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Found 781 with Last Name = 'newton' and Initial = 'g'
TargetAminopeptidase N(Homo sapiens (Human))
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50570849(CHEMBL4854733)
Affinity DataIC50:  1.5nMAssay Description:Inhibition of APN (unknown origin) using A-AMC as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Homo sapiens (Human))
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50570849(CHEMBL4854733)
Affinity DataIC50:  1.5nMAssay Description:Inhibition of APN (unknown origin) using A-AMC as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(RAT)
Rh£Ne-Poulenc Rorer Central Research

Curated by ChEMBL
LigandPNGBDBM50054959((4aS,4bR,5S,6aS,6bR,9aR)-4b-Fluoro-5-hydroxy-4a,6a...)
Affinity DataIC50:  1.60nMAssay Description:Steroid binding against the rat thymus glucocorticoid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(RAT)
Rh£Ne-Poulenc Rorer Central Research

Curated by ChEMBL
LigandPNGBDBM50054966((4aS,4bR,5S,6aS,6bR,8R,9aR)-4b-Fluoro-5-hydroxy-4a...)
Affinity DataIC50:  1.70nMAssay Description:Steroid binding against the rat thymus glucocorticoid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(RAT)
Rh£Ne-Poulenc Rorer Central Research

Curated by ChEMBL
LigandPNGBDBM50407988(CHEMBL2112857)
Affinity DataIC50:  1.80nMAssay Description:Steroid binding against the rat thymus glucocorticoid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(RAT)
Rh£Ne-Poulenc Rorer Central Research

Curated by ChEMBL
LigandPNGBDBM50054953((4aS,4bR,5S,6aS,6bR,8R,9aR)-4b-Fluoro-5-hydroxy-4a...)
Affinity DataIC50:  2.10nMAssay Description:Steroid binding against the rat thymus glucocorticoid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(RAT)
Rh£Ne-Poulenc Rorer Central Research

Curated by ChEMBL
LigandPNGBDBM50054955((4aS,4bR,5S,6aS,6bR,8R,9aR,12S)-4b,12-Difluoro-5-h...)
Affinity DataIC50:  2.20nMAssay Description:Steroid binding against the rat thymus glucocorticoid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(RAT)
Rh£Ne-Poulenc Rorer Central Research

Curated by ChEMBL
LigandPNGBDBM50054964((4aS,4bR,5S,6aS,6bR,8R,9aR,12S)-4b,12-Difluoro-6b-...)
Affinity DataIC50:  2.20nMAssay Description:Steroid binding against the rat thymus glucocorticoid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(RAT)
Rh£Ne-Poulenc Rorer Central Research

Curated by ChEMBL
LigandPNGBDBM50054961((4aS,4bR,5S,6aS,6bR,9aR,12S)-4b,12-Difluoro-5-hydr...)
Affinity DataIC50:  2.20nMAssay Description:Steroid binding against the rat thymus glucocorticoid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(RAT)
Rh£Ne-Poulenc Rorer Central Research

Curated by ChEMBL
LigandPNGBDBM50369181(TIPREDANE)
Affinity DataIC50:  2.30nMAssay Description:Steroid binding against the rat thymus glucocorticoid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Homo sapiens (Human))
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50570850(CHEMBL4877339)
Affinity DataIC50:  2.30nMAssay Description:Inhibition of APN (unknown origin) using A-AMC as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Homo sapiens (Human))
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50570850(CHEMBL4877339)
Affinity DataIC50:  2.30nMAssay Description:Inhibition of APN (unknown origin) using A-AMC as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(RAT)
Rh£Ne-Poulenc Rorer Central Research

Curated by ChEMBL
LigandPNGBDBM50054960((4aS,4bR,5S,6aS,6bR,8R,9aR,12S)-4b,12-Difluoro-5-h...)
Affinity DataIC50:  2.40nMAssay Description:Steroid binding against the rat thymus glucocorticoid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(RAT)
Rh£Ne-Poulenc Rorer Central Research

Curated by ChEMBL
LigandPNGBDBM50354850(BUDESONIDE | US10869929, Compound Budesonide | US1...)
Affinity DataIC50:  2.90nMAssay Description:Steroid binding against the rat thymus glucocorticoid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidase 1(Dermatophagoides pteronyssinus (European house dus...)
Domainex

Curated by ChEMBL
LigandPNGBDBM50031688(CHEMBL3360299)
Affinity DataIC50:  3nMAssay Description:Inhibition of house dust mite Derp-1 after 20 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidase 1(Dermatophagoides pteronyssinus (European house dus...)
Domainex

Curated by ChEMBL
LigandPNGBDBM50031689(CHEMBL3360298)
Affinity DataIC50:  3nMAssay Description:Inhibition of house dust mite Derp-1 after 20 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(RAT)
Rh£Ne-Poulenc Rorer Central Research

