Affinity DataKi: 0.200nMAssay Description:Binding towards dopamine receptor D4 expressed in CHO-K1 cells using [3H]spiperone More data for this Ligand-Target Pair
TargetNociceptin receptor(Homo sapiens (Human))
Louisiana State University
Curated by PDSP Ki Database
Louisiana State University
Curated by PDSP Ki Database
Affinity DataKi: 0.300nMAssay Description:Evaluated for binding towards Dopamine receptor D2 using [3H]-spiperone as radioligand, in cloned mammalian receptors expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
TargetNociceptin receptor(Homo sapiens (Human))
Louisiana State University
Curated by PDSP Ki Database
Louisiana State University
Curated by PDSP Ki Database
Affinity DataKi: 0.700nMAssay Description:Evaluated for binding towards Dopamine receptor D2 using [3H]-N-0437 as radioligand from rat striatal membraneMore data for this Ligand-Target Pair
Affinity DataKi: 0.700nMAssay Description:Evaluated for binding towards Dopamine receptor D2 using [3H]-N-0437 as radioligand from rat striatal membraneMore data for this Ligand-Target Pair
Affinity DataKi: 2.20nMAssay Description:Binding towards dopamine receptor D4 expressed in CHO-K1 cells using [3H]spiperone More data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Binding towards Dopamine receptor D3 expressed in CHO-K1 cells using [3H]spiperone More data for this Ligand-Target Pair
Affinity DataKi: 6.30nMAssay Description:In vitro binding affinity for muscarinic M1 receptor by displacing [3H]-Pirenzepine binding on rat brain homogenate.More data for this Ligand-Target Pair
Affinity DataKi: 6.40nMAssay Description:Binding towards Dopamine receptor D3 expressed in CHO-K1 cells using [3H]spiperone More data for this Ligand-Target Pair
Affinity DataKi: 7.70nMAssay Description:In vitro binding affinity for muscarinic M1 receptor by displacing [3H]-Pirenzepine binding on rat brain homogenate.More data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:In vitro binding affinity for muscarinic M1 receptor by displacing [3H]-Pirenzepine binding on rat brain homogenate.More data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:Binding affinity for sigma receptor using 2 nM of [3H]-DTG as radioligand, in membranes from brain minus cerebellumMore data for this Ligand-Target Pair
Affinity DataKi: 15nMAssay Description:In vitro binding affinity for muscarinic M1 receptor by displacing [3H]-Pirenzepine binding on rat brain homogenate.More data for this Ligand-Target Pair
Affinity DataKi: 18nMAssay Description:Evaluated for binding towards Dopamine receptor D2 using [3H]-spiperone as radioligand, in cloned mammalian receptors expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 21nMAssay Description:In vitro binding affinity for muscarinic M1 receptor by displacing [3H]-Pirenzepine binding on rat brain homogenate.More data for this Ligand-Target Pair
Affinity DataKi: 24nMAssay Description:In vitro binding affinity for muscarinic M1 receptor by displacing [3H]-Pirenzepine binding on rat brain homogenate.More data for this Ligand-Target Pair
Affinity DataKi: 26nMAssay Description:Binding towards Dopamine receptor D3 expressed in CHO-K1 cells using [3H]spiperone More data for this Ligand-Target Pair
Affinity DataKi: 26nMAssay Description:In vitro binding affinity for muscarinic M1 receptor by displacing [3H]-Pirenzepine binding on rat brain homogenate.More data for this Ligand-Target Pair
Affinity DataKi: 27nMAssay Description:In vitro binding affinity for muscarinic M1 receptor by displacing [3H]-Pirenzepine binding on rat brain homogenate.More data for this Ligand-Target Pair
Affinity DataKi: 30nMAssay Description:In vitro binding affinity for muscarinic M1 receptor by displacing [3H]-Pirenzepine binding on rat brain homogenate.More data for this Ligand-Target Pair
Affinity DataKi: 32nMAssay Description:In vitro binding affinity for muscarinic M1 receptor by displacing [3H]-Pirenzepine binding on rat brain homogenate.More data for this Ligand-Target Pair
Affinity DataKi: 32nMAssay Description:Binding towards Dopamine receptor D2 using [3H]-spiperone from rat striatal membraneMore data for this Ligand-Target Pair
Affinity DataKi: 32nMAssay Description:Binding towards Dopamine receptor D2 expressed in CHO-K1 cells using [3H]-U-86,170More data for this Ligand-Target Pair
Affinity DataKi: 35nMAssay Description:In vitro binding affinity for muscarinic M1 receptor by displacing [3H]-Pirenzepine binding on rat brain homogenate.More data for this Ligand-Target Pair
