows' and Initial = 'rp'
TargetStromelysin-1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50121950(2-[2-(3'-Cyano-biphenyl-4-sulfonyl)-ethoxy]-naphth...)
Affinity DataIC50:  62nMAssay Description:Inhibition of Stromelysin (MMP-3)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50121945(2-[3-(4'-Methoxy-biphenyl-4-sulfonyl)-propyl]-naph...)
Affinity DataIC50:  400nMAssay Description:Inhibition of Stromelysin (MMP-3)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50121944(2-[3-(4'-Methoxy-biphenyl-4-yl)-3-oxo-propyl]-naph...)
Affinity DataIC50:  450nMAssay Description:Inhibition of Stromelysin (MMP-3)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50121946(2-[2-(4'-Methoxy-biphenyl-4-sulfonyl)-ethoxy]-naph...)
Affinity DataIC50:  460nMAssay Description:Inhibition of Stromelysin (MMP-3)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50121959(2-[2-(4'-Chloro-biphenyl-4-yloxy)-ethyl]-naphthale...)
Affinity DataIC50:  640nMAssay Description:Inhibition of Stromelysin (MMP-3)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50121942(2-[2-(4'-Chloro-biphenyl-4-sulfonyl)-ethoxy]-napht...)
Affinity DataIC50:  670nMAssay Description:Inhibition of Stromelysin (MMP-3)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50121951(2-[(4'-Trifluoromethoxy-biphenyl-4-sulfonylamino)-...)
Affinity DataIC50:  690nMAssay Description:Inhibition of Stromelysin (MMP-3)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50121961(2-[4-(4'-Methoxy-biphenyl-4-yl)-4-oxo-butyl]-napht...)
Affinity DataIC50:  1.50E+3nMAssay Description:Inhibition of Stromelysin (MMP-3)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50121954(2-[2-(4'-Chloro-biphenyl-4-sulfonyl)-ethyl]-naphth...)
Affinity DataIC50:  3.70E+3nMAssay Description:Inhibition of Stromelysin (MMP-3)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50121948(2-[2-(4'-Methoxy-biphenyl-4-sulfonylamino)-ethyl]-...)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibition of Stromelysin (MMP-3)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50121947(2-(4'-Cyano-biphenyl-4-yloxymethyl)-naphthalene-1-...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of Stromelysin (MMP-3)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50121962(2-[3-(4'-Cyano-biphenyl-4-yloxy)-propoxy]-naphthal...)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibition of Stromelysin (MMP-3)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50015152(CHEMBL115468 | N-hydroxy-1-naphthamide | Naphthale...)
Affinity DataIC50:  5.00E+4nMAssay Description:Inhibition of Stromelysin (MMP-3)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase XIAP [241-356](Homo sapiens (Human))
Abbott Laboratories

LigandPNGBDBM13179((2S)-1-[(2S)-2-cyclohexyl-2-[(2S)-2-(dimethylamino...)
Affinity DataKd: >1.00E+3nMpH: 7.4 T: 2°CAssay Description:A fluorescence polarization anisotropy (FPA) competition assay was used to determine the affinities of compounds to BIR3 protein. Fluorescence polari...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase XIAP [241-356](Homo sapiens (Human))
Abbott Laboratories

LigandPNGBDBM13180((2S)-1-[(2S)-3,3-dimethyl-2-[(2R)-2-(methylamino)p...)
Affinity DataKd: >1.00E+3nMpH: 7.4 T: 2°CAssay Description:A fluorescence polarization anisotropy (FPA) competition assay was used to determine the affinities of compounds to BIR3 protein. Fluorescence polari...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase XIAP [241-356](Homo sapiens (Human))
Abbott Laboratories

LigandPNGBDBM13181((2S)-2-amino-N-(5,7-dimethyl-1,8-naphthyridin-2-yl...)
Affinity DataKd:  2.00E+4nMpH: 7.4 T: 2°CAssay Description:A fluorescence polarization anisotropy (FPA) competition assay was used to determine the affinities of compounds to BIR3 protein. Fluorescence polari...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase XIAP [241-356](Homo sapiens (Human))
Abbott Laboratories

LigandPNGBDBM13182((2S)-2-amino-N-[5-(4-butoxyphenyl)-1,3,4-thiadiazo...)
Affinity DataKd:  2.50E+4nMpH: 7.4 T: 2°CAssay Description:A fluorescence polarization anisotropy (FPA) competition assay was used to determine the affinities of compounds to BIR3 protein. Fluorescence polari...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase XIAP [241-356](Homo sapiens (Human))
Abbott Laboratories

LigandPNGBDBM13183((2S)-2-amino-N-(5-benzoyl-1H-1,3-benzodiazol-2-yl)...)
Affinity DataKd:  3.00E+4nMpH: 7.4 T: 2°CAssay Description:A fluorescence polarization anisotropy (FPA) competition assay was used to determine the affinities of compounds to BIR3 protein. Fluorescence polari...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase XIAP [241-356](Homo sapiens (Human))
Abbott Laboratories