Curated by ChEMBL
LigandPNGBDBM50054952((4aS,4bR,5S,6aS,6bR,8R,9aR)-4b-Fluoro-5-hydroxy-6b...)
Affinity DataIC50:  3.20nMAssay Description:Steroid binding against the rat thymus glucocorticoid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(RAT)
Rh£Ne-Poulenc Rorer Central Research

Curated by ChEMBL
LigandPNGBDBM50054962((4aS,4bR,5S,6aS,6bR,8R,9aR)-4b-Fluoro-6b-fluoromet...)
Affinity DataIC50:  3.30nMAssay Description:Steroid binding against the rat thymus glucocorticoid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(RAT)
Rh£Ne-Poulenc Rorer Central Research

Curated by ChEMBL
LigandPNGBDBM50054963((4aS,4bR,5S,6aS,6bR,8R,9aR)-6b-Ethylsulfanyl-4b-fl...)
Affinity DataIC50:  3.30nMAssay Description:Steroid binding against the rat thymus glucocorticoid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Homo sapiens (Human))
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50076744(CHEMBL3416733)
Affinity DataIC50:  3.60nMAssay Description:Inhibition of APN (unknown origin) using A-AMC as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Homo sapiens (Human))
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50076744(CHEMBL3416733)
Affinity DataIC50:  3.70nMAssay Description:Inhibition of APN (unknown origin) using A-AMC as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidase 1(Dermatophagoides pteronyssinus (European house dus...)
Domainex

Curated by ChEMBL
LigandPNGBDBM50031685(CHEMBL3360301)
Affinity DataIC50:  4nMAssay Description:Inhibition of house dust mite Derp-1 after 20 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidase 1(Dermatophagoides pteronyssinus (European house dus...)
Domainex

Curated by ChEMBL
LigandPNGBDBM50031684(CHEMBL3360302)
Affinity DataIC50:  4nMAssay Description:Inhibition of house dust mite Derp-1 after 20 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidase 1(Dermatophagoides pteronyssinus (European house dus...)
Domainex

Curated by ChEMBL
LigandPNGBDBM50031695(CHEMBL3360292)
Affinity DataIC50:  4nMAssay Description:Inhibition of house dust mite Derp-1 after 20 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidase 1(Dermatophagoides pteronyssinus (European house dus...)
Domainex

Curated by ChEMBL
LigandPNGBDBM50031687(CHEMBL3360300)
Affinity DataIC50:  4nMAssay Description:Inhibition of house dust mite Derp-1 after 20 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(RAT)
Rh£Ne-Poulenc Rorer Central Research

Curated by ChEMBL
LigandPNGBDBM50407989(CHEMBL2112850)
Affinity DataIC50:  4.30nMAssay Description:Steroid binding against the rat thymus glucocorticoid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(RAT)
Rh£Ne-Poulenc Rorer Central Research

Curated by ChEMBL
LigandPNGBDBM50354849(CCI-18781 | Cutivate | FLUTICASONE PROPIONATE | Fl...)
Affinity DataIC50:  5nMAssay Description:Steroid binding against the rat thymus glucocorticoid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidase 1(Dermatophagoides pteronyssinus (European house dus...)
Domainex

Curated by ChEMBL
LigandPNGBDBM50031690(CHEMBL3360297)
Affinity DataIC50:  5nMAssay Description:Inhibition of house dust mite Derp-1 after 20 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(RAT)
Rh£Ne-Poulenc Rorer Central Research

Curated by ChEMBL
LigandPNGBDBM50407990(CHEMBL2112858)
Affinity DataIC50:  5.30nMAssay Description:Steroid binding against the rat thymus glucocorticoid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(RAT)
Rh£Ne-Poulenc Rorer Central Research

Curated by ChEMBL
LigandPNGBDBM50054967((4aS,4bR,5S,6aS,6bR,8R,9aR)-4b-Fluoro-5-hydroxy-6b...)
Affinity DataIC50:  5.5nMAssay Description:Steroid binding against the rat thymus glucocorticoid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidase 1(Dermatophagoides pteronyssinus (European house dus...)
Domainex

Curated by ChEMBL
LigandPNGBDBM50031693(CHEMBL3360294)
Affinity DataIC50:  6nMAssay Description:Inhibition of house dust mite Derp-1 after 20 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidase 1(Dermatophagoides pteronyssinus (European house dus...)
Domainex

Curated by ChEMBL
LigandPNGBDBM50031713(CHEMBL3360282)
Affinity DataIC50:  6nMAssay Description:Inhibition of house dust mite Derp-1 after 20 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidase 1(Dermatophagoides pteronyssinus (European house dus...)
Domainex

Curated by ChEMBL
LigandPNGBDBM50031632(CHEMBL3359790)
Affinity DataIC50:  6nMAssay Description:Inhibition of house dust mite Derp-1 after 20 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidase 1(Dermatophagoides pteronyssinus (European house dus...)
Domainex

