Affinity DataKi: 0.00420nMAssay Description:Ability to inhibit [125I]ET1 binding to human cloned endothelin A receptor expressed on CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.0150nMAssay Description:Ability to inhibit [125I]ET1 binding to human cloned endothelin A receptor expressed on CHO cellsMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Yoshitomi Pharmaceutical Industries
Curated by ChEMBL
Yoshitomi Pharmaceutical Industries
Curated by ChEMBL
Affinity DataKi: 2.90nMAssay Description:Binding affinity towards 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Yoshitomi Pharmaceutical Industries
Curated by ChEMBL
Yoshitomi Pharmaceutical Industries
Curated by ChEMBL
Affinity DataKi: 3.80nMAssay Description:Binding affinity towards 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Yoshitomi Pharmaceutical Industries
Curated by ChEMBL
Yoshitomi Pharmaceutical Industries
Curated by ChEMBL
Affinity DataKi: 4.60nMAssay Description:In vitro inhibition of human trypsin.More data for this Ligand-Target Pair
Affinity DataKi: 5.5nMAssay Description:Binding affinity towards Dopamine receptor D2More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Yoshitomi Pharmaceutical Industries
Curated by ChEMBL
Yoshitomi Pharmaceutical Industries
Curated by ChEMBL
Affinity DataKi: 6nMAssay Description:Binding affinity towards 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Yoshitomi Pharmaceutical Industries
Curated by ChEMBL
Yoshitomi Pharmaceutical Industries
Curated by ChEMBL
Affinity DataKi: 6.40nMAssay Description:In vitro inhibition of human Coagulation factor X.More data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Yoshitomi Pharmaceutical Industries
Curated by ChEMBL
Yoshitomi Pharmaceutical Industries
Curated by ChEMBL
Affinity DataKi: 7.90nMAssay Description:Inhibition of class C beta-lactamase derived from Enterobacter cloacae P99More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Yoshitomi Pharmaceutical Industries
Curated by ChEMBL
Yoshitomi Pharmaceutical Industries
Curated by ChEMBL
Affinity DataKi: 33nMAssay Description:Binding affinity towards 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
TargetSerotonin 2 (5-HT2) receptor(Homo sapiens (Human))
Yoshitomi Pharmaceutical Industries
Curated by ChEMBL
Yoshitomi Pharmaceutical Industries
Curated by ChEMBL
Affinity DataKi: 37nMAssay Description:Inhibition of GC1 extended spectrum class C beta-lactamaseMore data for this Ligand-Target Pair
Affinity DataKi: 41nMAssay Description:Ability to inhibit [125I]-ET-1 binding to human cloned ETB receptors expressed on CHO cellsMore data for this Ligand-Target Pair
TargetSerotonin 2 (5-HT2) receptor(Homo sapiens (Human))
Yoshitomi Pharmaceutical Industries
Curated by ChEMBL
Yoshitomi Pharmaceutical Industries
Curated by ChEMBL
Affinity DataKi: 48nMAssay Description:Inhibition of GC1 extended spectrum class C beta-lactamaseMore data for this Ligand-Target Pair
Affinity DataKi: 49nMAssay Description:Binding affinity towards Dopamine receptor D2More data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Yoshitomi Pharmaceutical Industries
Curated by ChEMBL
Yoshitomi Pharmaceutical Industries
Curated by ChEMBL
Affinity DataKi: 69nMAssay Description:In vitro inhibition of human trypsin.More data for this Ligand-Target Pair
Affinity DataKi: 81nMAssay Description:Ability to inhibit [125I]ET1 binding to human cloned endothelin A receptor expressed on CHO cellsMore data for this Ligand-Target Pair
TargetSerotonin 2 (5-HT2) receptor(Homo sapiens (Human))
Yoshitomi Pharmaceutical Industries
Curated by ChEMBL
Yoshitomi Pharmaceutical Industries
Curated by ChEMBL
Affinity DataKi: 130nMAssay Description:In vitro inhibition of human thrombin.More data for this Ligand-Target Pair
Affinity DataKi: 130nMAssay Description:Ability to inhibit [125I]-ET-1 binding to human cloned ETB receptors expressed on CHO cellsMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Yoshitomi Pharmaceutical Industries
Curated by ChEMBL
Yoshitomi Pharmaceutical Industries
Curated by ChEMBL
Affinity DataKi: 140nMAssay Description:Binding affinity towards 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 140nMAssay Description:Ability to inhibit [125I]-ET-1 binding to human cloned ETB receptors expressed on CHO cellsMore data for this Ligand-Target Pair
TargetSerotonin 2 (5-HT2) receptor(Homo sapiens (Human))
Yoshitomi Pharmaceutical Industries
Curated by ChEMBL
Yoshitomi Pharmaceutical Industries
Curated by ChEMBL
Affinity DataKi: 160nMAssay Description:Inhibition of GC1 extended spectrum class C beta-lactamaseMore data for this Ligand-Target Pair
Affinity DataKi: 170nMAssay Description:Binding affinity towards Dopamine receptor D2More data for this Ligand-Target Pair
Affinity DataKi: 340nMAssay Description:Binding affinity towards Dopamine receptor D2More data for this Ligand-Target Pair
TargetSerotonin 2 (5-HT2) receptor(Homo sapiens (Human))
Yoshitomi Pharmaceutical Industries
Curated by ChEMBL
Yoshitomi Pharmaceutical Industries
Curated by ChEMBL
Affinity DataKi: >1.00E+3nMAssay Description:In vitro inhibition of human Coagulation factor X.More data for this Ligand-Target Pair
TargetSerotonin 2 (5-HT2) receptor(Homo sapiens (Human))
Yoshitomi Pharmaceutical Industries
Curated by ChEMBL
Yoshitomi Pharmaceutical Industries
Curated by ChEMBL