LigandPNGBDBM13184((2S)-2-amino-N-[4-(4-chloro-3-methylphenyl)-1,3-th...)
Affinity DataKd:  3.00E+4nMpH: 7.4 T: 2°CAssay Description:A fluorescence polarization anisotropy (FPA) competition assay was used to determine the affinities of compounds to BIR3 protein. Fluorescence polari...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase XIAP [241-356](Homo sapiens (Human))
Abbott Laboratories

LigandPNGBDBM13185((2S)-2-amino-N-{5-methyl-4-[(2,4,6-trimethylphenyl...)
Affinity DataKd:  2.00E+3nMpH: 7.4 T: 2°CAssay Description:A fluorescence polarization anisotropy (FPA) competition assay was used to determine the affinities of compounds to BIR3 protein. Fluorescence polari...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase XIAP [241-356](Homo sapiens (Human))
Abbott Laboratories

LigandPNGBDBM13186((2S)-2-amino-N-(5-methyl-4-phenyl-1,3-thiazol-2-yl...)
Affinity DataKd:  1.50E+4nMpH: 7.4 T: 2°CAssay Description:A fluorescence polarization anisotropy (FPA) competition assay was used to determine the affinities of compounds to BIR3 protein. Fluorescence polari...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase XIAP [241-356](Homo sapiens (Human))
Abbott Laboratories

LigandPNGBDBM13187((2S)-2-amino-N-(5-tert-butyl-4-phenyl-1,3-thiazol-...)
Affinity DataKd:  4.80E+3nMAssay Description:A fluorescence polarization anisotropy (FPA) competition assay was used to determine the affinities of compounds to BIR3 protein. Fluorescence polari...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase XIAP [241-356](Homo sapiens (Human))
Abbott Laboratories

LigandPNGBDBM13188((2S)-2-amino-N-(4-methyl-5-phenyl-1,3-thiazol-2-yl...)
Affinity DataKd:  1.50E+4nMAssay Description:A fluorescence polarization anisotropy (FPA) competition assay was used to determine the affinities of compounds to BIR3 protein. Fluorescence polari...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase XIAP [241-356](Homo sapiens (Human))
Abbott Laboratories

LigandPNGBDBM13189((2S)-2-amino-N-(4,5-diphenyl-1,3-thiazol-2-yl)prop...)
Affinity DataKd:  1.10E+3nMAssay Description:A fluorescence polarization anisotropy (FPA) competition assay was used to determine the affinities of compounds to BIR3 protein. Fluorescence polari...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase XIAP [241-356](Homo sapiens (Human))
Abbott Laboratories

LigandPNGBDBM13190((2S)-2-amino-N-[4-(4-bromophenyl)-5-phenyl-1,3-thi...)
Affinity DataKd:  740nMAssay Description:A fluorescence polarization anisotropy (FPA) competition assay was used to determine the affinities of compounds to BIR3 protein. Fluorescence polari...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase XIAP [241-356](Homo sapiens (Human))
Abbott Laboratories

LigandPNGBDBM13191((2S)-2-amino-N-[4-(4-benzylphenyl)-5-phenyl-1,3-th...)
Affinity DataKd:  1.20E+3nMAssay Description:A fluorescence polarization anisotropy (FPA) competition assay was used to determine the affinities of compounds to BIR3 protein. Fluorescence polari...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase XIAP [241-356](Homo sapiens (Human))
Abbott Laboratories

LigandPNGBDBM13192((2S)-2-amino-N-[5-benzyl-4-(3-benzylphenyl)-1,3-th...)
Affinity DataKd: >1.00E+5nMAssay Description:A fluorescence polarization anisotropy (FPA) competition assay was used to determine the affinities of compounds to BIR3 protein. Fluorescence polari...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase XIAP [241-356](Homo sapiens (Human))
Abbott Laboratories

LigandPNGBDBM13193((2S)-2-amino-N-[5-benzyl-4-(phenoxymethyl)-1,3-thi...)
Affinity DataKd:  4.10E+3nMAssay Description:A fluorescence polarization anisotropy (FPA) competition assay was used to determine the affinities of compounds to BIR3 protein. Fluorescence polari...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase XIAP [241-356](Homo sapiens (Human))
Abbott Laboratories

LigandPNGBDBM13194((2S)-2-amino-N-{5-benzyl-4-[(benzyloxy)methyl]-1,3...)
Affinity DataKd:  4.10E+3nMAssay Description:A fluorescence polarization anisotropy (FPA) competition assay was used to determine the affinities of compounds to BIR3 protein. Fluorescence polari...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase XIAP [241-356](Homo sapiens (Human))
Abbott Laboratories

LigandPNGBDBM13195((2S)-2-amino-N-{5-benzyl-4-[(naphthalen-1-yloxy)me...)
Affinity DataKd:  2.10E+4nMAssay Description:A fluorescence polarization anisotropy (FPA) competition assay was used to determine the affinities of compounds to BIR3 protein. Fluorescence polari...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase XIAP [241-356](Homo sapiens (Human))
Abbott Laboratories