Curated by ChEMBL
LigandPNGBDBM50031635(CHEMBL3359786)
Affinity DataIC50:  6nMAssay Description:Inhibition of house dust mite Derp-1 after 20 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidase 1(Dermatophagoides pteronyssinus (European house dus...)
Domainex

Curated by ChEMBL
LigandPNGBDBM103023(US8541363, PVA-039)
Affinity DataIC50:  6.30nMAssay Description:The fluorogenic substrate used for measuring Der p 1 proteolytic activity was 2-aminobenzoylvalylalanylnorleucylseryl-(3-nitro)tyrosinyl aspartamide....More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPeptidase 1(Dermatophagoides pteronyssinus (European house dus...)
Domainex

Curated by ChEMBL
LigandPNGBDBM50031668(CHEMBL3359782)
Affinity DataIC50:  7nMAssay Description:Inhibition of house dust mite Derp-1 after 20 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidase 1(Dermatophagoides pteronyssinus (European house dus...)
Domainex

Curated by ChEMBL
LigandPNGBDBM103022(US8541363, PVA-037)
Affinity DataIC50:  7.85nMAssay Description:The fluorogenic substrate used for measuring Der p 1 proteolytic activity was 2-aminobenzoylvalylalanylnorleucylseryl-(3-nitro)tyrosinyl aspartamide....More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPeptidase 1(Dermatophagoides pteronyssinus (European house dus...)
Domainex

Curated by ChEMBL
LigandPNGBDBM50031711(CHEMBL3360284)
Affinity DataIC50:  8nMAssay Description:Inhibition of house dust mite Derp-1 after 20 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidase 1(Dermatophagoides pteronyssinus (European house dus...)
Domainex

Curated by ChEMBL
LigandPNGBDBM50031719(CHEMBL3359772)
Affinity DataIC50:  8nMAssay Description:Inhibition of house dust mite Derp-1 after 20 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Homo sapiens (Human))
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50570851(CHEMBL4853049)
Affinity DataIC50:  8.60nMAssay Description:Inhibition of APN (unknown origin) using A-AMC as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Homo sapiens (Human))
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50570851(CHEMBL4853049)
Affinity DataIC50:  8.70nMAssay Description:Inhibition of APN (unknown origin) using A-AMC as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeptidase 1(Dermatophagoides pteronyssinus (European house dus...)
Domainex

Curated by ChEMBL
LigandPNGBDBM50031714(CHEMBL3360281)
Affinity DataIC50:  9nMAssay Description:Inhibition of house dust mite Derp-1 after 20 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidase 1(Dermatophagoides pteronyssinus (European house dus...)
Domainex

Curated by ChEMBL
LigandPNGBDBM50031697(CHEMBL3360290)
Affinity DataIC50:  9nMAssay Description:Inhibition of house dust mite Derp-1 after 20 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidase 1(Dermatophagoides pteronyssinus (European house dus...)
Domainex

Curated by ChEMBL
LigandPNGBDBM50031694(CHEMBL3360293)
Affinity DataIC50:  10nMAssay Description:Inhibition of house dust mite Derp-1 after 20 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidase 1(Dermatophagoides pteronyssinus (European house dus...)
Domainex

Curated by ChEMBL
LigandPNGBDBM50031700(CHEMBL3360287)
Affinity DataIC50:  11nMAssay Description:Inhibition of house dust mite Derp-1 after 20 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndoplasmic reticulum aminopeptidase 2(Homo sapiens (Human))
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50076744(CHEMBL3416733)
Affinity DataIC50:  11nMAssay Description:Inhibition of recombinant human ERAP2 using R-AMC as substrate incubated for 5 to 10 mins by fluorescence based assayMore data for this Ligand-Target Pair
TargetPeptidase 1(Dermatophagoides pteronyssinus (European house dus...)
Domainex

Curated by ChEMBL
LigandPNGBDBM50031682(CHEMBL3359775)
Affinity DataIC50:  12nMAssay Description:Inhibition of house dust mite Derp-1 after 20 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(RAT)
Rh£Ne-Poulenc Rorer Central Research

Curated by ChEMBL
LigandPNGBDBM50054957((4aS,4bR,5S,6aS,6bR,8R,9aR)-4b-Fluoro-5-hydroxy-4a...)
Affinity DataIC50:  12nMAssay Description:Steroid binding against the rat thymus glucocorticoid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidase 1(Dermatophagoides pteronyssinus (European house dus...)
Domainex

Curated by ChEMBL
LigandPNGBDBM103021(US8541363, PVA-038)
Affinity DataIC50:  13nMAssay Description:Inhibition of house dust mite Derp-1 after 20 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidase 1(Dermatophagoides pteronyssinus (European house dus...)
Domainex

Curated by ChEMBL
LigandPNGBDBM50031673(CHEMBL3359780)
Affinity DataIC50:  13nMAssay Description:Inhibition of house dust mite Derp-1 after 20 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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