Affinity DataKi: >1.00E+3nMAssay Description:In vitro inhibition of human thrombin.More data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Yoshitomi Pharmaceutical Industries
Curated by ChEMBL
Yoshitomi Pharmaceutical Industries
Curated by ChEMBL
Affinity DataKi: >1.00E+3nMAssay Description:In vitro inhibition of human plasmin.More data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Yoshitomi Pharmaceutical Industries
Curated by ChEMBL
Yoshitomi Pharmaceutical Industries
Curated by ChEMBL
Affinity DataKi: >1.00E+3nMAssay Description:In vitro inhibition of human Coagulation factor X.More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Yoshitomi Pharmaceutical Industries
Curated by ChEMBL
Yoshitomi Pharmaceutical Industries
Curated by ChEMBL
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity towards 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity towards Dopamine receptor D2More data for this Ligand-Target Pair
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity towards Dopamine receptor D2More data for this Ligand-Target Pair
TargetSerotonin 2 (5-HT2) receptor(Homo sapiens (Human))
Yoshitomi Pharmaceutical Industries
Curated by ChEMBL
Yoshitomi Pharmaceutical Industries
Curated by ChEMBL
Affinity DataKi: >1.00E+3nMAssay Description:Inhibition of class C beta-lactamase derived from Enterobacter cloacae P99More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Yoshitomi Pharmaceutical Industries
Curated by ChEMBL
Yoshitomi Pharmaceutical Industries
Curated by ChEMBL
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity towards 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
TargetSerotonin 2 (5-HT2) receptor(Homo sapiens (Human))
Yoshitomi Pharmaceutical Industries
Curated by ChEMBL
Yoshitomi Pharmaceutical Industries
Curated by ChEMBL
Affinity DataKi: >1.00E+3nMAssay Description:Inhibition of GC1 extended spectrum class C beta-lactamaseMore data for this Ligand-Target Pair
TargetSerotonin 2 (5-HT2) receptor(Homo sapiens (Human))
Yoshitomi Pharmaceutical Industries
Curated by ChEMBL
Yoshitomi Pharmaceutical Industries
Curated by ChEMBL
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity towards 5-hydroxytryptamine 2 receptorMore data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Yoshitomi Pharmaceutical Industries
Curated by ChEMBL
Yoshitomi Pharmaceutical Industries
Curated by ChEMBL
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity towards Alpha-1 adrenergic receptorMore data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Yoshitomi Pharmaceutical Industries
Curated by ChEMBL
Yoshitomi Pharmaceutical Industries
Curated by ChEMBL
Affinity DataKi: >1.00E+3nMAssay Description:Inhibition of class C beta-lactamase derived from Enterobacter cloacae P99More data for this Ligand-Target Pair
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity towards Dopamine receptor D2More data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Yoshitomi Pharmaceutical Industries
Curated by ChEMBL
Yoshitomi Pharmaceutical Industries
Curated by ChEMBL
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity towards Alpha-1 adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity towards Dopamine receptor D2More data for this Ligand-Target Pair
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity towards Dopamine receptor D2More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Yoshitomi Pharmaceutical Industries
Curated by ChEMBL
Yoshitomi Pharmaceutical Industries
Curated by ChEMBL
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity towards 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Yoshitomi Pharmaceutical Industries
Curated by ChEMBL
Yoshitomi Pharmaceutical Industries
Curated by ChEMBL
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity towards 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
Affinity DataIC50: <0.00100nMAssay Description:In vitro inhibition of [125 I]ET-1 binding to Endothelin A receptor in porcine aortic membrane.More data for this Ligand-Target Pair
Affinity DataIC50: 0.00110nMAssay Description:In vitro inhibition of [125I]-ET-1 binding to Endothelin A receptor in porcine aortic membrane from endothelial cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 0.00170nMAssay Description:In vitro inhibition of [125I]-ET-1 binding to Endothelin A receptor in porcine aortic membrane from endothelial cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 0.00170nMAssay Description:In vitro inhibition of [125I]-ET-1 binding to Endothelin A receptor in porcine aortic membrane from endothelial cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 0.00250nMAssay Description:In vitro inhibition of [125 I]ET-1 binding to Endothelin A receptor in porcine aortic membrane.More data for this Ligand-Target Pair
Affinity DataIC50: 0.00260nMAssay Description:Ability to inhibit [125I]ET1 binding to endothelin A receptor in porcine aortic membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 0.00390nMAssay Description:In vitro inhibition of [125 I]ET-1 binding to Endothelin A receptor in porcine aortic membrane.More data for this Ligand-Target Pair
Affinity DataIC50: 0.00390nMAssay Description:In vitro inhibition of [125I]-ET-1 binding to Endothelin A receptor in porcine aortic membrane from endothelial cellsMore data for this Ligand-Target Pair