LigandPNGBDBM13196((2S)-2-amino-N-{5-benzyl-4-[(naphthalen-2-yloxy)me...)
Affinity DataKd:  1.40E+4nMAssay Description:A fluorescence polarization anisotropy (FPA) competition assay was used to determine the affinities of compounds to BIR3 protein. Fluorescence polari...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase XIAP [241-356](Homo sapiens (Human))
Abbott Laboratories

LigandPNGBDBM13197((2S)-2-amino-N-{5-benzyl-4-[(2,3-dihydro-1H-inden-...)
Affinity DataKd:  2.20E+4nMAssay Description:A fluorescence polarization anisotropy (FPA) competition assay was used to determine the affinities of compounds to BIR3 protein. Fluorescence polari...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase XIAP [241-356](Homo sapiens (Human))
Abbott Laboratories

LigandPNGBDBM13198((2S)-2-amino-N-{5-thia-3-azatricyclo[7.4.0.0^{2,6}...)
Affinity DataKd:  7.10E+3nMAssay Description:A fluorescence polarization anisotropy (FPA) competition assay was used to determine the affinities of compounds to BIR3 protein. Fluorescence polari...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase XIAP [241-356](Homo sapiens (Human))
Abbott Laboratories

LigandPNGBDBM13199((2S)-2-amino-N-{5-thia-3-azatricyclo[7.4.0.0^{2,6}...)
Affinity DataKd:  5.60E+3nMAssay Description:A fluorescence polarization anisotropy (FPA) competition assay was used to determine the affinities of compounds to BIR3 protein. Fluorescence polari...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50121943(4'-Hydroxy-biphenyl-4-carbonitrile | CHEMBL114523)
Affinity DataKd:  2.00E+4nMAssay Description:Binding to stromelysin (MMP-3) in place of acetohydroxamic acid.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50015152(CHEMBL115468 | N-hydroxy-1-naphthamide | Naphthale...)
Affinity DataKd:  5.00E+4nMAssay Description:Binding to stromelysin (MMP-3) in place of acetohydroxamic acid.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50056900(2-Carbamoylphenol | 2-Carboxamidophenol | 2-Hydrox...)
Affinity DataKd: >2.50E+7nMAssay Description:Binding to stromelysin (MMP-3) in place of acetohydroxamic acid.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50121952(CHEMBL153081 | Ethyl hydroxycarbamate)
Affinity DataKd: >2.50E+7nMAssay Description:Binding to stromelysin (MMP-3) in place of acetohydroxamic acid.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50017811(CHEMBL467 | HU | US10155732, Compound HU | hydroxy...)
Affinity DataKd: >2.50E+7nMAssay Description:Binding to stromelysin (MMP-3) in place of acetohydroxamic acid.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50121955(4-Phenyl-pyridine | CHEMBL109074 | US11634391, Com...)
Affinity DataKd:  1.70E+5nMAssay Description:Binding to stromelysin (MMP-3) in the presence of acetohydroxamic acidMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50121958(4,4'-Biphenyldiol | 4,4'-Dihydroxybiphenyl | 4,4'-...)
Affinity DataKd:  1.50E+5nMAssay Description:Binding to stromelysin (MMP-3) in the presence of 1-NapthohydroxamateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50121956(4,4,4-Trifluoro-3-oxo-butyric acid ethyl ester | C...)
Affinity DataKd: >2.50E+7nMAssay Description:Binding to stromelysin (MMP-3) in place of acetohydroxamic acid.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50121957(CHEMBL152603 | Thiophen-2-yl-methanethiol)
Affinity DataKd:  1.50E+5nMAssay Description:Binding to stromelysin (MMP-3) in place of acetohydroxamic acid.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50121953(2-mercaptoethanecarboxylic acid | 3-mercaptopropan...)
Affinity DataKd:  3.00E+6nMAssay Description:Binding to stromelysin (MMP-3) in place of acetohydroxamic acid.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50099857(ACETOHYDROXAMIC ACID (AHA) | AHA | Acethydroxamsae...)
Affinity DataKd:  1.70E+7nMAssay Description:Binding to stromelysin (MMP-3) in place of acetohydroxamic acid.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50121955(4-Phenyl-pyridine | CHEMBL109074 | US11634391, Com...)
Affinity DataKd:  9.00E+5nMAssay Description:Binding to stromelysin (MMP-3) in the presence of 1-NapthohydroxamateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50121958(4,4'-Biphenyldiol | 4,4'-Dihydroxybiphenyl | 4,4'-...)
Affinity DataKd:  1.60E+5nMAssay Description:Binding to stromelysin (MMP-3) in the presence of acetohydroxamic acidMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM26193(2-Hydroxybenzoate, I | 2-hydroxybenzoic acid | CHE...)
Affinity DataKd: >2.50E+7nMAssay Description:Binding to stromelysin (MMP-3) in place of acetohydroxamic acid.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50015184(BENZHYDROXAMIC ACID | BENZOHYDROXAMATE | CHEMBL163...)
Affinity DataKd:  7.00E+6nMAssay Description:Binding to stromelysin (MMP-3) in place of acetohydroxamic acid.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50026891(1-Pyridin-2-yl-ethanone | CHEMBL11945)
Affinity DataKd: >2.50E+7nMAssay Description:Binding to stromelysin (MMP-3) in place of acetohydroxamic acid.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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