Affinity DataKi: 36nMAssay Description:In vitro binding affinity for muscarinic M1 receptor by displacing [3H]-Pirenzepine binding on rat brain homogenate.More data for this Ligand-Target Pair
Affinity DataKi: 37nMAssay Description:In vitro binding affinity for muscarinic M1 receptor by displacing [3H]-Pirenzepine binding on rat brain homogenate.More data for this Ligand-Target Pair
Affinity DataKi: 37nMAssay Description:In vitro binding affinity for muscarinic M1 receptor by displacing [3H]-Pirenzepine binding on rat brain homogenate.More data for this Ligand-Target Pair
Affinity DataKi: 40nMAssay Description:Binding towards Dopamine receptor D2 expressed in CHO-K1 cells using [3H]-U-86,170More data for this Ligand-Target Pair
Affinity DataKi: 40nMAssay Description:In vitro binding affinity for muscarinic M1 receptor by displacing [3H]-Pirenzepine binding on rat brain homogenate.More data for this Ligand-Target Pair
Affinity DataKi: 44nMAssay Description:In vitro binding affinity for muscarinic M1 receptor by displacing [3H]-Pirenzepine binding on rat brain homogenate.More data for this Ligand-Target Pair
Affinity DataKi: 48nMAssay Description:Binding towards dopamine receptor D4 expressed in CHO-K1 cells using [3H]spiperone More data for this Ligand-Target Pair
Affinity DataKi: 57nMAssay Description:In vitro binding affinity for muscarinic M1 receptor by displacing [3H]-Pirenzepine binding on rat brain homogenate.More data for this Ligand-Target Pair
Affinity DataKi: 68nMAssay Description:Binding towards Dopamine receptor D3 expressed in CHO-K1 cells using [3H]spiperone More data for this Ligand-Target Pair
Affinity DataKi: 70nMAssay Description:Evaluated for binding towards Dopamine receptor D2 using [3H]-N-0437 as radioligand from rat striatal membraneMore data for this Ligand-Target Pair
Affinity DataKi: 70nMAssay Description:Binding towards Dopamine receptor D2 expressed in CHO-K1 cells using [3H]-U-86,170More data for this Ligand-Target Pair
Affinity DataKi: 70nMAssay Description:Binding towards Dopamine receptor D3 expressed in CHO-K1 cells using [3H]spiperone More data for this Ligand-Target Pair
Affinity DataKi: 77nMAssay Description:In vitro binding affinity for muscarinic M1 receptor by displacing [3H]-Pirenzepine binding on rat brain homogenate.More data for this Ligand-Target Pair
Affinity DataKi: 84nMAssay Description:In vitro binding affinity for muscarinic M1 receptor by displacing [3H]-Pirenzepine binding on rat brain homogenate.More data for this Ligand-Target Pair
Affinity DataKi: 84nMAssay Description:In vitro binding affinity for muscarinic M1 receptor by displacing [3H]-Pirenzepine binding on rat brain homogenate.More data for this Ligand-Target Pair
Affinity DataKi: 100nMAssay Description:Evaluated for binding towards Dopamine receptor D2 using [3H]-N-0437 as radioligand from rat striatal membraneMore data for this Ligand-Target Pair
Affinity DataKi: 100nMAssay Description:In vitro binding affinity for muscarinic M1 receptor by displacing [3H]-Pirenzepine binding on rat brain homogenate.More data for this Ligand-Target Pair
Affinity DataKi: 117nMAssay Description:Binding towards dopamine receptor D4 expressed in CHO-K1 cells using [3H]spiperone More data for this Ligand-Target Pair
Affinity DataKi: 120nMAssay Description:In vitro binding affinity for muscarinic M1 receptor by displacing [3H]-Pirenzepine binding on rat brain homogenate.More data for this Ligand-Target Pair
Affinity DataKi: 120nMAssay Description:In vitro binding affinity for muscarinic M1 receptor by displacing [3H]-Pirenzepine binding on rat brain homogenate.More data for this Ligand-Target Pair
Affinity DataKi: 130nMAssay Description:Binding towards dopamine receptor D4 expressed in CHO-K1 cells using [3H]spiperone More data for this Ligand-Target Pair
Affinity DataKi: 135nMAssay Description:Evaluated for binding towards Dopamine receptor D2 using [3H]-N-0437 as radioligand from rat striatal membraneMore data for this Ligand-Target Pair
Affinity DataKi: 140nMAssay Description:In vitro binding affinity for muscarinic M1 receptor by displacing [3H]-Pirenzepine binding on rat brain homogenate.More data for this Ligand-Target Pair
Affinity DataKi: 145nMAssay Description:Binding towards Dopamine receptor D2 expressed in CHO-K1 cells using [3H]-U-86,170More data for this Ligand-Target Pair
Affinity DataKi: 158nMAssay Description:Binding towards Dopamine receptor D2 expressed in CHO-K1 cells using [3H]-U-86,170More data for this Ligand-Target Pair